flumazenil and oxazepam

flumazenil has been researched along with oxazepam in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19907 (26.92)18.7374
1990's8 (30.77)18.2507
2000's6 (23.08)29.6817
2010's5 (19.23)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Hönack, D; Löscher, W1
Martin, WR; Pruitt, TA; Sloan, JW; Wala, EP1
Roth, SH; Sewell, RD; Tan, KS3
de la Garza, R; Evans, S; Johanson, CE1
Martin, WR; McNicholas, LF; Sloan, JW; Wala, E1
Galletly, DC; Maling, T; Short, TG1
File, SE; Wilks, LJ1
Jenck, F; Martin, JR; Moreau, JL1
Marinelli, FC; Pals, JK; Thibault, GE; Weinberg, AD1
Martin, WR; Sloan, JW; Wala, EP1
Sloan, JW; Wala, EP1
Jing, X; Sloan, JW; Wala, EP1
Blanc, F; Butterworth, RF; Fabbro-Peray, P; Lavoie, J; Layrargues, GP; Mousseau, DD; Perney, P1
Brewer, C; Gerra, G; Giusti, F; Moi, G; Zaimovic, A1
Lamas, E; Pellón, R; Rodríguez, C; Ruíz, A1
Goeders, NE; Guerin, GF; Spence, AL1

Reviews

1 review(s) available for flumazenil and oxazepam

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for flumazenil and oxazepam

ArticleYear
Intravenous flumazenil versus oxazepam tapering in the treatment of benzodiazepine withdrawal: a randomized, placebo-controlled study.
    Addiction biology, 2002, Volume: 7, Issue:4

    Topics: Adult; Anti-Anxiety Agents; Antidotes; Benzodiazepines; Blood Pressure; Cognition Disorders; Diagnostic and Statistical Manual of Mental Disorders; Drug Administration Schedule; Female; Flumazenil; Heart Rate; Humans; Injections, Intravenous; Male; MMPI; Oxazepam; Personality Disorders; Substance Withdrawal Syndrome; Wechsler Scales

2002

Other Studies

24 other study(ies) available for flumazenil and oxazepam

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Withdrawal precipitation by benzodiazepine receptor antagonists in dogs chronically treated with diazepam or the novel anxiolytic and anticonvulsant beta-carboline abecarnil.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Carbolines; Diazepam; Dogs; Female; Flumazenil; GABA-A Receptor Antagonists; Oxazepam; Substance Withdrawal Syndrome

1992
The effects of flumazenil-precipitated abstinence on the pharmacokinetics of chronic oxazepam in dogs.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 35, Issue:2

    Topics: Administration, Oral; Animals; Biological Availability; Dogs; Drug Interactions; Female; Flumazenil; Injections, Intravenous; Oxazepam; Substance-Related Disorders

1990
Benzodiazepines produce contrasting effects on the active membrane properties of an invertebrate neuron.
    Neuropharmacology, 1985, Volume: 24, Issue:2

    Topics: Action Potentials; Animals; Anti-Anxiety Agents; Astacoidea; Benzodiazepinones; Electric Conductivity; Flumazenil; Flurazepam; In Vitro Techniques; Membrane Potentials; Neurons, Afferent; Oxazepam

1985
Discriminative stimulus properties of oxazepam in the pigeon.
    Life sciences, 1987, Jan-05, Volume: 40, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Columbidae; Discrimination Learning; Flumazenil; Oxazepam; Pentobarbital; Pyridazines

1987
Precipitation of abstinence in nordiazepam- and diazepam-dependent dogs.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Analysis of Variance; Animals; Diazepam; Dogs; Flumazenil; Nordazepam; Oxazepam; Pyrazoles; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1988
Ventricular arrhythmia precipitated by flumazenil.
    British medical journal (Clinical research ed.), 1988, Apr-09, Volume: 296, Issue:6628

    Topics: Adult; Chloral Hydrate; Electrocardiography; Female; Flumazenil; Heart Ventricles; Humans; Oxazepam; Tachycardia

1988
Does the behavioural activation detected after a single dose of a benzodiazepine reflect a withdrawal response?
    Life sciences, 1988, Volume: 42, Issue:23

    Topics: Animals; Behavior, Animal; Benzodiazepines; Flumazenil; Lorazepam; Male; Mice; Motor Activity; Oxazepam

1988
Synaptic and non-synaptic actions of benzodiazepines on the crayfish sensory neuron.
    European journal of pharmacology, 1984, Jun-15, Volume: 102, Issue:1

    Topics: Action Potentials; Animals; Anti-Anxiety Agents; Astacoidea; Benzodiazepinones; Flumazenil; Flurazepam; In Vitro Techniques; Mechanoreceptors; Membrane Potentials; Neurons, Afferent; Oxazepam; Receptors, Neurotransmitter

1984
Evidence for excitatory and depressant non-receptor-mediated membrane effects of benzodiazepines in the crayfish.
    Neuroscience letters, 1984, Mar-09, Volume: 45, Issue:1

    Topics: Animals; Astacoidea; Benzodiazepines; Benzodiazepinones; Cell Membrane; Electrophysiology; Flumazenil; Flurazepam; Neurons, Afferent; Oxazepam; Physical Stimulation

1984
Precipitated withdrawal in squirrel monkeys after repeated daily oral administration of alprazolam, diazepam, flunitrazepam or oxazepam.
    Psychopharmacology, 1995, Volume: 118, Issue:3

    Topics: Administration, Oral; Alprazolam; Animals; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Female; Flumazenil; Flunitrazepam; Male; Muscle Relaxation; Oxazepam; Saimiri; Sleep; Substance Withdrawal Syndrome; Substance-Related Disorders; Tremor

1995
Oxazepam overdose associated with ethanol ingestion: treatment with a benzodiazepine antagonist.
    American journal of critical care : an official publication, American Association of Critical-Care Nurses, 1994, Volume: 3, Issue:6

    Topics: Alcohol Drinking; Benzodiazepines; Drug Interactions; Drug Overdose; Flumazenil; Humans; Male; Middle Aged; Oxazepam

1994
Pharmacokinetics of nordiazepam in physical dependence and precipitated abstinence in dogs.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:4

    Topics: Administration, Oral; Animals; Blood Proteins; Diazepam; Dogs; Female; Flumazenil; Hydrolysis; Injections, Intravenous; Nordazepam; Oxazepam; Protein Binding; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
Flumazenil, diazepam, nordiazepam and oxazepam interactions on plasma protein binding.
    Pharmacological research, 1995, Volume: 32, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Biotransformation; Blood Proteins; Diazepam; Dogs; Drug Interactions; Flumazenil; In Vitro Techniques; Nordazepam; Oxazepam; Protein Binding

1995
The effect of chronic benzodiazepines exposure on body weight in rats.
    Pharmacological research, 1998, Volume: 37, Issue:3

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Flunitrazepam; GABA Modulators; Male; Nordazepam; Oxazepam; Rats; Rats, Sprague-Dawley; Sex Factors; Time Factors; Weight Gain

1998
Plasma and CSF benzodiazepine receptor ligand concentrations in cirrhotic patients with hepatic encephalopathy: relationship to severity of encephalopathy and to pharmaceutical benzodiazepine intake.
    Metabolic brain disease, 1998, Volume: 13, Issue:3

    Topics: Animals; Benzodiazepines; Binding, Competitive; Cell Fractionation; Cerebellum; Chronic Disease; Clonazepam; Diazepam; Flumazenil; GABA Modulators; Hepatic Encephalopathy; Humans; Isoquinolines; Liver Cirrhosis; Oxazepam; Radioligand Assay; Rats; Receptors, GABA-A; Tritium

1998
Pharmacological analysis of the effects of benzodiazepines on punished schedule-induced polydipsia in rats.
    Behavioural pharmacology, 2007, Volume: 18, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Chlordiazepoxide; Diazepam; Dose-Response Relationship, Drug; Drinking; Electroshock; Fear; Flumazenil; Food Deprivation; GABA Modulators; Imidazoles; Male; Oxazepam; Punishment; Pyrimidines; Rats; Rats, Wistar; Receptors, GABA-A; Reinforcement Schedule

2007
The differential effects of alprazolam and oxazepam on methamphetamine self-administration in rats.
    Drug and alcohol dependence, 2016, Sep-01, Volume: 166

    Topics: Alprazolam; Amphetamine-Related Disorders; Animals; Dose-Response Relationship, Drug; Flumazenil; Isoquinolines; Male; Methamphetamine; Oxazepam; Premedication; Rats; Rats, Wistar; Receptors, GABA-A; Self Administration

2016