flunitrazepam and isoxazoles

flunitrazepam has been researched along with isoxazoles in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19909 (60.00)18.7374
1990's3 (20.00)18.2507
2000's2 (13.33)29.6817
2010's1 (6.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Karobath, M; Lippitsch, M1
Karasawa, T; Mimaki, T; Suzuki, Y; Tagawa, T; Yabuuchi, H1
Damgaard, I; Saederup, E; Schousboe, A; Squires, RF1
Allan, AM; Gallaher, EJ; Gionet, SE; Harris, RA1
Chweh, AY; Kupferberg, HJ; Swinyard, EA; Wolf, HH1
Shavrin, AS; Zharkovskaia, TA; Zharkovskiĭ, AM1
Zarkovsky, AM1
Karobath, M; Supavilai, P2
Benson, DI; Klepner, CA; Squires, RF1
Saederup, E; Squires, RF1
Alkana, RL; Bolger, MB; Brinton, RD; Davies, DL; Finn, DA1
Blednov, YA; Boehm, SL; Harris, RA; Peden, L1
Brust, P; Deuther-Conrad, W; Ebert, B; Friemel, A; Hutson, PH; Nieber, K1
France, CP; Gerak, LR1

Other Studies

15 other study(ies) available for flunitrazepam and isoxazoles

ArticleYear
THIP and isoguvacine are partial agonists of GABA-stimulated benzodiazepine receptor binding.
    European journal of pharmacology, 1979, Oct-15, Volume: 58, Issue:4

    Topics: Animals; Benzodiazepines; Cerebral Cortex; Drug Synergism; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Isonicotinic Acids; Isoxazoles; Muscimol; Oxazoles; Rats; Receptors, Drug

1979
Interaction of zonisamide with benzodiazepine and GABA receptors in rat brain.
    Medical journal of Osaka University, 1990, Volume: 39, Issue:1-4

    Topics: Animals; Anticonvulsants; Brain; Dose-Response Relationship, Drug; Flunitrazepam; Isoxazoles; Male; Muscimol; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-A; Synaptic Membranes; Zonisamide

1990
Development of benzodiazepine and picrotoxin (t-butylbicyclophosphorothionate) binding sites in rat cerebellar granule cells in culture.
    Journal of neurochemistry, 1990, Volume: 54, Issue:2

    Topics: Animals; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cells, Cultured; Cerebellum; Flunitrazepam; Granulocytes; Isoxazoles; Pyrazoles; Pyridazines; Pyridines; Rats

1990
Genetic selection for benzodiazepine ataxia produces functional changes in the gamma-aminobutyric acid receptor chloride channel complex.
    Brain research, 1988, Jun-14, Volume: 452, Issue:1-2

    Topics: Animals; Ataxia; Chlorides; Diazepam; Ethanol; Flunitrazepam; Ion Channels; Isoxazoles; Mice; Muscimol; Phenobarbital; Receptors, GABA-A; Time Factors

1988
Effect of GABA agonists on the neurotoxicity and anticonvulsant activity of benzodiazepines.
    Life sciences, 1985, Feb-25, Volume: 36, Issue:8

    Topics: Animals; Anticonvulsants; Benzodiazepines; Drug Synergism; Electroshock; Flunitrazepam; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Muscimol; Nervous System; Receptors, GABA-A

1985
[Changes in the ligand affinity of benzodiazepine receptors in the presence of 4,5,6,7-tetrahydroisoxazolo(5,4-c)pyridin-3-ol (THIP)].
    Biulleten' eksperimental'noi biologii i meditsiny, 1987, Volume: 103, Issue:2

    Topics: Animals; Brain; Depression, Chemical; Dose-Response Relationship, Drug; Flunitrazepam; In Vitro Techniques; Isoxazoles; Ligands; Male; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Bicuculline-sensitive and insensitive effects of THIP on the binding of [3H]flunitrazepam.
    Neuropharmacology, 1987, Volume: 26, Issue:7A

    Topics: Animals; Bicuculline; Brain; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Isoxazoles; Male; Osmolar Concentration; Oxazoles; Rats; Rats, Inbred Strains; Sodium Chloride; Tritium

1987
Action of pyrazolopyridines as modulators of [3H]flunitrazepam binding to the gaba/benzodiazepine receptor complex of the cerebellum.
    European journal of pharmacology, 1981, Mar-12, Volume: 70, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Bicuculline; Binding Sites; Cerebellum; Chlorides; Etazolate; Flunitrazepam; Isoxazoles; Male; Muscimol; Nicotinic Acids; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Tritium

1981
The effect of temperature and chloride ions on the stimulation of [3H]flunitrazepam binding by the muscimol analogues THIP and piperidine-4-sulfonic acid.
    Neuroscience letters, 1980, Oct-02, Volume: 19, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; Isonicotinic Acids; Isoxazoles; Oxazoles; Piperidines; Rats; Stimulation, Chemical; Temperature; Tritium

1980
Multiple benzodiazepine receptor complexes: some benzodiazepine recognition sites are coupled to GABA receptors and ionophores.
    Advances in biochemical psychopharmacology, 1980, Volume: 21

    Topics: Animals; Anions; Benzodiazepines; Bicuculline; Brain; Buffers; Flunitrazepam; gamma-Aminobutyric Acid; Haplorhini; Hot Temperature; Ionophores; Isonicotinic Acids; Isoxazoles; Macromolecular Substances; Papio; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter

1980
gamma-aminobutyric acid receptors modulate cation binding sites coupled to independent benzodiazepine, picrotoxin, and anion binding sites.
    Molecular pharmacology, 1982, Volume: 22, Issue:2

    Topics: Animals; Binding Sites; Brain; Calcium Chloride; Electrolytes; Flunitrazepam; In Vitro Techniques; Isoxazoles; Picrotoxin; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Sodium Chloride

1982
In vivo and in vitro hyperbaric studies in mice suggest novel sites of action for ethanol.
    Psychopharmacology, 1999, Volume: 141, Issue:4

    Topics: Allosteric Regulation; Analysis of Variance; Animals; Diazepam; Ethanol; Flunitrazepam; GABA Modulators; Hyperbaric Oxygenation; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Pentobarbital; Pregnanolone; Receptors, GABA-A

1999
Deletion of the fyn-kinase gene alters sensitivity to GABAergic drugs: dependence on beta2/beta3 GABAA receptor subunits.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 309, Issue:3

    Topics: Animals; Binding Sites; Flunitrazepam; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Gene Deletion; Isoxazoles; Mice; Protein Subunits; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fyn; Receptors, GABA-A; Reflex; Tritium

2004
Postnatal development and kinetics of [3H]gaboxadol binding in rat brain: in vitro homogenate binding and quantitative autoradiography.
    Brain research, 2007, Sep-19, Volume: 1170

    Topics: Aging; Animals; Animals, Newborn; Autoradiography; Binding, Competitive; Brain; Brain Chemistry; Flunitrazepam; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Subcellular Fractions

2007
Discriminative stimulus effects of pregnanolone in rhesus monkeys.
    Psychopharmacology, 2014, Volume: 231, Issue:1

    Topics: Animals; Conditioning, Operant; Data Interpretation, Statistical; Discrimination, Psychological; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Flumazenil; Flunitrazepam; GABA Modulators; Gonadal Steroid Hormones; Hypnotics and Sedatives; Isoxazoles; Macaca mulatta; Male; Midazolam; Pregnanolone; Receptors, GABA-A; Reinforcement Schedule

2014