flunitrazepam has been researched along with bicuculline in 79 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 35 (44.30) | 18.7374 |
1990's | 33 (41.77) | 18.2507 |
2000's | 11 (13.92) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Chou, WH; McMahon, T; Messing, RO; Newton, PM; Qi, ZH; Shokat, KM; Song, M; Wallace, MJ; Wang, D; Zhang, C | 1 |
Haefely, W; Polc, P | 1 |
Dudai, Y | 1 |
Hales, TG; Kim, H; Longoni, B; Olsen, RW; Tobin, AJ | 1 |
Hirouchi, M; Kuriyama, K; Ohkuma, S | 1 |
Wilson, MA | 1 |
Miller, CL; Quinn, MR | 1 |
Biggio, G; Concas, A; Gessa, GL; Peduto, VA; Santoro, G | 1 |
Dawson, RM; Poretski, M | 1 |
Lummis, SC; Rauh, JJ; Sattelle, DB; Wong, JF | 1 |
Airaksinen, MM; MacDonald, E; Rägo, L; Saano, V | 1 |
De Luca, C; De Medici, D; Massotti, M | 1 |
Albers, HE; Liou, SY; Shibata, S; Ueki, S | 1 |
Crabbe, JC; Diggs, HE; Farrell, E; Feller, DJ; Merrill, C | 1 |
Quinn, MR | 1 |
Danielou, G; Lloyd, GK; Thuret, F | 1 |
Costa, E; Mienville, JM; Vicini, S | 2 |
David, JA; Pinnock, RD; Sattelle, DB; Wafford, KA | 1 |
Chiu, TH; Rosenberg, HC; Tietz, EI | 1 |
Jacqmin, P; Jacquot, C; Lesne, M; Rouch, C; Trouvin, JH | 1 |
Gossuin, A; Laterre, C; Maloteaux, JM; Octave, JN; Trouet, A | 1 |
Cox, DH; Guidotti, A; Santi, MR | 1 |
Barone, D; Colombo, G; Gallico, L; Sala, A; Tarzia, G; Winters, G | 1 |
McCabe, RT; Olsen, RW; Wamsley, JK; Yezuita, JP | 1 |
Ho, IK; Hoskins, B; Ito, Y; Lim, DK | 1 |
Collins, AC; Freund, RK; Jungschaffer, DA; Wehner, JM | 1 |
Gobbi, M; Mennini, T; Perin, L; Salmona, M | 1 |
Abalis, IM; Eldefrawi, AT; Eldefrawi, ME | 1 |
Kuriyama, K; Taguchi, J | 1 |
Bold, JM; Gardner, CR; Walker, RJ | 1 |
Lee, RJ; Lomax, P; McCabe, RT; Olsen, RW; Wamsley, JK | 1 |
Haefely, W; Möhler, H; Richards, JG; Schoch, P | 1 |
Kontro, P; Malminen, O | 1 |
McCabe, RT; Wamsley, JK | 1 |
Alho, H; Costa, E; Mienville, JM; Santi, MR; Vaccarino, FM; Vicini, S | 1 |
Crabbe, JC; Feller, DJ; Harris, RA | 1 |
Zarkovsky, AM | 1 |
Hösli, E; Hösli, L; Möhler, H; Richards, JG | 1 |
Drexler, G; Karobath, M; Supavilai, P | 1 |
Karobath, M; Supavilai, P | 1 |
Dehaven, R; Pong, SS; Wang, CC | 1 |
Collins, RJ; Daniels, EG; Sethy, VH | 1 |
Benson, DI; Klepner, CA; Squires, RF | 1 |
Malick, JB; Regan, JW; Roeske, WR; Yamamura, HI; Yamamura, SH | 1 |
Brinton, RE; Gee, KW; Yamamura, HI | 1 |
Hösli, E; Hösli, L | 1 |
Gähwiler, BH; Maurer, R; Wüthrich, HJ | 1 |
Regan, JW; Roeske, WR; Yamamura, HI | 1 |
Bormann, J; Feigenspan, A | 1 |
Nabeshima, A; Saito, T; Takahata, N; Toki, S | 1 |
Niles, LP; Tenn, CC | 1 |
Bormann, J; Feigenspan, A; Wässle, H | 1 |
Inglefield, JR; Kellogg, CK | 1 |
Cancedda, E; Corda, MG; Giorgi, O; Lecca, D; Orlandi, M | 1 |
Belelli, D; Chen, R; Lambert, JJ; Lan, NC; Peters, JA; Reyes, A | 1 |
Dunn, SM; Thuynsma, RP | 1 |
Liljequist, S; Tabakoff, B | 1 |
Barton, JM; Olson, MS; Svetlov, SI | 1 |
Simmonds, MA; Zhong, Y | 2 |
Fueta, Y; Janjua, NA; Mita, T; Murai, Y; Ohmori, O; Ohno, K; Ono, T | 1 |
Davies, PA; Hales, TG; Hanna, MC; Kirkness, EF | 1 |
Pomés, A; Rodríguez-Farré, E; Suñol, C; Vale, C | 1 |
Belachew, S; Coucke, P; Goffin, F; Lefebvre, PP; Malgrange, B; Moonen, G; Rigo, JM; Van de Water, TR; Xhauflaire, G | 1 |
Bristow, DR; Brown, MJ; Coldwell, MC; Wood, MD | 1 |
Buckingham, SD; Rauh, J; Sattelle, DB; Schnee, M | 1 |
Higashi, H; Nagata, K; Park, JS; Yoshimura, M | 1 |
Chéry, N; de Koninck, Y | 2 |
Crites, GJ; Goldenberg, R; Harrawood, D; Malatynska, E; Matheson, GK; Schindler, NL; Tunnicliff, G; Weinzapfel, D; Yochum, A | 1 |
Findlay, GS; Harris, RA; Harrison, NL; Ueno, S | 2 |
Baufreton, J; Bioulac, B; Dovero, S; Dufy, B; Garret, M; Taupignon, A | 1 |
Caruso, RR; Castro, NG; Costa, PR; da Silva, AJ; Lopes, DV; Noël, F | 1 |
García, DA; Nolan, MV; Perillo, MA; Sánchez, ME; Turina, AV | 1 |
Ariwodola, OJ; Weiner, JL | 1 |
Baur, R; Senn, M; Séquin, U; Sigel, E; Simmen, U | 1 |
Dzirkale, Z; Klusa, V; Krigere, L; Mezhapuke, R; Muceniece, R; Rumaks, J; Saleniece, K; Zharkova, O | 1 |
1 review(s) available for flunitrazepam and bicuculline
Article | Year |
---|---|
Benzodiazepine receptors resolved.
Topics: Animals; Antibodies, Monoclonal; Autoradiography; Benzodiazepines; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Clonazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Histocytochemistry; Humans; Immunologic Techniques; Ionophores; Muscimol; Neurons; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Spinal Cord; Synapses; Tissue Distribution | 1986 |
78 other study(ies) available for flunitrazepam and bicuculline
Article | Year |
---|---|
Protein kinase C epsilon regulates gamma-aminobutyrate type A receptor sensitivity to ethanol and benzodiazepines through phosphorylation of gamma2 subunits.
Topics: Adenosine Triphosphate; Allosteric Regulation; Animals; Benzodiazepines; Cells, Cultured; Enzyme Activation; Ethanol; Hippocampus; Humans; Mice; Mice, Knockout; Mutation; Phosphorylation; Protein Kinase C-epsilon; Protein Kinase Inhibitors; Protein Subunits; Pyridines; Receptors, GABA-A; Sensitivity and Specificity; Serine; Zolpidem | 2007 |
Effects of two benzodiazepines, phenobarbitone, and baclofen on synaptic transmission in the cat cuneate nucleus.
Topics: Aminobutyrates; Aminooxyacetic Acid; Animals; Anti-Anxiety Agents; Baclofen; Bicuculline; Cats; Diazepam; Drug Interactions; Evoked Potentials; Flunitrazepam; Glutamate Decarboxylase; Medulla Oblongata; Neural Inhibition; Phenobarbital; Picrotoxin; Propionates; Semicarbazides; Synapses; Synaptic Transmission | 1976 |
Modulation of benzodiazepine binding sites in calf cortex by an endogenous factor and GABAergic ligands.
Topics: Animals; Anti-Anxiety Agents; Bicuculline; Cattle; Cerebral Cortex; Cycloleucine; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Nerve Tissue Proteins; Receptors, Drug | 1979 |
Immortalized hypothalamic GT1-7 neurons express functional gamma-aminobutyric acid type A receptors.
Topics: Anesthetics; Animals; Barbiturates; Base Sequence; Bicuculline; Cell Line, Transformed; Cell Membrane; Chloride Channels; Diazepam; Electrophysiology; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Hypothalamus; Membrane Proteins; Mice; Molecular Sequence Data; Muscimol; Neurons; Peptides; Polymerase Chain Reaction; Receptors, GABA-A; RNA, Messenger; Sensitivity and Specificity; Steroids; Tritium; Tumor Cells, Cultured; Zinc | 1992 |
Muscimol-induced reduction of GABAA receptor alpha 1-subunit mRNA in primary cultured cerebral cortical neurons.
Topics: Animals; Bicuculline; Blotting, Northern; Cells, Cultured; Cerebral Cortex; Flunitrazepam; Mice; Muscimol; Neurons; Peptide Fragments; Receptors, GABA-A; Ribonucleases; RNA, Messenger | 1992 |
Influences of gender, gonadectomy, and estrous cycle on GABA/BZ receptors and benzodiazepine responses in rats.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Bicuculline; Brain; Brain Chemistry; Diazepam; Estrus; Female; Flunitrazepam; Male; Orchiectomy; Ovariectomy; Radioimmunoassay; Radioligand Assay; Rats; Receptors, GABA-A; Sex Characteristics | 1992 |
Taurine allosterically modulates flunitrazepam binding to synaptic membranes.
Topics: Animals; Bicuculline; Binding, Competitive; Cerebral Cortex; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Sprague-Dawley; Synaptic Membranes; Taurine; Temperature | 1992 |
Biochemical and electrophysiologic evidence that propofol enhances GABAergic transmission in the rat brain.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Male; Membrane Proteins; Propofol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Transmission | 1991 |
The interaction of tacrine with benzodiazepine and GABA binding sites of guinea pig brain.
Topics: Animals; Bicuculline; Binding, Competitive; Brain Chemistry; Cerebral Cortex; Flunitrazepam; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Kinetics; Radioligand Assay; Receptors, GABA-A; Tacrine | 1991 |
Pharmacology of insect GABA receptors.
Topics: Acetylcholine; Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Female; Flunitrazepam; gamma-Aminobutyric Acid; Houseflies; Insecticides; Male; Membrane Proteins; Nervous System; Neurons; Periplaneta; Pregnanes; Receptors, GABA-A; Synapses | 1991 |
The effect of medetomidine on GABA and benzodiazepine receptors in vivo: lack of anxiolytic but some evidence of possible stress-protective activity.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Bicuculline; Brain; Cerebral Cortex; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Imidazoles; Kidney; Male; Medetomidine; Muscimol; Myocardium; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Stimulation, Chemical; Stress, Physiological; Tritium | 1991 |
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem | 1990 |
Effects of GABA and anxiolytics on the single unit discharge of suprachiasmatic neurons in rat hypothalamic slices.
Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Baclofen; Bicuculline; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Hypothalamus; In Vitro Techniques; Muscimol; Neurons; Piperazines; Rats; Receptors, GABA-A; Suprachiasmatic Nucleus | 1990 |
Effect of chronic ivermectin treatment on GABA receptor function in ethanol withdrawal-seizure prone and resistant mice.
Topics: Animals; Bicuculline; Brain Chemistry; Ethanol; Flunitrazepam; Ivermectin; Mice; Ovum; Oxyuroidea; Receptors, GABA-A; Seizures | 1990 |
Taurine allosterically modulates binding sites of the GABAA receptor.
Topics: Allosteric Regulation; Animals; Bicuculline; Flunitrazepam; In Vitro Techniques; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Taurine; Temperature | 1990 |
The activity of zolpidem and other hypnotics within the gamma-aminobutyric acid (GABAA) receptor supramolecular complex, as determined by 35S-t-butylbicyclophosphorothionate (35S-TBPS) binding to rat cerebral cortex membranes.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Zolpidem | 1990 |
Flunitrazepam action on the GABA-Cl ionophore complex in rat cortical neurons in culture: a patch-clamp study.
Topics: Animals; Bicuculline; Cerebral Cortex; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Neurons; Osmolar Concentration; Rats | 1986 |
GABA receptors on the cell-body membrane of an identified insect motor neuron.
Topics: Androstanes; Animals; Azasteroids; Bicuculline; Chlorides; Cockroaches; Dibenzazepines; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Membrane Potentials; Microelectrodes; Motor Neurons; Nipecotic Acids; Periplaneta; Picrotoxin; Receptors, GABA-A | 1988 |
Chloride channel modulation through the benzodiazepine recognition site.
Topics: Animals; Bicuculline; Carbolines; Cells, Cultured; Chlorides; Convulsants; Flumazenil; Flunitrazepam; Ion Channels; Neurons; Receptors, GABA-A | 1988 |
Regional GABA/benzodiazepine receptor/chloride channel coupling after acute and chronic benzodiazepine treatment.
Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Bicuculline; Brain; Chlorides; Diazepam; Flunitrazepam; Flurazepam; gamma-Aminobutyric Acid; Ion Channels; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stimulation, Chemical | 1989 |
Benzodiazepine receptors are involved in tabernanthine-induced tremor: in vitro and in vivo evidence.
Topics: Alkaloids; Animals; Behavior, Animal; Bicuculline; Binding, Competitive; Female; Flunitrazepam; Ibogaine; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes; Tremor | 1987 |
GABA induces down-regulation of the benzodiazepine-GABA receptor complex in the rat cultured neurons.
Topics: Animals; Bicuculline; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Neurons; Radioligand Assay; Rats; Receptors, GABA-A | 1987 |
Heterogeneity of gamma-aminobutyric acid/benzodiazepine/beta-carboline receptor complex in rat spinal cord.
Topics: Animals; Bicuculline; Binding, Competitive; Carbolines; Cerebellum; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Receptors, GABA-A; Spinal Cord; Synaptic Membranes | 1988 |
3-(1-Iminoethyl)-4,5-cycloalkylpyridine-2,6-diol derivatives. A novel class of benzodiazepine receptor antagonists and partial agonists.
Topics: Animals; Bicuculline; Binding, Competitive; Chemical Phenomena; Chemistry; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Mice; Muscle Relaxants, Central; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1987 |
Osmotic shock: a method to eliminate endogenous gamma-aminobutyric acid and account for the influence on benzodiazepine binding affinity in autoradiographic studies.
Topics: Animals; Autoradiography; Benzodiazepines; Bicuculline; Binding Sites; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Male; Osmotic Pressure; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
Bicuculline up-regulation of GABAA receptors in rat brain.
Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Corpus Striatum; Flunitrazepam; Frontal Lobe; gamma-Aminobutyric Acid; Male; Muscimol; Octoxynol; Polyethylene Glycols; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra; Synaptic Membranes | 1988 |
Evidence for modulation of GABAergic neurotransmission by nicotine.
Topics: Action Potentials; Allylglycine; Animals; Bicuculline; Brain Chemistry; Female; Flunitrazepam; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hippocampus; In Vitro Techniques; Mice; Mice, Inbred DBA; Nicotine; Receptors, GABA-A | 1988 |
Rapid internalization of benzodiazepine receptors in the rat cortex induced by handling.
Topics: Animals; Bicuculline; Carbolines; Cerebral Cortex; Corticosterone; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Ligands; Male; Rats; Receptors, GABA-A; Stress, Physiological; Synaptic Membranes; Viscosity | 1988 |
Actions of avermectin B1a on the gamma-aminobutyric acidA receptor and chloride channels in rat brain.
Topics: Animals; Bicuculline; Binding, Competitive; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Flunitrazepam; Ivermectin; Kinetics; Male; Membrane Proteins; Muscimol; Rats; Receptors, GABA-A | 1986 |
Functional coupling of gamma-aminobutyric acid (GABA)A and benzodiazepine type II receptors: analysis using purified GABA/benzodiazepine receptor complex from bovine cerebral cortex.
Topics: Animals; Antipsychotic Agents; Bicuculline; Cattle; Cerebral Cortex; Flumazenil; Flunitrazepam; In Vitro Techniques; Kinetics; Muscimol; Pyridazines; Receptors, GABA-A | 1987 |
Central effects of nicotinamide and inosine which are not mediated through benzodiazepine receptors.
Topics: Action Potentials; Animals; Benzodiazepinones; Bicuculline; Binding, Competitive; Brain; Chlordiazepoxide; Convulsants; Female; Flumazenil; Flunitrazepam; In Vitro Techniques; Inosine; Male; Membranes; Niacinamide; Purkinje Cells; Rats; Rats, Inbred Strains; Receptors, GABA-A; Social Behavior | 1985 |
Benzodiazepine/gamma-aminobutyric acid receptor deficit in the midbrain of the seizure-susceptible gerbil.
Topics: Animals; Bicuculline; Diazepam; Disease Models, Animal; Flunitrazepam; Gerbillinae; Mesencephalon; Muscimol; Pentobarbital; Receptors, GABA-A; Seizures | 1985 |
Modulation of the GABA-benzodiazepine receptor complex by taurine in rat brain membranes.
Topics: Animals; Bicuculline; Brain; Flunitrazepam; gamma-Aminobutyric Acid; Male; Rats; Receptors, GABA-A; Taurine | 1986 |
Autoradiographic localization of subcomponents of the macromolecular GABA receptor complex.
Topics: Animals; Autoradiography; Baclofen; Bicuculline; Binding, Competitive; Brain Chemistry; Flunitrazepam; Macromolecular Substances; Muscimol; Rats; Receptors, GABA-A; Tissue Distribution; Tritium | 1986 |
Modulation of gamma-aminobutyric acid-mediated inhibitory synaptic currents in dissociated cortical cell cultures.
Topics: Animals; Bicuculline; Carbolines; Cells, Cultured; Cerebral Cortex; Electric Conductivity; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Potentials; Neural Inhibition; Rats; Synapses | 1986 |
Differences in GABA activity between ethanol withdrawal seizure prone and resistant mice.
Topics: Animals; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Ethanol; Female; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Picrotoxin; Seizures; Substance Withdrawal Syndrome | 1988 |
Bicuculline-sensitive and insensitive effects of THIP on the binding of [3H]flunitrazepam.
Topics: Animals; Bicuculline; Brain; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Isoxazoles; Male; Osmolar Concentration; Oxazoles; Rats; Rats, Inbred Strains; Sodium Chloride; Tritium | 1987 |
Autoradiographic localization of binding sites for [3H]gamma-aminobutyrate, [3H]muscimol,(+)[3H]bicuculline methiodide and [3H] flunitrazepam in cultures of rat cerebellum and spinal cord.
Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Autoradiography; Bicuculline; Binding Sites; Cells, Cultured; Cerebellum; Female; Fetus; Flunitrazepam; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Pregnancy; Rats; Receptors, Drug; Spinal Cord; Tritium | 1980 |
Modulation by picrotoxin and IPTBO of 3H-flunitrazepam binding to the GABA/benzodiazepine receptor complex of rat cerebellum.
Topics: Animals; Anti-Anxiety Agents; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Male; Membranes; Organophosphorus Compounds; Picrotoxin; Rats; Receptors, Drug; Receptors, GABA-A; Temperature | 1981 |
Action of pyrazolopyridines as modulators of [3H]flunitrazepam binding to the gaba/benzodiazepine receptor complex of the cerebellum.
Topics: Animals; Anti-Anxiety Agents; Bicuculline; Binding Sites; Cerebellum; Chlorides; Etazolate; Flunitrazepam; Isoxazoles; Male; Muscimol; Nicotinic Acids; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Tritium | 1981 |
Stimulation of benzodiazepine binding to rat brain membranes and solubilized receptor complex by avermectin B1a and gamma-aminobutyric acid.
Topics: Animals; Anthelmintics; Anti-Anxiety Agents; Bicuculline; Brain; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Ivermectin; Lactones; Male; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Synaptic Membranes | 1981 |
Determination of biological activity of adinazolam and its metabolites.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Bicuculline; Brain; Cell Membrane; Flunitrazepam; In Vitro Techniques; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1984 |
Multiple benzodiazepine receptor complexes: some benzodiazepine recognition sites are coupled to GABA receptors and ionophores.
Topics: Animals; Anions; Benzodiazepines; Bicuculline; Brain; Buffers; Flunitrazepam; gamma-Aminobutyric Acid; Haplorhini; Hot Temperature; Ionophores; Isonicotinic Acids; Isoxazoles; Macromolecular Substances; Papio; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter | 1980 |
gamma-Aminobutyric acid enhancement of CL 218,872 affinity and evidence of benzodiazepine receptor heterogeneity.
Topics: Animals; Bicuculline; Binding, Competitive; Brain; Cattle; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kidney; Kinetics; Pyridazines; Receptors, Drug; Receptors, GABA-A; Retina | 1981 |
PK 8165 and PK 9084, two quinoline derivatives with anxiolytic properties, antagonize the anticonvulsant effects of diazepam.
Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Brain; Diazepam; Drug Antagonism; Flunitrazepam; gamma-Aminobutyric Acid; Male; Mice; Quinolines; Receptors, Cell Surface; Receptors, GABA-A; Seizures | 1983 |
Autoradiographic localization of binding sites for inhibitory amino acids and their antagonists in cultured rat CNS.
Topics: Amino Acids; Animals; Animals, Newborn; Autoradiography; Bicuculline; Brain Stem; Cells, Cultured; Cerebellum; Female; Fetus; Flunitrazepam; gamma-Aminobutyric Acid; Muscimol; Neuroglia; Neurons; Pregnancy; Rats; Receptors, Cell Surface; Spinal Cord; Tritium | 1983 |
Pitrazepin, a novel GABAA antagonist.
Topics: Animals; Baclofen; Bicuculline; Binding, Competitive; Culture Techniques; Dibenzazepines; Flunitrazepam; GABA Antagonists; Hippocampus; Hypothalamus; Membrane Potentials; Muscimol; Neurons; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Muscarinic | 1984 |
The benzodiazepine receptor: its development and its modulation by gamma-aminobutyric acid.
Topics: Age Factors; Aminobutyrates; Animals; Benzodiazepines; Bicuculline; Brain Chemistry; Female; Fetus; Flunitrazepam; gamma-Aminobutyric Acid; Mice; Mice, Inbred Strains; Pregnancy; Receptors, Drug | 1980 |
Differential pharmacology of GABAA and GABAC receptors on rat retinal bipolar cells.
Topics: Animals; Bicuculline; Binding Sites; Cells, Cultured; Chickens; Chloride Channels; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; GABA-A Receptor Antagonists; Hexachlorocyclohexane; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Pyridazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Retina; Sesterterpenes; Signal Transduction | 1994 |
[Changes in GABAA/benzodiazepine receptor complex function in the pentobarbital-dependent rat. II: Strain differences between Lewis and Wistar-Kyoto rats].
Topics: Animals; Bicuculline; Brain; Chlorine; Ethanol; Female; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Lew; Rats, Inbred WKY; Receptors, GABA-A; Substance-Related Disorders | 1995 |
Central-type benzodiazepine receptors mediate the antidopaminergic effect of clonazepam and melatonin in 6-hydroxydopamine lesioned rats: involvement of a GABAergic mechanism.
Topics: Animals; Apomorphine; Behavior, Animal; Bicuculline; Clonazepam; Corpus Striatum; Dopamine Agonists; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Isoquinolines; Male; Melatonin; Oxidopamine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 1995 |
Pharmacology of GABA receptor Cl- channels in rat retinal bipolar cells.
Topics: Animals; Animals, Newborn; Bicuculline; Cells, Cultured; Chloride Channels; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Membrane Potentials; Membrane Proteins; Neurons; Pentobarbital; Photoreceptor Cells; Picrotoxin; Pregnanediones; Rats; Receptors, GABA-A; Sesterterpenes; Strychnine | 1993 |
Hypothalamic GABAA receptor blockade modulates cerebral cortical systems sensitive to acute stressors.
Topics: Animals; Behavior, Animal; Bicuculline; Brain Chemistry; Cerebral Cortex; Chlorides; Dopamine; Flunitrazepam; Frontal Lobe; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hypothalamus; Male; Rats; Stress, Psychological | 1994 |
Allosteric modulation of [35S]TBPS-binding in the cerebral cortex of the rat during postnatal development.
Topics: Aging; Allosteric Regulation; Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Convulsants; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stereoisomerism; Sulfur Radioisotopes | 1994 |
Cloning and functional expression of a Drosophila gamma-aminobutyric acid receptor.
Topics: Amino Acid Sequence; Animals; Base Sequence; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cloning, Molecular; Convulsants; DNA Primers; DNA, Complementary; Drosophila melanogaster; Female; Flunitrazepam; gamma-Aminobutyric Acid; Gene Expression; Macromolecular Substances; Molecular Sequence Data; Muscimol; Oocytes; Pentobarbital; Picrotoxin; Polymerase Chain Reaction; Receptors, GABA; Receptors, GABA-A; Transcription, Genetic; Xenopus laevis | 1994 |
Reconstitution of purified GABAA receptors: ligand binding and chloride transporting properties.
Topics: Animals; Bicuculline; Biological Transport; Brain Chemistry; Cattle; Chlorides; Chromatography, Affinity; Dose-Response Relationship, Drug; Flow Injection Analysis; Flunitrazepam; Ligands; Liposomes; Membrane Proteins; Muscimol; Picrotoxin; Quinolinium Compounds; Receptors, GABA-A | 1994 |
Bicuculline-produced regional differences in the modulation of 35S-TBPS binding by GABA, pentobarbital and diazepam in mouse cerebellum and cortex.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebellum; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Phenobarbital; Receptors, GABA-A | 1993 |
The specific binding of the platelet-activating factor (PAF) receptor antagonist WEB 2086 and the benzodiazepine flunitrazepam to rat hepatocytes.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Azepines; Benzodiazepinones; Bicuculline; Cells, Cultured; Clonazepam; Convulsants; Flunitrazepam; Kinetics; Liver; Male; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Triazoles; Tritium | 1996 |
Pharmacological characterisation of multiple components in the enhancement by pregnanolone and propofol of [3H]flunitrazepam binding to GABAA receptors.
Topics: Anesthetics, Intravenous; Animals; Bicuculline; Flunitrazepam; GABA Agonists; GABA Modulators; In Vitro Techniques; Male; Muscimol; Pregnanolone; Progesterone; Propofol; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Membranes | 1996 |
Granule cell disinhibition in dentate gyrus of genetically seizure susceptible El mice.
Topics: Aging; Animals; Anticonvulsants; Bicuculline; Chromatography, High Pressure Liquid; Dentate Gyrus; Electrophysiology; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Phenobarbital; Seizures | 1997 |
Insensitivity to anaesthetic agents conferred by a class of GABA(A) receptor subunit.
Topics: Amino Acid Sequence; Anesthetics, Intravenous; Animals; Bicuculline; Brain; Cell Line; Consensus Sequence; DNA, Complementary; Flumazenil; Flunitrazepam; GABA Agents; gamma-Aminobutyric Acid; Humans; Molecular Sequence Data; Muscimol; Pentobarbital; Picrotoxin; Pregnanolone; Propofol; Rats; Receptors, GABA-A; Recombinant Proteins; RNA, Messenger; Transfection | 1997 |
Allosteric interactions between gamma-aminobutyric acid, benzodiazepine and picrotoxinin binding sites in primary cultures of cerebellar granule cells. Differential effects induced by gamma- and delta-hexachlorocyclohexane.
Topics: Animals; Bicuculline; Cells, Cultured; Cerebellum; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hexachlorocyclohexane; Isomerism; Kinetics; Rats; Receptors, GABA-A | 1997 |
Diazepam-insensitive GABAA receptors on postnatal spiral ganglion neurones in culture.
Topics: Animals; Animals, Newborn; Baclofen; Bicuculline; Carbolines; Cells, Cultured; Convulsants; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Spiral Ganglion; Zinc | 1997 |
Measurement of GABAA receptor function in rat cultured cerebellar granule cells by the Cytosensor microphysiometer.
Topics: Animals; Benzodiazepines; Bicuculline; Cell Count; Cells, Cultured; Cerebellum; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hydrogen-Ion Concentration; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 1997 |
Interactions between loreclezole, chlormethiazole and pentobarbitone at GABA(A) receptors: functional and binding studies.
Topics: Animals; Anticonvulsants; Bicuculline; Chlormethiazole; Flunitrazepam; In Vitro Techniques; Male; Medulla Oblongata; Pentobarbital; Rats; Rats, Wistar; Receptors, GABA-A; Triazoles | 1997 |
Pharmacology of skeletal muscle GABA-gated chloride channels in the cockroach Periplaneta americana.
Topics: Animals; Bicuculline; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Flunitrazepam; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channel Gating; Isonicotinic Acids; Male; Motor Neurons; Muscle, Skeletal; Periplaneta; Picrotoxin; Receptors, GABA; Sesterterpenes | 1997 |
Bicuculline-resistant, Cl- dependent GABA response in the rat spinal dorsal horn.
Topics: Animals; Bicuculline; Chloride Channels; Evoked Potentials; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Male; Neurons; Picrotoxin; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Gelatinosa; Thiopental | 1999 |
Junctional versus extrajunctional glycine and GABA(A) receptor-mediated IPSCs in identified lamina I neurons of the adult rat spinal cord.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Bicuculline; Evoked Potentials; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Male; Neurons; Patch-Clamp Techniques; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glycine; Spinal Cord; Strychnine; Sucrose; Tetrodotoxin | 1999 |
Effects of treatment with GABA(A) receptor subunit antisense oligodeoxynucleotides on GABA-stimulated 36Cl- influx in the rat cerebral cortex.
Topics: Animals; Base Sequence; Bicuculline; Cerebral Cortex; Chlorides; Flunitrazepam; gamma-Aminobutyric Acid; Male; Oligodeoxyribonucleotides, Antisense; Open Reading Frames; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reverse Transcriptase Polymerase Chain Reaction | 2000 |
GABA(B) receptors are the first target of released GABA at lamina I inhibitory synapses in the adult rat spinal cord.
Topics: Age Factors; Animals; Benzylamines; Bicuculline; Flunitrazepam; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Glycine Agents; Male; Membrane Potentials; Neural Inhibition; Patch-Clamp Techniques; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Receptors, Glycine; Spinal Cord; Strychnine; Synapses | 2000 |
Allosteric modulation in spontaneously active mutant gamma-aminobutyric acid(A) receptors [corrected].
Topics: Allosteric Regulation; Amino Acid Substitution; Animals; Bicuculline; Cells, Cultured; Female; Flunitrazepam; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Humans; Ion Channel Gating; Mutagenesis, Site-Directed; Oocytes; Pentobarbital; Picrotoxin; Protein Structure, Tertiary; Receptors, GABA-A; Steroids; Xenopus laevis | 2000 |
Allosteric modulation in spontaneously active mutant gamma-aminobutyric acidA receptors.
Topics: Allosteric Regulation; Animals; Bicuculline; Electric Conductivity; Female; Flunitrazepam; GABA Antagonists; GABA Modulators; Patch-Clamp Techniques; Pentobarbital; Picrotoxin; Pregnanolone; Protein Isoforms; Receptors, GABA-A; Xenopus laevis | 2001 |
Activation of GABA(A) receptors in subthalamic neurons in vitro: properties of native receptors and inhibition mechanisms.
Topics: Animals; Bicarbonates; Bicuculline; Chlorides; Diazepam; Electrophysiology; Flunitrazepam; GABA Agonists; GABA Antagonists; GABA Modulators; Membrane Potentials; Muscimol; Neural Inhibition; Neurons; Organ Culture Techniques; Pentobarbital; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Sesterterpenes; Subthalamic Nucleus | 2001 |
Characterization of a new synthetic isoflavonoid with inverse agonist activity at the central benzodiazepine receptor.
Topics: Analysis of Variance; Animals; Bicuculline; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Female; Flavonoids; Flunitrazepam; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Hippocampus; Isoflavones; Kinetics; Male; Membrane Potentials; Midazolam; Neurons; Pregnancy; Rats; Rats, Wistar; Receptors, GABA-A; Synaptosomes; Time Factors; Tritium | 2004 |
Surface activity of thymol: implications for an eventual pharmacological activity.
Topics: Air; Animals; Bicuculline; Cell Membrane; Chickens; Flunitrazepam; GABA Antagonists; Glycine max; Kinetics; Lipid Bilayers; Micelles; Octoxynol; Phosphatidylcholines; Protein Binding; Pyrimidinones; Spectrophotometry; Surface-Active Agents; Thymol; Time Factors; Water | 2004 |
Ethanol potentiation of GABAergic synaptic transmission may be self-limiting: role of presynaptic GABA(B) receptors.
Topics: Animals; Autoreceptors; Baclofen; Bicuculline; Central Nervous System Depressants; Electric Stimulation; Electrophysiology; Ethanol; Flunitrazepam; GABA-A Receptor Antagonists; Hippocampus; In Vitro Techniques; Male; Morpholines; Neural Inhibition; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission | 2004 |
Novel plant substances acting as beta subunit isoform-selective positive allosteric modulators of GABAA receptors.
Topics: Allosteric Regulation; Animals; Araliaceae; Bicuculline; Flumazenil; Flunitrazepam; GABA Modulators; Picrotoxin; Plant Extracts; Receptors, GABA-A; Xenopus laevis | 2005 |
Betulin binds to gamma-aminobutyric acid receptors and exerts anticonvulsant action in mice.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Anticonvulsants; Antineoplastic Agents; Betulinic Acid; Bicuculline; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Muscle Tonus; Pentacyclic Triterpenes; Postural Balance; Receptors, GABA; Seizures; Triterpenes | 2008 |