flumazenil and zk 93426

flumazenil has been researched along with zk 93426 in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-199013 (48.15)18.7374
1990's11 (40.74)18.2507
2000's2 (7.41)29.6817
2010's1 (3.70)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clayton, T; Cook, JM; Cromer, BA; Ma, C; Majumder, S; Namjoshi, OA; Petrou, S; Platt, DM; Roth, BL; VanLinn, ML; Yin, W1
Lucki, I; Rowan, GA1
Hönack, D; Löscher, W1
Jackson, HC; Nutt, DJ; Ramsay, E1
Jackson, HC; Nutt, DJ1
Fassbender, CP; Hönack, D; Löscher, W1
Lister, RG2
Randall, JI; Rodgers, RJ1
Biggio, G; Corda, MG; Fernández, A; Giorgi, O1
File, SE; Pellow, S2
Braestrup, C; Petersen, EN; Scheel-Krüger, J1
File, SE; Jensen, LH; Pellow, S1
File, SE; Herberg, LJ; Montgomery, AM; Pellow, S; Stephens, DN1
Jensen, LH; Petersen, EN1
Biggio, G; Carcangiu, P; Corda, MG; Giorgi, O; Mereu, G1
Braestrup, C; Honoré, T; Jensen, LH; Kehr, W; Petersen, EN; Schmiechen, R; Schneider, H; Seidelmann, D; Stephens, DN1
Miczek, KA; Tornatzky, W; Weerts, EM2
Kapetanovic, IM; Kupferberg, HJ; Torchin, CD1
Andrews, N; File, SE1
Barakat, MT; Dean, PM1
Acri, JB; Barrett, JE; Gleeson, S; Witkin, JM1
Allen, A; Braun, MR; Cason, CR; Craig, KS; DeLong, J; June, HL; Murphy, JM; Torres, L; Zuccarelli, D1
Cook, JM; DeLorey, TM; He, X; Lameh, J; Lin, RC; Loew, GH; McBrady, B1
Camerman, A; Camerman, N; Hempel, A; Mastropaolo, D1

Other Studies

27 other study(ies) available for flumazenil and zk 93426

ArticleYear
Design, synthesis, and subtype selectivity of 3,6-disubstituted β-carbolines at Bz/GABA(A)ergic receptors. SAR and studies directed toward agents for treatment of alcohol abuse.
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Alcoholism; Animals; Benzodiazepines; Binding Sites; Carbolines; Cell Line; Computer Simulation; GABA-A Receptor Antagonists; Humans; Protein Subunits; Rats; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship

2010
Discriminative stimulus properties of the benzodiazepine receptor antagonist flumazenil.
    Psychopharmacology, 1992, Volume: 107, Issue:1

    Topics: Analysis of Variance; Animals; Anticonvulsants; Behavior, Animal; Benzodiazepines; Carbolines; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Antagonists; Male; Pyrazoles; Rats; Rats, Inbred Strains

1992
Withdrawal precipitation by benzodiazepine receptor antagonists in dogs chronically treated with diazepam or the novel anxiolytic and anticonvulsant beta-carboline abecarnil.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Carbolines; Diazepam; Dogs; Female; Flumazenil; GABA-A Receptor Antagonists; Oxazepam; Substance Withdrawal Syndrome

1992
Effect of the cyclopyrrolones suriclone and RP 59037 on body temperature in mice.
    European journal of pharmacology, 1992, May-27, Volume: 216, Issue:1

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Benzodiazepines; Body Temperature; Carbolines; Drug Interactions; Flumazenil; Indoles; Isoindoles; Male; Mice; Naphthyridines; Piperazines; Receptors, GABA-A; Sulfur Compounds

1992
Effect of benzodiazepine and beta-carboline antagonists and partial agonists on loprazolam- and ZK 93423-induced hypothermia.
    European journal of pharmacology, 1991, Feb-07, Volume: 193, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Hypothermia, Induced; Male; Mice

1991
Physical dependence on diazepam in the dog: precipitation of different abstinence syndromes by the benzodiazepine receptor antagonists Ro 15-1788 and ZK 93426.
    British journal of pharmacology, 1989, Volume: 97, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Carbolines; Diazepam; Dogs; Female; Flumazenil; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1989
Reversal of the intrinsic effects of Ro 15-4513 on exploratory behavior by two benzodiazepine receptor antagonists.
    Neuroscience letters, 1987, Aug-31, Volume: 79, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Exploratory Behavior; Flumazenil; Male; Mice; Motor Activity; Receptors, GABA-A

1987
Are the analgesic effects of social defeat mediated by benzodiazepine receptors?
    Physiology & behavior, 1987, Volume: 41, Issue:3

    Topics: Analgesia; Animals; Behavior, Animal; Carbolines; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Pyrazoles; Receptors, GABA-A; Social Behavior

1987
The abstinence syndrome in diazepam-dependent cats is precipitated by Ro 15-1788 and Ro 15-4513 but not by the benzodiazepine receptor antagonist ZK 93426.
    Neuroscience letters, 1988, May-26, Volume: 88, Issue:2

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Cats; Diazepam; Flumazenil; Receptors, GABA-A; Substance Withdrawal Syndrome

1988
Partial reversal of ethanol-induced reductions in exploration by two benzodiazepine antagonists (flumazenil and ZK 93426).
    Brain research bulletin, 1988, Volume: 21, Issue:5

    Topics: Animals; Carbolines; Diazepam; Dose-Response Relationship, Drug; Ethanol; Exploratory Behavior; Flumazenil; Male; Mice; Receptors, GABA-A

1988
Anxiolytic and anxiogenic drug effects on exploratory activity in an elevated plus-maze: a novel test of anxiety in the rat.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Convulsants; Exploratory Behavior; Flumazenil; Male; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats

1986
Evidence that the anticonflict effect of midazolam in amygdala is mediated by the specific benzodiazepine receptors.
    Neuroscience letters, 1985, Feb-04, Volume: 53, Issue:3

    Topics: Amygdala; Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Conflict, Psychological; Flumazenil; Male; Midazolam; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Actions of the beta-carboline ZK 93426 in an animal test of anxiety and the holeboard: interactions with Ro 15-1788.
    Journal of neural transmission, 1986, Volume: 65, Issue:2

    Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Drug Synergism; Exploratory Behavior; Flumazenil; Interpersonal Relations; Male; Rats; Receptors, GABA-A

1986
Do the intrinsic actions of benzodiazepine receptor antagonists imply the existence of an endogenous ligand for benzodiazepine receptors?
    Advances in biochemical psychopharmacology, 1986, Volume: 41

    Topics: Animals; Anxiety; Behavior, Animal; Benzodiazepinones; Carbolines; Convulsants; Diazepam Binding Inhibitor; Electroshock; Exploratory Behavior; Flumazenil; Humans; Ligands; Nerve Tissue Proteins; Receptors, GABA-A

1986
Effect on hypothalamic self-stimulation of the novel beta-carbolines ZK 93 426 (a benzodiazepine receptor antagonist) and ZK 91 296 (a putative partial agonist).
    Journal of neural transmission, 1986, Volume: 66, Issue:2

    Topics: Animals; Benzodiazepinones; Carbolines; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Hypothalamus; Injections, Intraperitoneal; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Self Stimulation

1986
Chronic treatment with lorazepam and FG 7142 may change the effects of benzodiazepine receptor agonists, antagonists and inverse agonists by different mechanisms.
    European journal of pharmacology, 1987, Jan-20, Volume: 133, Issue:3

    Topics: Animals; Carbolines; Drug Interactions; Drug Tolerance; Female; Flumazenil; Lorazepam; Mice; Pentylenetetrazole; Receptors, GABA-A

1987
The beta-carboline ZK 93423 inhibits reticulata neurons: an effect reversed by benzodiazepine antagonists.
    Life sciences, 1987, Apr-06, Volume: 40, Issue:14

    Topics: Action Potentials; Animals; Carbolines; Diazepam; Flumazenil; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1987
Evaluation of the beta-carboline ZK 93 426 as a benzodiazepine receptor antagonist.
    Psychopharmacology, 1984, Volume: 83, Issue:3

    Topics: Animals; Anticonvulsants; Ataxia; Benzodiazepinones; Binding, Competitive; Carbolines; Diazepam; Discrimination, Psychological; Drinking; Exploratory Behavior; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Mice; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Sleep

1984
"Anxiolytic" and "anxiogenic" benzodiazepines and beta-carbolines: effects on aggressive and social behavior in rats and squirrel monkeys.
    Psychopharmacology, 1993, Volume: 110, Issue:4

    Topics: Aggression; Animals; Anti-Anxiety Agents; Anxiety; Azides; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Motor Activity; Rats; Saimiri; Social Behavior; Species Specificity

1993
Prevention of the pro-aggressive effects of alcohol in rats and squirrel monkeys by benzodiazepine receptor antagonists.
    Psychopharmacology, 1993, Volume: 111, Issue:2

    Topics: Aggression; Animals; Carbolines; Dominance-Subordination; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Feeding Behavior; Female; Flumazenil; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Male; Motor Activity; Postural Balance; Rats; Saimiri

1993
A system for testing the development and reversal of anticonvulsant tolerance to benzodiazepines in mice.
    Epilepsy research, 1993, Volume: 16, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Carbolines; Diazepam; Drug Tolerance; Flumazenil; Flunitrazepam; Infusion Pumps, Implantable; Infusions, Parenteral; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Seizures; Solvents; Time Factors

1993
F 2692: flumazenil-reversible anxiolytic effects but inactive on [3H]-Ro 15-4513 binding.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:1

    Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding, Competitive; Carbolines; Cerebellum; Diazepam; Flumazenil; GABA-A Receptor Antagonists; In Vitro Techniques; Interpersonal Relations; Male; Membranes; Motor Activity; Pyridazines; Rats; Receptors, GABA-A

1994
The atom assignment problem in automated de novo drug design. 5. Tests for envelope-directed fragment placement based on molecular similarity.
    Journal of computer-aided molecular design, 1995, Volume: 9, Issue:5

    Topics: Binding Sites; Carbolines; Computer-Aided Design; Drug Design; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; Humans; Models, Molecular; Molecular Structure; Protein Binding; Protein Conformation; Receptors, GABA-A; Structure-Activity Relationship

1995
Blockade of behavioral effects of bretazenil by flumazenil and ZK 93,426 in pigeons.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 56, Issue:1

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Carbolines; Columbidae; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; GABA Antagonists; GABA Modulators; Male; Midazolam; Punishment; Receptors, GABA

1997
High-affinity benzodiazepine antagonists reduce responding maintained by ethanol presentation in ethanol-preferring rats.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:3

    Topics: Animals; Carbolines; Dose-Response Relationship, Drug; Ethanol; Flumazenil; GABA-A Receptor Antagonists; Male; Pyrazoles; Rats; Reinforcement, Psychology; Saccharin

1998
Influence of benzodiazepine binding site ligands on fear-conditioned contextual memory.
    European journal of pharmacology, 2001, Aug-24, Volume: 426, Issue:1-2

    Topics: Animals; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; Conditioning, Psychological; Convulsants; Fear; Flumazenil; GABA Antagonists; GABA Modulators; Imidazoles; Ligands; Male; Memory; Mice; Mice, Inbred C57BL; Motor Activity; N-Methylscopolamine; Piperazines; Quinolines; Receptors, GABA-A; Scopolamine; Silanes; Tritium

2001
Ethyl 5-isopropoxy-4-methyl-beta-carboline-3-carboxylate: structural determinants of benzodiazepine-receptor antagonism.
    Acta crystallographica. Section C, Crystal structure communications, 2005, Volume: 61, Issue:Pt 4

    Topics: Carbolines; Crystallography, X-Ray; Flumazenil; GABA Modulators; Hydrogen Bonding; Molecular Structure

2005