flunitrazepam and phenobarbital

flunitrazepam has been researched along with phenobarbital in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-199016 (55.17)18.7374
1990's9 (31.03)18.2507
2000's3 (10.34)29.6817
2010's1 (3.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Deweer, E1
Delvaux, V; Devroye, Y; Taziaux, P1
Haefely, W; Polc, P1
Jovanović, UJ1
Cantanna, R; da Rin Betta, V1
Allan, AM; Baier, LD; Zhang, X1
Gallaher, EJ; Phillips, TJ1
Allan, AM; Draski, LJ; Mayes, GG1
Breimer, DD; de Boer, AG; van Hoogdalem, E1
Machen, VL; Swaiman, KF1
Fares, F; Gavish, M; Pick, CG; Weizman, A; Yanai, J2
Allan, AM; Gallaher, EJ; Gionet, SE; Harris, RA1
Endo, Y; Kokubu, M; Ohtomo, F; Shinya, N1
Fanelli, RJ; Iadarola, MJ; McNamara, JO; Wilson, WA1
Garrett, KM; Tabakoff, B1
Laird, H; Mimaki, T; Yabuuchi, H; Yamamura, HI1
Barbi, S; Beccia, F; Ferraro, M; Pala, F; Sabato, AF1
Garrett, KM; Liljequist, S; Tabakoff, B1
Costa, MF; Fages, C; Gonnard, P; Rolland, B; Tardy, M1
Braestrup, C; Kehr, W; Nielsen, M; Paschelke, G; Petersen, EN1
Dasheiff, RM; Fanelli, RJ; Kraus, VM; McNamara, JO1
Liljequist, S; Tabakoff, B1
Fueta, Y; Janjua, NA; Mita, T; Murai, Y; Ohmori, O; Ohno, K; Ono, T1
van Luijtelaar, EL1
Lu, YQ; Yu, R1

Reviews

1 review(s) available for flunitrazepam and phenobarbital

ArticleYear
Pharmacokinetics of rectal drug administration, Part I. General considerations and clinical applications of centrally acting drugs.
    Clinical pharmacokinetics, 1991, Volume: 21, Issue:1

    Topics: Administration, Rectal; Antiemetics; Atropine; Carbamazepine; Clonazepam; Delayed-Action Preparations; Diazepam; Flunitrazepam; Humans; Hydromorphone; Intestinal Absorption; Methadone; Methohexital; Midazolam; Morphine; Pharmacokinetics; Phenobarbital; Valproic Acid

1991

Trials

3 trial(s) available for flunitrazepam and phenobarbital

ArticleYear
[Can the severe and chronic insomniac escape from barbiturates? A double blind, long-term clinical study of a new hypnotic].
    Bruxelles medical, 1975, Volume: 55, Issue:3

    Topics: Anti-Anxiety Agents; Clinical Trials as Topic; Drug Evaluation; Flunitrazepam; Humans; Phenobarbital; Placebos; Sleep Initiation and Maintenance Disorders

1975
[Comparison between a new hypnotic Flunitrazepam (Ro 5-4200), and a barbiturate by double-blind method].
    Revue medicale de Liege, 1976, Aug-15, Volume: 31, Issue:16

    Topics: Anti-Anxiety Agents; Clinical Trials as Topic; Drug Evaluation; Flunitrazepam; Humans; Hypnotics and Sedatives; Phenobarbital

1976
[Vigilance pattern and sleep quality under the effect of flunitrazepam].
    Klinische Anasthesiologie und Intensivtherapie, 1978, Issue:17

    Topics: Adult; Anti-Anxiety Agents; Attention; Clinical Trials as Topic; Diazepam; Electroencephalography; Female; Flunitrazepam; Humans; Male; Phenobarbital; Placebos; Sleep; Sleep Wake Disorders

1978

Other Studies

25 other study(ies) available for flunitrazepam and phenobarbital

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Effects of two benzodiazepines, phenobarbitone, and baclofen on synaptic transmission in the cat cuneate nucleus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1976, Volume: 294, Issue:2

    Topics: Aminobutyrates; Aminooxyacetic Acid; Animals; Anti-Anxiety Agents; Baclofen; Bicuculline; Cats; Diazepam; Drug Interactions; Evoked Potentials; Flunitrazepam; Glutamate Decarboxylase; Medulla Oblongata; Neural Inhibition; Phenobarbital; Picrotoxin; Propionates; Semicarbazides; Synapses; Synaptic Transmission

1976
[Tetanus: 10 years of experience].
    Minerva anestesiologica, 1978, Volume: 44, Issue:12

    Topics: Adolescent; Adult; Aged; Child; Child, Preschool; Diazepam; Female; Flunitrazepam; Humans; Infant; Intubation, Intratracheal; Male; Middle Aged; Pancuronium; Phenobarbital; Tetanus; Tracheotomy

1978
Effects of lorazepam tolerance and withdrawal on GABAA receptor-operated chloride channels.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:2

    Topics: Animals; Appetite Depressants; Binding Sites; Brain; Carbolines; Chloride Channels; Chlorides; Diazepam; Drug Interactions; Ethanol; Flunitrazepam; Ion Channels; Lorazepam; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Phenobarbital; Receptors, GABA-A

1992
Locomotor responses to benzodiazepines, barbiturates and ethanol in diazepam-sensitive (DS) and -resistant (DR) mice.
    Psychopharmacology, 1992, Volume: 107, Issue:1

    Topics: Analysis of Variance; Animals; Diazepam; Dose-Response Relationship, Drug; Ethanol; Female; Flumazenil; Flunitrazepam; Male; Mice; Motor Activity; Pentobarbital; Phenobarbital

1992
gamma-Aminobutyric acid-activated chloride channels in rats selectively bred for differential acute sensitivity to alcohol.
    Alcoholism, clinical and experimental research, 1991, Volume: 15, Issue:2

    Topics: Alcohol Drinking; Animals; Chloride Channels; Diazepam; Female; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Proteins; Muscimol; Pentobarbital; Phenobarbital; Phenotype; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Selection, Genetic

1991
Effects of phenobarbital and phenytoin on cortical glial cells in culture.
    Brain & development, 1991, Volume: 13, Issue:4

    Topics: Animals; Animals, Newborn; Benzodiazepinones; Cells, Cultured; Cerebral Cortex; Flunitrazepam; Mice; Neuroglia; Phenobarbital; Phenytoin; Radioligand Assay

1991
Effect of prenatal and neonatal chronic exposure to phenobarbital on central and peripheral benzodiazepine receptors.
    Brain research, 1990, Jan-01, Volume: 506, Issue:1

    Topics: Aging; Animals; Brain; Female; Flunitrazepam; Male; Mice; Muscimol; Phenobarbital; Pregnancy; Prenatal Exposure Delayed Effects; Receptors, GABA-A

1990
Genetic selection for benzodiazepine ataxia produces functional changes in the gamma-aminobutyric acid receptor chloride channel complex.
    Brain research, 1988, Jun-14, Volume: 452, Issue:1-2

    Topics: Animals; Ataxia; Chlorides; Diazepam; Ethanol; Flunitrazepam; Ion Channels; Isoxazoles; Mice; Muscimol; Phenobarbital; Receptors, GABA-A; Time Factors

1988
Chronic phenobarbital administration affects GABA and benzodiazepine receptors in the brain and periphery.
    European journal of pharmacology, 1989, Oct-10, Volume: 169, Issue:2-3

    Topics: Animals; Brain Chemistry; Flunitrazepam; Hippocampus; In Vitro Techniques; Isoquinolines; Kidney; Male; Membranes; Mice; Muscimol; Myocardium; Olfactory Bulb; Peripheral Nerves; Phenobarbital; Receptors, GABA-A

1989
Relationship between the pharmacological effects of benzodiazepines and their in vivo binding sites in the brain of rats.
    Higashi Nihon shigaku zasshi, 1989, Volume: 8, Issue:2

    Topics: Animals; Brain Stem; Cerebral Cortex; Diazepam; Flunitrazepam; Hypothalamus; Phenobarbital; Rats; Receptors, GABA-A

1989
Comparison of the effects of diphenylbarbituric acid, phenobarbital, pentobarbital and secobarbital on GABA-mediated inhibition and benzodiazepine binding.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:1

    Topics: Animals; Benzodiazepines; Electrophysiology; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Male; Pentobarbital; Phenobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Secobarbital; Time Factors

1985
Effects of prenatal phenobarbital on benzodiazepine receptor development.
    Journal of neurochemistry, 1986, Volume: 47, Issue:4

    Topics: Animals; Brain; Cerebellum; Diencephalon; Female; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Phenobarbital; Pregnancy; Prenatal Exposure Delayed Effects; Pyridazines; Receptors, GABA-A; Telencephalon

1986
Effects of seizures and antiepileptic drugs on benzodiazepine receptors in rat brain.
    Pediatric pharmacology (New York, N.Y.), 1984, Volume: 4, Issue:4

    Topics: Acoustic Stimulation; Aminooxyacetic Acid; Animals; Anticonvulsants; Brain; Cerebral Cortex; Flunitrazepam; Male; Phenobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Valproic Acid

1984
The effect of five drugs in coma doses on neurotransmitter amino acids in the brains of guinea pigs.
    Resuscitation, 1983, Volume: 10, Issue:4

    Topics: Amino Acids; Animals; Brain; Brain Chemistry; Central Nervous System Agents; Central Nervous System Depressants; Diazepam; Flunitrazepam; Guinea Pigs; Neurotransmitter Agents; Phenobarbital; Phenytoin; Pregnanediones

1983
Specific effects of chronic phenobarbital administration on high- and low-affinity benzodiazepine receptors in mouse cerebellum and forebrain.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Animals; Anti-Anxiety Agents; Brain; Cerebellum; Flunitrazepam; Kinetics; Membranes; Mice; Mice, Inbred C57BL; Phenobarbital; Pyridazines; Receptors, GABA-A; Time Factors

1984
Benzodiazepine receptors on primary cultures of mouse astrocytes.
    Journal of neurochemistry, 1981, Volume: 36, Issue:4

    Topics: Animals; Anticonvulsants; Astrocytes; Binding, Competitive; Cell Membrane; Cells, Cultured; Diazepam; Flunitrazepam; Mice; Phenobarbital; Receptors, Drug; Receptors, GABA-A

1981
Does the reversal of the anticonflict effect of phenobarbital by beta-CCE and FG 7142 indicate benzodiazepine receptor-mediated anxiogenic properties?
    European journal of pharmacology, 1982, Aug-27, Volume: 82, Issue:3-4

    Topics: Animals; Anxiety; Carbolines; Conflict, Psychological; Diazepam; Flunitrazepam; Humans; Indoles; Male; Phenobarbital; Punishment; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A

1982
Benzodiazepine receptor declines in hippocampal formation following limbic seizures.
    Brain research, 1983, Oct-31, Volume: 277, Issue:2

    Topics: Afferent Pathways; Animals; Diazepam; Dominance, Cerebral; Flunitrazepam; Hippocampus; Limbic System; Male; Phenobarbital; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1983
Bicuculline-produced regional differences in the modulation of 35S-TBPS binding by GABA, pentobarbital and diazepam in mouse cerebellum and cortex.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Phenobarbital; Receptors, GABA-A

1993
Granule cell disinhibition in dentate gyrus of genetically seizure susceptible El mice.
    Brain research, 1997, Jan-16, Volume: 745, Issue:1-2

    Topics: Aging; Animals; Anticonvulsants; Bicuculline; Chromatography, High Pressure Liquid; Dentate Gyrus; Electrophysiology; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Phenobarbital; Seizures

1997
Spike-wave discharges and sleep spindles in rats.
    Acta neurobiologiae experimentalis, 1997, Volume: 57, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Anti-Anxiety Agents; Clonidine; Electroencephalography; Flunitrazepam; Frontal Lobe; Hypnotics and Sedatives; Male; Phenobarbital; Rats; Rats, Inbred Strains; Sleep; Thalamus

1997
Synergistic protection of allopregnanolone and phenobarbital against maximal electroshock seizures in mice.
    Acta pharmacologica Sinica, 2001, Volume: 22, Issue:4

    Topics: Animals; Anticonvulsants; Cerebral Cortex; Drug Synergism; Electroshock; Flunitrazepam; GABA Modulators; Male; Mice; Mice, Inbred C57BL; Phenobarbital; Pregnanolone; Seizures

2001