flumazenil and yohimbine

flumazenil has been researched along with yohimbine in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19906 (27.27)18.7374
1990's6 (27.27)18.2507
2000's5 (22.73)29.6817
2010's5 (22.73)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Sun, H1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Benson, GJ; Gross, ME; Olson, WA; Thurmon, JC; Tranquilli, WJ1
Fukuda, N; Wada, T1
Chopin, P; File, SE; Pellow, S2
Idemudia, SO; Lal, H; Mathis, DA1
Assié, MB; Briley, M; Charveron, M; Stenger, A1
Clark, JD; Hatch, RC; Kitzman, JV; Zahner, JM1
Chapouthier, G; Jacquot, F; Sara, S; Save, E; Venault, P1
Kohno, SI; Matsumoto, K; Ojima, K; Watanabe, H1
Castro, JL; Ramirez, A; Ricci, D; Taira, CA1
Calle, PP; Cook, RA; James, SB; Kalk, P; MacLaughlin, K; Raphael, BL; Stetter, MD1
Iyo, M; Kakiuchi, T; Matsunaga, T; Mori, N; Nishiyama, S; Sekine, Y; Tsukada, H1
Doherty, T; Miller, BF; Miller, KV; Muller, LI; Osborn, DA; Warren, RJ1
Eskandari, MH; Vesal, N1
Vesal, N; Zare, P1
Evenden, J; Jonak, G; Ross, L; Zhou, J1
Ishola, IO; Olayemi, SO; Umeh, EA; Yemitan, OK1
Alba-Betancourt, C; Alonso-Castro, AJ; Gasca-Martínez, D; Pérez-Gutiérrez, S; Rocha-González, E; Ruiz-Arredondo, A; Zapata-Morales, JR1

Trials

2 trial(s) available for flumazenil and yohimbine

ArticleYear
Sedative effects of midazolam and xylazine with or without ketamine and detomidine alone following intranasal administration in Ring-necked Parakeets.
    Journal of the American Veterinary Medical Association, 2006, Feb-01, Volume: 228, Issue:3

    Topics: Administration, Intranasal; Adrenergic alpha-Antagonists; Animals; Cross-Over Studies; Dose-Response Relationship, Drug; Drug Combinations; Female; Flumazenil; Heart Rate; Hypnotics and Sedatives; Imidazoles; Ketamine; Male; Midazolam; Parakeets; Prospective Studies; Respiration; Time Factors; Treatment Outcome; Xylazine; Yohimbine

2006
Clinical evaluation of intranasal benzodiazepines, alpha-agonists and their antagonists in canaries.
    Veterinary anaesthesia and analgesia, 2006, Volume: 33, Issue:3

    Topics: Administration, Intranasal; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anesthesia; Animals; Behavior, Animal; Benzodiazepines; Canaries; Diazepam; Drug Therapy, Combination; Female; Flumazenil; Hypnotics and Sedatives; Imidazoles; Male; Midazolam; Prospective Studies; Xylazine; Yohimbine

2006

Other Studies

20 other study(ies) available for flumazenil and yohimbine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Capture hydrolysis signals in the microsomal stability assay: molecular mechanisms of the alkyl ester drug and prodrug metabolism.
    Bioorganic & medicinal chemistry letters, 2012, Jan-15, Volume: 22, Issue:2

    Topics: Carboxylic Acids; Cytochrome P-450 Enzyme System; Esters; Humans; Hydrolysis; Microsomes; Models, Molecular; Molecular Structure; Prodrugs; Quantum Theory; Signal Transduction

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Yohimbine/flumazenil antagonism of hemodynamic alterations induced by a combination of midazolam, xylazine, and butorphanol in dogs.
    Journal of the American Veterinary Medical Association, 1992, Dec-15, Volume: 201, Issue:12

    Topics: Anesthesia; Anesthetics; Animals; Blood Pressure; Butorphanol; Cardiac Output; Dogs; Female; Flumazenil; Heart Rate; Hemodynamics; Male; Midazolam; Stroke Volume; Vascular Resistance; Xylazine; Yohimbine

1992
Effects of DN-2327, a new anxiolytic, diazepam and buspirone on exploratory activity of the rat in an elevated plus-maze.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Buspirone; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Exploratory Behavior; Flumazenil; Isoindoles; Male; Naphthyridines; Pentylenetetrazole; Rats; Rats, Inbred Strains; Spiro Compounds; Yohimbine

1991
The effects of yohimbine on exploratory and locomotor behaviour are attributable to its effects at noradrenaline and not at benzodiazepine receptors.
    Neuropharmacology, 1986, Volume: 25, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Benzodiazepinones; Chlordiazepoxide; Clonidine; Drug Interactions; Exploratory Behavior; Flumazenil; Male; Motor Activity; Rats; Receptors, GABA-A; Yohimbine

1986
Are the anxiogenic effects of yohimbine mediated by its action at benzodiazepine receptors?
    Neuroscience letters, 1985, Mar-22, Volume: 55, Issue:1

    Topics: Animals; Arousal; Benzodiazepinones; Brain; Chlordiazepoxide; Clonidine; Dose-Response Relationship, Drug; Flumazenil; Male; Rats; Receptors, Adrenergic, alpha; Receptors, GABA-A; Social Behavior; Social Environment; Yohimbine

1985
Enhancement of a diazepam withdrawal symptom by bicuculline and yohimbine.
    Neuropharmacology, 1987, Volume: 26, Issue:12

    Topics: Animals; Bicuculline; Diazepam; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; Male; Rats; Substance Withdrawal Syndrome; Yohimbine

1987
Benzodiazepine agonist-type activity of raubasine, a rauwolfia serpentina alkaloid.
    European journal of pharmacology, 1984, Nov-13, Volume: 106, Issue:2

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Binding, Competitive; Brain; Diazepam; Flumazenil; Flurazepam; In Vitro Techniques; Kinetics; Male; Mice; Rats; Receptors, GABA-A; Secologanin Tryptamine Alkaloids; Yohimbine

1984
Comparison of five preanesthetic medicaments in thiopental-anesthetized cats: antagonism by selected compounds.
    American journal of veterinary research, 1984, Volume: 45, Issue:11

    Topics: 4-Aminopyridine; Acepromazine; Aminopyridines; Anesthesia, General; Animals; Arousal; Benzodiazepinones; Cats; Central Nervous System Stimulants; Convulsants; Diazepam; Drug Antagonism; Female; Flumazenil; Ketamine; Male; Meperidine; Naloxone; Pentobarbital; Preanesthetic Medication; Sodium Chloride; Xylazine; Yohimbine

1984
Anxiogenic-like effects of yohimbine and idazoxan in two behavioral situations in mice.
    Life sciences, 1993, Volume: 52, Issue:7

    Topics: Adrenergic alpha-Antagonists; Animals; Anxiety; Behavior, Animal; Choice Behavior; Clonidine; Conditioning, Classical; Conflict, Psychological; Dioxanes; Flumazenil; Idazoxan; Male; Mice; Yohimbine

1993
Flumazenil but not FG7142 reverses the decrease in pentobarbital sleep caused by activation of central noradrenergic systems in mice.
    Brain research, 1997, Apr-18, Volume: 754, Issue:1-2

    Topics: Animals; Appetite Depressants; Carbolines; Cerebral Ventricles; Flumazenil; Injections, Intravenous; Injections, Intraventricular; Male; Methoxamine; Mice; Mice, Inbred Strains; Pentobarbital; Sleep; Yohimbine

1997
Central benzodiazepine involvement in clonidine cardiovascular actions.
    Canadian journal of physiology and pharmacology, 1999, Volume: 77, Issue:11

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Atropine Derivatives; Blood Pressure; Carbolines; Cardiovascular Agents; Clonidine; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Heart Rate; Infusions, Intravenous; Injections, Intraventricular; Male; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, GABA-A; Stereotaxic Techniques; Time Factors; Yohimbine

1999
Immobilization of babirusa (Babyrousa babyrussa) with xylazine and tiletamine/zolazepam and reversal with yohimbine and flumazenil.
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 1999, Volume: 30, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anesthetics, Dissociative; Animals; Animals, Zoo; Anti-Anxiety Agents; Antidotes; Body Temperature; Female; Flumazenil; GABA Modulators; Heart Rate; Immobilization; Injections, Intramuscular; Injections, Intravenous; Male; Oxygen; Preanesthetic Medication; Respiration; Retrospective Studies; Swine; Tiletamine; Xylazine; Yohimbine; Zolazepam

1999
Yohimbine increases the binding potential for [11C]flumazenil in the monkey brain.
    Journal of neural transmission (Vienna, Austria : 1996), 2001, Volume: 108, Issue:12

    Topics: Adrenergic alpha-Antagonists; Animals; Behavior, Animal; Binding Sites; Binding, Competitive; Brain; Carbon Radioisotopes; Flumazenil; GABA Modulators; Hippocampus; Macaca mulatta; Male; Receptors, GABA-A; Tomography, Emission-Computed; Up-Regulation; Vocalization, Animal; Yohimbine

2001
Effectiveness of antagonists for tiletamine-zolazepam/xylazine immobilization in female white-tailed deer.
    Journal of wildlife diseases, 2004, Volume: 40, Issue:3

    Topics: Adrenergic alpha-Agonists; Anesthetics; Animals; Deer; Dose-Response Relationship, Drug; Drug Combinations; Female; Flumazenil; GABA Modulators; Imidazoles; Immobilization; Random Allocation; Tiletamine; Time Factors; Tolazoline; Xylazine; Yohimbine; Zolazepam

2004
A novel operant conflict procedure using incrementing shock intensities to assess the anxiolytic and anxiogenic effects of drugs.
    Behavioural pharmacology, 2009, Volume: 20, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Aripiprazole; Benzodiazepines; Chlordiazepoxide; Conditioning, Operant; Conflict, Psychological; Dextroamphetamine; Diazepam; Electroshock; Flumazenil; Male; Piperazines; Punishment; Pyridazines; Quinolones; Rats; Rats, Sprague-Dawley; Triazoles; Yohimbine

2009
Antidepressant and anxiolytic effects of the methanol root extract of Capparis thonningii: involvement of monoaminergic, cholinergic and GABAergic systems.
    Drug research, 2015, Volume: 65, Issue:4

    Topics: Adrenergic Antagonists; Animals; Anti-Anxiety Agents; Antidepressive Agents; Atropine; Behavior, Animal; Biogenic Monoamines; Capparis; Cholinergic Agents; Cholinergic Neurons; Cyproheptadine; Dopamine Antagonists; Female; Flumazenil; GABA Agents; gamma-Aminobutyric Acid; Immobility Response, Tonic; Male; Metergoline; Methanol; Mice; Muscarinic Antagonists; Plant Extracts; Plant Roots; Prazosin; Serotonin Antagonists; Sulpiride; Yohimbine

2015
Neuropharmacological effects of d-pinitol and its possible mechanisms of action.
    Journal of food biochemistry, 2019, Volume: 43, Issue:12

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Antidepressive Agents; Flumazenil; Hypnotics and Sedatives; Inositol; Mice; Mice, Inbred BALB C; Neuropharmacology; Pentylenetetrazole; Seizures; Yohimbine

2019