flunitrazepam and alpidem

flunitrazepam has been researched along with alpidem in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19901 (11.11)18.7374
1990's4 (44.44)18.2507
2000's1 (11.11)29.6817
2010's2 (22.22)24.3611
2020's1 (11.11)2.80

Authors

AuthorsStudies
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Bendinelli, S; Castellano, S; Cosconati, S; Costa, B; Da Pozzo, E; Da Settimo, F; Greco, G; Martini, C; Milite, C; Novellino, E; Pugliesi, I; Rizzetto, E; Sbardella, G; Stefancich, G; Taliani, S1
Baglini, E; Barresi, E; Costa, B; Da Pozzo, E; Da Settimo, F; Martini, C; Robello, M; Salerno, S; Taliani, S1
Constantidinis, J; Javoy-Agid, F; Lloyd, GK; Lowenthal, A1
De Luca, C; De Medici, D; Massotti, M1
Arbilla, S; Langer, SZ1
Mehta, AK; Shank, RP1
Anzini, M; Basile, AS; Bruni, G; Cappelli, A; Giorgi, G; Langer, T; Romeo, MR; Vomero, S1
Betti, L; Bistocchi, M; Giannaccini, G; Gori, M; Lucacchini, A1

Reviews

1 review(s) available for flunitrazepam and alpidem

ArticleYear
An update into the medicinal chemistry of translocator protein (TSPO) ligands.
    European journal of medicinal chemistry, 2021, Jan-01, Volume: 209

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Anticonvulsants; Apoptosis; Benzimidazoles; Benzodiazepines; Cell Proliferation; Diazepam; Humans; Imidazoles; Membrane Potential, Mitochondrial; Mitochondria; Mitochondrial ADP, ATP Translocases; Mitochondrial Membranes; Mitochondrial Permeability Transition Pore; Oxidative Stress; Protein Binding; Pyridines; Quinolines; Receptors, GABA; Structure-Activity Relationship; Voltage-Dependent Anion Channels

2021

Other Studies

8 other study(ies) available for flunitrazepam and alpidem

ArticleYear
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.
    Journal of medicinal chemistry, 2012, May-10, Volume: 55, Issue:9

    Topics: Animals; Binding, Competitive; Carrier Proteins; Cell Line, Tumor; Cell Survival; Inhibitory Concentration 50; Molecular Structure; Quinazolines; Rats; Receptors, GABA-A; Structure-Activity Relationship

2012
GABAA receptor complex function in frontal cortex membranes from control and neurological patients.
    European journal of pharmacology, 1991, May-02, Volume: 197, Issue:1

    Topics: Adult; Aged; Alzheimer Disease; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Clonazepam; Female; Flunitrazepam; Humans; Huntington Disease; Imidazoles; In Vitro Techniques; Kinetics; Male; Membranes; Middle Aged; Nervous System Diseases; Parkinson Disease; Pyridines; Receptors, GABA-A

1991
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
    Psychopharmacology, 1990, Volume: 102, Issue:4

    Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem

1990
Imidazopyridines as a tool for the characterization of benzodiazepine receptors: a proposal for a pharmacological classification as omega receptor subtypes.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:4

    Topics: Animals; Brain Chemistry; Flunitrazepam; GABA-A Receptor Antagonists; Imidazoles; In Vitro Techniques; Isoquinolines; Kidney; Ligands; Pyridazines; Pyridines; Rats; Receptors, GABA-A; Spinal Cord; Terminology as Topic; Zolpidem

1988
Characterization of a benzodiazepine receptor site with exceptionally high affinity for Ro 15-4513 in the rat CNS.
    Brain research, 1995, Dec-18, Volume: 704, Issue:2

    Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Central Nervous System; Cerebellum; Chlorides; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; GABA Modulators; Hippocampus; Imidazoles; Male; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Spinal Cord; Tritium

1995
Molecular basis of peripheral vs central benzodiazepine receptor selectivity in a new class of peripheral benzodiazepine receptor ligands related to alpidem.
    Journal of medicinal chemistry, 1996, Oct-11, Volume: 39, Issue:21

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Cerebral Cortex; Drug Design; Flunitrazepam; Imidazoles; Isoquinolines; Models, Molecular; Protein Conformation; Pyridines; Rats; Receptors, GABA-A; Structure-Activity Relationship

1996
[3H]Ro 15-1788 binding sites to brain membrane of the saltwater Mugil cephalus.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2001, Volume: 128, Issue:3

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Female; Fishes; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Imidazoles; Ionophores; Male; Pyridines; Receptors, GABA-A; Synaptosomes; Tritium; Zolpidem

2001