flunitrazepam and alphaxalone

flunitrazepam has been researched along with alphaxalone in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19904 (22.22)18.7374
1990's13 (72.22)18.2507
2000's1 (5.56)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bowers, BJ; Wehner, JM1
Prince, RJ; Simmonds, MA3
Kokka, N; Olsen, RW; Sapp, DW; Witte, U1
Bolger, MB; Chen, JS; Gee, KW; Lan, NC1
Barbi, S; Beccia, F; Ferraro, M; Pala, F; Sabato, AF1
Bormann, J; Feigenspan, A; Wässle, H1
Harris, BD; Moody, EJ; Skolnick, P; Wong, G1
Hadingham, KL; Harkness, PC; Horne, AL; Kemp, JA; Whiting, P1
Biggio, G; Ghiani, CA; Maciocco, E; Sanna, E; Serra, M; Tuligi, G1
Fiszer de Plazas, S; Pignataro, L1
Maitra, R; Reynolds, JN1
Asproni, B; Biggio, G; Busonero, F; Cerri, R; Maciocco, E; Mascia, MP; Pau, A; Sanna, E; Talani, G1
David, JA; Pinnock, RD; Sattelle, DB; Wafford, KA1
Eichinger, A; Sieghart, W1
Olsen, RW; Yang, JS1
Ai, J; Kahnberg, P; Nielsen, M; Saederup, E; Squires, RF; Sterner, O; Witt, MR1

Other Studies

18 other study(ies) available for flunitrazepam and alphaxalone

ArticleYear
Biochemical and behavioral effects of steroids on GABAA receptor function in long- and short-sleep mice.
    Brain research bulletin, 1992, Volume: 29, Issue:1

    Topics: Anesthetics; Animals; Behavior, Animal; Brain Chemistry; Chlorides; Desoxycorticosterone; Ethanol; Flunitrazepam; Male; Mice; Mice, Inbred Strains; Pentobarbital; Pregnanediones; Pregnenolone; Receptors, GABA-A; Sleep; Species Specificity; Steroids

1992
Temperature and anion dependence of allosteric interactions at the gamma-aminobutyric acid-benzodiazepine receptor.
    Biochemical pharmacology, 1992, Oct-06, Volume: 44, Issue:7

    Topics: Animals; Anions; Binding, Competitive; Brain Chemistry; Drug Interactions; Flunitrazepam; Male; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Wistar; Receptors, GABA-A; Temperature

1992
Sex differences in sensitivity to pentylenetetrazol but not in GABAA receptor binding.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:2

    Topics: Anesthetics; Animals; Anticonvulsants; Autoradiography; Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Diazepam; Electroshock; Ethanol; Female; Flunitrazepam; Male; Muscimol; Orchiectomy; Ovariectomy; Pentylenetetrazole; Pregnanediones; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Sex Characteristics

1992
Propofol potentiates the binding of [3H]flunitrazepam to the GABAA receptor complex.
    Brain research, 1992, Nov-20, Volume: 596, Issue:1-2

    Topics: Animals; Binding, Competitive; Drug Synergism; Flunitrazepam; Male; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Wistar; Receptors, GABA-A; Tritium

1992
Differential responses of expressed recombinant human gamma-aminobutyric acidA receptors to neurosteroids.
    Journal of neurochemistry, 1991, Volume: 57, Issue:5

    Topics: Allosteric Regulation; Animals; Binding, Competitive; Brain; Cell Line; Flunitrazepam; Humans; Kinetics; Macromolecular Substances; Muscimol; Pregnanediones; Pregnanes; Progesterone; Rats; Receptors, GABA-A; Recombinant Proteins; Spinal Cord; Transfection

1991
The effect of five drugs in coma doses on neurotransmitter amino acids in the brains of guinea pigs.
    Resuscitation, 1983, Volume: 10, Issue:4

    Topics: Amino Acids; Animals; Brain; Brain Chemistry; Central Nervous System Agents; Central Nervous System Depressants; Diazepam; Flunitrazepam; Guinea Pigs; Neurotransmitter Agents; Phenobarbital; Phenytoin; Pregnanediones

1983
Pharmacology of GABA receptor Cl- channels in rat retinal bipolar cells.
    Nature, 1993, Jan-14, Volume: 361, Issue:6408

    Topics: Animals; Animals, Newborn; Bicuculline; Cells, Cultured; Chloride Channels; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Membrane Potentials; Membrane Proteins; Neurons; Pentobarbital; Photoreceptor Cells; Picrotoxin; Pregnanediones; Rats; Receptors, GABA-A; Sesterterpenes; Strychnine

1993
Different subunit requirements for volatile and nonvolatile anesthetics at gamma-aminobutyric acid type A receptors.
    Molecular pharmacology, 1995, Volume: 47, Issue:2

    Topics: Anesthetics; Binding Sites; Cell Line; Flunitrazepam; Halothane; Humans; Isoflurane; Pentobarbital; Pregnanediones; Receptors, GABA-A

1995
Differential antagonism by epipregnanolone of alphaxalone and pregnanolone potentiation of [3H]flunitrazepam binding suggests more than one class of binding site for steroids at GABAA receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:1

    Topics: Anesthetics; Animals; Brain; Flunitrazepam; In Vitro Techniques; Male; Membranes; Pregnanediones; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A

1993
The influence of the gamma 2L subunit on the modulation of responses to GABAA receptor activation.
    British journal of pharmacology, 1993, Volume: 108, Issue:3

    Topics: Anesthetics; Animals; Fibroblasts; Flunitrazepam; gamma-Aminobutyric Acid; L Cells; Mice; Pentobarbital; Pregnanediones; Receptors, GABA-A; Recombinant Proteins; Transfection

1993
Biochemical evaluations of the effects of loreclezole and propofol on the GABAA receptor in rat brain.
    Biochemical pharmacology, 1996, Jun-14, Volume: 51, Issue:11

    Topics: Anesthetics; Animals; Anticonvulsants; Brain; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Muscimol; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes; Triazoles; Tritium

1996
Epipregnanolone acts as a partial agonist on a common neurosteroid modulatory site of the GABA(A) receptor complex in avian CNS.
    Neurochemical research, 1997, Volume: 22, Issue:2

    Topics: Animals; Chickens; Drug Synergism; Flunitrazepam; GABA Agonists; Pregnanediones; Pregnanolone; Receptors, GABA; Tritium

1997
Modulation of GABA(A) receptor function by neuroactive steroids: evidence for heterogeneity of steroid sensitivity of recombinant GABA(A) receptor isoforms.
    Canadian journal of physiology and pharmacology, 1998, Volume: 76, Issue:9

    Topics: Animals; Dose-Response Relationship, Drug; Female; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Humans; Pregnanediones; Pregnanolone; Protein Isoforms; Receptors, GABA-A; Recombinant Proteins; Steroids; Xenopus laevis

1998
Ethyl 2-(4-bromophenyl)-1-(2,4-dichlorophenyl)-1H-4-imidazolecarboxylate is a novel positive modulator of GABAA receptors.
    European journal of pharmacology, 2005, Jun-15, Volume: 516, Issue:3

    Topics: Animals; Binding, Competitive; Cell Membrane; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Etomidate; Female; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Glycine; Humans; Hydrocarbons, Halogenated; Imidazoles; Male; Membrane Potentials; Oocytes; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Glycine; Receptors, Serotonin, 5-HT3; Serotonin; Tritium; Xenopus laevis

2005
GABA receptors on the cell-body membrane of an identified insect motor neuron.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1988, Jan-22, Volume: 232, Issue:1269

    Topics: Androstanes; Animals; Azasteroids; Bicuculline; Chlorides; Cockroaches; Dibenzazepines; Dose-Response Relationship, Drug; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Membrane Potentials; Microelectrodes; Motor Neurons; Nipecotic Acids; Periplaneta; Picrotoxin; Receptors, GABA-A

1988
Differential degradation of different benzodiazepine binding proteins by incubation of membranes from cerebellum or hippocampus with trypsin.
    Journal of neurochemistry, 1985, Volume: 45, Issue:1

    Topics: Affinity Labels; Androstanes; Animals; Azasteroids; Cell Membrane; Cerebellum; Electrophoresis, Polyacrylamide Gel; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Molecular Weight; Peptide Fragments; Photochemistry; Rats; Receptors, GABA-A; Trypsin

1985
gamma-Aminobutyric acid receptor-regulated 36Cl- flux in mouse cortical slices.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: Androstanes; Animals; Azasteroids; Barbiturates; Cerebral Cortex; Chlorides; Dose-Response Relationship, Drug; Electrophysiology; Flunitrazepam; Male; Mathematics; Mice; Muscimol; Receptors, GABA-A

1987
Honokiol and magnolol increase the number of [3H] muscimol binding sites three-fold in rat forebrain membranes in vitro using a filtration assay, by allosterically increasing the affinities of low-affinity sites.
    Neurochemical research, 1999, Volume: 24, Issue:12

    Topics: Allosteric Regulation; Androstanes; Animals; Azasteroids; Binding Sites; Biphenyl Compounds; Cell Membrane; Central Nervous System Depressants; Cerebellum; Diflunisal; Drugs, Chinese Herbal; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Lignans; Muscimol; Picrotoxin; Propofol; Prosencephalon; Rats; Receptors, GABA-A; Tritium

1999