flumazenil and ro 5-4864

flumazenil has been researched along with ro 5-4864 in 69 studies

Research

Studies (69)

TimeframeStudies, this research(%)All Research%
pre-199041 (59.42)18.7374
1990's21 (30.43)18.2507
2000's4 (5.80)29.6817
2010's3 (4.35)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bendinelli, S; Castellano, S; Cosconati, S; Costa, B; Da Pozzo, E; Da Settimo, F; Greco, G; Martini, C; Milite, C; Novellino, E; Pugliesi, I; Rizzetto, E; Sbardella, G; Stefancich, G; Taliani, S1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Järvinen, A; Männistö, PT; Rägo, L1
Bitran, D; Ison, JR; Kellogg, CK; Sullivan, AT1
Da-Cunha, C; Ferreira, MB; Izquierdo, I; Jerusalinsky, D; Medina, JH; Wolfman, C1
Izquierdo, I; Medina, JH; Pereira, ME1
Elgoyhen, AB; Kazanietz, MG1
Knudsen, J; Nielsen, M1
Berkovich, A; Campagnone, M; Guidotti, A; Hensley, P; McPhie, P1
Hashemi, FS; Niles, LP1
Adler-Graschinsky, E; Elgoyhen, B1
Brouillet, E; Chavoix, C; de la Sayette, V; Dodd, RH; Fournier, D; Guibert, B; Hantraye, P; Khalili-Varasteh, M; Kunimoto, M; Naquet, R1
Griffin, K; Hong, T; Levy, JV1
Chiesi, M; Erne, P; Fulbright, J; Hermsmeyer, K; Longoni, S1
Berg, DK; McEachern, AE1
Daval, JL; Deckert, J; Marangos, PJ; Morgan, PF; Nakajima, T1
File, SE; Pellow, S5
Casals-Stenzel, J; Weber, KH1
O'Regan, MH; Phillis, JW1
Dubroeucq, MC; Gauthier, A; Guérémy, C; Le Fur, G; Mizoule, J; Renault, C; Uzan, A1
Consolo, S; Forloni, G; Garattini, S; Kolasa, K; Ladinsky, H1
Cooper, SJ; Gilbert, DB1
Abraham, CJ; De Blas, AL; Haney, SA; Park, D; Rayner, CA; Sangameswaran, L1
Cole, R; De Vellis, J; Noble, EP; Syapin, PJ1
Fares, F; Gavish, M1
Basile, AS; Skolnick, P1
Simmonds, MA1
Lingjaerde, O1
Lucantoni, D; Massotti, M1
Bryere, P; Naquet, R; Valin, A1
Kunert-Radek, J; Pawlikowski, M; Stepień, H2
Lafaille, F; Lal, S; Nair, NP; Quirion, R; Suranyi-Cadotte, B1
Kulkarni, SK; Kunchandy, J1
Teo, WL; Wong, PT1
Glushakov, PG1
Kunert-Radek, J; Pawlikowski, M; Radek, A; Stepien, H1
Belin, C; Carriot, T; Dubroeucq, MC; Guérémy, C; Le Fur, G; Mestre, M; Renault, C; Uzan, A1
Brown, C; Martin, IL1
Phillis, JW1
Chen Chow, S; Davies, LP; Johnston, GA; Skerritt, JH1
Garattini, S; Mennini, T1
File, SE; Green, AR; Nutt, DJ; Vincent, ND1
Coffin, VL; Phillis, JW; Wu, PH1
Lloyd, HG; Morgan, PF; Stone, TW1
Ramanjaneyulu, R; Ticku, MK1
Hirsch, JD1
Cuparencu, B; Horák, J1
Antonenko, YN; Kinnally, KW; McEnery, MW; Snyder, SH; Tedeschi, H; Zorov, DB1
Chen, JS; Gee, KW; Johnson, D; Lan, NC1
Matthews, EK; Ratcliffe, SL1
Chang, CC; Chiou, LC1
Lichtensteiger, W; Ramseier, H; Schlumpf, M1
Neu, JM; Niles, LP; Tenn, CC1
Cespuglio, R; Miachon, S1
Leeuwin, RS; van Hamme, J; van Wilgenburg, H; Zeegers, A1
Kulkarni, SK; Reddy, DS1
Katukov, VIu; Lesnichuk, SA; Porodenko, NV; Severin, ES1
Kawaguchi, M; Okubo, M1
Bender, AS; Norenberg, MD1
Kaur, G; Kulkarni, SK; Raghavendra, V1
Bruni, F; Ciciani, G; Costa, B; Costagli, C; Costanzo, A; Guerrini, G; Martini, C; Selleri, S1
Biggio, G; Latrofa, A; Papi, G; Pisu, MG; Porcu, P; Serra, M; Trapani, G1
Dehne, MG; Engel, J; Fuchs, M; Gonter, J; Hempelmann, G; Krüll, M; Matejec, R; Menges, T; Mühling, J; Nickolaus, KA; Sablotzki, A; Welters, ID; Wolff, M1
Chen, SL; Liu, XG; Wei, XH; Zang, Y; Zheng, WH1

Reviews

5 review(s) available for flumazenil and ro 5-4864

ArticleYear
Memory modulation by brain benzodiazepines.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 1991, Volume: 24, Issue:9

    Topics: Animals; Avoidance Learning; Benzodiazepines; Benzodiazepinones; Brain; Brain Chemistry; Convulsants; Down-Regulation; Flumazenil; Habituation, Psychophysiologic; Memory; Muscimol; Rats

1991
The role of adenosine in the central actions of the benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1988, Volume: 12, Issue:4

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Arousal; Benzodiazepinones; Brain; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Neural Inhibition; Neurons; Purkinje Cells; Rats; Receptors, GABA-A

1988
Behavioural actions of Ro 5-4864: a peripheral-type benzodiazepine?
    Life sciences, 1984, Jul-16, Volume: 35, Issue:3

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Binding Sites; Brain; Convulsants; Drug Interactions; Flumazenil; Humans; Isoquinolines; Kidney; Phenytoin; Picrotoxin; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A

1984
Multiple sites of action for anxiogenic drugs: behavioural, electrophysiological and biochemical correlations.
    Psychopharmacology, 1984, Volume: 83, Issue:4

    Topics: Action Potentials; Animals; Anxiety; Behavior, Animal; Benzodiazepinones; Binding Sites; Brain Chemistry; Carbolines; Cats; Flumazenil; Humans; Mice; Rats; Receptors, GABA-A

1984
Adenosine's role in the central actions of the benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1984, Volume: 8, Issue:4-6

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Brain; Cats; Cell Line; Cerebral Cortex; Diazepam; Flumazenil; Rats; Synaptosomes; Thioinosine

1984

Other Studies

64 other study(ies) available for flumazenil and ro 5-4864

ArticleYear
Synthesis and biological evaluation of 4-phenylquinazoline-2-carboxamides designed as a novel class of potent ligands of the translocator protein.
    Journal of medicinal chemistry, 2012, May-10, Volume: 55, Issue:9

    Topics: Animals; Binding, Competitive; Carrier Proteins; Cell Line, Tumor; Cell Survival; Inhibitory Concentration 50; Molecular Structure; Quinazolines; Rats; Receptors, GABA-A; Structure-Activity Relationship

2012
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Effects of central and peripheral type benzodiazepine ligands on thyrotropin and prolactin secretion.
    Neuropeptides, 1992, Volume: 21, Issue:3

    Topics: Animals; Benzodiazepinones; Carbolines; Clonazepam; Cold Temperature; Diazepam; Flumazenil; Hypothalamo-Hypophyseal System; Isoquinolines; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Secretory Rate; Thyrotropin; Thyrotropin-Releasing Hormone

1992
Modulation of noise-potentiated acoustic startle via the benzodiazepine--gamma-aminobutyric acid receptor complex.
    Behavioral neuroscience, 1991, Volume: 105, Issue:5

    Topics: Acoustic Stimulation; Animals; Auditory Perception; Benzodiazepinones; Brain; Convulsants; Diazepam; Flumazenil; GABA-A Receptor Antagonists; Male; Neurons; Rats; Receptors, GABA-A; Reflex, Startle

1991
Benzodiazepine receptor ligand influences on acquisition: suggestion of an endogenous modulatory mechanism mediated by benzodiazepine receptors.
    Behavioral and neural biology, 1990, Volume: 54, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Arousal; Avoidance Learning; Benzodiazepinones; Brain; Carbolines; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Flumazenil; Habituation, Psychophysiologic; Memory; Mental Recall; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Retention, Psychology

1990
Relaxant effect of benzodiazepines on uterine rings isolated from estrogen-treated rats.
    European journal of pharmacology, 1990, Aug-28, Volume: 185, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Bicuculline; Clonazepam; Convulsants; Diazepam; Estradiol; Estrogens; Female; Flumazenil; In Vitro Techniques; Isoquinolines; Muscle, Smooth; Potassium Chloride; Propranolol; Rats; Rats, Inbred Strains; Uterine Contraction

1990
Diazepam-binding inhibitor: a neuropeptide and/or an acyl-CoA ester binding protein?
    The Biochemical journal, 1990, Feb-01, Volume: 265, Issue:3

    Topics: Acyl Coenzyme A; Adrenal Cortex; Amino Acid Sequence; Animals; Benzodiazepinones; Brain; Carboxylic Acids; Carrier Proteins; Cattle; Diazepam; Diazepam Binding Inhibitor; Esters; Flumazenil; Liver; Molecular Sequence Data; Nerve Tissue Proteins; Neuropeptides; Peptide Fragments; Rats

1990
A natural processing product of rat diazepam binding inhibitor, triakontatetraneuropeptide (diazepam binding inhibitor 17-50) contains an alpha-helix, which allows discrimination between benzodiazepine binding site subtypes.
    Molecular pharmacology, 1990, Volume: 37, Issue:2

    Topics: Amino Acid Sequence; Animals; Benzodiazepinones; Binding, Competitive; Circular Dichroism; Flumazenil; In Vitro Techniques; Models, Molecular; Molecular Sequence Data; Neuropeptides; Peptide Fragments; Protein Conformation; Rats; Receptors, GABA-A; Structure-Activity Relationship

1990
Pharmacological inhibition of forskolin-stimulated adenylate cyclase activity in rat brain by melatonin, its analogs, and diazepam.
    Biochemical pharmacology, 1990, Dec-15, Volume: 40, Issue:12

    Topics: Adenylyl Cyclases; Animals; Benzodiazepinones; Brain; Brain Mapping; Cell Membrane; Colforsin; Corpus Striatum; Diazepam; Dose-Response Relationship, Drug; Enzyme Activation; Flumazenil; In Vitro Techniques; Male; Melatonin; Rats; Rats, Inbred Strains

1990
Diminution by benzodiazepines of the chronotropic responses to noradrenaline in rat isolated atria.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Colforsin; Cyclic AMP; Diazepam; Female; Flumazenil; Heart; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains

1989
Anticonvulsant activity of the diaryltriazine, LY81067: studies using electroencephalographic recording and positron emission tomography.
    Neuropharmacology, 1989, Volume: 28, Issue:4

    Topics: Animals; Anticonvulsants; Behavior, Animal; Benzodiazepinones; Brain; Convulsants; Electroencephalography; Epilepsy; Flumazenil; Injections, Intravenous; Male; Papio; Tomography, Emission-Computed; Triazines

1989
The benzodiazepine receptor ligands RO 5-4864 and RO 15-1788 do not block the inhibition of PAF-induced platelet aggregation seen with the hetrazepine WEB2086.
    Biochemical and biophysical research communications, 1989, Apr-14, Volume: 160, Issue:1

    Topics: Adenosine Triphosphate; Animals; Azepines; Benzodiazepinones; Blood Platelets; Female; Flumazenil; Male; Platelet Activating Factor; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Rabbits; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Receptors, GABA-A; Triazines; Triazoles

1989
Relaxation of rat vascular muscle by peripheral benzodiazepine modulators.
    The Journal of clinical investigation, 1989, Volume: 84, Issue:2

    Topics: Animals; Benzodiazepinones; Calcium; Calcium Channel Blockers; Flumazenil; Guanylate Cyclase; In Vitro Techniques; Isoquinolines; Potassium; Rats; Rats, Inbred WKY; Receptors, GABA-A; Vasodilation

1989
Benzodiazepine interactions with GABAA receptors on chick ciliary ganglion neurons.
    Molecular pharmacology, 1988, Volume: 34, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Cell Membrane; Cells, Cultured; Chick Embryo; Flumazenil; Flunitrazepam; Ganglia, Parasympathetic; Membrane Potentials; Receptors, GABA-A; Spinal Cord

1988
Regional ontogenetic profile of central and peripheral benzodiazepine receptors in the guinea pig brain.
    Neuroscience letters, 1988, Sep-23, Volume: 92, Issue:1

    Topics: Aging; Animals; Benzodiazepinones; Brain; Flumazenil; Guinea Pigs; Receptors, GABA-A

1988
Anxiolytic and anxiogenic drug effects on exploratory activity in an elevated plus-maze: a novel test of anxiety in the rat.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Convulsants; Exploratory Behavior; Flumazenil; Male; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats

1986
Triazolodiazepines: dissociation of their Paf (platelet activating factor) antagonistic and CNS activity.
    British journal of pharmacology, 1987, Volume: 90, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Azepines; Benzodiazepinones; Central Nervous System; Flumazenil; Guinea Pigs; Humans; Hypnotics and Sedatives; In Vitro Techniques; Platelet Activating Factor; Platelet Aggregation; Receptors, GABA-A; Tidal Volume; Triazolam

1987
Opposite effects of two ligands for peripheral type benzodiazepine binding sites, PK 11195 and RO5-4864, in a conflict situation in the rat.
    Life sciences, 1985, Mar-18, Volume: 36, Issue:11

    Topics: Animals; Benzodiazepinones; Carbolines; Conditioning, Operant; Conflict, Psychological; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Flumazenil; Isoquinolines; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
The anxiogenic action of RO 5-4864 in the social interaction test: effect of chlordiazepoxide, RO 15-1788 and CGS 8216.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 328, Issue:3

    Topics: Animals; Anxiety; Benzodiazepinones; Chlordiazepoxide; Convulsants; Drug Interactions; Flumazenil; Humans; Male; Motor Activity; Pyrazoles; Rats; Receptors, GABA-A; Social Behavior

1985
Blockade of the diazepam-induced increase in rat striatal acetylcholine content by the specific benzodiazepine antagonists ethyl-beta-carboline-3-carboxylate and Ro 15-1788.
    Brain research, 1985, Jun-17, Volume: 336, Issue:2

    Topics: Acetylcholine; Animals; Benzodiazepines; Benzodiazepinones; Brain Chemistry; Carbolines; Corpus Striatum; Diazepam; Female; Flumazenil; Indoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Clonazepam-induced hyperphagia in nondeprived rats: tests of pharmacological specificity with Ro5-4864, Ro5-3663, Ro15-1788 and CGS 9896.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:5

    Topics: Animals; Benzodiazepinones; Clonazepam; Drug Interactions; Feeding Behavior; Flumazenil; Humans; Hyperphagia; Male; Pyrazoles; Rats; Receptors, GABA-A

1985
Monoclonal antibodies to benzodiazepines.
    Journal of neurochemistry, 1985, Volume: 45, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Antibodies, Monoclonal; Benzodiazepines; Benzodiazepinones; Diazepam; Flumazenil; Flunitrazepam; Flurazepam; Mice; Mice, Inbred BALB C; Receptors, GABA-A; Structure-Activity Relationship

1985
Benzodiazepine binding characteristics of embryonic rat brain neurons grown in culture.
    Journal of neurochemistry, 1985, Volume: 45, Issue:6

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cells, Cultured; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Neurons; Pyridazines; Rats; Receptors, GABA-A

1985
Solubilization of peripheral benzodiazepine-binding sites from rat kidney.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1985, Volume: 5, Issue:11

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Carbolines; Chlordiazepoxide; Clonazepam; Diazepam; Digitonin; Flumazenil; Flurazepam; Guanidine; Guanidines; Hot Temperature; Isoquinolines; Kidney; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Solubility; Time Factors; Urea

1985
Subcellular localization of "peripheral-type" binding sites for benzodiazepines in rat brain.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: Animals; Benzodiazepinones; Binding Sites; Brain; Cell Nucleus; Flumazenil; Male; Mitochondria; Myelin Sheath; Rats; Rats, Inbred Strains; Receptors, GABA-A; Subcellular Fractions; Synaptosomes

1986
Antagonism of flurazepam and other effects of Ro15-1788, PK8165 and Ro5-4864 on the GABA-A receptor complex in rat cuneate nucleus.
    European journal of pharmacology, 1985, Oct-29, Volume: 117, Issue:1

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Drug Synergism; Flumazenil; Flurazepam; In Vitro Techniques; Male; Medulla Oblongata; Muscimol; Pentobarbital; Picrotoxin; Quinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Effects of the benzodiazepine receptor ligands midazolam, Ro 15-1788, and Ro 5-4864, alone and in combinations, on platelet serotonin uptake.
    Pharmacopsychiatry, 1986, Volume: 19, Issue:1

    Topics: Benzodiazepines; Benzodiazepinones; Blood Platelets; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Humans; In Vitro Techniques; Kinetics; Midazolam; Receptors, GABA-A; Serotonin

1986
The peripheral benzodiazepine receptor ligand Ro 5-4864 induces supraspinal convulsions in rabbits. Reversal by the central benzodiazepine antagonist Ro 15-1788.
    Psychopharmacology, 1986, Volume: 88, Issue:3

    Topics: Animals; Benzodiazepinones; Convulsants; Electrodes, Implanted; Electroencephalography; Flumazenil; Male; Rabbits; Receptors, GABA-A; Seizures

1986
Convulsant effect of Ro 5-4864, a peripheral type benzodiazepine, on the baboon (Papio papio).
    Neuroscience letters, 1986, May-15, Volume: 66, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Isoquinolines; Papio; Receptors, GABA-A; Seizures

1986
Rat hypothalamus contains an antimitogenic factor acting via benzodiazepine receptors.
    Experimental and clinical endocrinology, 1986, Volume: 88, Issue:3

    Topics: Animals; Benzodiazepinones; Flumazenil; Hypothalamus; Ligands; Lymphocyte Activation; Male; Mice; Mice, Inbred BALB C; Mitogens; Peptides; Rats; Receptors, GABA-A; Tissue Extracts

1986
Coexistence of central and peripheral benzodiazepine binding sites in the human pineal gland.
    Life sciences, 1987, Apr-13, Volume: 40, Issue:15

    Topics: Aged; Benzodiazepinones; Binding, Competitive; Cell Membrane; Clonazepam; Female; Flumazenil; Flunitrazepam; Humans; Isoquinolines; Male; Middle Aged; Pineal Gland; Receptors, GABA-A

1987
Naloxone-sensitive and GABAA receptor mediated analgesic response of benzodiazepines in mice.
    Methods and findings in experimental and clinical pharmacology, 1987, Volume: 9, Issue:2

    Topics: Analgesics; Animals; Benzodiazepines; Benzodiazepinones; Bicuculline; Female; Flumazenil; Male; Mice; Naloxone; Phenytoin; Reaction Time; Receptors, GABA-A

1987
Enhancement of estradiol-induced DNA synthesis in the anterior pituitary gland by the peripheral-type benzodiazepine receptor ligand Ro 5-4864.
    Journal of neural transmission, 1986, Volume: 66, Issue:3-4

    Topics: Animals; Benzodiazepinones; DNA; Drug Synergism; Estradiol; Flumazenil; Male; Mitosis; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Valproic Acid

1986
Diazepam-sensitive specific binding of phenytoin in rat brain.
    Journal of receptor research, 1986, Volume: 6, Issue:3-4

    Topics: Animals; Benzodiazepinones; Binding Sites; Cell Membrane; Cerebral Cortex; Clonazepam; Diazepam; Flumazenil; Male; Phenytoin; Rats; Rats, Inbred Strains

1986
[Effect of RO 15-1788 and RO 5-4684 on the evoked activity of neurons in hippocampal sections].
    Biulleten' eksperimental'noi biologii i meditsiny, 1987, Volume: 104, Issue:12

    Topics: Animals; Benzodiazepinones; Evoked Potentials; Flumazenil; Hippocampus; In Vitro Techniques; Rats

1987
Inhibition of cell proliferation of human gliomas by benzodiazepines in vitro.
    Acta neurologica Scandinavica, 1988, Volume: 77, Issue:3

    Topics: Astrocytoma; Benzodiazepines; Benzodiazepinones; Cell Division; Clonazepam; Diazepam; Female; Flumazenil; Glioma; Humans; Male; Middle Aged; Thymidine; Tumor Cells, Cultured

1988
Electrophysiological and pharmacological characterization of peripheral benzodiazepine receptors in a guinea pig heart preparation.
    Life sciences, 1984, Aug-27, Volume: 35, Issue:9

    Topics: Action Potentials; Animals; Benzodiazepinones; Clonazepam; Convulsants; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Flumazenil; Guinea Pigs; Heart; In Vitro Techniques; Isoquinolines; Myocardial Contraction; Myocardium; Receptors, Cell Surface; Receptors, GABA-A

1984
Autoradiographic localisation of benzodiazepine receptors in the rat pituitary gland.
    European journal of pharmacology, 1984, Jul-20, Volume: 102, Issue:3-4

    Topics: Animals; Autoradiography; Benzodiazepinones; Clonazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Purines interact with 'central' but not 'peripheral' benzodiazepine binding sites.
    Neuroscience letters, 1982, Dec-23, Volume: 34, Issue:1

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Diazepam; Flumazenil; Purines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Synaptosomes

1982
RO5-4864, a ligand for benzodiazepine micromolar and peripheral binding sites: antagonism and enhancement of behavioural effects.
    Psychopharmacology, 1983, Volume: 80, Issue:2

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Drug Interactions; Flumazenil; Male; Motor Activity; Phenytoin; Picrotoxin; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Benzodiazepines receptor binding in vivo: pharmacokinetic and pharmacological significance.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Adrenal Glands; Animals; Benzodiazepinones; Brain; Carbolines; Corticosterone; Diazepam; Flumazenil; Flunitrazepam; Kinetics; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
On the convulsant action of Ro 5-4864 and the existence of a micromolar benzodiazepine binding site in rat brain.
    Psychopharmacology, 1984, Volume: 82, Issue:3

    Topics: Animals; Benzodiazepinones; Binding Sites; Brain; Convulsants; Diazepam; Electroshock; Flumazenil; Male; Mice; Pentylenetetrazole; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1984
Inhibition of adenosine uptake into rat brain synaptosomes by prostaglandins, benzodiazepines and other centrally active compounds.
    General pharmacology, 1983, Volume: 14, Issue:5

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Brain; Calmodulin; Carbolines; Flumazenil; Hydroxyzine; Imidazoles; Male; Prostaglandins; Pyrazoles; Rats; Rats, Inbred Strains; Sulfonamides; Synaptosomes

1983
Inhibition of adenosine accumulation by a CNS benzodiazepine antagonist (Ro 15-1788) and a peripheral benzodiazepine receptor ligand (Ro 05-4864).
    Neuroscience letters, 1983, Oct-31, Volume: 41, Issue:1-2

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Central Nervous System; Diazepam; Flumazenil; Flurazepam; Hexobendine; Male; Rats; Synaptosomes; Time Factors

1983
RO5-4864 inhibits the binding of [35S]t-butylbicyclophosphorothionate to rat brain membranes.
    Life sciences, 1984, Feb-13, Volume: 34, Issue:7

    Topics: Androstanes; Animals; Azasteroids; Benzodiazepinones; Bicuculline; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cell Membrane; Cerebellum; Cerebral Cortex; Dose-Response Relationship, Drug; Flumazenil; Hippocampus; Male; Picrotoxin; Radioligand Assay; Rats

1984
Peripheral and central-type benzodiazepine binding sites in mammalian ocular tissues.
    Experimental eye research, 1984, Volume: 38, Issue:1

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Eye; Female; Flumazenil; Flunitrazepam; Macaca mulatta; Male; Rabbits; Rats; Rats, Inbred Strains

1984
Effects of 4'-chlordiazepam on glycemia and serum lipids in hyperlipidemic rats: interactions with PK 11195 and flumazenil.
    Research communications in molecular pathology and pharmacology, 1995, Volume: 89, Issue:1

    Topics: Animals; Benzodiazepinones; Blood Glucose; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Hypolipidemic Agents; Isoquinolines; Lipids; Male; Rats; Rats, Wistar; Receptors, GABA-A

1995
Mitochondrial benzodiazepine receptor linked to inner membrane ion channels by nanomolar actions of ligands.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Feb-15, Volume: 90, Issue:4

    Topics: Animals; Benzodiazepinones; Clonazepam; Convulsants; Flumazenil; Intracellular Membranes; Ion Channels; Isoquinolines; Male; Membrane Potentials; Mitochondria, Heart; Protoporphyrins; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Submitochondrial Particles

1993
Differential effects of 4'-chlorodiazepam on expressed human GABAA receptors.
    Journal of neurochemistry, 1995, Volume: 64, Issue:2

    Topics: Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Clonazepam; Flumazenil; Humans; Quinolines; Receptors, GABA; Transfection

1995
Modification of the photodynamic action of delta-aminolaevulinic acid (ALA) on rat pancreatoma cells by mitochondrial benzodiazepine receptor ligands.
    British journal of cancer, 1995, Volume: 71, Issue:2

    Topics: Aminolevulinic Acid; Animals; Benzodiazepines; Benzodiazepinones; Cell Division; Cell Survival; Clonazepam; Flumazenil; Isoquinolines; Ligands; Mitochondria; Oxygen; Pancreatic Neoplasms; Photochemotherapy; Protoporphyrins; Radiation-Protective Agents; Radiation-Sensitizing Agents; Rats; Receptors, GABA-A; Singlet Oxygen; Tumor Cells, Cultured

1995
Pharmacological relevance of peripheral type benzodiazepine receptors on motor nerve and skeletal muscle.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Benzodiazepinones; Diaphragm; Electric Stimulation; Electrophysiology; Female; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Microelectrodes; Motor Endplate; Motor Neurons; Muscle Contraction; Muscles; Neostigmine; Phrenic Nerve

1994
In vitro inhibition of cellular immune responses by benzodiazepines and PK 11195. Effects on mitogen- and alloantigen-driven lymphocyte proliferation and on IL-1, IL-2 synthesis and IL-2 receptor expression.
    Immunopharmacology and immunotoxicology, 1993, Volume: 15, Issue:5

    Topics: Animals; B-Lymphocytes; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Female; Flumazenil; Immunity, Cellular; In Vitro Techniques; Interleukin-1; Interleukin-2; Isoquinolines; Lymphocyte Activation; Male; Mice; Mice, Inbred A; Mice, Inbred C57BL; Neuroimmunomodulation; Receptors, GABA-A; T-Lymphocytes

1993
PK 11195 blockade of benzodiazepine-induced inhibition of forskolin-stimulated adenylate cyclase activity in the striatum.
    British journal of pharmacology, 1996, Volume: 119, Issue:2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Benzodiazepines; Benzodiazepinones; Colforsin; Corpus Striatum; Diazepam; Drug Interactions; Flumazenil; GABA-A Receptor Antagonists; Guanosine Triphosphate; Indoles; Isoquinolines; Kinetics; Male; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Stimulation, Chemical; Virulence Factors, Bordetella

1996
Prevention of ACTH- and adrenalectomy-induced muricidal behavior: by benzodiazepinic ligands.
    Peptides, 1997, Volume: 18, Issue:2

    Topics: Adrenalectomy; Adrenocorticotropic Hormone; Aggression; Animals; Benzodiazepinones; Clonazepam; Flumazenil; GABA Modulators; Isoquinolines; Male; Mice; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A; Time Factors

1997
Modification of cardiac actions of RO 05-4864 by PK 11195 and flumazenil in the perfused rat heart.
    Life sciences, 1997, Volume: 61, Issue:17

    Topics: Animals; Benzodiazepinones; Drug Interactions; Female; Flumazenil; Heart; Isoquinolines; Myocardial Contraction; Rats; Rats, Wistar; Regional Blood Flow

1997
Reversal of benzodiazepine inverse agonist FG 7142-induced anxiety syndrome by neurosteroids in mice.
    Methods and findings in experimental and clinical pharmacology, 1997, Volume: 19, Issue:10

    Topics: Animals; Anxiety; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; Isoquinolines; Male; Maze Learning; Mice; Mice, Inbred BALB C; Motor Activity; Progesterone; Receptors, GABA-A; Steroids

1997
[Characteristics of human lymphocyte benzodiazepine receptors].
    Biulleten' eksperimental'noi biologii i meditsiny, 1998, Volume: 126, Issue:10

    Topics: Adult; Baclofen; Benzodiazepinones; Binding, Competitive; Diazepam; Flumazenil; GABA Agonists; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Ligands; Lymphocytes; Male; Receptors, GABA-A

1998
Inhibitory regulation of amylase release in rat parotid acinar cells by benzodiazepine receptors.
    European journal of pharmacology, 1998, Oct-23, Volume: 359, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amylases; Animals; Atropine; Benzodiazepinones; Carbachol; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoproterenol; Male; Muscarinic Agonists; Muscarinic Antagonists; Parotid Gland; Propranolol; Rats; Rats, Wistar; Receptors, GABA-A

1998
Effect of benzodiazepines and neurosteroids on ammonia-induced swelling in cultured astrocytes.
    Journal of neuroscience research, 1998, Dec-01, Volume: 54, Issue:5

    Topics: Ammonia; Astrocytes; Atrial Natriuretic Factor; Benzodiazepines; Benzodiazepinones; Brain Edema; Cell Size; Clonazepam; Dehydroepiandrosterone Sulfate; Desoxycorticosterone; Diazepam; Diazepam Binding Inhibitor; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoquinolines; Nerve Tissue Proteins; Neuropeptides; Peptide Fragments; Pregnanolone; Pregnenolone; Protoporphyrins; Receptors, GABA-A; Steroids; Up-Regulation

1998
Anti-depressant action of melatonin in chronic forced swimming-induced behavioral despair in mice, role of peripheral benzodiazepine receptor modulation.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2000, Volume: 10, Issue:6

    Topics: Alprazolam; Analysis of Variance; Animals; Anti-Anxiety Agents; Antioxidants; Benzodiazepinones; Bicuculline; Convulsants; Depression; Disease Models, Animal; Drug Interactions; Drug Therapy, Combination; Flumazenil; GABA Agents; Immobilization; Isoquinolines; Male; Melatonin; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Receptors, GABA-A; Swimming; Time Factors

2000
2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective peripheral benzodiazepine receptor ligands.
    Bioorganic & medicinal chemistry, 2001, Volume: 9, Issue:10

    Topics: Acetamides; Animals; Benzodiazepinones; Binding Sites; Cerebral Cortex; Clonazepam; Flumazenil; Glioma; Intracellular Membranes; Isoquinolines; Kidney; Ligands; Magnetic Resonance Spectroscopy; Molecular Structure; Pyrazoles; Pyrimidines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Thermodynamics; Tumor Cells, Cultured

2001
Binding of [3H]CB 34, a selective ligand for peripheral benzodiazepine receptors, to rat brain membranes.
    European journal of pharmacology, 2001, Dec-07, Volume: 432, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Female; Flumazenil; Imidazoles; Indoleacetic Acids; Isoquinolines; Ligands; Membrane Proteins; Membranes; Nordazepam; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tritium

2001
Benzodiazepine receptor-dependent modulation of neutrophil (PMN) free amino- and alpha-keto acid profiles or immune functions.
    Amino acids, 2005, Volume: 28, Issue:1

    Topics: Adult; Amino Acids; Benzodiazepinones; Cells, Cultured; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Humans; Hydrogen Peroxide; Isoquinolines; Keto Acids; Male; Midazolam; Naloxone; Neutrophils; Peroxidase; Receptors, GABA-A; Superoxides

2005
Inhibition of Neuropathic Pain by a Single Intraperitoneal Injection of Diazepam in the Rat: Possible Role of Neurosteroids.
    The Chinese journal of physiology, 2016, 02-29, Volume: 59, Issue:1

    Topics: Animals; Benzodiazepinones; Carrier Proteins; Diazepam; Flumazenil; Injections, Intraperitoneal; Interleukin-1beta; Male; Neuralgia; Neurotransmitter Agents; Pregnenolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

2016