flunitrazepam has been researched along with cl 218872 in 67 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 50 (74.63) | 18.7374 |
1990's | 13 (19.40) | 18.2507 |
2000's | 4 (5.97) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Cook, JM; Cox, ED; Diaz-Arauzo, H; Harris, B; Huang, Q; Ma, C; McKernan, R; Reddy, MS; Skolnick, P | 1 |
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S | 1 |
Hirouchi, M; Kohno, Y; Kuriyama, K; Mizutani, H | 1 |
Bacon, E; de Barry, J; Gombos, G | 1 |
De Luca, C; De Medici, D; Massotti, M | 1 |
Ito, M; Mikawa, H; Mutoh, K; Oguro, K; Shiraishi, H; Shirasaka, Y; Tsuda, H | 1 |
Damgaard, I; Saederup, E; Schousboe, A; Squires, RF | 1 |
De Robertis, E; de Stein, ML; Medina, JH | 1 |
Moffett, JR; Namboodiri, A; Neale, JH | 1 |
Lüddens, H; Pritchett, DB; Seeburg, PH | 1 |
Faull, RL; Villiger, JW | 2 |
Benavides, J; Dubois, A; Morel, E; Peny, B; Perrault, G; Scatton, B; Zivkovic, B | 1 |
Cortés, R; Palacios, JM; Probst, A; Zezula, J | 1 |
Arbilla, S; Langer, SZ | 1 |
Garrett, KM; Tabakoff, B | 2 |
Barnett, A; Golden, JS; Wamsley, JK; Yamamura, HI | 2 |
Komiskey, HL | 1 |
Kuriyama, K; Taguchi, J | 1 |
Massotti, M; Valerio, A | 1 |
Beer, B; Garrett, KM; Lippa, AS; Meyerson, LR; Tabakoff, B; Wennogle, LP | 1 |
Biggio, G; Corda, MG; Porceddu, ML; Sanna, E | 1 |
Kito, S; Miyoshi, R; Mizuno, K | 1 |
Sieghart, W | 3 |
Eichinger, A; Sieghart, W | 2 |
Bobillier, P; Kopp, N; Manchon, M; Miachon, S | 1 |
Herblin, WF | 1 |
Hyde, L; Khatami, S; Salafsky, B; Shibuya, T; Watanabe, Y | 1 |
Eichinger, A; Möhler, H; Richards, JG; Sieghart, W | 1 |
Faull, RL; Holford, NH; Villiger, JW | 1 |
Drexler, G; Karobath, M; Sieghart, W; Supavilai, P | 1 |
Gee, KW; Morelli, M; Yamamura, HI | 1 |
Beer, B; Coupet, J; Dubnick, B; Greenblatt, EN; Klepner, CA; Lippa, AS | 1 |
Drexler, G; Mayer, A; Sieghart, W | 1 |
Goldberg, ME; Malick, JB; Patel, JB; Salama, AI | 1 |
Gee, KW; Yamamura, HI | 2 |
Keane, P; Morre, M | 1 |
Pan, HS; Penney, JB; Young, AB | 1 |
Jones, BJ; Oakley, NR; Straughan, DW | 1 |
Garrett, KM; Liljequist, S; Tabakoff, B | 1 |
Beer, B; Kuhar, MJ; Lippa, AS; Niehoff, D; Young, WS | 1 |
Beer, B; Lippa, AS; Meyerson, LR; Sano, MC; Vogel, RA | 1 |
Malick, JB; Regan, JW; Roeske, WR; Yamamura, HI; Yamamura, SH | 1 |
Horst, WD; Kuhar, MJ; Mashal, RD; Niehoff, DL; O'Brien, RA; Palacios, JM | 1 |
Beer, B; Lippa, AS; Meyerson, LR | 1 |
Brown, CL; Doble, A; Martin, IL | 1 |
Chisholm, J; Kellogg, C; Lippa, A | 1 |
Niehoff, DL; Whitehouse, PJ | 1 |
Kuhar, MJ; Mashal, RD; Niehoff, DL | 1 |
Kuhar, MJ; Lo, MM; Niehoff, DL; Snyder, SH | 1 |
Squires, RF | 1 |
Cancedda, E; Corda, MG; Giorgi, O; Lecca, D; Serra, GP | 1 |
Bannwarth, W; Benke, D; Fritschy, JM; Mohler, H; Trzeciak, A | 1 |
Erickson, A; Hendrickson, A; March, D; Richards, G; Shaw, C | 1 |
March, D; Shaw, CA | 1 |
Machado, A; Ruano, D; Vitorica, J | 1 |
de Plazas, SF; Gravielle, MC | 1 |
Hadingham, KL; Palmer, KJ; Thompson, SA; Wafford, KA; Whiting, PJ | 1 |
Bromidge, FA; Casula, MA; Hadingham, KL; Martin, K; Maubach, K; Pillai, GV; Seabrook, GR; Whiting, PJ; Wingrove, PB | 1 |
Safo, P; Thompson, SA; Wafford, KA; Wheat, L; Whiting, PJ; Wingrove, PB | 1 |
Cook, JM; Lelas, S; Rowlett, JK; Spealman, RD; Yin, W | 1 |
6 review(s) available for flunitrazepam and cl 218872
Article | Year |
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The separation of 3H-benzodiazepine binding sites in brain and of benzodiazepine pharmacological properties.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Autoradiography; Brain; Flunitrazepam; Humans; Hypnotics and Sedatives; In Vitro Techniques; Kinetics; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Novel non-benzodiazepine anxiolytics.
Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Benzodiazepinones; Conflict, Psychological; Flumazenil; Flunitrazepam; Hypnotics and Sedatives; Mice; Piperazines; Pyrazoles; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
[Is the benzodiazepine binding site a receptor?].
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Binding, Competitive; Brain; Brain Chemistry; Carbolines; Cats; Flunitrazepam; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Structure-Activity Relationship | 1983 |
Molecular substrates of anxiety: clues from the heterogeneity of benzodiazepine receptors.
Topics: Aging; Animals; Anxiety; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Chemical Phenomena; Chemistry, Physical; Flunitrazepam; Humans; Muscles; Pentylenetetrazole; Pyridazines; Receptors, Drug; Receptors, GABA-A; Tissue Distribution; Triazoles | 1982 |
Multiple benzodiazepine receptors: structures in the brain or structures in the mind? A critical review.
Topics: Affinity Labels; Animals; Behavior, Animal; Benzodiazepines; Binding Sites; Binding, Competitive; Brain; Carbolines; Cell Membrane; Chemical Phenomena; Chemistry; Chemistry, Physical; Flunitrazepam; Kinetics; Models, Biological; Photochemistry; Protein Conformation; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A; Solubility; Temperature | 1983 |
Benzodiazepine receptor multiplicity.
Topics: Animals; Brain; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
61 other study(ies) available for flunitrazepam and cl 218872
Article | Year |
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Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423)
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Binding, Competitive; Carbolines; Cell Line; Cerebral Cortex; Drug Design; GABA Agonists; Humans; Male; Mice; Muscle Relaxation; Rats; Receptors, GABA-A; Recombinant Proteins; Seizures; Structure-Activity Relationship | 1998 |
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship | 2000 |
Characteristics of the association of brotizolam, a thieno-triazolo diazepine derivative, with the benzodiazepine receptor: a selective and high affinity ligand of the central type I benzodiazepine receptor.
Topics: Animals; Anti-Anxiety Agents; Azepines; Brain; Dose-Response Relationship, Drug; Flunitrazepam; Hypnotics and Sedatives; In Vitro Techniques; Nitrazepam; Pyridazines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Synaptic Membranes; Tritium | 1992 |
Differential ontogenesis of type I and II benzodiazepine receptors in mouse cerebellum.
Topics: Aging; Animals; Cerebellum; Flunitrazepam; Mice; Models, Biological; Pyridazines; Pyridines; Receptors, GABA-A; Zolpidem | 1991 |
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem | 1990 |
Decreased benzodiazepine receptor binding in epileptic El mice: a quantitative autoradiographic study.
Topics: Animals; Autoradiography; Binding, Competitive; Disease Models, Animal; Epilepsy; Flunitrazepam; In Vitro Techniques; Mice; Mice, Inbred Strains; Physical Stimulation; Pyridazines; Receptors, GABA-A; Tritium | 1990 |
Development of benzodiazepine and picrotoxin (t-butylbicyclophosphorothionate) binding sites in rat cerebellar granule cells in culture.
Topics: Animals; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cells, Cultured; Cerebellum; Flunitrazepam; Granulocytes; Isoxazoles; Pyrazoles; Pyridazines; Pyridines; Rats | 1990 |
n-[3H]butyl-beta-carboline-3-carboxylate, a putative endogenous ligand, binds preferentially to subtype 1 of central benzodiazepine receptors.
Topics: Animals; Brain; Carbolines; Cell Nucleus; Cerebral Cortex; Flunitrazepam; gamma-Aminobutyric Acid; Microsomes; Mitochondria; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes | 1989 |
Two forms of the GABAA receptor distinguished by anion-exchange chromatography.
Topics: Animals; Brain Chemistry; Cell Membrane; Chromatography, High Pressure Liquid; Flunitrazepam; Muscimol; Octoxynol; Polyethylene Glycols; Potassium Chloride; Pyridazines; Rats; Receptors, GABA-A; Solubility | 1989 |
Type I and type II GABAA-benzodiazepine receptors produced in transfected cells.
Topics: Cell Line; Diazepam; Flumazenil; Flunitrazepam; Humans; Molecular Weight; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Transfection | 1989 |
Multiple benzodiazepine receptors in the human basal ganglia: a detailed pharmacological and anatomical study.
Topics: Adolescent; Adult; Aged; Autoradiography; Basal Ganglia; Binding, Competitive; Carbolines; Caudate Nucleus; Child; Child, Preschool; Female; Flunitrazepam; Globus Pallidus; Humans; Male; Middle Aged; Putamen; Pyridazines; Receptors, GABA-A | 1988 |
In vivo interaction of zolpidem with central benzodiazepine (BZD) binding sites (as labeled by [3H]Ro 15-1788) in the mouse brain. Preferential affinity of zolpidem for the omega 1 (BZD1) subtype.
Topics: Animals; Autoradiography; Binding Sites; Brain; Flumazenil; Flunitrazepam; Hypnotics and Sedatives; In Vitro Techniques; Male; Mice; Pyridazines; Pyridines; Receptors, GABA-A; Zolpidem | 1988 |
Benzodiazepine receptor sites in the human brain: autoradiographic mapping.
Topics: Aged; Aged, 80 and over; Autoradiography; Brain; Brain Mapping; Female; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Postmortem Changes; Pyridazines; Receptors, GABA-A | 1988 |
Imidazopyridines as a tool for the characterization of benzodiazepine receptors: a proposal for a pharmacological classification as omega receptor subtypes.
Topics: Animals; Brain Chemistry; Flunitrazepam; GABA-A Receptor Antagonists; Imidazoles; In Vitro Techniques; Isoquinolines; Kidney; Ligands; Pyridazines; Pyridines; Rats; Receptors, GABA-A; Spinal Cord; Terminology as Topic; Zolpidem | 1988 |
Benzodiazepine receptors in the human hippocampal formation: a pharmacological and quantitative autoradiographic study.
Topics: Adolescent; Adult; Aged; Autoradiography; Binding, Competitive; Carbolines; Child; Child, Preschool; Female; Flunitrazepam; Humans; Male; Middle Aged; Pyridazines; Receptors, GABA-A | 1988 |
The development of type I and type II benzodiazepine receptors in the mouse cortex and cerebellum.
Topics: Aging; Animals; Anti-Anxiety Agents; Binding, Competitive; Cerebellum; Cerebral Cortex; Female; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Mice; Nerve Tissue Proteins; Pyridazines; Receptors, GABA-A; Synaptic Membranes | 1985 |
Autoradiographic demonstration of the selectivity of two 1-N-trifluoroethyl benzodiazepines for the BZD-1 receptors in the rat brain.
Topics: Animals; Anti-Anxiety Agents; Autoradiography; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Brain; Computers; Flunitrazepam; In Vitro Techniques; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Quazepam, a sedative-hypnotic selective for the benzodiazepine type 1 receptor: autoradiographic localization in rat and human brain.
Topics: Animals; Anti-Anxiety Agents; Autoradiography; Benzodiazepines; Binding, Competitive; Brain; Flunitrazepam; Humans; Hypnotics and Sedatives; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Aging: effect on ex-vivo benzodiazepine binding after a diazepam injection.
Topics: Aging; Animals; Anti-Anxiety Agents; Binding, Competitive; Brain; Diazepam; Flunitrazepam; Kinetics; Male; Pyridazines; Rats; Rats, Inbred F344; Receptors, GABA-A | 1987 |
Functional coupling of gamma-aminobutyric acid (GABA)A and benzodiazepine type II receptors: analysis using purified GABA/benzodiazepine receptor complex from bovine cerebral cortex.
Topics: Animals; Antipsychotic Agents; Bicuculline; Cattle; Cerebral Cortex; Flumazenil; Flunitrazepam; In Vitro Techniques; Kinetics; Muscimol; Pyridazines; Receptors, GABA-A | 1987 |
Electroencephalographic changes after short-term exposure to agonists of benzodiazepine receptors in the rat.
Topics: Animals; Anti-Anxiety Agents; Brain; Clonazepam; Electroencephalography; Flunitrazepam; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Heterogeneity of brain benzodiazepine receptors: effects of physiological conditions.
Topics: Animals; Binding, Competitive; Brain; Cerebellum; Cerebral Cortex; Electrophoresis, Polyacrylamide Gel; Flunitrazepam; Kinetics; Male; Mice; Pyridazines; Receptors, GABA-A; Temperature | 1985 |
Increase in nigral type II benzodiazepine recognition sites following striatonigral denervation.
Topics: Animals; Carbolines; Corpus Striatum; Denervation; Flunitrazepam; Kainic Acid; Male; Neural Pathways; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra | 1985 |
Autoradiographic studies on benzodiazepine receptor subtypes in the rat brain.
Topics: Animals; Autoradiography; Brain Chemistry; Carbolines; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Benzodiazepine receptors: multiple receptors or multiple conformations?
Topics: Animals; Binding Sites; Brain; Brain Chemistry; Carbolines; Chemical Phenomena; Chemistry; Flunitrazepam; Humans; Kinetics; Models, Chemical; Molecular Conformation; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A | 1985 |
Postnatal development of proteins associated with different benzodiazepine receptors.
Topics: Age Factors; Animals; Azides; Benzodiazepines; Cerebral Cortex; Electrophoresis, Polyacrylamide Gel; Flunitrazepam; Membrane Proteins; Molecular Weight; Pyridazines; Rats; Receptors, GABA-A | 1986 |
Autoradiographic and quantitative study of benzodiazepine-binding sites in human hippocampus.
Topics: Adolescent; Adult; Aged; Anxiety; Autoradiography; Benzodiazepines; Binding Sites; Binding, Competitive; Clonazepam; Female; Flunitrazepam; Hippocampus; Humans; Male; Middle Aged; Pyridazines; Receptors, GABA-A; Tritium | 1985 |
Characterization of benzodiazepine binding sites after short-wave photo-affinity labeling with flunitrazepam.
Topics: Affinity Labels; Animals; Binding Sites; Carbolines; Cell Membrane; Cerebral Cortex; Flunitrazepam; Male; Photochemistry; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Ultraviolet Rays | 1986 |
The neonatal development of benzodiazepine receptor subtypes in the rat cerebral cortex and cerebellum.
Topics: Age Factors; Animals; Animals, Newborn; Cerebellum; Cerebral Cortex; Female; Flunitrazepam; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Comparison of benzodiazepine receptors in cerebellum and inferior colliculus.
Topics: Aging; Animals; Animals, Newborn; Carbolines; Cell Membrane; Cerebellum; Clonazepam; Diazepam; Flunitrazepam; Inferior Colliculi; Pyridazines; Rats; Receptors, GABA-A | 1986 |
Effects of prenatal phenobarbital on benzodiazepine receptor development.
Topics: Animals; Brain; Cerebellum; Diencephalon; Female; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Phenobarbital; Pregnancy; Prenatal Exposure Delayed Effects; Pyridazines; Receptors, GABA-A; Telencephalon | 1986 |
Photoaffinity labeling of benzodiazepine receptor proteins with the partial inverse agonist [3H]Ro 15-4513: a biochemical and autoradiographic study.
Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Brain; Carbolines; Cell Membrane; Cerebellum; Flunitrazepam; Hippocampus; Molecular Weight; Photochemistry; Pyridazines; Rats; Receptors, GABA-A | 1987 |
Benzodiazepine receptors in the human cerebellar cortex: a quantitative autoradiographic and pharmacological study demonstrating the predominance of type I receptors.
Topics: Adult; Autoradiography; Binding, Competitive; Carbolines; Cerebellar Cortex; Female; Flunitrazepam; Humans; Male; Pyridazines; Receptors, GABA-A | 1987 |
Photoaffinity labeling of different benzodiazepine receptors at physiological temperature.
Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cell Membrane; Cerebellum; Flunitrazepam; Hippocampus; Photochemistry; Pyridazines; Rats; Receptors, GABA-A; Temperature | 1984 |
Properties of benzodiazepine receptors in rat retina.
Topics: Animals; Anthelmintics; Anti-Anxiety Agents; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Ivermectin; Lactones; Molecular Weight; Pyridazines; Rats; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Retina | 1982 |
The effect of temperature on CL 218872 and propyl beta-carboline-3-carboxylate inhibition of [3H]-flunitrazepam binding in rat brain.
Topics: Animals; Anti-Anxiety Agents; Binding Sites; Carbolines; Cerebral Cortex; Diazepam; Flunitrazepam; Hippocampus; Indoles; Kinetics; Male; Pyridazines; Rats; Rats, Inbred Strains | 1982 |
Properties of [3H]flunitrazepam binding to different benzodiazepine binding proteins.
Topics: Animals; Anti-Anxiety Agents; Carbolines; Cerebellum; Flunitrazepam; Hippocampus; In Vitro Techniques; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Tritium | 1983 |
Association of proteins irreversibly labeled by 3H-flunitrazepam with different benzodiazepine.
Topics: Anti-Anxiety Agents; Cerebellum; Flunitrazepam; Hippocampus; Humans; In Vitro Techniques; Proteins; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Selective anxiolytics: are the actions related to partial "agonist" activity or a preferential affinity for benzodiazepine receptor subtypes?
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Cerebral Cortex; Drug Interactions; Flunitrazepam; Male; Postural Balance; Pyrazoles; Pyridazines; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Reflex; Temperature | 1983 |
Characterization of benzodiazepine receptor changes in substantia nigra, globus pallidus and entopeduncular nucleus after striatal lesions.
Topics: Animals; Binding, Competitive; Corpus Striatum; Flunitrazepam; Globus Pallidus; Glutamates; Glutamic Acid; Kainic Acid; Male; Pyridazines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra; Time Factors | 1984 |
The benzodiazepine receptor ligand CL218,872 has both anxiolytic and sedative properties in rodents.
Topics: Aggression; Animals; Anti-Anxiety Agents; Arousal; Brain; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; Humans; Male; Mice; Mice, Inbred Strains; Motor Activity; Motor Skills; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Specific effects of chronic phenobarbital administration on high- and low-affinity benzodiazepine receptors in mouse cerebellum and forebrain.
Topics: Animals; Anti-Anxiety Agents; Brain; Cerebellum; Flunitrazepam; Kinetics; Membranes; Mice; Mice, Inbred C57BL; Phenobarbital; Pyridazines; Receptors, GABA-A; Time Factors | 1984 |
Multiple benzodiazepine receptor localization by light microscopic radiohistochemistry.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cerebellum; Flunitrazepam; Mesencephalon; Pyridazines; Rats; Receptors, Drug; Receptors, GABA-A; Structure-Activity Relationship | 1981 |
Differential ontogeny of type 1 and type 2 benzodiazepine receptors.
Topics: Animals; Brain; Female; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Pregnancy; Protein Binding; Pyridazines; Rats; Receptors, Drug; Receptors, GABA-A | 1981 |
gamma-Aminobutyric acid enhancement of CL 218,872 affinity and evidence of benzodiazepine receptor heterogeneity.
Topics: Animals; Bicuculline; Binding, Competitive; Brain; Cattle; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kidney; Kinetics; Pyridazines; Receptors, Drug; Receptors, GABA-A; Retina | 1981 |
Binding of a radiolabeled triazolopyridazine to a subtype of benzodiazepine receptor in the rat cerebellum.
Topics: Animals; Anions; Cerebellum; Flunitrazepam; gamma-Aminobutyric Acid; Male; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A | 1982 |
Regional heterogeneity of benzodiazepine receptors at 37 degrees C: an in vitro study in various regions of the rat brain.
Topics: Animals; Binding, Competitive; Brain; Carbolines; Cerebellum; Cerebral Cortex; Flunitrazepam; Hippocampus; Male; Pons; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Temperature | 1982 |
Development of benzodiazepine binding subtypes in three regions of rat brain.
Topics: Aging; Animals; Binding, Competitive; Brain; Cerebellum; Cerebral Cortex; Flunitrazepam; Hippocampus; Muridae; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Multiple benzodiazepine receptors: autoradiographic localization in normal human amygdala.
Topics: Adolescent; Adult; Aged; Amygdala; Animals; Autoradiography; Female; Flunitrazepam; Humans; Male; Middle Aged; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Species Specificity | 1983 |
Benzodiazepine receptors: preferential stimulation of Type 1 receptors by pentobarbital.
Topics: Animals; Cerebellum; Cerebral Cortex; Flunitrazepam; In Vitro Techniques; Male; Pentobarbital; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Autoradiographic differentiation of multiple benzodiazepine receptors by detergent solubilization and pharmacologic specificity.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Corpus Striatum; Flunitrazepam; Neural Pathways; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra | 1983 |
Modulation of [35S]TBPS binding by ligands with preferential affinity for benzodiazepine BZ1 sites in the cerebral cortex of newborn and adult rats.
Topics: Age Factors; Animals; Animals, Newborn; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Female; Flunitrazepam; Male; Pregnancy; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zolpidem | 1995 |
Distribution, prevalence, and drug binding profile of gamma-aminobutyric acid type A receptor subtypes differing in the beta-subunit variant.
Topics: Animals; Brain Chemistry; Carbolines; Flumazenil; Flunitrazepam; Genetic Variation; Immunohistochemistry; Male; Microscopy, Confocal; Molecular Weight; Precipitin Tests; Protein Conformation; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tissue Distribution; Zolpidem | 1994 |
Coincidental appearance of the alpha 1 subunit of the GABA-A receptor and the type I benzodiazepine receptor near birth in macaque monkey visual cortex.
Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Antibodies, Monoclonal; Autoradiography; Binding, Competitive; Female; Flunitrazepam; Hypnotics and Sedatives; Immunohistochemistry; Ligands; Macaca nemestrina; Pregnancy; Pyridazines; Pyridines; Receptors, GABA-A; Visual Cortex; Zolpidem | 1994 |
Fetal, neonatal and adult expression of benzodiazepine receptor subtypes in human visual cortex.
Topics: Adult; Aged; Aging; Anti-Anxiety Agents; Autoradiography; Embryonic and Fetal Development; Flunitrazepam; Humans; Infant, Newborn; Male; Middle Aged; Pyridazines; Receptors, GABA-A; Visual Cortex | 1993 |
Absence of modifications of the pharmacological properties of the GABAA receptor complex during aging, as assessed in 3- and 24-month-old rat cerebral cortex.
Topics: Affinity Labels; Aging; Animals; Anti-Anxiety Agents; Binding, Competitive; Cerebral Cortex; Flunitrazepam; Hypnotics and Sedatives; In Vitro Techniques; Male; Membrane Proteins; Muscimol; Photochemistry; Pyridazines; Pyridines; Rats; Rats, Inbred F344; Rats, Wistar; Receptors, GABA-A; Zolpidem | 1993 |
Ontogeny of two different benzodiazepine binding sites in the chick optic lobe.
Topics: Animals; Anti-Anxiety Agents; Binding Sites; Chickens; Flunitrazepam; Kinetics; Pyridazines; Receptors, GABA-A; Tectum Mesencephali | 1995 |
Expression and pharmacology of human GABAA receptors containing gamma 3 subunits.
Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Base Sequence; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Molecular Sequence Data; Pyrazoles; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Proteins; Sequence Homology, Amino Acid; Triazolam; Xenopus; Zolpidem | 1995 |
Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor.
Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; DNA, Complementary; Female; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Humans; Imidazoles; Isoleucine; Ligands; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Protein Binding; Protein Structure, Tertiary; Protein Subunits; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Fusion Proteins; Sequence Alignment; Structure-Activity Relationship; Threonine; Transfection; Xenopus laevis; Zolpidem | 2001 |
Mechanism of alpha-subunit selectivity of benzodiazepine pharmacology at gamma-aminobutyric acid type A receptors.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Cell Line; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Mutation; Oocytes; Protein Subunits; Pyridazines; Pyridines; Radioligand Assay; Receptors, GABA-A; Tritium; Xenopus laevis; Zolpidem | 2002 |
Discriminative stimulus effects of zolpidem in squirrel monkeys: role of GABA(A)/alpha1 receptors.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Carbolines; Discrimination Learning; Dose-Response Relationship, Drug; Flunitrazepam; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; Injections, Intravenous; Male; Pyridazines; Pyridines; Receptors, GABA-A; Saimiri; Zolpidem | 2003 |