flumazenil and piperidines

flumazenil has been researched along with piperidines in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19904 (17.39)18.7374
1990's3 (13.04)18.2507
2000's6 (26.09)29.6817
2010's9 (39.13)24.3611
2020's1 (4.35)2.80

Authors

AuthorsStudies
Borsini, F; D'Aranno, V; Lecci, A; Mancinelli, A; Meli, A; Stasi, MA; Volterra, G1
Insel, TR; Winslow, JT1
Kumasaka, Y; Ueki, S; Yamamoto, T1
Le Bihan, C; Simon, P; Soubrié, P; Thiébot, MH1
Comar, D; Maziere, M; Turner, JH1
Allikmets, LKh; Maĭmets, MO; Nurk, AM; Riago, LK; Vasar, EE1
Brown, RE; Dastur, FN; McGregor, IS; McLellan, RA1
Pennell, PB1
Bergström, M; Hillered, L; Långström, B; Marklund, N; Sihver, S; Watanabe, Y1
Abe, K; Hatazawa, J; Hosoi, R; Inoue, O; Kashiwagi, Y; Tokumura, M1
Bernöster, K; Dost, R; Egerland, U; Langen, B; Rundfeldt, C; Unverferth, K1
Hendrikse, NH; Ishiwata, K; Kawamura, K; Yanai, K1
Langen, B; Rundfeldt, C1
Baburin, I; Hamburger, M; Hering, S; Kim, HJ; Strommer, B; Zaugg, J1
Gerónimo Pardo, M; Mateo Cerdán, CM; Moreno Salcedo, JM1
Anastasiou, E; Andreotti, B; Chapsa, C; Karakosta, A; Pouliou, A1
Brito, GA; Cavalheiro, EA; da Costa, MA; da Cruz, GM; da Graça Naffah-Mazzacoratti, M; de Andrade, GM; de Barros Viana, GS; Felipe, CF; Leal, LK; Menezes, ML; Scorza, FA; Tavares, AF1
Kawamata, M; Kawamata, T; Koike, Y; Yamamoto, K1
Jang, YP; Jung, JW; Kim, DH; Ko, ES; Lee, JH; Lee, S; Oh, WB; Ryu, JH; Seo, YT1
Hashimoto, T; Hatayama, Y; Nakamichi, K; Yoshida, N1
Arnason, JT; Cal, V; Cayer, C; Harris, CS; Kent, P; Liu, R; Merali, Z1
Arnulf, I; Dodet, P; Leu-Semenescu, S1
Shimizu, T; Takasusuki, T; Yamaguchi, S1

Reviews

2 review(s) available for flumazenil and piperidines

ArticleYear
PET: cholinergic neuroreceptor mapping.
    Advances in neurology, 2000, Volume: 83

    Topics: Benzilates; Brain; Calcium Channel Blockers; Epilepsy, Temporal Lobe; Flumazenil; GABA Modulators; Humans; Piperidines; Receptors, Cholinergic; Tomography, Emission-Computed

2000
Precision Medicine for Idiopathic Hypersomnia.
    Sleep medicine clinics, 2019, Volume: 14, Issue:3

    Topics: Central Nervous System Stimulants; Clarithromycin; Flumazenil; GABA Modulators; Humans; Idiopathic Hypersomnia; Mazindol; Modafinil; Orexins; Piperidines; Polysomnography; Precision Medicine; Sleep; Sodium Oxybate; Wakefulness; Wakefulness-Promoting Agents

2019

Trials

2 trial(s) available for flumazenil and piperidines

ArticleYear
Flumazenil expedites recovery from sevoflurane/remifentanil anaesthesia when administered to healthy unpremedicated patients.
    European journal of anaesthesiology, 2010, Volume: 27, Issue:11

    Topics: Adult; Aged; Anesthesia Recovery Period; Anesthetics, Inhalation; Anesthetics, Intravenous; Double-Blind Method; Elective Surgical Procedures; Female; Flumazenil; GABA Modulators; Humans; Male; Methyl Ethers; Middle Aged; Piperidines; Remifentanil; Sevoflurane

2010
Remimazolam Compared to Propofol for Total Intravenous Anesthesia with Remifentanil on the Recovery of Psychomotor Function: A Randomized Controlled Trial.
    Advances in therapy, 2023, Volume: 40, Issue:10

    Topics: Anesthesia, Intravenous; Anesthetics, Intravenous; Flumazenil; Humans; Piperidines; Propofol; Remifentanil

2023

Other Studies

19 other study(ies) available for flumazenil and piperidines

ArticleYear
Effect of serotoninergic drugs on stress-induced hyperthermia (SIH) in mice.
    Journal of neural transmission. General section, 1990, Volume: 82, Issue:3

    Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Body Temperature Regulation; Buspirone; Diazepam; Ergolines; Fenclonine; Fever; Flumazenil; Imidazoles; Male; Mice; Ondansetron; Piperazines; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Stress, Psychological; Tetrahydronaphthalenes

1990
Serotonergic and catecholaminergic reuptake inhibitors have opposite effects on the ultrasonic isolation calls of rat pups.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1990, Volume: 3, Issue:1

    Topics: Animals; Body Temperature; Catecholamines; Citalopram; Clomipramine; Desipramine; Flumazenil; Mazindol; Motor Activity; Naltrexone; Nortriptyline; Paroxetine; Piperidines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Stress, Psychological; Ultrasonics; Vocalization, Animal

1990
Behavioral analysis of zopiclone on the basis of their discriminative stimulus properties in the rat.
    Japanese journal of pharmacology, 1989, Volume: 51, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Behavior, Animal; Benzodiazepines; Bicuculline; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Hypnotics and Sedatives; Male; Muscimol; Naphthyridines; Pentylenetetrazole; Piperazines; Piperidines; Rats; Rats, Inbred WKY; Ritanserin; Serotonin Antagonists; Sulfur Compounds

1989
Benzodiazepines reduce the tolerance to reward delay in rats.
    Psychopharmacology, 1985, Volume: 86, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Choice Behavior; Diazepam; Flumazenil; Male; Piperidines; Rats; Rats, Inbred Strains; Reward; Serotonin Antagonists; Synaptic Transmission; Zimeldine

1985
Localization of 11C-radiopharmaceuticals in the Greene melanoma of hamsters.
    European journal of nuclear medicine, 1985, Volume: 10, Issue:9-10

    Topics: Animals; Benzodiazepinones; Carbon Radioisotopes; Chlorpromazine; Cricetinae; Flumazenil; Flunitrazepam; Gallium Radioisotopes; Isotope Labeling; Ketanserin; Melanoma; Mesocricetus; Methionine; Neoplasm Transplantation; Pimozide; Piperidines; Quinuclidinyl Benzilate; Radionuclide Imaging; Tissue Distribution

1985
[Effect of an imidazobenzodiazepine (RO 15-1788) on aggressive behavior in mice].
    Biulleten' eksperimental'noi biologii i meditsiny, 1984, Volume: 98, Issue:10

    Topics: Aggression; Animals; Apomorphine; Benzodiazepinones; Brain; Catalepsy; Dose-Response Relationship, Drug; Flumazenil; Haloperidol; Humans; Hydroxyindoleacetic Acid; Male; Mice; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin

1984
Cannabinoid modulation of rat pup ultrasonic vocalizations.
    European journal of pharmacology, 1996, Oct-10, Volume: 313, Issue:1-2

    Topics: Analysis of Variance; Animals; Animals, Newborn; Behavior, Animal; Benzazepines; Body Temperature; Cannabinoids; Cyclohexanols; Dopamine Antagonists; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Hypothermia; Motor Activity; Naloxone; Narcotic Antagonists; Piperidines; Pyrazoles; Rats; Rimonabant; Vocalization, Animal

1996
Changes in mACh, NMDA and GABA(A) receptor binding after lateral fluid-percussion injury: in vitro autoradiography of rat brain frozen sections.
    Journal of neurochemistry, 2001, Volume: 78, Issue:3

    Topics: Animals; Autoradiography; Binding Sites; Brain; Brain Injuries; Cerebral Cortex; Dizocilpine Maleate; Flumazenil; Frozen Sections; Hippocampus; Humans; Kinetics; Male; Nitriles; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Muscarinic; Receptors, N-Methyl-D-Aspartate; Tomography, Emission-Computed

2001
Discrepancy between cell injury and benzodiazepine receptor binding after transient middle cerebral artery occlusion in rats.
    Synapse (New York, N.Y.), 2004, Sep-15, Volume: 53, Issue:4

    Topics: Animals; Autoradiography; Benzazepines; Benzilates; Binding Sites; Binding, Competitive; Cerebral Cortex; Cerebral Infarction; Corpus Striatum; Disease Models, Animal; Down-Regulation; Flumazenil; Infarction, Middle Cerebral Artery; Male; Nerve Degeneration; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D1; Receptors, GABA-A; Receptors, Muscarinic; Reperfusion Injury; Sensitivity and Specificity; Tritium

2004
Characterization in rats of the anxiolytic potential of ELB139 [1-(4-chlorophenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-on], a new agonist at the benzodiazepine binding site of the GABAA receptor.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Binding Sites; Binding, Competitive; Conflict, Psychological; Diazepam; Drug Tolerance; Flumazenil; Flunitrazepam; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Light; Male; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Rats; Rats, Wistar

2005
In vivo evaluation of P-glycoprotein modulation of 8 PET radioligands used clinically.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 2007, Volume: 48, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Brain; Cyclosporine; Donepezil; Flumazenil; Indans; Ligands; Male; Mice; Piperidines; Positron-Emission Tomography; Radioisotopes; Sensory Receptor Cells; Verapamil; Xanthines

2007
ELB139 an agonist at the benzodiazepine binding site increases 5-HT in the striatum and prefrontal cortex of rats: a microdialysis study.
    Pharmacology, biochemistry, and behavior, 2007, Volume: 86, Issue:1

    Topics: Animals; Chromatography, High Pressure Liquid; Dopamine; Electrochemistry; Flumazenil; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; Imidazoles; Injections, Intraperitoneal; Male; Microdialysis; Neostriatum; Piperidines; Prefrontal Cortex; Raphe Nuclei; Rats; Rats, Wistar; Serotonin

2007
HPLC-based activity profiling: discovery of piperine as a positive GABA(A) receptor modulator targeting a benzodiazepine-independent binding site.
    Journal of natural products, 2010, Feb-26, Volume: 73, Issue:2

    Topics: Alkaloids; Animals; Benzodiazepines; Benzodioxoles; Binding Sites; Chloride Channels; Chromatography, High Pressure Liquid; Female; Flumazenil; Fruit; GABA Modulators; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Oocytes; Piper nigrum; Piperidines; Polyunsaturated Alkamides; Rats; Receptors, GABA-A; Xenopus laevis

2010
[Transient decerebrate rigidity from hypoxemia during administration of propofol, midazolam-flumazenil, and remifentanil-naloxone].
    Revista espanola de anestesiologia y reanimacion, 2010, Volume: 57, Issue:2

    Topics: Airway Obstruction; Anesthetics, Intravenous; Bradycardia; Cardiotonic Agents; Cholangiopancreatography, Endoscopic Retrograde; Choledocholithiasis; Decerebrate State; Flumazenil; GABA Agonists; Humans; Hypnotics and Sedatives; Hypoxia; Intraoperative Complications; Intubation, Intratracheal; Male; Midazolam; Middle Aged; Naloxone; Piperidines; Propofol; Remifentanil; Sleep Apnea, Obstructive

2010
Piperine decreases pilocarpine-induced convulsions by GABAergic mechanisms.
    Pharmacology, biochemistry, and behavior, 2013, Volume: 104

    Topics: Alkaloids; Amino Acids; Animals; Anticonvulsants; Antioxidants; Atropine; Benzodioxoles; Biogenic Monoamines; Brain; Diazepam; Disease Models, Animal; Epilepsy; Flumazenil; gamma-Aminobutyric Acid; Humans; Male; Memantine; Mice; Nimodipine; Nitrites; Pilocarpine; Piperidines; Polyunsaturated Alkamides; Seizures; Tumor Necrosis Factor-alpha

2013
[Improvement of consciousness by administration of flumazenil in a patient with unexpectedly delayed emergence from general anesthesia].
    Masui. The Japanese journal of anesthesiology, 2013, Volume: 62, Issue:4

    Topics: Anesthesia Recovery Period; Anesthesia, General; Consciousness; Female; Flumazenil; Humans; Middle Aged; Piperidines; Propofol; Remifentanil

2013
Involvement of histaminergic system in the anxiolytic-like activities of Morus alba leaves in mice.
    Biological & pharmaceutical bulletin, 2013, Volume: 36, Issue:11

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Flumazenil; GABA-A Receptor Antagonists; Histamine H3 Antagonists; Histidine Decarboxylase; Male; Mice; Mice, Inbred ICR; Morus; Piperazines; Piperidines; Plant Extracts; Plant Leaves; Pyridines; Serotonin Antagonists

2013
Procognitive effect of AC-3933 in aged mice, and synergistic effect of combination with donepezil in scopolamine-treated mice.
    European journal of pharmacology, 2014, Dec-15, Volume: 745

    Topics: Aging; Animals; Donepezil; Drug Synergism; Flumazenil; GABA-A Receptor Agonists; Indans; Male; Maze Learning; Memory Disorders; Mice; Mice, Inbred C57BL; Naphthyridines; Nootropic Agents; Oxadiazoles; Piperidines; Rats; Scopolamine

2014
Sacred Maya incense, copal (Protium copal - Burseraceae), has antianxiety effects in animal models.
    Journal of ethnopharmacology, 2018, Apr-24, Volume: 216

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Burseraceae; Carrier Proteins; Ceremonial Behavior; Disease Models, Animal; Endocannabinoids; Enzyme Inhibitors; Exploratory Behavior; Fear; Flumazenil; Humans; Male; Maze Learning; Monoacylglycerol Lipases; Phytotherapy; Piperidines; Plant Extracts; Plants, Medicinal; Pyrazoles; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, GABA-A; Resins, Plant; Signal Transduction; Social Behavior

2018