flumazenil and scopolamine hydrobromide

flumazenil has been researched along with scopolamine hydrobromide in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19904 (16.00)18.7374
1990's8 (32.00)18.2507
2000's6 (24.00)29.6817
2010's7 (28.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Topliss, JG; Yoshida, F1
Adkison, KK; Humphreys, JE; Mahar Doan, KM; Polli, JW; Serabjit-Singh, CJ; Shampine, LJ; Webster, LO; Wring, SA1
Lombardo, F; Obach, RS; Waters, NJ1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
McNamara, RK; Skelton, RW1
Forster, MJ; Lal, H; Prather, PL1
Ichihara, K; Kameyama, T; Nabeshima, T; Tohyama, K1
Bilsky, EJ; Marglin, SH; Reid, LD1
Kameyama, T; Nabeshima, T; Tohyama, K1
Kulkarni, SK; Sharma, AC1
Haigh, JR; Lines, CR; Poppleton, P; Preston, GC; Traub, M; Ward, C1
Fuxe, K; Ogren, SO1
Sansone, M1
Kulkarni, SK; Shaji, AV1
Bishop, KI; Curran, HV1
Kaneko, T; Kikusui, T; Tonohiro, T1
Cook, JM; DeLorey, TM; He, X; Lameh, J; Lin, RC; Loew, GH; McBrady, B1
Del Río, J; Diez-Ariza, M; García-Alloza, M; Lasheras, B; Ramírez, MJ; Redondo, C1
Akanmu, MA; Bamitale, KD; Ukponmwan, OE1
Hashimoto, T; Hatayama, Y; Nakamichi, K; Yoshida, N1

Reviews

1 review(s) available for flumazenil and scopolamine hydrobromide

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for flumazenil and scopolamine hydrobromide

ArticleYear
An investigation of the effects of benzodiazepine receptor ligands and of scopolamine on conceptual priming.
    Psychopharmacology, 1998, Volume: 140, Issue:3

    Topics: Adolescent; Adult; Female; Flumazenil; GABA Modulators; Humans; Lorazepam; Male; Memory; Middle Aged; Muscarinic Antagonists; Neuropsychological Tests; Scopolamine

1998

Other Studies

23 other study(ies) available for flumazenil and scopolamine hydrobromide

ArticleYear
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Passive permeability and P-glycoprotein-mediated efflux differentiate central nervous system (CNS) and non-CNS marketed drugs.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Cell Line; Cell Membrane Permeability; Central Nervous System Agents; Dogs; Drug Delivery Systems; Permeability; Pharmaceutical Preparations

2002
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Assessment of a cholinergic contribution to chlordiazepoxide-induced deficits of place learning in the Morris water maze.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:3

    Topics: Acetylcholine; Animals; Chlordiazepoxide; Drug Interactions; Flumazenil; Learning; Male; Memory; Physostigmine; Rats; Receptors, Cholinergic; Receptors, GABA-A; Scopolamine

1992
Learning and memory-enhancing effects of Ro 15-4513: a comparison with flumazenil.
    Neuropharmacology, 1992, Volume: 31, Issue:3

    Topics: Amnesia; Animals; Avoidance Learning; Azides; Benzodiazepines; Discrimination Learning; Flumazenil; Learning; Memory; Mice; Mice, Inbred ICR; Scopolamine; Stimulation, Chemical

1992
Attenuation of benzodiazepine-induced passive avoidance deficit by post-training administration of muscimol: interaction with the cholinergic neuronal system.
    European journal of pharmacology, 1990, Jul-17, Volume: 182, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Bicuculline; Chlordiazepoxide; Flumazenil; Male; Mice; Mice, Inbred Strains; Muscimol; Neurons; Parasympathetic Nervous System; Receptors, Cholinergic; Receptors, GABA-A; Scopolamine

1990
Using antagonists to assess neurochemical coding of a drug's ability to establish a conditioned place preference.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:3

    Topics: Analgesics; Animals; Brain Chemistry; Conditioning, Operant; Flumazenil; Habituation, Psychophysiologic; Male; Morphine; Naloxone; Naltrexone; Rats; Rats, Inbred Strains; Scopolamine

1990
Effects of DM-9384, a pyrrolidone derivative, on alcohol- and chlordiazepoxide-induced amnesia in mice.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:2

    Topics: Amnesia; Animals; Avoidance Learning; Bicuculline; Central Nervous System Agents; Chlordiazepoxide; Drug Interactions; Ethanol; Flumazenil; Male; Mice; Pyrrolidinones; Retention, Psychology; Scopolamine

1990
Evidence for GABA-BZ receptor modulation in short-term memory passive avoidance task paradigm in mice.
    Methods and findings in experimental and clinical pharmacology, 1990, Volume: 12, Issue:3

    Topics: Animals; Avoidance Learning; Carbolines; Electroshock; Female; Flumazenil; gamma-Aminobutyric Acid; Male; Memory, Short-Term; Mice; Physostigmine; Receptors, GABA-A; Scopolamine

1990
Scopolamine and benzodiazepine models of dementia: cross-reversals by Ro 15-1788 and physostigmine.
    Psychopharmacology, 1989, Volume: 98, Issue:4

    Topics: Acoustic Stimulation; Adult; Anti-Anxiety Agents; Attention; Cognition Disorders; Dementia; Disease Models, Animal; Female; Flumazenil; Humans; Male; Memory Disorders; Photic Stimulation; Physostigmine; Psychomotor Performance; Pupil; Reaction Time; Scopolamine

1989
D1- and D2-receptor antagonists induce catalepsy via different efferent striatal pathways [corrected].
    Neuroscience letters, 1988, Mar-10, Volume: 85, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Catalepsy; Corpus Striatum; Dose-Response Relationship, Drug; Flumazenil; Injections, Intraperitoneal; Male; Muscimol; Raclopride; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Scopolamine

1988
Scopolamine-induced locomotor stimulation in mice: effect of diazepam and a benzodiazepine antagonist.
    Psychopharmacology, 1982, Volume: 77, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Flumazenil; Male; Mice; Mice, Inbred BALB C; Motor Activity; Scopolamine

1982
Evidence of GABAergic modulation in melatonin-induced short-term memory deficits and food consumption.
    Methods and findings in experimental and clinical pharmacology, 1998, Volume: 20, Issue:4

    Topics: Animals; Antioxidants; Diazepam; Eating; Female; Flumazenil; GABA Modulators; Latency Period, Psychological; Male; Maze Learning; Melatonin; Memory Disorders; Memory, Short-Term; Mice; Muscarinic Antagonists; Rats; Rats, Wistar; Receptors, GABA; Scopolamine; Triazolam

1998
The allocentric place discrimination task is selectively and highly dependent on the central muscarinic system in rats.
    Pharmacology, biochemistry, and behavior, 2000, Jan-01, Volume: 65, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Diazepam; Discrimination Learning; Dizocilpine Maleate; Flumazenil; Male; Mecamylamine; Ondansetron; Rats; Rats, Inbred F344; Receptors, Muscarinic; Scopolamine; Swimming

2000
Influence of benzodiazepine binding site ligands on fear-conditioned contextual memory.
    European journal of pharmacology, 2001, Aug-24, Volume: 426, Issue:1-2

    Topics: Animals; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; Conditioning, Psychological; Convulsants; Fear; Flumazenil; GABA Antagonists; GABA Modulators; Imidazoles; Ligands; Male; Memory; Mice; Mice, Inbred C57BL; Motor Activity; N-Methylscopolamine; Piperazines; Quinolines; Receptors, GABA-A; Scopolamine; Silanes; Tritium

2001
Flumazenil and tacrine increase the effectiveness of ondansetron on scopolamine-induced impairment of spatial learning in rats.
    Psychopharmacology, 2003, Volume: 169, Issue:1

    Topics: Animals; Cholinesterase Inhibitors; Drug Therapy, Combination; Flumazenil; Learning; Male; Maze Learning; Memory; Muscarinic Antagonists; Ondansetron; Rats; Rats, Wistar; Receptors, GABA-A; Scopolamine; Serotonin Antagonists; Tacrine

2003
Neuropharmacological profile of aqueous extract of Anaphe venata larva (Notondotidae) in rats.
    African journal of traditional, complementary, and alternative medicines : AJTCAM, 2011, Volume: 8, Issue:3

    Topics: Amphetamine; Animals; Ataxia; Behavior, Animal; Dose-Response Relationship, Drug; Flumazenil; Grooming; Injections, Intraperitoneal; Larva; Locomotion; Moths; Naloxone; Neuropharmacology; Neurotransmitter Agents; Rats; Scopolamine; Stereotyped Behavior; Thiamine; Water

2011
Procognitive effect of AC-3933 in aged mice, and synergistic effect of combination with donepezil in scopolamine-treated mice.
    European journal of pharmacology, 2014, Dec-15, Volume: 745

    Topics: Aging; Animals; Donepezil; Drug Synergism; Flumazenil; GABA-A Receptor Agonists; Indans; Male; Maze Learning; Memory Disorders; Mice; Mice, Inbred C57BL; Naphthyridines; Nootropic Agents; Oxadiazoles; Piperidines; Rats; Scopolamine

2014