flunitrazepam and beta-carboline-3-carboxylic acid ethyl ester

flunitrazepam has been researched along with beta-carboline-3-carboxylic acid ethyl ester in 52 studies

Research

Studies (52)

TimeframeStudies, this research(%)All Research%
pre-199043 (82.69)18.7374
1990's4 (7.69)18.2507
2000's3 (5.77)29.6817
2010's2 (3.85)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cook, JM; Cox, ED; Diaz-Arauzo, H; Harris, B; Huang, Q; Ma, C; McKernan, R; Reddy, MS; Skolnick, P1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Clayton, T; Cook, J; DeLorey, TM; Furtmüller, R; Halliwell, RF; Harris, D; Huck, S; Sahbaie, P; Sieghart, W1
Anzini, M; Betti, L; Biggio, G; Braile, C; Cappelli, A; Castriconi, F; Di Capua, A; Di Cesare Mannelli, L; Frosini, M; Ghelardini, C; Giannaccini, G; Giorgi, G; Giuliani, G; Grisci, G; Lucacchini, A; Mascia, MP; Paolino, M; Ricci, L; Valenti, S; Vomero, S1
Kuriyama, K; Taguchi, J1
Meliksetyan, MB1
Biggio, G; Corda, MG; Giorgi, O; Gritti, I; Mariotti, M; Ongini, E1
Cooper, SJ; Deckert, J; Estall, LB; Marangos, PJ1
Friedl, W; Hebebrand, J; Propping, P; Rabe, S1
Faull, RL; Villiger, JW1
Gobbi, M; Mennini, T; Perin, L; Salmona, M1
Clow, A; Glover, V; Sandler, M1
Chiu, TH; Rosenberg, HC; Tietz, EI1
Kempner, ES; Paul, SM; Schwartz, RD; Skolnick, P; Thomas, JW1
Biggio, G; Corda, MG; Porceddu, ML; Sanna, E1
Hammond, JR1
Sieghart, W2
Belonogoff, OB; Zuzin, VN1
Barbaccia, ML; Costa, E; Ravizza, L1
Herblin, WF1
Cohen, RM; Havoundjian, H; Paul, SM; Skolnick, P1
Hammond, JR; Martin, IL1
Chang, LR; Lee, HK; Tao, PL1
Insel, T; Marangos, PJ; Tamborska, E1
Eichinger, A; Möhler, H; Richards, JG; Sieghart, W1
Poshivalov, VP; Rozhanets, VV; Sukhotina, IA1
Dodd, RH; Ouannès, C; Potier, MC; Potier, P; Prado de Carvalho, L; Rossier, J1
Faull, RL; Holford, NH; Villiger, JW1
Eichinger, A; Sieghart, W1
Biggio, G; Concas, A; Corda, MG; Mele, S; Montaldo, S; Serra, M1
Saano, V1
Drexler, G; Mayer, A; Sieghart, W1
De Robertis, E; Medina, JH; Novas, ML2
Cardinali, DP; Lowenstein, PR1
Braestrup, C; Nielsen, M; Olsen, CE1
Hirsch, JD; Lydigsen, JL1
Cain, M; Paul, SM; Rice, KC; Skolnick, P; Williams, EF1
Braestrup, C; Kehr, W; Nielsen, M; Paschelke, G; Petersen, EN1
Beer, B; Lippa, AS; Meyerson, LR1
Horton, RW; Prestwich, SA; Stapleton, SR1
Airaksinen, MM; Saano, V1
Tallman, JF; Thomas, JW1
Aprison, MH; Ghetti, B; Rea, MA; Vaccarino, FM; Wade, SE1
Garattini, S; Mennini, T1
Braestrup, C; Honoré, T; Jensen, LH; Nielsen, M; Petersen, EN1
Keys, C; Loew, G; Spangler, D; Toll, L1
Jun, X; Katsura, M; Kuriyama, K; Ohkuma, S1
Hosoi, R; Inoue, O; Kobayashi, K; Watanabe, Y1
Delatte, MS; Gerak, LR; Leonard, ST; Moerschbaecher, JM; Winsauer, PJ1
Abe, K; Hosoi, R; Inoue, O; Momosaki, S1

Reviews

2 review(s) available for flunitrazepam and beta-carboline-3-carboxylic acid ethyl ester

ArticleYear
Molecular substrates of anxiety: clues from the heterogeneity of benzodiazepine receptors.
    Life sciences, 1982, Oct-04, Volume: 31, Issue:14

    Topics: Aging; Animals; Anxiety; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Chemical Phenomena; Chemistry, Physical; Flunitrazepam; Humans; Muscles; Pentylenetetrazole; Pyridazines; Receptors, Drug; Receptors, GABA-A; Tissue Distribution; Triazoles

1982
Benzodiazepine receptor ligands with negative efficacy: chloride channel coupling.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Barbiturates; Brain; Carbolines; Chlorides; Flunitrazepam; Humans; Ion Channels; Ligands; Membranes; Receptors, Cell Surface; Receptors, GABA-A

1983

Other Studies

50 other study(ies) available for flunitrazepam and beta-carboline-3-carboxylic acid ethyl ester

ArticleYear
Synthesis and evaluation of analogues of the partial agonist 6-(propyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (6-PBC) and the full agonist 6-(benzyloxy)-4-(methoxymethyl)-beta-carboline-3-carboxylic acid ethyl ester (Zk 93423)
    Journal of medicinal chemistry, 1998, Jul-02, Volume: 41, Issue:14

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Binding, Competitive; Carbolines; Cell Line; Cerebral Cortex; Drug Design; GABA Agonists; Humans; Male; Mice; Muscle Relaxation; Rats; Receptors, GABA-A; Recombinant Proteins; Seizures; Structure-Activity Relationship

1998
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.
    Journal of medicinal chemistry, 2008, Jul-10, Volume: 51, Issue:13

    Topics: Animals; Behavior, Animal; Benzodiazepines; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Databases, Factual; Electrophysiology; Female; Ligands; Male; Memory; Mice; Models, Molecular; Molecular Structure; Oocytes; Protein Isoforms; Protein Subunits; Quantitative Structure-Activity Relationship; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis

2008
Design, Synthesis, and Biological Evaluation of Imidazo[1,5-a]quinoline as Highly Potent Ligands of Central Benzodiazepine Receptors.
    Journal of medicinal chemistry, 2016, Apr-14, Volume: 59, Issue:7

    Topics: Amnesia; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Binding Sites; Brain; Cattle; Drug Design; Humans; Ischemia; Ligands; Male; Mice; Models, Molecular; Neuroprotective Agents; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Structure-Activity Relationship; Synaptosomes

2016
Functional modulation of cerebral gamma-aminobutyric acidA receptor/benzodiazepine receptor/chloride ion channel complex with ethyl beta-carboline-3-carboxylate: presence of independent binding site for ethyl beta-carboline-3-carboxylate.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:2

    Topics: Animals; Baclofen; Binding Sites; Brain; Carbolines; Cells, Cultured; Chloride Channels; Chlorides; Drug Interactions; Flunitrazepam; Male; Membrane Proteins; Mice; Muscimol; Receptors, GABA-A; Tritium

1990
Non-benzodiazepine, Ag-dependent, brain-specific binding sites for [3H]beta-carboline-3-carboxylic acid ethyl ester.
    European journal of pharmacology, 1989, Dec-07, Volume: 173, Issue:2-3

    Topics: Animals; Binding Sites; Brain; Carbolines; Diazepam; Flunitrazepam; In Vitro Techniques; Kinetics; Male; Membranes; Rats; Receptors, GABA-A; Silver

1989
Binding sites for [3H]2-oxo-quazepam in the brain of the cat: evidence for heterogeneity of benzodiazepine recognition sites.
    Neuropharmacology, 1989, Volume: 28, Issue:7

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Brain Chemistry; Carbolines; Cats; Flunitrazepam; Male; Receptors, GABA-A

1989
CGS 8216 treatment decreases central-type benzodiazepine receptors in rat brain.
    European journal of pharmacology, 1987, Oct-27, Volume: 142, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Convulsants; Flunitrazepam; Male; Pyrazoles; Rats; Receptors, GABA-A

1987
Phylogenetic conservation of the benzodiazepine binding sites: pharmacological evidence.
    Neuropharmacology, 1988, Volume: 27, Issue:2

    Topics: Affinity Labels; Animals; Anura; Binding, Competitive; Brain; Carbolines; Ducks; Fishes; Flunitrazepam; Guinea Pigs; Humans; Male; Photochemistry; Phylogeny; Radioligand Assay; Rats; Receptors, GABA-A; Species Specificity; Swine

1988
Multiple benzodiazepine receptors in the human basal ganglia: a detailed pharmacological and anatomical study.
    Neuroscience, 1988, Volume: 24, Issue:2

    Topics: Adolescent; Adult; Aged; Autoradiography; Basal Ganglia; Binding, Competitive; Carbolines; Caudate Nucleus; Child; Child, Preschool; Female; Flunitrazepam; Globus Pallidus; Humans; Male; Middle Aged; Putamen; Pyridazines; Receptors, GABA-A

1988
Rapid internalization of benzodiazepine receptors in the rat cortex induced by handling.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Bicuculline; Carbolines; Cerebral Cortex; Corticosterone; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Ligands; Male; Rats; Receptors, GABA-A; Stress, Physiological; Synaptic Membranes; Viscosity

1988
Triazolam, an anomalous benzodiazepine receptor ligand: in vitro characterization of alprazolam and triazolam binding.
    Journal of neurochemistry, 1985, Volume: 45, Issue:2

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Carbolines; Clonazepam; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Triazolam

1985
Pre- versus postsynaptic localization of benzodiazepine and beta-carboline binding sites.
    Journal of neurochemistry, 1985, Volume: 44, Issue:5

    Topics: Animals; Carbolines; Cerebellum; Cerebral Cortex; Flunitrazepam; Hippocampus; Indoles; Male; Polyethylene Glycols; Rats; Receptors, GABA-A; Solubility; Synaptic Membranes

1985
Radiation inactivation studies of the benzodiazepine/gamma-aminobutyric acid/chloride ionophore receptor complex.
    Journal of neurochemistry, 1985, Volume: 45, Issue:1

    Topics: Animals; Barbiturates; Benzodiazepines; Benzodiazepinones; Binding Sites; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Flumazenil; Flunitrazepam; Ionophores; Male; Molecular Weight; Muscimol; Picrotoxin; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Increase in nigral type II benzodiazepine recognition sites following striatonigral denervation.
    European journal of pharmacology, 1985, Jun-07, Volume: 112, Issue:2

    Topics: Animals; Carbolines; Corpus Striatum; Denervation; Flunitrazepam; Kainic Acid; Male; Neural Pathways; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1985
Photoaffinity labelling of benzodiazepine receptors: lack of effect on ligand binding to the nucleoside transport system.
    Journal of neurochemistry, 1985, Volume: 45, Issue:4

    Topics: Affinity Labels; Animals; Benzodiazepinones; Biological Transport, Active; Carbolines; Cerebral Cortex; Dipyridamole; Flumazenil; Flunitrazepam; Guinea Pigs; Nucleosides; Photochemistry; Receptors, GABA-A; Thioinosine

1985
Benzodiazepine receptors: multiple receptors or multiple conformations?
    Journal of neural transmission, 1985, Volume: 63, Issue:3-4

    Topics: Animals; Binding Sites; Brain; Brain Chemistry; Carbolines; Chemical Phenomena; Chemistry; Flunitrazepam; Humans; Kinetics; Models, Chemical; Molecular Conformation; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A

1985
Differences in the properties of bovine brain benzodiazepine receptors in the cerebellum and hippocampus revealed after reduction of disulphide bonds.
    Neuroscience letters, 1985, Nov-11, Volume: 61, Issue:3

    Topics: Animals; Brain Chemistry; Carbolines; Cattle; Cerebellum; Cerebral Cortex; Dithiothreitol; Flunitrazepam; Hippocampus; Oxidation-Reduction; Receptors, GABA-A

1985
Maprotiline: an antidepressant with an unusual pharmacological profile.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:2

    Topics: Animals; Anthracenes; Brain; Carbolines; Desipramine; Flunitrazepam; In Vitro Techniques; Male; Maprotiline; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, GABA-A; Receptors, Serotonin; Tritium

1986
Characterization of benzodiazepine binding sites after short-wave photo-affinity labeling with flunitrazepam.
    Life sciences, 1986, Feb-10, Volume: 38, Issue:6

    Topics: Affinity Labels; Animals; Binding Sites; Carbolines; Cell Membrane; Cerebral Cortex; Flunitrazepam; Male; Photochemistry; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Ultraviolet Rays

1986
Differential sensitivity of "central" and "peripheral" type benzodiazepine receptors to phospholipase A2.
    Journal of neurochemistry, 1986, Volume: 46, Issue:3

    Topics: Animals; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Kidney; Male; Myocardium; Pentobarbital; Phospholipases; Phospholipases A; Phospholipases A2; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
Comparison of benzodiazepine receptors in cerebellum and inferior colliculus.
    Journal of neurochemistry, 1986, Volume: 47, Issue:3

    Topics: Aging; Animals; Animals, Newborn; Carbolines; Cell Membrane; Cerebellum; Clonazepam; Diazepam; Flunitrazepam; Inferior Colliculi; Pyridazines; Rats; Receptors, GABA-A

1986
Solubilization of the benzodiazepine/gamma-aminobutyric acid receptor complex: comparison of the detergents octylglucopyranoside and 3-[(3-cholamidopropyl)-dimethylammonio]1-propanesulfonate (CHAPS).
    Journal of neurochemistry, 1986, Volume: 47, Issue:4

    Topics: Animals; Carbolines; Cerebellum; Chlorides; Cholic Acids; Drug Stability; Flunitrazepam; gamma-Aminobutyric Acid; Glucosides; Glycosides; Male; Phospholipids; Pyrazoles; Rats; Receptors, GABA-A; Solubility; Synaptic Membranes

1986
Heterogeneity of [3H]ethyl beta-carboline-3-carboxylate binding sites and [3H]gamma-aminobutyric acid binding sites.
    The Chinese journal of physiology, 1986, Volume: 29, Issue:1

    Topics: Animals; Binding, Competitive; Carbolines; Cattle; Cerebral Cortex; Detergents; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Molecular Weight; Muscimol; Photolysis; Radioligand Assay; Receptors, GABA-A; Receptors, Neurotransmitter; Synaptosomes

1986
'Peripheral' and 'central' type benzodiazepine receptors in Maudsley rats.
    European journal of pharmacology, 1986, Jul-31, Volume: 126, Issue:3

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Brain; Carbolines; Female; Flunitrazepam; Kinetics; Male; Rats; Rats, Mutant Strains; Receptors, GABA-A; Tissue Distribution

1986
Photoaffinity labeling of benzodiazepine receptor proteins with the partial inverse agonist [3H]Ro 15-4513: a biochemical and autoradiographic study.
    Journal of neurochemistry, 1987, Volume: 48, Issue:1

    Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Brain; Carbolines; Cell Membrane; Cerebellum; Flunitrazepam; Hippocampus; Molecular Weight; Photochemistry; Pyridazines; Rats; Receptors, GABA-A

1987
[Independent benzodiazepine and beta-carboline binding sites in the brain of aggressive and anxious-defensive mice].
    Biulleten' eksperimental'noi biologii i meditsiny, 1987, Volume: 103, Issue:6

    Topics: Aggression; Animals; Anxiety; Binding Sites; Brain; Carbolines; Diazepam; Flunitrazepam; Ligands; Male; Mice; Receptors, GABA-A; Tritium

1987
Synthesis of beta-carboline-benzodiazepine hybrid molecules: use of the known structural requirements for benzodiazepine and beta-carboline binding in designing a novel, high-affinity ligand for the benzodiazepine receptor.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:7

    Topics: Animals; Benzodiazepines; Carbolines; Flunitrazepam; Ligands; Mice; Molecular Conformation; Receptors, GABA-A

1987
Benzodiazepine receptors in the human cerebellar cortex: a quantitative autoradiographic and pharmacological study demonstrating the predominance of type I receptors.
    Brain research, 1987, May-19, Volume: 411, Issue:2

    Topics: Adult; Autoradiography; Binding, Competitive; Carbolines; Cerebellar Cortex; Female; Flunitrazepam; Humans; Male; Pyridazines; Receptors, GABA-A

1987
Photoaffinity labeling of different benzodiazepine receptors at physiological temperature.
    Journal of neurochemistry, 1984, Volume: 43, Issue:6

    Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cell Membrane; Cerebellum; Flunitrazepam; Hippocampus; Photochemistry; Pyridazines; Rats; Receptors, GABA-A; Temperature

1984
Evidence for the presence of benzodiazepine receptor subclasses in different areas of the human brain.
    Neuroscience letters, 1984, Dec-21, Volume: 52, Issue:3

    Topics: Adult; Aged; Brain; Brain Chemistry; Carbolines; Cerebellum; Cerebral Cortex; Female; Flunitrazepam; Hippocampus; Humans; Male; Middle Aged; Radioligand Assay; Receptors, GABA-A

1984
Tofizopam selectively increases the affinity of benzo-diazepine binding sites for [3H]flunitrazepam but not for beta [3H] carboline-3-carboxylic acid ethyl ester.
    Pharmacological research communications, 1982, Volume: 14, Issue:10

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Brain; Carbolines; Cerebellum; Female; Flunitrazepam; Indoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission

1982
Properties of [3H]flunitrazepam binding to different benzodiazepine binding proteins.
    European journal of pharmacology, 1983, Apr-08, Volume: 88, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Carbolines; Cerebellum; Flunitrazepam; Hippocampus; In Vitro Techniques; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Tritium

1983
Heterogeneity of benzodiazepine receptors: experimental differences between [3H]flunitrazepam and [3H]ethyl-beta-carboline-3-carboxylate binding sites in rat brain membranes.
    Journal of neurochemistry, 1983, Volume: 41, Issue:3

    Topics: Age Factors; Animals; Anti-Anxiety Agents; Benzylamines; Brain; Carbolines; Flunitrazepam; Hydroxydopamines; Indoles; Male; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Tissue Distribution

1983
Characterization of flunitrazepam and beta-carboline high affinity binding in bovine pineal gland.
    Neuroendocrinology, 1983, Volume: 37, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding Sites; Carbolines; Cattle; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Kinetics; Pentobarbital; Pineal Gland; Rats; Species Specificity

1983
Urinary and brain beta-carboline-3-carboxylates as potent inhibitors of brain benzodiazepine receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1980, Volume: 77, Issue:4

    Topics: Binding, Competitive; Brain; Carbolines; Diazepam; Flunitrazepam; Humans; Indoles; Ligands; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Structure-Activity Relationship; Synaptic Membranes

1980
Binding of beta-carboline-3-carboxylic acid ethyl ester to mouse brain benzodiazepine receptors in vivo.
    European journal of pharmacology, 1981, Jul-10, Volume: 72, Issue:4

    Topics: Animals; Binding, Competitive; Brain; Carbolines; Flunitrazepam; Indoles; Membranes; Mice; Mice, Inbred ICR; Receptors, Drug; Receptors, GABA-A

1981
Binding of [3H]ethyl-beta-carboline-3-carboxylate to brain benzodiazepine receptors: effect of drugs and anions.
    FEBS letters, 1981, Sep-28, Volume: 132, Issue:2

    Topics: Animals; Barbiturates; Benzodiazepines; Brain; Carbolines; Cerebellum; Cerebral Cortex; Diazepam; Flunitrazepam; Indoles; Male; Pyrazoles; Pyridines; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A; Sodium Chloride

1981
Does the reversal of the anticonflict effect of phenobarbital by beta-CCE and FG 7142 indicate benzodiazepine receptor-mediated anxiogenic properties?
    European journal of pharmacology, 1982, Aug-27, Volume: 82, Issue:3-4

    Topics: Animals; Anxiety; Carbolines; Conflict, Psychological; Diazepam; Flunitrazepam; Humans; Indoles; Male; Phenobarbital; Punishment; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A

1982
Regional heterogeneity of benzodiazepine binding sites in rat brain.
    European journal of pharmacology, 1982, Oct-22, Volume: 84, Issue:3-4

    Topics: Animals; Binding, Competitive; Brain; Carbolines; Cerebellum; Chlorides; Diazepam; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Kinetics; Rats; Receptors, Cell Surface; Receptors, GABA-A

1982
Binding of beta-carbolines and caffeine on benzodiazepine receptors: correlations to convulsions and tremor.
    Acta pharmacologica et toxicologica, 1982, Volume: 51, Issue:4

    Topics: Animals; Brain; Caffeine; Carbolines; Flunitrazepam; Harmaline; Harmine; Indoles; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Tremor

1982
Photoaffinity labeling of benzodiazepine receptors causes altered agonist-antagonist interactions.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1983, Volume: 3, Issue:2

    Topics: Animals; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Flunitrazepam; Kinetics; Ligands; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Loss of Purkinje cell-associated benzodiazepine receptors spares a high affinity subpopulation: a study with pcd mutant mice.
    Journal of neuroscience research, 1983, Volume: 9, Issue:3

    Topics: Animals; Benzodiazepines; Carbolines; Cell Membrane; Flunitrazepam; Kinetics; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Purkinje Cells; Receptors, Cell Surface; Receptors, GABA-A

1983
Chronic RO 15-1788 treatment increases the number of benzodiazepine receptors in rat cerebral cortex and hippocampus.
    European journal of pharmacology, 1983, May-20, Volume: 90, Issue:1

    Topics: Animals; Benzodiazepinones; Carbolines; Cerebral Cortex; Female; Flumazenil; Flunitrazepam; Hippocampus; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
Benzodiazepines receptor binding in vivo: pharmacokinetic and pharmacological significance.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Adrenal Glands; Animals; Benzodiazepinones; Brain; Carbolines; Corticosterone; Diazepam; Flumazenil; Flunitrazepam; Kinetics; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Computer-assisted determination of benzodiazepine receptor heterogeneity.
    European journal of pharmacology, 1984, Mar-23, Volume: 99, Issue:2-3

    Topics: Animals; Binding, Competitive; Brain Chemistry; Carbolines; Computers; Diazepam; Flunitrazepam; In Vitro Techniques; Male; Models, Biological; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1984
Down-regulation of benzodiazepine receptors by ethyl beta-carboline-3-carboxylate in cerebrocortical neurons.
    European journal of pharmacology, 1996, Feb-29, Volume: 298, Issue:1

    Topics: Animals; Carbolines; Cells, Cultured; Cerebral Cortex; Dose-Response Relationship, Drug; Down-Regulation; Flumazenil; Flunitrazepam; Mice; Receptors, GABA-A

1996
Discrepancy of benzodiazepine receptor occupancy between 3H-flumazenil and 125I-iomazenil in intact mouse brain.
    Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:3-4

    Topics: Animals; Binding, Competitive; Brain; Carbolines; Flumazenil; Flunitrazepam; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Male; Mice; Nitrazepam; Receptors, GABA-A; Triazolam; Tritium

1999
Relative potency and effectiveness of flunitrazepam, ethanol, and beta-CCE for disrupting the acquisition and retention of response sequences in rats.
    Behavioural pharmacology, 2009, Volume: 20, Issue:1

    Topics: Allosteric Regulation; Animals; Behavior, Animal; Carbolines; Conditioning, Operant; Dose-Response Relationship, Drug; Ethanol; Flunitrazepam; Learning; Male; Memory; Rats; Rats, Long-Evans; Receptors, GABA-A; Reinforcement Schedule; Retention, Psychology

2009
Remarkable selectivity of the in vivo binding of [3H]Ro15-4513 to α5 subtype of benzodiazepine receptor in the living mouse brain.
    Synapse (New York, N.Y.), 2010, Volume: 64, Issue:12

    Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Male; Mice; Protein Subunits; Receptors, GABA-A; Tritium

2010