flumazenil and nordazepam

flumazenil has been researched along with nordazepam in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19905 (22.73)18.7374
1990's10 (45.45)18.2507
2000's6 (27.27)29.6817
2010's1 (4.55)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Adkison, KK; Humphreys, JE; Mahar Doan, KM; Polli, JW; Serabjit-Singh, CJ; Shampine, LJ; Webster, LO; Wring, SA1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Lombardo, F; Obach, RS; Waters, NJ1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Basile, AS; Harrison, PM; Hughes, RD; Jones, EA; Murata, Y; Pannell, L; Skolnick, P; Williams, R1
Dickey, KM; Martin, WR; Sloan, JW; Wala, E1
Campisi, M; Iseppi, D; Laganà, G; Stacca, R; Tassi, A1
Hole, K; Rosland, JH1
Appel, M; Bron, HN; Hooymans, PM; Janknegt, R1
Fassbender, CP; Hönack, D; Löscher, W1
Spealman, RD2
Martin, WR; McNicholas, LF; Sloan, JW; Wala, E1
Jing, X; Sloan, JW; Wala, EP2
Martin, WR; Sloan, JW; Wala, EP1
Sloan, JW; Wala, EP1
Camaris, C; Little, D1
Alzieu, M; Becquemont, L; Delhotal Landes, B; Guglielminotti, J; Guidet, B; Maury, E; Offenstadt, G1
Arditti, J; Bourdon, JH; de Haro, L; Hayek-Lanthois, M; Iliadis, A; Valli, M1
Biggio, G; Latrofa, A; Papi, G; Pisu, MG; Porcu, P; Serra, M; Trapani, G1

Other Studies

22 other study(ies) available for flumazenil and nordazepam

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Passive permeability and P-glycoprotein-mediated efflux differentiate central nervous system (CNS) and non-CNS marketed drugs.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Cell Line; Cell Membrane Permeability; Central Nervous System Agents; Dogs; Drug Delivery Systems; Permeability; Pharmaceutical Preparations

2002
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Elevated brain concentrations of 1,4-benzodiazepines in fulminant hepatic failure.
    The New England journal of medicine, 1991, Aug-15, Volume: 325, Issue:7

    Topics: Adult; Aged; Benzodiazepines; Brain Chemistry; Chromatography; Diazepam; Flumazenil; Frontal Lobe; gamma-Aminobutyric Acid; Hepatic Encephalopathy; Humans; Mass Spectrometry; Middle Aged; Nordazepam; Receptors, GABA-A; Synaptic Transmission

1991
Chronic administration of and dependence on halazepam, diazepam, and nordiazepam in the dog.
    Drug and alcohol dependence, 1991, Volume: 28, Issue:3

    Topics: Administration, Oral; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Dogs; Dose-Response Relationship, Drug; Flumazenil; Neurologic Examination; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders

1991
[Antagonism with flumazenil of sedation by benzodiazepine during loco-regional anesthesia].
    Minerva anestesiologica, 1990, Volume: 56, Issue:9

    Topics: Adult; Anesthesia, Local; Anti-Anxiety Agents; Benzodiazepines; Conscious Sedation; Female; Flumazenil; Humans; Male; Middle Aged; Nerve Block; Nordazepam

1990
Benzodiazepine-induced antagonism of opioid antinociception may be abolished by spinalization or blockade of the benzodiazepine receptor.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:3

    Topics: Analgesics; Animals; Anti-Anxiety Agents; Diazepam; Flumazenil; Male; Mice; Midazolam; Morphine; Narcotics; Nordazepam; Psychomotor Performance; Reaction Time; Receptors, GABA-A; Receptors, Opioid; Skin Temperature; Spinal Cord

1990
Efficacy of flumazenil in COPD patient with therapeutic diazepam levels.
    Lancet (London, England), 1989, Feb-18, Volume: 1, Issue:8634

    Topics: Aged; Diazepam; Drug Evaluation; Flumazenil; Humans; Lung Diseases, Obstructive; Male; Nordazepam

1989
Physical dependence on diazepam in the dog: precipitation of different abstinence syndromes by the benzodiazepine receptor antagonists Ro 15-1788 and ZK 93426.
    British journal of pharmacology, 1989, Volume: 97, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Carbolines; Diazepam; Dogs; Female; Flumazenil; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1989
Disruption of schedule-controlled behavior by Ro 15-1788 one day after acute treatment with benzodiazepines.
    Psychopharmacology, 1986, Volume: 88, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Chlordiazepoxide; Conditioning, Operant; Convulsants; Diazepam; Flumazenil; Male; Nordazepam; Reinforcement Schedule; Saimiri

1986
Discriminative-stimulus effects of midazolam in squirrel monkeys: comparison with other drugs and antagonism by Ro 15-1788.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Azabicyclo Compounds; Barbital; Benzodiazepines; Benzodiazepinones; Buspirone; Caffeine; Chlordiazepoxide; Cinanserin; Clozapine; Conditioning, Operant; Cyproheptadine; Diazepam; Diphenhydramine; Discrimination Learning; Electroshock; Flumazenil; Male; Midazolam; Muscimol; Nordazepam; Pentobarbital; Piperazines; Pyridazines; Pyrimidines; Saimiri; Tripelennamine

1985
Precipitation of abstinence in nordiazepam- and diazepam-dependent dogs.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Analysis of Variance; Animals; Diazepam; Dogs; Flumazenil; Nordazepam; Oxazepam; Pyrazoles; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1988
Flunitrazepam and nordiazepam slowly released from silastic capsules induce physical dependence in rat.
    Drug and alcohol dependence, 1995, Volume: 39, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Antidotes; Biological Availability; Delayed-Action Preparations; Diazepam; Drug Implants; Female; Flumazenil; Flunitrazepam; Nordazepam; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Substance-Related Disorders

1995
Pharmacokinetics of nordiazepam in physical dependence and precipitated abstinence in dogs.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:4

    Topics: Administration, Oral; Animals; Blood Proteins; Diazepam; Dogs; Female; Flumazenil; Hydrolysis; Injections, Intravenous; Nordazepam; Oxazepam; Protein Binding; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
Flumazenil, diazepam, nordiazepam and oxazepam interactions on plasma protein binding.
    Pharmacological research, 1995, Volume: 32, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Biotransformation; Blood Proteins; Diazepam; Dogs; Drug Interactions; Flumazenil; In Vitro Techniques; Nordazepam; Oxazepam; Protein Binding

1995
A fatality due to moclobemide.
    Journal of forensic sciences, 1997, Volume: 42, Issue:5

    Topics: Antidepressive Agents; Benzamides; Diazepam; Fatal Outcome; Female; Flumazenil; Humans; Liver; Middle Aged; Moclobemide; Nordazepam; Trifluoperazine

1997
The effect of chronic benzodiazepines exposure on body weight in rats.
    Pharmacological research, 1998, Volume: 37, Issue:3

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Flunitrazepam; GABA Modulators; Male; Nordazepam; Oxazepam; Rats; Rats, Sprague-Dawley; Sex Factors; Time Factors; Weight Gain

1998
Prolonged sedation requiring mechanical ventilation and continuous flumazenil infusion after routine doses of clorazepam for alcohol withdrawal syndrome.
    Intensive care medicine, 1999, Volume: 25, Issue:12

    Topics: Aged; Alcohol Withdrawal Seizures; Anticonvulsants; Antidotes; Bronchitis; Clorazepate Dipotassium; Coma; Fatal Outcome; Flumazenil; Humans; Infusions, Intravenous; Liver Diseases; Male; Middle Aged; Nordazepam; Pneumonia; Respiration, Artificial

1999
Diazepam poisoning with one-month monitoring of diazepam and nordiazepam blood levels.
    Veterinary and human toxicology, 2001, Volume: 43, Issue:3

    Topics: Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Flumazenil; Humans; Male; Middle Aged; Nordazepam; Poisoning; Suicide, Attempted; Treatment Outcome

2001
Binding of [3H]CB 34, a selective ligand for peripheral benzodiazepine receptors, to rat brain membranes.
    European journal of pharmacology, 2001, Dec-07, Volume: 432, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Female; Flumazenil; Imidazoles; Indoleacetic Acids; Isoquinolines; Ligands; Membrane Proteins; Membranes; Nordazepam; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tritium

2001