flumazenil and tiagabine

flumazenil has been researched along with tiagabine in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19901 (11.11)18.7374
1990's1 (11.11)18.2507
2000's3 (33.33)29.6817
2010's4 (44.44)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Greentree, SG; Pertwee, RG; Swift, PA1
al-Tikriti, MS; Baldwin, RM; Bradberry, C; Bremner, JD; During, M; Malison, RT; Seibyl, JP; Sybirska, E; Zea-Ponce, Y; Zoghbi, S1
Cho, RY; Frankle, WG; Lewis, DA; Litschge, M; Mason, NS; Mathis, CA; Narendran, R; Price, JC; Vora, S1
Chen, CM; Cho, RY; Frankle, WG; Himes, M; Lewis, DA; Mason, NS; Mathis, CA; Narendran, R; Walker, C1
Cho, RY; Frankle, WG; Himes, ML; Lewis, DA; Mason, NS; Narendran, R; Paris, J; Prasad, KM; Walker, C1

Reviews

1 review(s) available for flumazenil and tiagabine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

8 other study(ies) available for flumazenil and tiagabine

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Drugs which stimulate or facilitate central GABAergic transmission interact synergistically with delta-9-tetrahydrocannabinol to produce marked catalepsy in mice.
    Neuropharmacology, 1988, Volume: 27, Issue:12

    Topics: Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Catalepsy; Dronabinol; Drug Synergism; Flumazenil; Flupenthixol; Flurazepam; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Nipecotic Acids; Receptors, GABA-A; Strychnine; Taurine; Tiagabine

1988
[123I]iomazenil SPECT imaging demonstrates significant benzodiazepine receptor reserve in human and nonhuman primate brain.
    Neuropharmacology, 1993, Volume: 32, Issue:7

    Topics: Adult; Animals; Binding, Competitive; Brain; Dialysis; Female; Flumazenil; gamma-Aminobutyric Acid; Half-Life; Humans; Hypnotics and Sedatives; Iodine Radioisotopes; Lorazepam; Male; Nipecotic Acids; Ovariectomy; Papio; Receptors, GABA-A; Tiagabine; Tomography, Emission-Computed, Single-Photon

1993
Tiagabine increases [11C]flumazenil binding in cortical brain regions in healthy control subjects.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:3

    Topics: Adult; Brain Mapping; Cerebral Cortex; Cognition; Cortical Synchronization; Feasibility Studies; Female; Flumazenil; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; gamma-Aminobutyric Acid; Humans; Magnetic Resonance Imaging; Male; Middle Aged; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Positron-Emission Tomography; Receptors, GABA-A; Tiagabine

2009
[11C]flumazenil binding is increased in a dose-dependent manner with tiagabine-induced elevations in GABA levels.
    PloS one, 2012, Volume: 7, Issue:2

    Topics: Adult; Carbon Isotopes; Cognition; Dose-Response Relationship, Drug; Electroencephalography; Electrophysiology; Female; Flumazenil; GABA Modulators; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Humans; Ligands; Male; Models, Statistical; Nipecotic Acids; Positron-Emission Tomography; Regression Analysis; Tiagabine

2012
In vivo measurement of GABA transmission in healthy subjects and schizophrenia patients.
    The American journal of psychiatry, 2015, Nov-01, Volume: 172, Issue:11

    Topics: Adult; Carbon Radioisotopes; Case-Control Studies; Cerebral Cortex; Female; Flumazenil; GABA Modulators; GABA Plasma Membrane Transport Proteins; Gamma Rhythm; gamma-Aminobutyric Acid; Humans; Male; Neuropsychological Tests; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Positron-Emission Tomography; Schizophrenia; Schizophrenic Psychology; Synaptic Transmission; Temporal Lobe; Tiagabine; Young Adult

2015