flunitrazepam and naloxone

flunitrazepam has been researched along with naloxone in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-199014 (56.00)18.7374
1990's6 (24.00)18.2507
2000's3 (12.00)29.6817
2010's2 (8.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Chang, TK; Ensom, MH; Kiang, TK1
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Dick, W; Knoche, E; Milewski, P; Traub, E1
Dick, W; Milewski, P1
Baasch, K; Reist, F; Schaer, H1
Fuji, K; Miyamoto, K; Okuda, T; Suekane, K; Wakita, K1
Achtari, R; Baasch, K; Schaer, H1
Hofer, P; Scollo-Lavizzari, G1
Pan, HS; Penney, JB; Young, AB1
Bidlack, JM; Denton, RR1
Gibert-Rahola, J; Leonsegui, I; Maldonado, R; Micó, JA; Saavedra, MC1
Bittiger, H; Dooley, DJ1
Pitt-Miller, P1
Bhanot, R; Eskes, G; Moger, WH; Wilkinson, DA; Wilkinson, M1
Agoston, S; Langrehr, D; Schmutzler, S; Uges, D1
Castellano, C; Filibeck, U; Pavone, F1
Bhanot, R; Brawer, JR; Wilkinson, DA; Wilkinson, M1
Chen, A; Culling, A; Davis, TP; Schoemaker, H; Yamamura, HI1
Acuña-Castroviejo, D; Castillo, JL; del Aguila, CM; Fernández, B; Gomar, MD2
Ackermann, RF; Chugani, HT; Engel, J; Rocha, L1
Chugani, HT; Engel, J; Rocha, L; Tatsukawa, K1
Kolik, LG; Nadorova, AV; Seredenin, SB; Yarkova, MA1

Reviews

1 review(s) available for flunitrazepam and naloxone

ArticleYear
UDP-glucuronosyltransferases and clinical drug-drug interactions.
    Pharmacology & therapeutics, 2005, Volume: 106, Issue:1

    Topics: Clinical Trials as Topic; Drug Interactions; Enzyme Activation; Enzyme Induction; Glucuronides; Glucuronosyltransferase; Humans; Pharmaceutical Preparations; Pharmacogenetics; Polymorphism, Genetic

2005

Trials

4 trial(s) available for flunitrazepam and naloxone

ArticleYear
[Clinical studies on the usefulness of naloxone after short lasting anaesthesias with narcotic analgesics (author's transl)].
    Der Anaesthesist, 1978, Volume: 27, Issue:6

    Topics: Analgesics, Opioid; Anesthesia, General; Dose-Response Relationship, Drug; Female; Fentanyl; Flunitrazepam; Humans; Male; Naloxone; Pentazocine; Respiration Disorders

1978
[Administration and dosage of flunitrazepam in combination with analgesics].
    Klinische Anasthesiologie und Intensivtherapie, 1978, Issue:17

    Topics: Adult; Aged; Analgesics; Anesthesia; Anti-Anxiety Agents; Blood Gas Analysis; Blood Pressure; Clinical Trials as Topic; Drug Combinations; Female; Fentanyl; Flunitrazepam; Humans; Male; Middle Aged; Naloxone; Pentazocine; Preanesthetic Medication; Pulse; Pupil; Respiration; Time Factors

1978
[Respiratory depression after fentanyl and antagonism by naloxone (author's transl)].
    Der Anaesthesist, 1978, Volume: 27, Issue:6

    Topics: Adolescent; Adult; Aged; Anesthesia, General; Fentanyl; Flunitrazepam; Humans; Meperidine; Middle Aged; Naloxone; Pulmonary Ventilation; Respiration Disorders; Unconsciousness; Wakefulness

1978
[Antagonism of flunitrazepam and fentanyl by flumazenil, naloxone or nalbuphine].
    Der Anaesthesist, 1990, Volume: 39, Issue:1

    Topics: Adult; Double-Blind Method; Fentanyl; Flumazenil; Flunitrazepam; Humans; Middle Aged; Morphinans; Nalbuphine; Naloxone; Randomized Controlled Trials as Topic; Respiratory Insufficiency

1990

Other Studies

20 other study(ies) available for flunitrazepam and naloxone

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Suppressant effects of midazolam on responses of spinal dorsal horn neurones in rabbits.
    Neuropharmacology, 1992, Volume: 31, Issue:1

    Topics: Animals; Bradykinin; Decerebrate State; Flunitrazepam; Microelectrodes; Midazolam; Naloxone; Neurons; Pain; Rabbits; Spinal Cord

1992
Benzodiazepine antagonist Ro 15-1788 in self-poisoning. Diagnostic and therapeutic use.
    Archives of internal medicine, 1985, Volume: 145, Issue:4

    Topics: Adult; Aged; Anti-Anxiety Agents; Antidotes; Benzodiazepinones; Coma; Diazepam; Electroencephalography; Female; Flumazenil; Flunitrazepam; Humans; Male; Middle Aged; Naloxone; Suicide, Attempted

1985
Gamma-aminobutyric acid and benzodiazepine receptor changes induced by unilateral 6-hydroxydopamine lesions of the medial forebrain bundle.
    Journal of neurochemistry, 1985, Volume: 45, Issue:5

    Topics: Animals; Autoradiography; Benzodiazepines; Brain; Dopamine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Flunitrazepam; Hydroxydopamines; Kinetics; Muscimol; Naloxone; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spiperone; Tritium

1985
A monoclonal antibody capable of modulating opioid binding to rat neural membranes.
    The Journal of biological chemistry, 1985, Dec-15, Volume: 260, Issue:29

    Topics: Animals; Antibodies, Monoclonal; Cell Line; Cyclazocine; Dihydromorphine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Flunitrazepam; Immunoglobulin M; Kinetics; Male; Mice; Mice, Inbred BALB C; Molecular Weight; Naloxone; Narcotics; Nerve Tissue; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Opioid

1985
Comparative study in mice of flunitrazepam vs. diazepam on morphine withdrawal syndrome.
    Progress in neuro-psychopharmacology & biological psychiatry, 1988, Volume: 12, Issue:6

    Topics: Animals; Behavior, Animal; Diazepam; Flunitrazepam; Male; Mice; Mice, Inbred Strains; Morphine; Morphine Dependence; Naloxone; Substance Withdrawal Syndrome

1988
Characterization of neurotransmitter receptors in the rat hippocampal formation.
    Journal of neurochemistry, 1982, Volume: 38, Issue:6

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Dihydroalprenolol; Flunitrazepam; Hippocampus; Kinetics; Male; Naloxone; Prazosin; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter

1982
Reversal of flunitrazepam-induced drowsiness with naloxone.
    Anaesthesia, 1982, Volume: 37, Issue:12

    Topics: Adult; Anesthesia, Intravenous; Anti-Anxiety Agents; Female; Flunitrazepam; Humans; Male; Middle Aged; Naloxone; Sleep Stages

1982
Photoperiodic modification of opiate but not beta-adrenergic or benzodiazepine binding sites in hamster brain.
    Biology of reproduction, 1983, Volume: 28, Issue:4

    Topics: Alprenolol; Animals; Anti-Anxiety Agents; Binding Sites; Body Weight; Brain; Cricetinae; Dihydroalprenolol; Flunitrazepam; Male; Naloxone; Organ Size; Periodicity; Photic Stimulation; Testis

1983
[Rohypnol poisoning as a cause of postanesthetic coma and the success of 4-aminopyridine therapy].
    Der Anaesthesist, 1984, Volume: 33, Issue:6

    Topics: 4-Aminopyridine; Adult; Aminopyridines; Anesthesia; Coma; Female; Flunitrazepam; Humans; Naloxone; Physostigmine; Postoperative Complications

1984
Naltrexone-reversible effects of flunitrazepam on locomotor activity and passive avoidance behaviour in mice.
    European journal of pharmacology, 1984, Sep-03, Volume: 104, Issue:1-2

    Topics: Animals; Avoidance Learning; Flunitrazepam; Male; Memory; Mice; Mice, Inbred C57BL; Motor Activity; Naloxone; Naltrexone

1984
Prolonged estrogen treatment induces changes in opiate, benzodiazepine and beta-adrenergic binding sites in female rat hypothalamus.
    Brain research bulletin, 1983, Volume: 11, Issue:3

    Topics: Amygdala; Animals; Binding Sites; Cerebral Cortex; Dihydroalprenolol; Estradiol; Female; Flunitrazepam; Hypothalamus; Naloxone; Rats; Rats, Inbred Strains

1983
Isolation and characterization of in vitro endorphin metabolism in the brain.
    Proceedings of the Western Pharmacology Society, 1982, Volume: 25

    Topics: Animals; Brain; Chromatography, High Pressure Liquid; Endorphins; Flunitrazepam; Humans; In Vitro Techniques; Naloxone; Quinuclidinyl Benzilate; Rats; Spiperone

1982
Melatonin counteracts pinealectomy-dependent decreases in rat brain [3H]flunitrazepam binding through an opioid mechanism.
    Neuroscience letters, 1993, Dec-24, Volume: 164, Issue:1-2

    Topics: Animals; Brain; Endorphins; Flunitrazepam; Ganglionectomy; Injections, Intraventricular; Male; Melatonin; Membranes; Naloxone; Pineal Gland; Rats; Rats, Wistar; Superior Cervical Ganglion; Sympathetic Nervous System

1993
Chronic pretreatment with naloxone modifies benzodiazepine receptor binding in amygdaloid kindled rats.
    Epilepsy research, 1994, Volume: 17, Issue:2

    Topics: Amygdala; Animals; Autoradiography; Electric Stimulation; Electroencephalography; Flunitrazepam; Kindling, Neurologic; Male; Naloxone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1994
Benzodiazepine receptor binding following chronic treatment with naloxone, morphine and met-enkephalin in normal rats.
    Brain research, 1993, May-28, Volume: 612, Issue:1-2

    Topics: Animals; Brain; Densitometry; Enkephalin, Methionine; Flunitrazepam; Injections, Intraperitoneal; Injections, Intraventricular; Male; Morphine; Naloxone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1993
Intracerebroventricular injection of naloxone blocks melatonin-dependent brain [3H]flunitrazepam binding.
    Neuroreport, 1993, Volume: 4, Issue:7

    Topics: Adrenal Cortex Hormones; Animals; beta-Endorphin; Cerebral Cortex; Dose-Response Relationship, Drug; Flunitrazepam; Hypophysectomy; In Vitro Techniques; Injections, Intraventricular; Male; Melatonin; Naloxone; Rats; Rats, Wistar; Receptors, GABA-A

1993
Effects of phenazepam on the behavior of C57BL/6 and BALB/c mice in the open field test after naloxone pretreatment.
    Bulletin of experimental biology and medicine, 2013, Volume: 155, Issue:3

    Topics: Animals; Benzodiazepines; Exploratory Behavior; Flunitrazepam; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Motor Activity; Naloxone; Radioligand Assay; Species Specificity; Statistics, Nonparametric; Stress, Psychological

2013