flumazenil has been researched along with zk 93426 in 27 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 13 (48.15) | 18.7374 |
1990's | 11 (40.74) | 18.2507 |
2000's | 2 (7.41) | 29.6817 |
2010's | 1 (3.70) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Clayton, T; Cook, JM; Cromer, BA; Ma, C; Majumder, S; Namjoshi, OA; Petrou, S; Platt, DM; Roth, BL; VanLinn, ML; Yin, W | 1 |
Lucki, I; Rowan, GA | 1 |
Hönack, D; Löscher, W | 1 |
Jackson, HC; Nutt, DJ; Ramsay, E | 1 |
Jackson, HC; Nutt, DJ | 1 |
Fassbender, CP; Hönack, D; Löscher, W | 1 |
Lister, RG | 2 |
Randall, JI; Rodgers, RJ | 1 |
Biggio, G; Corda, MG; Fernández, A; Giorgi, O | 1 |
File, SE; Pellow, S | 2 |
Braestrup, C; Petersen, EN; Scheel-Krüger, J | 1 |
File, SE; Jensen, LH; Pellow, S | 1 |
File, SE; Herberg, LJ; Montgomery, AM; Pellow, S; Stephens, DN | 1 |
Jensen, LH; Petersen, EN | 1 |
Biggio, G; Carcangiu, P; Corda, MG; Giorgi, O; Mereu, G | 1 |
Braestrup, C; Honoré, T; Jensen, LH; Kehr, W; Petersen, EN; Schmiechen, R; Schneider, H; Seidelmann, D; Stephens, DN | 1 |
Miczek, KA; Tornatzky, W; Weerts, EM | 2 |
Kapetanovic, IM; Kupferberg, HJ; Torchin, CD | 1 |
Andrews, N; File, SE | 1 |
Barakat, MT; Dean, PM | 1 |
Acri, JB; Barrett, JE; Gleeson, S; Witkin, JM | 1 |
Allen, A; Braun, MR; Cason, CR; Craig, KS; DeLong, J; June, HL; Murphy, JM; Torres, L; Zuccarelli, D | 1 |
Cook, JM; DeLorey, TM; He, X; Lameh, J; Lin, RC; Loew, GH; McBrady, B | 1 |
Camerman, A; Camerman, N; Hempel, A; Mastropaolo, D | 1 |
27 other study(ies) available for flumazenil and zk 93426
Article | Year |
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Design, synthesis, and subtype selectivity of 3,6-disubstituted β-carbolines at Bz/GABA(A)ergic receptors. SAR and studies directed toward agents for treatment of alcohol abuse.
Topics: Alcoholism; Animals; Benzodiazepines; Binding Sites; Carbolines; Cell Line; Computer Simulation; GABA-A Receptor Antagonists; Humans; Protein Subunits; Rats; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship | 2010 |
Discriminative stimulus properties of the benzodiazepine receptor antagonist flumazenil.
Topics: Analysis of Variance; Animals; Anticonvulsants; Behavior, Animal; Benzodiazepines; Carbolines; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Antagonists; Male; Pyrazoles; Rats; Rats, Inbred Strains | 1992 |
Withdrawal precipitation by benzodiazepine receptor antagonists in dogs chronically treated with diazepam or the novel anxiolytic and anticonvulsant beta-carboline abecarnil.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Carbolines; Diazepam; Dogs; Female; Flumazenil; GABA-A Receptor Antagonists; Oxazepam; Substance Withdrawal Syndrome | 1992 |
Effect of the cyclopyrrolones suriclone and RP 59037 on body temperature in mice.
Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Benzodiazepines; Body Temperature; Carbolines; Drug Interactions; Flumazenil; Indoles; Isoindoles; Male; Mice; Naphthyridines; Piperazines; Receptors, GABA-A; Sulfur Compounds | 1992 |
Effect of benzodiazepine and beta-carboline antagonists and partial agonists on loprazolam- and ZK 93423-induced hypothermia.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Hypothermia, Induced; Male; Mice | 1991 |
Physical dependence on diazepam in the dog: precipitation of different abstinence syndromes by the benzodiazepine receptor antagonists Ro 15-1788 and ZK 93426.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Carbolines; Diazepam; Dogs; Female; Flumazenil; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors | 1989 |
Reversal of the intrinsic effects of Ro 15-4513 on exploratory behavior by two benzodiazepine receptor antagonists.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Exploratory Behavior; Flumazenil; Male; Mice; Motor Activity; Receptors, GABA-A | 1987 |
Are the analgesic effects of social defeat mediated by benzodiazepine receptors?
Topics: Analgesia; Animals; Behavior, Animal; Carbolines; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Pyrazoles; Receptors, GABA-A; Social Behavior | 1987 |
The abstinence syndrome in diazepam-dependent cats is precipitated by Ro 15-1788 and Ro 15-4513 but not by the benzodiazepine receptor antagonist ZK 93426.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Cats; Diazepam; Flumazenil; Receptors, GABA-A; Substance Withdrawal Syndrome | 1988 |
Partial reversal of ethanol-induced reductions in exploration by two benzodiazepine antagonists (flumazenil and ZK 93426).
Topics: Animals; Carbolines; Diazepam; Dose-Response Relationship, Drug; Ethanol; Exploratory Behavior; Flumazenil; Male; Mice; Receptors, GABA-A | 1988 |
Anxiolytic and anxiogenic drug effects on exploratory activity in an elevated plus-maze: a novel test of anxiety in the rat.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Convulsants; Exploratory Behavior; Flumazenil; Male; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats | 1986 |
Evidence that the anticonflict effect of midazolam in amygdala is mediated by the specific benzodiazepine receptors.
Topics: Amygdala; Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Conflict, Psychological; Flumazenil; Male; Midazolam; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Actions of the beta-carboline ZK 93426 in an animal test of anxiety and the holeboard: interactions with Ro 15-1788.
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Drug Synergism; Exploratory Behavior; Flumazenil; Interpersonal Relations; Male; Rats; Receptors, GABA-A | 1986 |
Do the intrinsic actions of benzodiazepine receptor antagonists imply the existence of an endogenous ligand for benzodiazepine receptors?
Topics: Animals; Anxiety; Behavior, Animal; Benzodiazepinones; Carbolines; Convulsants; Diazepam Binding Inhibitor; Electroshock; Exploratory Behavior; Flumazenil; Humans; Ligands; Nerve Tissue Proteins; Receptors, GABA-A | 1986 |
Effect on hypothalamic self-stimulation of the novel beta-carbolines ZK 93 426 (a benzodiazepine receptor antagonist) and ZK 91 296 (a putative partial agonist).
Topics: Animals; Benzodiazepinones; Carbolines; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Hypothalamus; Injections, Intraperitoneal; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Self Stimulation | 1986 |
Chronic treatment with lorazepam and FG 7142 may change the effects of benzodiazepine receptor agonists, antagonists and inverse agonists by different mechanisms.
Topics: Animals; Carbolines; Drug Interactions; Drug Tolerance; Female; Flumazenil; Lorazepam; Mice; Pentylenetetrazole; Receptors, GABA-A | 1987 |
The beta-carboline ZK 93423 inhibits reticulata neurons: an effect reversed by benzodiazepine antagonists.
Topics: Action Potentials; Animals; Carbolines; Diazepam; Flumazenil; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra | 1987 |
Evaluation of the beta-carboline ZK 93 426 as a benzodiazepine receptor antagonist.
Topics: Animals; Anticonvulsants; Ataxia; Benzodiazepinones; Binding, Competitive; Carbolines; Diazepam; Discrimination, Psychological; Drinking; Exploratory Behavior; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Mice; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Sleep | 1984 |
"Anxiolytic" and "anxiogenic" benzodiazepines and beta-carbolines: effects on aggressive and social behavior in rats and squirrel monkeys.
Topics: Aggression; Animals; Anti-Anxiety Agents; Anxiety; Azides; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Motor Activity; Rats; Saimiri; Social Behavior; Species Specificity | 1993 |
Prevention of the pro-aggressive effects of alcohol in rats and squirrel monkeys by benzodiazepine receptor antagonists.
Topics: Aggression; Animals; Carbolines; Dominance-Subordination; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Feeding Behavior; Female; Flumazenil; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Male; Motor Activity; Postural Balance; Rats; Saimiri | 1993 |
A system for testing the development and reversal of anticonvulsant tolerance to benzodiazepines in mice.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Carbolines; Diazepam; Drug Tolerance; Flumazenil; Flunitrazepam; Infusion Pumps, Implantable; Infusions, Parenteral; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Seizures; Solvents; Time Factors | 1993 |
F 2692: flumazenil-reversible anxiolytic effects but inactive on [3H]-Ro 15-4513 binding.
Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding, Competitive; Carbolines; Cerebellum; Diazepam; Flumazenil; GABA-A Receptor Antagonists; In Vitro Techniques; Interpersonal Relations; Male; Membranes; Motor Activity; Pyridazines; Rats; Receptors, GABA-A | 1994 |
The atom assignment problem in automated de novo drug design. 5. Tests for envelope-directed fragment placement based on molecular similarity.
Topics: Binding Sites; Carbolines; Computer-Aided Design; Drug Design; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; Humans; Models, Molecular; Molecular Structure; Protein Binding; Protein Conformation; Receptors, GABA-A; Structure-Activity Relationship | 1995 |
Blockade of behavioral effects of bretazenil by flumazenil and ZK 93,426 in pigeons.
Topics: Animals; Behavior, Animal; Benzodiazepinones; Carbolines; Columbidae; Conditioning, Operant; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; GABA Antagonists; GABA Modulators; Male; Midazolam; Punishment; Receptors, GABA | 1997 |
High-affinity benzodiazepine antagonists reduce responding maintained by ethanol presentation in ethanol-preferring rats.
Topics: Animals; Carbolines; Dose-Response Relationship, Drug; Ethanol; Flumazenil; GABA-A Receptor Antagonists; Male; Pyrazoles; Rats; Reinforcement, Psychology; Saccharin | 1998 |
Influence of benzodiazepine binding site ligands on fear-conditioned contextual memory.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; Conditioning, Psychological; Convulsants; Fear; Flumazenil; GABA Antagonists; GABA Modulators; Imidazoles; Ligands; Male; Memory; Mice; Mice, Inbred C57BL; Motor Activity; N-Methylscopolamine; Piperazines; Quinolines; Receptors, GABA-A; Scopolamine; Silanes; Tritium | 2001 |
Ethyl 5-isopropoxy-4-methyl-beta-carboline-3-carboxylate: structural determinants of benzodiazepine-receptor antagonism.
Topics: Carbolines; Crystallography, X-Ray; Flumazenil; GABA Modulators; Hydrogen Bonding; Molecular Structure | 2005 |