flunitrazepam and chlordiazepoxide

flunitrazepam has been researched along with chlordiazepoxide in 34 studies

Research

Studies (34)

TimeframeStudies, this research(%)All Research%
pre-199024 (70.59)18.7374
1990's4 (11.76)18.2507
2000's4 (11.76)29.6817
2010's2 (5.88)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Dudai, Y; Yavin, E; Yavin, Z1
Beck, O; Borg, S; Hjemdahl, P; Lafolie, P; Odelius, G; Wirbing, P1
Rothe, T; Schliebs, R1
Akaike, N; Kaneda, M; Oyama, Y; Wakamori, M1
Celentano, JJ; Farb, DH; Gibbs, TT; Gyenes, M; Mierlak, D1
Barrett, JE; Mansbach, RS; Skolnick, P; Weissman, BA; Witkin, JM1
Avnimelech-Gigus, N; Feldon, J; Gavish, M; Myslobodsky, M1
Bold, JM; Gardner, CR; Walker, RJ1
Baraldi, PG; Borea, PA; Guarneri, M; Manfredini, S; Periotto, V; Simoni, D1
Ambrose, F; Barbaz, B; Bittiger, H; Iyengar, S; Neale, RF; Petrack, B; Rinehart, RK; Steel, DJ; Williams, M; Wood, PL1
Fioretti, P; Galbani, P; Gambacciani, M; Melis, GB; Ronca-Testoni, S1
Thomas, WA1
Kanto, JH1
Olive, G; Rey, E1
Baron, JC; Berger, G; Cepeda, C; Comar, D; Godot, JM; Mazière, M; Menini, C; Naquet, R1
Hamon, M; Soubríe, P; Thiébot, MH1
Abbracchio, MP; Balduini, W; Cagiano, R; Cattabeni, F; Coen, E; Cuomo, V; Lombardelli, G; Peruzzi, G; Ragusa, MC1
Blanchard, JC; Boireau, A; Julou, L2
Abbracchio, MP; Balduini, W; Cattabeni, F; Coen, E; Lombardelli, G; Peruzzi, G1
Cepeda, C; Comar, D; Crouzel, M; Guibert, B; Hantraye, P; Kaijima, M; Maziere, M; Naquet, R; Prenant, C; Sastre, J1
Jeevanjee, F; Johnson, AM; Loudon, JM; Nicholass, JM1
Klieser, E; Lehmann, E; Wolfrum, C1
Breese, GR; Frye, GD; Koepke, KM; Kuhn, CM; Mailman, RB; Mueller, RA; Vogel, RA; Wilson, JH1
Hamon, M; Jobert, A; Soubrié, P; Thiébot, MH1
Catarzi, D; Cecchi, L; Colotta, V; Conti, G; Filacchioni, G; Giusti, L; Lucacchini, A; Martini, C1
Catarzi, D; Cecchi, L; Colotta, V; Filacchioni, G; Giusti, L; Lucacchini, A; Martini, C; Melani, F1
Hiramatsu, M; Ishihara, S; Kameyama, T; Nabeshima, T1
Fiacco, TT; Galler, JR; Rosene, DL; Shultz, PL; Shumsky, JS; Tonkiss, J; Vincitore, M1
Dirse, V; Ivanauskas, L; Kiliuviene, G; Zevzikovas, A1
Gunn, J; Kriger, S; Terrell, AR1

Reviews

2 review(s) available for flunitrazepam and chlordiazepoxide

ArticleYear
Use of benzodiazepines during pregnancy, labour and lactation, with particular reference to pharmacokinetic considerations.
    Drugs, 1982, Volume: 23, Issue:5

    Topics: Anti-Anxiety Agents; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Female; Flunitrazepam; Humans; Infant, Newborn; Labor, Obstetric; Lactation; Lorazepam; Maternal-Fetal Exchange; Nitrazepam; Oxazepam; Pregnancy

1982
[Benzodiazepines and pregnancy. Transplacental passage, labor and lactation].
    L'Encephale, 1983, Volume: 9, Issue:4 Suppl 2

    Topics: Anti-Anxiety Agents; Biotransformation; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Female; Flunitrazepam; Humans; Kinetics; Lorazepam; Maternal-Fetal Exchange; Milk, Human; Nitrazepam; Oxazepam; Postpartum Period; Pregnancy

1983

Other Studies

32 other study(ies) available for flunitrazepam and chlordiazepoxide

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Binding of [3H]flunitrazepam to differentiating rat cerebral cells in culture.
    Brain research, 1979, Nov-16, Volume: 177, Issue:2

    Topics: Age Factors; Animals; Anti-Anxiety Agents; Brain; Chlordiazepoxide; Culture Techniques; Diazepam; Flunitrazepam; Neurons; Rats; Receptors, Drug

1979
Detection of benzodiazepine intake in therapeutic doses by immunoanalysis of urine: two techniques evaluated and modified for improved performance.
    Clinical chemistry, 1992, Volume: 38, Issue:2

    Topics: Adult; Alprazolam; Benzodiazepines; Chlordiazepoxide; False Negative Reactions; Flunitrazepam; Fluorescence Polarization Immunoassay; Humans; Immunoenzyme Techniques; Lorazepam; Male; Middle Aged; Nitrazepam; Triazolam

1992
Laminar distribution of benzodiazepine receptors in visual cortex of adult rat.
    General physiology and biophysics, 1989, Volume: 8, Issue:4

    Topics: Animals; Chlordiazepoxide; Flunitrazepam; Kinetics; Rats; Rats, Inbred Strains; Receptors, GABA-A; Visual Cortex

1989
Effects of chlordiazepoxide, chlorpromazine, diazepam, diphenylhydantoin, flunitrazepam and haloperidol on the voltage-dependent sodium current of isolated mammalian brain neurons.
    Brain research, 1989, Aug-14, Volume: 494, Issue:2

    Topics: Animals; Chlordiazepoxide; Chlorpromazine; Diazepam; Flunitrazepam; Haloperidol; Hippocampus; In Vitro Techniques; Membrane Potentials; Phenytoin; Psychotropic Drugs; Rats; Sodium

1989
Functional and structural correlates of GABA receptor modulation.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Benzodiazepines; Cations, Divalent; Cells, Cultured; Chickens; Chlordiazepoxide; Flunitrazepam; Kinetics; Receptors, GABA-A; Trypsin

1988
Behavioral studies with anxiolytic drugs. III. Antipunishment actions of buspirone in the pigeon do not involve benzodiazepine receptor mechanisms.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Buspirone; Chlordiazepoxide; Columbidae; Diazepam; Flumazenil; Flunitrazepam; Punishment; Pyrimidines; Receptors, GABA-A

1986
Prenatal chlordiazepoxide effects on metrazol seizures and benzodiazepine receptors density in adult albino rats.
    Life sciences, 1985, May-06, Volume: 36, Issue:18

    Topics: Animals; Brain; Cerebellum; Cerebral Cortex; Chlordiazepoxide; Drug Resistance; Female; Flunitrazepam; Pentylenetetrazole; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1985
Central effects of nicotinamide and inosine which are not mediated through benzodiazepine receptors.
    British journal of pharmacology, 1985, Volume: 84, Issue:3

    Topics: Action Potentials; Animals; Benzodiazepinones; Bicuculline; Binding, Competitive; Brain; Chlordiazepoxide; Convulsants; Female; Flumazenil; Flunitrazepam; In Vitro Techniques; Inosine; Male; Membranes; Niacinamide; Purkinje Cells; Rats; Rats, Inbred Strains; Receptors, GABA-A; Social Behavior

1985
Synthesis and interaction of 5-(substituted-phenyl)-3-methyl-6,7-dihydropyrazolo[4,3-e] [1,4]diazepin-8(7H)-ones with benzodiazepine receptors in rat cerebral cortex.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:5

    Topics: Animals; Azepines; Binding, Competitive; Cerebral Cortex; Chlordiazepoxide; Diazepam; Flunitrazepam; In Vitro Techniques; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship

1985
Benzodiazepine interactions with central thyroid-releasing hormone binding sites: characterization and physiological significance.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Amygdala; Animals; Benzodiazepines; Brain; Cerebral Cortex; Chlordiazepoxide; Corpus Striatum; Cyclic GMP; Flunitrazepam; Kinetics; Male; Membranes; Midazolam; Pentobarbital; Pyrazoles; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Thyrotropin-Releasing Hormone; Sleep; Thiazolidines; Thyrotropin; Thyrotropin-Releasing Hormone

1986
Evidence of specific benzodiazepine binding to myometrial membrane preparations from human pregnant uterus.
    Acta obstetricia et gynecologica Scandinavica, 1986, Volume: 65, Issue:4

    Topics: Adult; Benzodiazepines; Benzodiazepinones; Cell Membrane; Chlordiazepoxide; Diazepam; Female; Flunitrazepam; Humans; Lorazepam; Myometrium; Pregnancy; Receptors, Cell Surface

1986
Peptide derivatives as prodrugs.
    Biochemical Society transactions, 1986, Volume: 14, Issue:2

    Topics: Amino Acids; Animals; Bacteria; Biological Availability; Biological Transport, Active; Chlordiazepoxide; Diazepam; Flunitrazepam; Flurazepam; Humans; Kinetics; Nitrazepam; Papio; Rats

1986
Positron tomography. A new method for in vivo brain studies of benzodiazepine, in animal and in man.
    Advances in biochemical psychopharmacology, 1981, Volume: 26

    Topics: Animals; Brain; Chlordiazepoxide; Flunitrazepam; Humans; Kinetics; Papio; Receptors, Drug; Receptors, GABA-A; Tomography, Emission-Computed

1981
Attenuation of induced-anxiety in rats by chlordiazepoxide: role of raphe dorsalis benzodiazepine binding sites and serotoninergic neurons.
    Neuroscience, 1982, Volume: 7, Issue:9

    Topics: 5,7-Dihydroxytryptamine; Animals; Arousal; Brain Stem; Chlordiazepoxide; Conditioning, Operant; Dose-Response Relationship, Drug; Flunitrazepam; Ganglia, Spinal; Male; Metergoline; Neurons; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Receptors, Serotonin; Serotonin; Tryptophan Hydroxylase

1982
Early postnatal chlordiazepoxide administration: permanent behavioural effects in the mature rat and possible involvement of the GABA-benzodiazepine system.
    Psychopharmacology, 1983, Volume: 81, Issue:3

    Topics: Animals; Animals, Newborn; Avoidance Learning; Behavior, Animal; Brain Chemistry; Chlordiazepoxide; Female; Flunitrazepam; Kinetics; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
Brain receptors and zopiclone.
    Pharmacology, 1983, Volume: 27 Suppl 2

    Topics: Animals; Azabicyclo Compounds; Binding, Competitive; Brain; Cerebellum; Chlordiazepoxide; Diazepam; Flunitrazepam; Hippocampus; Hypnotics and Sedatives; In Vitro Techniques; Male; Mice; Nitrazepam; Piperazines; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A

1983
Chronic chlordiazepoxide treatment on adult and newborn rats: effect on the GABA-benzodiazepine receptor complex.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Aging; Animals; Animals, Newborn; Chlordiazepoxide; Female; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1983
[In vivo study of benzodiazepine receptors using positron emission tomography].
    L'Encephale, 1983, Volume: 9, Issue:4 Suppl 2

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Chlordiazepoxide; Flumazenil; Flunitrazepam; Kinetics; Lorazepam; Male; Papio; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Stereoisomerism

1983
Brain receptors and zopiclone.
    International pharmacopsychiatry, 1982, Volume: 17 Suppl 2

    Topics: Animals; Azabicyclo Compounds; Barbiturates; Binding, Competitive; Brain; Chlordiazepoxide; Cyclic GMP; Diazepam; Flunitrazepam; Hippocampus; Hypnotics and Sedatives; In Vitro Techniques; Male; Piperazines; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A

1982
Enhancement of [3H]flunitrazepam binding by mianserin, in vivo.
    Neuroscience letters, 1984, May-18, Volume: 46, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Convulsants; Dibenzazepines; Drinking Behavior; Flumazenil; Flunitrazepam; Kinetics; Male; Mianserin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1984
Single case experiments in psychopharmacological trials.
    Neuropsychobiology, 1984, Volume: 12, Issue:2-3

    Topics: Adult; Amitriptyline; Chlordiazepoxide; Clinical Trials as Topic; Drug Combinations; Female; Flunitrazepam; Heart Diseases; Humans; Male; Middle Aged; Psychopharmacology; Psychophysiologic Disorders; Psychotropic Drugs; Random Allocation; Sleep Wake Disorders

1984
Attenuation of the effects of punishment by ethanol: comparisons with chlordiazepoxide.
    Psychopharmacology, 1980, Volume: 71, Issue:2

    Topics: Animals; Avoidance Learning; Brain; Chlordiazepoxide; Conflict, Psychological; Ethanol; Flunitrazepam; Male; Membranes; Mice; Punishment; Rats

1980
Serotoninergic control of punished behavior: effects of intra-raphe microinjections of chlordiazepoxide, GABA and 5-HT on behavioral suppression in rats.
    Journal de physiologie, 1981, Volume: 77, Issue:2-3

    Topics: 5,7-Dihydroxytryptamine; Animals; Behavior, Animal; Chlordiazepoxide; Desipramine; Flunitrazepam; gamma-Aminobutyric Acid; Male; Punishment; Raphe Nuclei; Rats; Rats, Inbred Strains; Serotonin

1981
Tricyclic heteroaromatic systems pyrazolo[1,5-a]quinoxalines: synthesis and benzodiazepine receptor activity.
    Farmaco (Societa chimica italiana : 1989), 1993, Volume: 48, Issue:8

    Topics: Animals; Binding, Competitive; Cattle; Cerebral Cortex; Chlordiazepoxide; Flunitrazepam; In Vitro Techniques; Pyrazoles; Quinoxalines; Receptors, GABA-A

1993
Tricyclic heteroaromatic systems 1,2,4-triazolo[1,5-a]quinoxalines: synthesis and benzodiazepine receptor activity.
    Farmaco (Societa chimica italiana : 1989), 1993, Volume: 48, Issue:8

    Topics: Animals; Binding, Competitive; Cattle; Cerebral Cortex; Chlordiazepoxide; Flunitrazepam; In Vitro Techniques; Quinoxalines; Receptors, GABA-A; Triazoles

1993
Development of tolerance to anxiolytic effects of chlordiazepoxide in elevated plus-maze test and decrease of GABAA receptors.
    Journal of neural transmission. General section, 1993, Volume: 91, Issue:1

    Topics: Animals; Azides; Benzodiazepines; Binding, Competitive; Brain Chemistry; Chlordiazepoxide; Down-Regulation; Drug Tolerance; Exploratory Behavior; Flunitrazepam; Male; Mice; Receptors, GABA-A

1993
Chlordiazepoxide-induced spatial learning deficits: dose-dependent differences following prenatal malnutrition.
    Pharmacology, biochemistry, and behavior, 2000, Jan-01, Volume: 65, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Body Weight; Chlordiazepoxide; Chlorides; Dose-Response Relationship, Drug; Female; Flunitrazepam; Gene Expression Regulation, Developmental; Learning Disabilities; Motor Activity; Pregnancy; Pregnancy Complications; Protein Deficiency; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

2000
[Analysis of benzodiazepine derivative mixture by gas-liquid chromatography].
    Medicina (Kaunas, Lithuania), 2002, Volume: 38, Issue:3

    Topics: Anti-Anxiety Agents; Benzodiazepines; Chlordiazepoxide; Chromatography, Gas; Flunitrazepam; Humans; Medazepam; Models, Theoretical; Nitrazepam; Oxazepam

2002
Simultaneous determination and quantification of 12 benzodiazepines in serum or whole blood using UPLC/MS/MS.
    Methods in molecular biology (Clifton, N.J.), 2010, Volume: 603

    Topics: Alprazolam; Benzodiazepines; Chlordiazepoxide; Chromatography, Liquid; Clonazepam; Flunitrazepam; Humans; Lorazepam; Midazolam; Nordazepam; Oxazepam; Reproducibility of Results; Tandem Mass Spectrometry

2010