flumazenil has been researched along with methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate in 51 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 24 (47.06) | 18.7374 |
1990's | 17 (33.33) | 18.2507 |
2000's | 10 (19.61) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Dekermendjian, K; Kahnberg, P; Liljefors, T; Nielsen, M; Sterner, O; Witt, MR | 1 |
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Dudley, MW; Kane, JM; Kehne, JH; Miller, JA; Sorensen, SM | 1 |
Bernasconi, R; Leonhardt, T; Martin, P; Portet, C; Schmutz, M; Steulet, AF | 1 |
De Boer, SF; Katz, JL; Valentino, RJ | 1 |
Buck, KJ; Harris, RA; Heim, H | 1 |
De Boer, SF; Slangen, JL; Van der Gugten, J | 1 |
Buck, KJ; Harris, RA | 1 |
Blier, P; De Montigny, C; Lista, A | 1 |
Dragunow, M | 1 |
Costa, E; Mienville, JM; Vicini, S | 1 |
Gallager, DW; Wilson, MA | 2 |
Cooper, SJ; Estall, LB | 1 |
Cox, DH; Guidotti, A; Santi, MR | 1 |
Arbilla, S; Langer, SZ; Lista, A | 1 |
Moody, EJ; Skolnick, P | 1 |
Leidenheimer, NJ; Schechter, MD | 1 |
Klockgether, T; Schwarz, M; Sontag, KH; Turski, L | 1 |
Chan, CY; Farb, DH | 1 |
Barber, DJ; Cooper, SJ; Gilbert, DB; Moores, WR | 1 |
Havoundjian, H; Paul, SM; Reed, GF; Skolnick, P | 1 |
Jensen, LH; Petersen, EN | 1 |
Brouillet, E; Chavoix, C; Crouzel, M; Dodd, RH; Fukuda, H; Guibert, B; Hantraye, P; Mazière, M; Naquet, R; Prenant, C | 1 |
Alho, H; Costa, E; Mienville, JM; Santi, MR; Vaccarino, FM; Vicini, S | 1 |
Randall, JI; Rodgers, RJ | 1 |
Ableitner, A; Herz, A | 1 |
Little, HJ; Nutt, DJ; Sellars, N; Taylor, SC | 1 |
Braestrup, C; Honoré, T; Jensen, LH; Kehr, W; Petersen, EN; Schmiechen, R; Schneider, H; Seidelmann, D; Stephens, DN | 1 |
Borea, PA; Karobath, M; Supavilai, P | 1 |
Biggio, G; Concas, A; Salis, M; Serra, M | 1 |
Biggio, G; Concas, A; Fanni, B; Mereu, G; Serra, M | 1 |
Biggio, G; Mereu, G | 1 |
Braestrup, C; Honoré, T; Jensen, LH; Nielsen, M; Petersen, EN | 1 |
Carter, DB; Im, HK; Im, WB; McKinley, DD | 1 |
Kirby, LG; Lucki, I; Rowan, GA; Smith, RL | 1 |
Carlen, PL; Facciponte, G; Jahromi, SS; Pelletier, MR; Polc, P; Zhang, L | 1 |
Chimirri, A; De Sarro, A; De Sarro, G; Guisti, P; Lipartiti, M; Zappala, M | 1 |
Bowery, BJ; Dawson, GR; Easter, A; Seabrook, GR | 1 |
Chimirri, A; De Sarro, A; De Sarro, G; Giusti, P; McKernan, R; Quirk, K | 1 |
Castro, JL; Ramirez, A; Ricci, D; Taira, CA | 1 |
Costentin, J; Garcia de Mateos-Verchere, J; Leprince, J; Tonon, MC; Vaudry, H | 1 |
Breese, GR; Duncan, GE; Knapp, DJ; Moy, SS | 1 |
Beaujean, D; Do-Rego, JL; Leprince, J; Luu-The, V; Mensah-Nyagan, AG; Pelletier, G; Tonon, MC; Vaudry, H | 1 |
Cook, JM; DeLorey, TM; He, X; Lameh, J; Lin, RC; Loew, GH; McBrady, B | 1 |
Bokonjić, DR; Cook, JM; Obradović, DI; Savić, MM; Ugresić, ND; Yin, W | 1 |
Bokonjić, DR; Cook, JM; Obradović, DI; Sarma, PV; Savić, MM; Ugresić, ND | 1 |
France, CP; McMahon, LR | 1 |
Bostwick, R; Chen, T; Huston, J; Knappenberger, K; Liu, J; Norris, T; Wood, M | 1 |
Barbalho, CA; Canto-de-Souza, A; Nunes-de-Souza, RL | 1 |
1 review(s) available for flumazenil and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate
Article | Year |
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Behavioural pharmacology of food, water and salt intake in relation to drug actions at benzodiazepine receptors.
Topics: Animals; Anti-Anxiety Agents; Appetite; Appetite Depressants; Benzodiazepines; Benzodiazepinones; Carbolines; Chlordiazepoxide; Chlorides; Choice Behavior; Diazepam; Drinking Behavior; Feeding Behavior; Flumazenil; Food Deprivation; Food Preferences; gamma-Aminobutyric Acid; Ion Channels; Midazolam; Picrotoxin; Punishment; Pyrazoles; Receptors, GABA-A; Satiation; Sodium Chloride; Species Specificity | 1985 |
50 other study(ies) available for flumazenil and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate
Article | Year |
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Structure-activity relationships and molecular modeling analysis of flavonoids binding to the benzodiazepine site of the rat brain GABA(A) receptor complex.
Topics: Animals; Binding Sites; Brain; Flavonoids; In Vitro Techniques; Male; Models, Molecular; Molecular Conformation; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Reproducibility of Results; Structure-Activity Relationship | 1999 |
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship | 2000 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
MDL 26,479: a potential cognition enhancer with benzodiazepine inverse agonist-like properties.
Topics: Animals; Behavior, Animal; Benzodiazepines; Binding Sites; Carbolines; Cognition; Convulsants; Diazepam; Flumazenil; Hemicholinium 3; Hippocampus; In Vitro Techniques; Male; Mice; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Triazoles | 1992 |
Effects of benzodiazepine receptor ligands with different intrinsic activities on seizures induced by inhibition of GAD.
Topics: Animals; Anti-Anxiety Agents; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hippocampus; Isoniazid; Male; Mice; Mice, Inbred Strains; Pyrazoles; Reaction Time; Receptors, GABA-A; Seizures | 1992 |
Common mechanisms underlying the proconflict effects of corticotropin-releasing factor, a benzodiazepine inverse agonist and electric foot-shock.
Topics: Animals; Behavior, Animal; Carbolines; Chlordiazepoxide; Convulsants; Corticotropin-Releasing Hormone; Electroshock; Flumazenil; Injections, Intraventricular; Male; Punishment; Rats; Rats, Inbred Strains | 1992 |
Reversal of alcohol dependence and tolerance by a single administration of flumazenil.
Topics: Alcoholism; Animals; Ataxia; Behavior, Animal; Brain; Carbolines; Chlorides; Drug Administration Schedule; Drug Tolerance; Ethanol; Flumazenil; Hypothermia; Male; Mice; Mice, Inbred ICR; Neurons; Receptors, GABA-A | 1991 |
Effects of chlordiazepoxide, flumazenil and DMCM on plasma catecholamine and corticosterone concentrations in rats.
Topics: Animals; Carbolines; Catecholamines; Chlordiazepoxide; Corticosterone; Epinephrine; Flumazenil; Injections, Intraperitoneal; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1991 |
Benzodiazepine agonist and inverse agonist actions on GABAA receptor-operated chloride channels. I. Acute effects of ethanol.
Topics: Animals; Benzodiazepines; Brain; Carbolines; Chloride Channels; Chlorides; Convulsants; Ethanol; Flumazenil; Flunitrazepam; Injections, Intraperitoneal; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Tritium | 1990 |
The benzodiazepine receptor inverse agonist DMCM decreases serotonergic transmission in rat hippocampus: an in vivo electrophysiological study.
Topics: Animals; Carbolines; Diazepam; Electrophysiology; Flumazenil; Hippocampus; Neural Pathways; Pargyline; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synaptic Transmission | 1990 |
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines | 1990 |
Chloride channel modulation through the benzodiazepine recognition site.
Topics: Animals; Bicuculline; Carbolines; Cells, Cultured; Chlorides; Convulsants; Flumazenil; Flunitrazepam; Ion Channels; Neurons; Receptors, GABA-A | 1988 |
Responses of substantia nigra pars reticulata neurons to benzodiazepine ligands after acute and prolonged diazepam exposure. I. Modulation of gamma-aminobutyric acid sensitivity.
Topics: Animals; Carbolines; Diazepam; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Ligands; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra | 1989 |
Responses of substantia nigra pars reticulata neurons to benzodiazepine ligands after acute and prolonged diazepam exposure. II. Modulation of firing rate.
Topics: Animals; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra | 1989 |
Heterogeneity of gamma-aminobutyric acid/benzodiazepine/beta-carboline receptor complex in rat spinal cord.
Topics: Animals; Bicuculline; Binding, Competitive; Carbolines; Cerebellum; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Receptors, GABA-A; Spinal Cord; Synaptic Membranes | 1988 |
Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.
Topics: Animals; Benzodiazepines; Carbolines; Cerebral Cortex; Diazepam; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Monoamine Oxidase Inhibitors; Pargyline; Pyrazoles; Pyridazines; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin | 1988 |
The imidazobenzodiazepine Ro 15-4513 antagonizes methoxyflurane anesthesia.
Topics: Anesthesia, General; Animals; Azides; Benzodiazepines; Carbolines; Flumazenil; Male; Methoxyflurane; Mice; Receptors, GABA-A; Sleep | 1988 |
Discriminative stimulus properties of CGS 9896: interactions within the GABA/benzodiazepine receptor complex.
Topics: Animals; Carbolines; Chlordiazepoxide; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Male; Pentobarbital; Pentylenetetrazole; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1988 |
ZK 91296, an anticonvulsant beta-carboline which lacks muscle relaxant properties.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Electromyography; Electroshock; Flumazenil; Indoles; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle Relaxants, Central; Muscle Tonus; Phenobarbital; Rats; Rats, Inbred Strains | 1985 |
Modulation of neurotransmitter action: control of the gamma-aminobutyric acid response through the benzodiazepine receptor.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Chick Embryo; Electric Conductivity; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Neurotransmitter Agents; Picrotoxin; Pyridazines; Receptors, GABA-A | 1985 |
Benzodiazepine receptor ligands and the consumption of a highly palatable diet in non-deprived male rats.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Drug Interactions; Feeding Behavior; Flumazenil; Ligands; Male; Midazolam; Pyrazoles; Rats; Receptors, GABA-A | 1985 |
Protection against the lethal effects of pentobarbital in mice by a benzodiazepine receptor inverse agonist, 6,7-dimethoxy-4-ethyl-3-carbomethoxy-beta-carboline.
Topics: Animals; Carbolines; Flumazenil; Male; Mice; Mice, Inbred Strains; Pentobarbital; Receptors, GABA-A | 1987 |
Chronic treatment with lorazepam and FG 7142 may change the effects of benzodiazepine receptor agonists, antagonists and inverse agonists by different mechanisms.
Topics: Animals; Carbolines; Drug Interactions; Drug Tolerance; Female; Flumazenil; Lorazepam; Mice; Pentylenetetrazole; Receptors, GABA-A | 1987 |
Benzodiazepine receptors studied in living primates by positron emission tomography: inverse agonist interactions.
Topics: Animals; Binding, Competitive; Carbolines; Cerebral Cortex; Convulsants; Dose-Response Relationship, Drug; Electroencephalography; Flumazenil; Male; Papio; Receptors, GABA-A; Tomography, Emission-Computed | 1987 |
Modulation of gamma-aminobutyric acid-mediated inhibitory synaptic currents in dissociated cortical cell cultures.
Topics: Animals; Bicuculline; Carbolines; Cells, Cultured; Cerebral Cortex; Electric Conductivity; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Potentials; Neural Inhibition; Rats; Synapses | 1986 |
Benzodiazepine ligands, nociception and 'defeat' analgesia in male mice.
Topics: Analgesia; Animals; Appetite Depressants; Benzodiazepines; Carbolines; Chlordiazepoxide; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Nociceptors; Pyrazoles | 1987 |
Changes in local cerebral glucose utilization induced by the beta-carbolines FG 7142 and DMCM reveal brain structures involved in the control of anxiety and seizure activity.
Topics: Animals; Anxiety; Autoradiography; Brain; Carbolines; Convulsants; Deoxyglucose; Flumazenil; Glucose; Male; Rats; Rats, Inbred Strains; Seizures | 1987 |
A benzodiazepine agonist and contragonist have hypothermic effects in rodents.
Topics: Animals; Benzodiazepinones; Body Temperature; Carbolines; Convulsants; Flumazenil; Flurazepam; Hypothermia; Indoles; Male; Mice; Mice, Inbred Strains; Motor Activity; Rats; Rats, Inbred Strains | 1985 |
Evaluation of the beta-carboline ZK 93 426 as a benzodiazepine receptor antagonist.
Topics: Animals; Anticonvulsants; Ataxia; Benzodiazepinones; Binding, Competitive; Carbolines; Diazepam; Discrimination, Psychological; Drinking; Exploratory Behavior; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Mice; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Sleep | 1984 |
Differential modulation of etazolate or pentobarbital enhanced [3H] muscimol binding by benzodiazepine agonists and inverse agonists.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Etazolate; Flumazenil; Flunitrazepam; Kinetics; Muscimol; Nicotinic Acids; Oxazoles; Pentobarbital; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Increase of cyclic GMP in cerebellum by methyl-6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate (DMCM).
Topics: Animals; Benzodiazepinones; Carbolines; Cerebellar Cortex; Cyclic GMP; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Indoles; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Stimulation, Chemical | 1983 |
beta-Carbolines activate neurons in the substantia nigra pars reticulata: an effect reversed by diazepam and Ro15-1788.
Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Drug Interactions; Flumazenil; Indoles; Injections, Intravenous; Male; Rats; Rats, Inbred Strains; Substantia Nigra; Synaptic Transmission | 1983 |
Effect of agonists, inverse agonists, and antagonists of benzodiazepine receptors on the firing rate of substantia nigra pars reticulata neurons.
Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electrophysiology; Flumazenil; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra | 1983 |
Ligands for benzodiazepine receptors with positive and negative efficacy.
Topics: Animals; Benzodiazepinones; Carbolines; Flumazenil; Humans; Ligands; Radioligand Assay; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Interaction of beta-carboline inverse agonists for the benzodiazepine site with another site on GABAA receptors.
Topics: Barbiturates; Carbolines; Cell Line; Chloride Channels; Convulsants; Flumazenil; GABA Antagonists; GABA-A Receptor Agonists; Humans; Kidney; Patch-Clamp Techniques; Plasmids; Receptors, GABA-A; Steroids | 1995 |
Discriminative stimulus properties of the benzodiazepine receptor inverse agonist methyl-6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate (DMCM).
Topics: Animals; Carbolines; Convulsants; Discrimination, Psychological; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Generalization, Stimulus; Male; Rats; Rats, Sprague-Dawley; Saccharin; Taste | 1994 |
Benzodiazepine antagonists reduce epileptiform discharges in rat hippocampal slices.
Topics: Animals; Carbolines; Convulsants; Disease Models, Animal; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Leucine; Epilepsy; Flumazenil; Hippocampus; Kindling, Neurologic; Male; Rats; Rats, Wistar; Receptors, GABA-A; Structure-Activity Relationship; Synaptic Transmission | 1996 |
Azirino[1, 2-d][1, 4]benzodiazepine derivatives and related 1,4-benzodiazepines as anticonvulsant agents in DBA/2 mice.
Topics: Acoustic Stimulation; Animals; Anticonvulsants; Benzodiazepines; Binding, Competitive; Carbolines; Cell Membrane; Cerebellum; Cerebral Cortex; Chemical Phenomena; Chemistry, Physical; Convulsants; Flumazenil; GABA Modulators; Male; Mice; Mice, Inbred DBA; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures | 1996 |
Modulation of long-term potentiation in CA1 region of mouse hippocampal brain slices by GABAA receptor benzodiazepine site ligands.
Topics: Animals; Carbolines; Convulsants; Dizocilpine Maleate; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Mice; Quinolones; Receptors, GABA-A | 1997 |
Anticonvulsant activity of azirino[1,2-d][1,4]benzodiazepines and related 1,4-benzodiazepines in mice.
Topics: Animals; Anticonvulsants; Benzodiazepines; Carbolines; Cell Line; Convulsants; Flumazenil; GABA Modulators; Male; Membranes; Mice; Mice, Inbred DBA; Movement; Pentylenetetrazole; Radioligand Assay; Receptors, GABA-A; Seizures | 1997 |
Central benzodiazepine involvement in clonidine cardiovascular actions.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Atropine Derivatives; Blood Pressure; Carbolines; Cardiovascular Agents; Clonidine; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Heart Rate; Infusions, Intravenous; Injections, Intraventricular; Male; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, GABA-A; Stereotaxic Techniques; Time Factors; Yohimbine | 1999 |
Reduction of pentylenetetrazol-induced convulsions by the octadecaneuropeptide ODN.
Topics: Acoustic Stimulation; Amino Acid Sequence; Animals; Carbolines; Convulsants; Diazepam Binding Inhibitor; Electric Stimulation; Flumazenil; Injections, Intraventricular; Male; Mice; Mice, Inbred DBA; Molecular Sequence Data; Neuropeptides; Pentylenetetrazole; Peptide Fragments; Receptors, GABA-A; Seizures | 1999 |
Enhanced ultrasonic vocalization and Fos protein expression following ethanol withdrawal: effects of flumazenil.
Topics: Animals; Carbolines; Ethanol; Flumazenil; Male; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Substance Withdrawal Syndrome; Vocalization, Animal | 2000 |
The octadecaneuropeptide ODN stimulates neurosteroid biosynthesis through activation of central-type benzodiazepine receptors.
Topics: 17-alpha-Hydroxypregnenolone; 17-alpha-Hydroxyprogesterone; 3-Hydroxysteroid Dehydrogenases; Animals; Carbolines; Chromatography, High Pressure Liquid; Dehydroepiandrosterone; Diazepam Binding Inhibitor; Dihydrotestosterone; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hydroxysteroids; Hypothalamus; Immunohistochemistry; In Vitro Techniques; Ligands; Male; Neuroglia; Neurons; Neuropeptides; Peptide Fragments; Pregnenolone; Progesterone; Rana ridibunda; Receptors, GABA-A | 2001 |
Influence of benzodiazepine binding site ligands on fear-conditioned contextual memory.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; Conditioning, Psychological; Convulsants; Fear; Flumazenil; GABA Antagonists; GABA Modulators; Imidazoles; Ligands; Male; Memory; Mice; Mice, Inbred C57BL; Motor Activity; N-Methylscopolamine; Piperazines; Quinolines; Receptors, GABA-A; Scopolamine; Silanes; Tritium | 2001 |
Bidirectional effects of benzodiazepine binding site ligands in the elevated plus-maze: differential antagonism by flumazenil and beta-CCt.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding Sites; Carbolines; Drug Interactions; Flumazenil; GABA Modulators; Ligands; Male; Maze Learning; Mice; Midazolam; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Zolpidem | 2004 |
Bidirectional effects of benzodiazepine binding site ligands on active avoidance acquisition and retention: differential antagonism by flumazenil and beta-CCt.
Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Benzodiazepines; Binding Sites; Carbolines; Convulsants; Dose-Response Relationship, Drug; Flumazenil; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; Habituation, Psychophysiologic; Injections, Intraperitoneal; Ligands; Male; Midazolam; Motor Activity; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Retention, Psychology; Zolpidem | 2005 |
Negative GABA(A) modulators attenuate the discriminative stimulus effects of benzodiazepines and the neuroactive steroid pregnanolone in rhesus monkeys.
Topics: Animals; Benzodiazepines; Carbolines; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Female; Flumazenil; Macaca mulatta; Male; Midazolam; Pregnanolone; Receptors, GABA-A; Serotonin Antagonists; Serotonin Receptor Agonists | 2005 |
A high-throughput functional assay for characterization of gamma-aminobutyric acid(A) channel modulators using cryopreserved transiently transfected cells.
Topics: Carbolines; Cell Culture Techniques; Cell Line; Cell Membrane; Cryopreservation; Diazepam; DNA; Dose-Response Relationship, Drug; Drug Discovery; Flumazenil; Flunitrazepam; Fluorescent Dyes; Fluorobenzenes; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Receptors, GABA-A; Reproducibility of Results; Spectrometry, Fluorescence; Transfection; Triazoles; Tritium | 2008 |
Similar anxiolytic-like effects following intra-amygdala infusions of benzodiazepine receptor agonist and antagonist: evidence for the release of an endogenous benzodiazepine inverse agonist in mice exposed to elevated plus-maze test.
Topics: Amygdala; Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Carbolines; Catheterization; Exploratory Behavior; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Maze Learning; Mice; Microinjections; Midazolam; Motor Activity | 2009 |