flunitrazepam and cl 218872

flunitrazepam has been researched along with cl 218872 in 67 studies

Research

Studies (67)

TimeframeStudies, this research(%)All Research%
pre-199050 (74.63)18.7374
1990's13 (19.40)18.2507
2000's4 (5.97)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cook, JM; Cox, ED; Diaz-Arauzo, H; Harris, B; Huang, Q; Ma, C; McKernan, R; Reddy, MS; Skolnick, P1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Hirouchi, M; Kohno, Y; Kuriyama, K; Mizutani, H1
Bacon, E; de Barry, J; Gombos, G1
De Luca, C; De Medici, D; Massotti, M1
Ito, M; Mikawa, H; Mutoh, K; Oguro, K; Shiraishi, H; Shirasaka, Y; Tsuda, H1
Damgaard, I; Saederup, E; Schousboe, A; Squires, RF1
De Robertis, E; de Stein, ML; Medina, JH1
Moffett, JR; Namboodiri, A; Neale, JH1
Lüddens, H; Pritchett, DB; Seeburg, PH1
Faull, RL; Villiger, JW2
Benavides, J; Dubois, A; Morel, E; Peny, B; Perrault, G; Scatton, B; Zivkovic, B1
Cortés, R; Palacios, JM; Probst, A; Zezula, J1
Arbilla, S; Langer, SZ1
Garrett, KM; Tabakoff, B2
Barnett, A; Golden, JS; Wamsley, JK; Yamamura, HI2
Komiskey, HL1
Kuriyama, K; Taguchi, J1
Massotti, M; Valerio, A1
Beer, B; Garrett, KM; Lippa, AS; Meyerson, LR; Tabakoff, B; Wennogle, LP1
Biggio, G; Corda, MG; Porceddu, ML; Sanna, E1
Kito, S; Miyoshi, R; Mizuno, K1
Sieghart, W3
Eichinger, A; Sieghart, W2
Bobillier, P; Kopp, N; Manchon, M; Miachon, S1
Herblin, WF1
Hyde, L; Khatami, S; Salafsky, B; Shibuya, T; Watanabe, Y1
Eichinger, A; Möhler, H; Richards, JG; Sieghart, W1
Faull, RL; Holford, NH; Villiger, JW1
Drexler, G; Karobath, M; Sieghart, W; Supavilai, P1
Gee, KW; Morelli, M; Yamamura, HI1
Beer, B; Coupet, J; Dubnick, B; Greenblatt, EN; Klepner, CA; Lippa, AS1
Drexler, G; Mayer, A; Sieghart, W1
Goldberg, ME; Malick, JB; Patel, JB; Salama, AI1
Gee, KW; Yamamura, HI2
Keane, P; Morre, M1
Pan, HS; Penney, JB; Young, AB1
Jones, BJ; Oakley, NR; Straughan, DW1
Garrett, KM; Liljequist, S; Tabakoff, B1
Beer, B; Kuhar, MJ; Lippa, AS; Niehoff, D; Young, WS1
Beer, B; Lippa, AS; Meyerson, LR; Sano, MC; Vogel, RA1
Malick, JB; Regan, JW; Roeske, WR; Yamamura, HI; Yamamura, SH1
Horst, WD; Kuhar, MJ; Mashal, RD; Niehoff, DL; O'Brien, RA; Palacios, JM1
Beer, B; Lippa, AS; Meyerson, LR1
Brown, CL; Doble, A; Martin, IL1
Chisholm, J; Kellogg, C; Lippa, A1
Niehoff, DL; Whitehouse, PJ1
Kuhar, MJ; Mashal, RD; Niehoff, DL1
Kuhar, MJ; Lo, MM; Niehoff, DL; Snyder, SH1
Squires, RF1
Cancedda, E; Corda, MG; Giorgi, O; Lecca, D; Serra, GP1
Bannwarth, W; Benke, D; Fritschy, JM; Mohler, H; Trzeciak, A1
Erickson, A; Hendrickson, A; March, D; Richards, G; Shaw, C1
March, D; Shaw, CA1
Machado, A; Ruano, D; Vitorica, J1
de Plazas, SF; Gravielle, MC1
Hadingham, KL; Palmer, KJ; Thompson, SA; Wafford, KA; Whiting, PJ1
Bromidge, FA; Casula, MA; Hadingham, KL; Martin, K; Maubach, K; Pillai, GV; Seabrook, GR; Whiting, PJ; Wingrove, PB1
Safo, P; Thompson, SA; Wafford, KA; Wheat, L; Whiting, PJ; Wingrove, PB1
Cook, JM; Lelas, S; Rowlett, JK; Spealman, RD; Yin, W1

Reviews

6 review(s) available for flunitrazepam and cl 218872

ArticleYear
The separation of 3H-benzodiazepine binding sites in brain and of benzodiazepine pharmacological properties.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Autoradiography; Brain; Flunitrazepam; Humans; Hypnotics and Sedatives; In Vitro Techniques; Kinetics; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A

1983
Novel non-benzodiazepine anxiolytics.
    Neuropharmacology, 1983, Volume: 22, Issue:12B

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Benzodiazepinones; Conflict, Psychological; Flumazenil; Flunitrazepam; Hypnotics and Sedatives; Mice; Piperazines; Pyrazoles; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
[Is the benzodiazepine binding site a receptor?].
    L'Encephale, 1983, Volume: 9, Issue:4 Suppl 2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding Sites; Binding, Competitive; Brain; Brain Chemistry; Carbolines; Cats; Flunitrazepam; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Structure-Activity Relationship

1983
Molecular substrates of anxiety: clues from the heterogeneity of benzodiazepine receptors.
    Life sciences, 1982, Oct-04, Volume: 31, Issue:14

    Topics: Aging; Animals; Anxiety; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Chemical Phenomena; Chemistry, Physical; Flunitrazepam; Humans; Muscles; Pentylenetetrazole; Pyridazines; Receptors, Drug; Receptors, GABA-A; Tissue Distribution; Triazoles

1982
Multiple benzodiazepine receptors: structures in the brain or structures in the mind? A critical review.
    Life sciences, 1983, Apr-25, Volume: 32, Issue:17

    Topics: Affinity Labels; Animals; Behavior, Animal; Benzodiazepines; Binding Sites; Binding, Competitive; Brain; Carbolines; Cell Membrane; Chemical Phenomena; Chemistry; Chemistry, Physical; Flunitrazepam; Kinetics; Models, Biological; Photochemistry; Protein Conformation; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A; Solubility; Temperature

1983
Benzodiazepine receptor multiplicity.
    Neuropharmacology, 1983, Volume: 22, Issue:12B

    Topics: Animals; Brain; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A

1983

Other Studies

61 other study(ies) available for flunitrazepam and cl 218872

ArticleYear
Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423)
    Journal of medicinal chemistry, 1998, Jul-02, Volume: 41, Issue:14

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Binding, Competitive; Carbolines; Cell Line; Cerebral Cortex; Drug Design; GABA Agonists; Humans; Male; Mice; Muscle Relaxation; Rats; Receptors, GABA-A; Recombinant Proteins; Seizures; Structure-Activity Relationship

1998
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
Characteristics of the association of brotizolam, a thieno-triazolo diazepine derivative, with the benzodiazepine receptor: a selective and high affinity ligand of the central type I benzodiazepine receptor.
    Japanese journal of pharmacology, 1992, Volume: 59, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Azepines; Brain; Dose-Response Relationship, Drug; Flunitrazepam; Hypnotics and Sedatives; In Vitro Techniques; Nitrazepam; Pyridazines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord; Synaptic Membranes; Tritium

1992
Differential ontogenesis of type I and II benzodiazepine receptors in mouse cerebellum.
    Brain research. Developmental brain research, 1991, Feb-22, Volume: 58, Issue:2

    Topics: Aging; Animals; Cerebellum; Flunitrazepam; Mice; Models, Biological; Pyridazines; Pyridines; Receptors, GABA-A; Zolpidem

1991
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
    Psychopharmacology, 1990, Volume: 102, Issue:4

    Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem

1990
Decreased benzodiazepine receptor binding in epileptic El mice: a quantitative autoradiographic study.
    Neurochemical research, 1990, Volume: 15, Issue:9

    Topics: Animals; Autoradiography; Binding, Competitive; Disease Models, Animal; Epilepsy; Flunitrazepam; In Vitro Techniques; Mice; Mice, Inbred Strains; Physical Stimulation; Pyridazines; Receptors, GABA-A; Tritium

1990
Development of benzodiazepine and picrotoxin (t-butylbicyclophosphorothionate) binding sites in rat cerebellar granule cells in culture.
    Journal of neurochemistry, 1990, Volume: 54, Issue:2

    Topics: Animals; Benzodiazepines; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cells, Cultured; Cerebellum; Flunitrazepam; Granulocytes; Isoxazoles; Pyrazoles; Pyridazines; Pyridines; Rats

1990
n-[3H]butyl-beta-carboline-3-carboxylate, a putative endogenous ligand, binds preferentially to subtype 1 of central benzodiazepine receptors.
    Journal of neurochemistry, 1989, Volume: 52, Issue:3

    Topics: Animals; Brain; Carbolines; Cell Nucleus; Cerebral Cortex; Flunitrazepam; gamma-Aminobutyric Acid; Microsomes; Mitochondria; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes

1989
Two forms of the GABAA receptor distinguished by anion-exchange chromatography.
    FEBS letters, 1989, Apr-10, Volume: 247, Issue:1

    Topics: Animals; Brain Chemistry; Cell Membrane; Chromatography, High Pressure Liquid; Flunitrazepam; Muscimol; Octoxynol; Polyethylene Glycols; Potassium Chloride; Pyridazines; Rats; Receptors, GABA-A; Solubility

1989
Type I and type II GABAA-benzodiazepine receptors produced in transfected cells.
    Science (New York, N.Y.), 1989, Sep-22, Volume: 245, Issue:4924

    Topics: Cell Line; Diazepam; Flumazenil; Flunitrazepam; Humans; Molecular Weight; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Transfection

1989
Multiple benzodiazepine receptors in the human basal ganglia: a detailed pharmacological and anatomical study.
    Neuroscience, 1988, Volume: 24, Issue:2

    Topics: Adolescent; Adult; Aged; Autoradiography; Basal Ganglia; Binding, Competitive; Carbolines; Caudate Nucleus; Child; Child, Preschool; Female; Flunitrazepam; Globus Pallidus; Humans; Male; Middle Aged; Putamen; Pyridazines; Receptors, GABA-A

1988
In vivo interaction of zolpidem with central benzodiazepine (BZD) binding sites (as labeled by [3H]Ro 15-1788) in the mouse brain. Preferential affinity of zolpidem for the omega 1 (BZD1) subtype.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:3

    Topics: Animals; Autoradiography; Binding Sites; Brain; Flumazenil; Flunitrazepam; Hypnotics and Sedatives; In Vitro Techniques; Male; Mice; Pyridazines; Pyridines; Receptors, GABA-A; Zolpidem

1988
Benzodiazepine receptor sites in the human brain: autoradiographic mapping.
    Neuroscience, 1988, Volume: 25, Issue:3

    Topics: Aged; Aged, 80 and over; Autoradiography; Brain; Brain Mapping; Female; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Male; Middle Aged; Postmortem Changes; Pyridazines; Receptors, GABA-A

1988
Imidazopyridines as a tool for the characterization of benzodiazepine receptors: a proposal for a pharmacological classification as omega receptor subtypes.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:4

    Topics: Animals; Brain Chemistry; Flunitrazepam; GABA-A Receptor Antagonists; Imidazoles; In Vitro Techniques; Isoquinolines; Kidney; Ligands; Pyridazines; Pyridines; Rats; Receptors, GABA-A; Spinal Cord; Terminology as Topic; Zolpidem

1988
Benzodiazepine receptors in the human hippocampal formation: a pharmacological and quantitative autoradiographic study.
    Neuroscience, 1988, Volume: 26, Issue:3

    Topics: Adolescent; Adult; Aged; Autoradiography; Binding, Competitive; Carbolines; Child; Child, Preschool; Female; Flunitrazepam; Humans; Male; Middle Aged; Pyridazines; Receptors, GABA-A

1988
The development of type I and type II benzodiazepine receptors in the mouse cortex and cerebellum.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:6

    Topics: Aging; Animals; Anti-Anxiety Agents; Binding, Competitive; Cerebellum; Cerebral Cortex; Female; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Mice; Nerve Tissue Proteins; Pyridazines; Receptors, GABA-A; Synaptic Membranes

1985
Autoradiographic demonstration of the selectivity of two 1-N-trifluoroethyl benzodiazepines for the BZD-1 receptors in the rat brain.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Autoradiography; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Brain; Computers; Flunitrazepam; In Vitro Techniques; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Quazepam, a sedative-hypnotic selective for the benzodiazepine type 1 receptor: autoradiographic localization in rat and human brain.
    Clinical neuropharmacology, 1985, Volume: 8 Suppl 1

    Topics: Animals; Anti-Anxiety Agents; Autoradiography; Benzodiazepines; Binding, Competitive; Brain; Flunitrazepam; Humans; Hypnotics and Sedatives; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Aging: effect on ex-vivo benzodiazepine binding after a diazepam injection.
    Neurochemical research, 1987, Volume: 12, Issue:8

    Topics: Aging; Animals; Anti-Anxiety Agents; Binding, Competitive; Brain; Diazepam; Flunitrazepam; Kinetics; Male; Pyridazines; Rats; Rats, Inbred F344; Receptors, GABA-A

1987
Functional coupling of gamma-aminobutyric acid (GABA)A and benzodiazepine type II receptors: analysis using purified GABA/benzodiazepine receptor complex from bovine cerebral cortex.
    Neuropharmacology, 1987, Volume: 26, Issue:12

    Topics: Animals; Antipsychotic Agents; Bicuculline; Cattle; Cerebral Cortex; Flumazenil; Flunitrazepam; In Vitro Techniques; Kinetics; Muscimol; Pyridazines; Receptors, GABA-A

1987
Electroencephalographic changes after short-term exposure to agonists of benzodiazepine receptors in the rat.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Brain; Clonazepam; Electroencephalography; Flunitrazepam; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Heterogeneity of brain benzodiazepine receptors: effects of physiological conditions.
    Brain research bulletin, 1985, Volume: 14, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Cerebellum; Cerebral Cortex; Electrophoresis, Polyacrylamide Gel; Flunitrazepam; Kinetics; Male; Mice; Pyridazines; Receptors, GABA-A; Temperature

1985
Increase in nigral type II benzodiazepine recognition sites following striatonigral denervation.
    European journal of pharmacology, 1985, Jun-07, Volume: 112, Issue:2

    Topics: Animals; Carbolines; Corpus Striatum; Denervation; Flunitrazepam; Kainic Acid; Male; Neural Pathways; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1985
Autoradiographic studies on benzodiazepine receptor subtypes in the rat brain.
    Japanese journal of pharmacology, 1985, Volume: 38, Issue:3

    Topics: Animals; Autoradiography; Brain Chemistry; Carbolines; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Benzodiazepine receptors: multiple receptors or multiple conformations?
    Journal of neural transmission, 1985, Volume: 63, Issue:3-4

    Topics: Animals; Binding Sites; Brain; Brain Chemistry; Carbolines; Chemical Phenomena; Chemistry; Flunitrazepam; Humans; Kinetics; Models, Chemical; Molecular Conformation; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A

1985
Postnatal development of proteins associated with different benzodiazepine receptors.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: Age Factors; Animals; Azides; Benzodiazepines; Cerebral Cortex; Electrophoresis, Polyacrylamide Gel; Flunitrazepam; Membrane Proteins; Molecular Weight; Pyridazines; Rats; Receptors, GABA-A

1986
Autoradiographic and quantitative study of benzodiazepine-binding sites in human hippocampus.
    Neuroscience letters, 1985, Nov-20, Volume: 62, Issue:1

    Topics: Adolescent; Adult; Aged; Anxiety; Autoradiography; Benzodiazepines; Binding Sites; Binding, Competitive; Clonazepam; Female; Flunitrazepam; Hippocampus; Humans; Male; Middle Aged; Pyridazines; Receptors, GABA-A; Tritium

1985
Characterization of benzodiazepine binding sites after short-wave photo-affinity labeling with flunitrazepam.
    Life sciences, 1986, Feb-10, Volume: 38, Issue:6

    Topics: Affinity Labels; Animals; Binding Sites; Carbolines; Cell Membrane; Cerebral Cortex; Flunitrazepam; Male; Photochemistry; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Ultraviolet Rays

1986
The neonatal development of benzodiazepine receptor subtypes in the rat cerebral cortex and cerebellum.
    Yakubutsu, seishin, kodo = Japanese journal of psychopharmacology, 1985, Volume: 5, Issue:4

    Topics: Age Factors; Animals; Animals, Newborn; Cerebellum; Cerebral Cortex; Female; Flunitrazepam; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Comparison of benzodiazepine receptors in cerebellum and inferior colliculus.
    Journal of neurochemistry, 1986, Volume: 47, Issue:3

    Topics: Aging; Animals; Animals, Newborn; Carbolines; Cell Membrane; Cerebellum; Clonazepam; Diazepam; Flunitrazepam; Inferior Colliculi; Pyridazines; Rats; Receptors, GABA-A

1986
Effects of prenatal phenobarbital on benzodiazepine receptor development.
    Journal of neurochemistry, 1986, Volume: 47, Issue:4

    Topics: Animals; Brain; Cerebellum; Diencephalon; Female; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Phenobarbital; Pregnancy; Prenatal Exposure Delayed Effects; Pyridazines; Receptors, GABA-A; Telencephalon

1986
Photoaffinity labeling of benzodiazepine receptor proteins with the partial inverse agonist [3H]Ro 15-4513: a biochemical and autoradiographic study.
    Journal of neurochemistry, 1987, Volume: 48, Issue:1

    Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Brain; Carbolines; Cell Membrane; Cerebellum; Flunitrazepam; Hippocampus; Molecular Weight; Photochemistry; Pyridazines; Rats; Receptors, GABA-A

1987
Benzodiazepine receptors in the human cerebellar cortex: a quantitative autoradiographic and pharmacological study demonstrating the predominance of type I receptors.
    Brain research, 1987, May-19, Volume: 411, Issue:2

    Topics: Adult; Autoradiography; Binding, Competitive; Carbolines; Cerebellar Cortex; Female; Flunitrazepam; Humans; Male; Pyridazines; Receptors, GABA-A

1987
Photoaffinity labeling of different benzodiazepine receptors at physiological temperature.
    Journal of neurochemistry, 1984, Volume: 43, Issue:6

    Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cell Membrane; Cerebellum; Flunitrazepam; Hippocampus; Photochemistry; Pyridazines; Rats; Receptors, GABA-A; Temperature

1984
Properties of benzodiazepine receptors in rat retina.
    Experimental eye research, 1982, Volume: 34, Issue:6

    Topics: Animals; Anthelmintics; Anti-Anxiety Agents; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Ivermectin; Lactones; Molecular Weight; Pyridazines; Rats; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Retina

1982
The effect of temperature on CL 218872 and propyl beta-carboline-3-carboxylate inhibition of [3H]-flunitrazepam binding in rat brain.
    Biochemical and biophysical research communications, 1982, Apr-29, Volume: 105, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Binding Sites; Carbolines; Cerebral Cortex; Diazepam; Flunitrazepam; Hippocampus; Indoles; Kinetics; Male; Pyridazines; Rats; Rats, Inbred Strains

1982
Properties of [3H]flunitrazepam binding to different benzodiazepine binding proteins.
    European journal of pharmacology, 1983, Apr-08, Volume: 88, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Carbolines; Cerebellum; Flunitrazepam; Hippocampus; In Vitro Techniques; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Tritium

1983
Association of proteins irreversibly labeled by 3H-flunitrazepam with different benzodiazepine.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Anti-Anxiety Agents; Cerebellum; Flunitrazepam; Hippocampus; Humans; In Vitro Techniques; Proteins; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A

1983
Selective anxiolytics: are the actions related to partial "agonist" activity or a preferential affinity for benzodiazepine receptor subtypes?
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Cerebral Cortex; Drug Interactions; Flunitrazepam; Male; Postural Balance; Pyrazoles; Pyridazines; Quinolines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Reflex; Temperature

1983
Characterization of benzodiazepine receptor changes in substantia nigra, globus pallidus and entopeduncular nucleus after striatal lesions.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:3

    Topics: Animals; Binding, Competitive; Corpus Striatum; Flunitrazepam; Globus Pallidus; Glutamates; Glutamic Acid; Kainic Acid; Male; Pyridazines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra; Time Factors

1984
The benzodiazepine receptor ligand CL218,872 has both anxiolytic and sedative properties in rodents.
    Neuropharmacology, 1984, Volume: 23, Issue:7A

    Topics: Aggression; Animals; Anti-Anxiety Agents; Arousal; Brain; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; Humans; Male; Mice; Mice, Inbred Strains; Motor Activity; Motor Skills; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1984
Specific effects of chronic phenobarbital administration on high- and low-affinity benzodiazepine receptors in mouse cerebellum and forebrain.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Animals; Anti-Anxiety Agents; Brain; Cerebellum; Flunitrazepam; Kinetics; Membranes; Mice; Mice, Inbred C57BL; Phenobarbital; Pyridazines; Receptors, GABA-A; Time Factors

1984
Multiple benzodiazepine receptor localization by light microscopic radiohistochemistry.
    The Journal of pharmacology and experimental therapeutics, 1981, Volume: 216, Issue:2

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Cerebellum; Flunitrazepam; Mesencephalon; Pyridazines; Rats; Receptors, Drug; Receptors, GABA-A; Structure-Activity Relationship

1981
Differential ontogeny of type 1 and type 2 benzodiazepine receptors.
    Life sciences, 1981, May-21, Volume: 28, Issue:21

    Topics: Animals; Brain; Female; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Pregnancy; Protein Binding; Pyridazines; Rats; Receptors, Drug; Receptors, GABA-A

1981
gamma-Aminobutyric acid enhancement of CL 218,872 affinity and evidence of benzodiazepine receptor heterogeneity.
    Molecular pharmacology, 1981, Volume: 20, Issue:3

    Topics: Animals; Bicuculline; Binding, Competitive; Brain; Cattle; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kidney; Kinetics; Pyridazines; Receptors, Drug; Receptors, GABA-A; Retina

1981
Binding of a radiolabeled triazolopyridazine to a subtype of benzodiazepine receptor in the rat cerebellum.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 221, Issue:3

    Topics: Animals; Anions; Cerebellum; Flunitrazepam; gamma-Aminobutyric Acid; Male; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A

1982
Regional heterogeneity of benzodiazepine receptors at 37 degrees C: an in vitro study in various regions of the rat brain.
    Life sciences, 1982, Nov-01, Volume: 31, Issue:18

    Topics: Animals; Binding, Competitive; Brain; Carbolines; Cerebellum; Cerebral Cortex; Flunitrazepam; Hippocampus; Male; Pons; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Temperature

1982
Development of benzodiazepine binding subtypes in three regions of rat brain.
    Brain research, 1983, May-16, Volume: 267, Issue:2

    Topics: Aging; Animals; Binding, Competitive; Brain; Cerebellum; Cerebral Cortex; Flunitrazepam; Hippocampus; Muridae; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A

1983
Multiple benzodiazepine receptors: autoradiographic localization in normal human amygdala.
    Brain research, 1983, Oct-16, Volume: 276, Issue:2

    Topics: Adolescent; Adult; Aged; Amygdala; Animals; Autoradiography; Female; Flunitrazepam; Humans; Male; Middle Aged; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Species Specificity

1983
Benzodiazepine receptors: preferential stimulation of Type 1 receptors by pentobarbital.
    European journal of pharmacology, 1983, Aug-19, Volume: 92, Issue:1-2

    Topics: Animals; Cerebellum; Cerebral Cortex; Flunitrazepam; In Vitro Techniques; Male; Pentobarbital; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
Autoradiographic differentiation of multiple benzodiazepine receptors by detergent solubilization and pharmacologic specificity.
    Neuroscience letters, 1983, Aug-19, Volume: 39, Issue:1

    Topics: Animals; Autoradiography; Binding, Competitive; Brain; Corpus Striatum; Flunitrazepam; Neural Pathways; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra

1983
Modulation of [35S]TBPS binding by ligands with preferential affinity for benzodiazepine BZ1 sites in the cerebral cortex of newborn and adult rats.
    European journal of pharmacology, 1995, Jun-23, Volume: 290, Issue:1

    Topics: Age Factors; Animals; Animals, Newborn; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Female; Flunitrazepam; Male; Pregnancy; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zolpidem

1995
Distribution, prevalence, and drug binding profile of gamma-aminobutyric acid type A receptor subtypes differing in the beta-subunit variant.
    The Journal of biological chemistry, 1994, Oct-28, Volume: 269, Issue:43

    Topics: Animals; Brain Chemistry; Carbolines; Flumazenil; Flunitrazepam; Genetic Variation; Immunohistochemistry; Male; Microscopy, Confocal; Molecular Weight; Precipitin Tests; Protein Conformation; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tissue Distribution; Zolpidem

1994
Coincidental appearance of the alpha 1 subunit of the GABA-A receptor and the type I benzodiazepine receptor near birth in macaque monkey visual cortex.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 1994, Volume: 12, Issue:4

    Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Antibodies, Monoclonal; Autoradiography; Binding, Competitive; Female; Flunitrazepam; Hypnotics and Sedatives; Immunohistochemistry; Ligands; Macaca nemestrina; Pregnancy; Pyridazines; Pyridines; Receptors, GABA-A; Visual Cortex; Zolpidem

1994
Fetal, neonatal and adult expression of benzodiazepine receptor subtypes in human visual cortex.
    European journal of pharmacology, 1993, May-19, Volume: 236, Issue:2

    Topics: Adult; Aged; Aging; Anti-Anxiety Agents; Autoradiography; Embryonic and Fetal Development; Flunitrazepam; Humans; Infant, Newborn; Male; Middle Aged; Pyridazines; Receptors, GABA-A; Visual Cortex

1993
Absence of modifications of the pharmacological properties of the GABAA receptor complex during aging, as assessed in 3- and 24-month-old rat cerebral cortex.
    European journal of pharmacology, 1993, Jun-15, Volume: 246, Issue:1

    Topics: Affinity Labels; Aging; Animals; Anti-Anxiety Agents; Binding, Competitive; Cerebral Cortex; Flunitrazepam; Hypnotics and Sedatives; In Vitro Techniques; Male; Membrane Proteins; Muscimol; Photochemistry; Pyridazines; Pyridines; Rats; Rats, Inbred F344; Rats, Wistar; Receptors, GABA-A; Zolpidem

1993
Ontogeny of two different benzodiazepine binding sites in the chick optic lobe.
    Neuroreport, 1995, Oct-23, Volume: 6, Issue:15

    Topics: Animals; Anti-Anxiety Agents; Binding Sites; Chickens; Flunitrazepam; Kinetics; Pyridazines; Receptors, GABA-A; Tectum Mesencephali

1995
Expression and pharmacology of human GABAA receptors containing gamma 3 subunits.
    European journal of pharmacology, 1995, Nov-30, Volume: 291, Issue:3

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Base Sequence; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Molecular Sequence Data; Pyrazoles; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Proteins; Sequence Homology, Amino Acid; Triazolam; Xenopus; Zolpidem

1995
Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; DNA, Complementary; Female; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Humans; Imidazoles; Isoleucine; Ligands; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Protein Binding; Protein Structure, Tertiary; Protein Subunits; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Fusion Proteins; Sequence Alignment; Structure-Activity Relationship; Threonine; Transfection; Xenopus laevis; Zolpidem

2001
Mechanism of alpha-subunit selectivity of benzodiazepine pharmacology at gamma-aminobutyric acid type A receptors.
    European journal of pharmacology, 2002, Feb-15, Volume: 437, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Cell Line; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Mutation; Oocytes; Protein Subunits; Pyridazines; Pyridines; Radioligand Assay; Receptors, GABA-A; Tritium; Xenopus laevis; Zolpidem

2002
Discriminative stimulus effects of zolpidem in squirrel monkeys: role of GABA(A)/alpha1 receptors.
    Psychopharmacology, 2003, Volume: 165, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Carbolines; Discrimination Learning; Dose-Response Relationship, Drug; Flunitrazepam; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; Injections, Intravenous; Male; Pyridazines; Pyridines; Receptors, GABA-A; Saimiri; Zolpidem

2003