flumazenil and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate

flumazenil has been researched along with methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate in 51 studies

Research

Studies (51)

TimeframeStudies, this research(%)All Research%
pre-199024 (47.06)18.7374
1990's17 (33.33)18.2507
2000's10 (19.61)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dekermendjian, K; Kahnberg, P; Liljefors, T; Nielsen, M; Sterner, O; Witt, MR1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Dudley, MW; Kane, JM; Kehne, JH; Miller, JA; Sorensen, SM1
Bernasconi, R; Leonhardt, T; Martin, P; Portet, C; Schmutz, M; Steulet, AF1
De Boer, SF; Katz, JL; Valentino, RJ1
Buck, KJ; Harris, RA; Heim, H1
De Boer, SF; Slangen, JL; Van der Gugten, J1
Buck, KJ; Harris, RA1
Blier, P; De Montigny, C; Lista, A1
Dragunow, M1
Costa, E; Mienville, JM; Vicini, S1
Gallager, DW; Wilson, MA2
Cooper, SJ; Estall, LB1
Cox, DH; Guidotti, A; Santi, MR1
Arbilla, S; Langer, SZ; Lista, A1
Moody, EJ; Skolnick, P1
Leidenheimer, NJ; Schechter, MD1
Klockgether, T; Schwarz, M; Sontag, KH; Turski, L1
Chan, CY; Farb, DH1
Barber, DJ; Cooper, SJ; Gilbert, DB; Moores, WR1
Havoundjian, H; Paul, SM; Reed, GF; Skolnick, P1
Jensen, LH; Petersen, EN1
Brouillet, E; Chavoix, C; Crouzel, M; Dodd, RH; Fukuda, H; Guibert, B; Hantraye, P; Mazière, M; Naquet, R; Prenant, C1
Alho, H; Costa, E; Mienville, JM; Santi, MR; Vaccarino, FM; Vicini, S1
Randall, JI; Rodgers, RJ1
Ableitner, A; Herz, A1
Little, HJ; Nutt, DJ; Sellars, N; Taylor, SC1
Braestrup, C; Honoré, T; Jensen, LH; Kehr, W; Petersen, EN; Schmiechen, R; Schneider, H; Seidelmann, D; Stephens, DN1
Borea, PA; Karobath, M; Supavilai, P1
Biggio, G; Concas, A; Salis, M; Serra, M1
Biggio, G; Concas, A; Fanni, B; Mereu, G; Serra, M1
Biggio, G; Mereu, G1
Braestrup, C; Honoré, T; Jensen, LH; Nielsen, M; Petersen, EN1
Carter, DB; Im, HK; Im, WB; McKinley, DD1
Kirby, LG; Lucki, I; Rowan, GA; Smith, RL1
Carlen, PL; Facciponte, G; Jahromi, SS; Pelletier, MR; Polc, P; Zhang, L1
Chimirri, A; De Sarro, A; De Sarro, G; Guisti, P; Lipartiti, M; Zappala, M1
Bowery, BJ; Dawson, GR; Easter, A; Seabrook, GR1
Chimirri, A; De Sarro, A; De Sarro, G; Giusti, P; McKernan, R; Quirk, K1
Castro, JL; Ramirez, A; Ricci, D; Taira, CA1
Costentin, J; Garcia de Mateos-Verchere, J; Leprince, J; Tonon, MC; Vaudry, H1
Breese, GR; Duncan, GE; Knapp, DJ; Moy, SS1
Beaujean, D; Do-Rego, JL; Leprince, J; Luu-The, V; Mensah-Nyagan, AG; Pelletier, G; Tonon, MC; Vaudry, H1
Cook, JM; DeLorey, TM; He, X; Lameh, J; Lin, RC; Loew, GH; McBrady, B1
Bokonjić, DR; Cook, JM; Obradović, DI; Savić, MM; Ugresić, ND; Yin, W1
Bokonjić, DR; Cook, JM; Obradović, DI; Sarma, PV; Savić, MM; Ugresić, ND1
France, CP; McMahon, LR1
Bostwick, R; Chen, T; Huston, J; Knappenberger, K; Liu, J; Norris, T; Wood, M1
Barbalho, CA; Canto-de-Souza, A; Nunes-de-Souza, RL1

Reviews

1 review(s) available for flumazenil and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate

ArticleYear
Behavioural pharmacology of food, water and salt intake in relation to drug actions at benzodiazepine receptors.
    Neuroscience and biobehavioral reviews, 1985,Spring, Volume: 9, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Appetite; Appetite Depressants; Benzodiazepines; Benzodiazepinones; Carbolines; Chlordiazepoxide; Chlorides; Choice Behavior; Diazepam; Drinking Behavior; Feeding Behavior; Flumazenil; Food Deprivation; Food Preferences; gamma-Aminobutyric Acid; Ion Channels; Midazolam; Picrotoxin; Punishment; Pyrazoles; Receptors, GABA-A; Satiation; Sodium Chloride; Species Specificity

1985

Other Studies

50 other study(ies) available for flumazenil and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate

ArticleYear
Structure-activity relationships and molecular modeling analysis of flavonoids binding to the benzodiazepine site of the rat brain GABA(A) receptor complex.
    Journal of medicinal chemistry, 1999, Oct-21, Volume: 42, Issue:21

    Topics: Animals; Binding Sites; Brain; Flavonoids; In Vitro Techniques; Male; Models, Molecular; Molecular Conformation; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Reproducibility of Results; Structure-Activity Relationship

1999
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
MDL 26,479: a potential cognition enhancer with benzodiazepine inverse agonist-like properties.
    British journal of pharmacology, 1992, Volume: 107, Issue:1

    Topics: Animals; Behavior, Animal; Benzodiazepines; Binding Sites; Carbolines; Cognition; Convulsants; Diazepam; Flumazenil; Hemicholinium 3; Hippocampus; In Vitro Techniques; Male; Mice; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Triazoles

1992
Effects of benzodiazepine receptor ligands with different intrinsic activities on seizures induced by inhibition of GAD.
    Epilepsy research. Supplement, 1992, Volume: 8

    Topics: Animals; Anti-Anxiety Agents; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hippocampus; Isoniazid; Male; Mice; Mice, Inbred Strains; Pyrazoles; Reaction Time; Receptors, GABA-A; Seizures

1992
Common mechanisms underlying the proconflict effects of corticotropin-releasing factor, a benzodiazepine inverse agonist and electric foot-shock.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:1

    Topics: Animals; Behavior, Animal; Carbolines; Chlordiazepoxide; Convulsants; Corticotropin-Releasing Hormone; Electroshock; Flumazenil; Injections, Intraventricular; Male; Punishment; Rats; Rats, Inbred Strains

1992
Reversal of alcohol dependence and tolerance by a single administration of flumazenil.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:3

    Topics: Alcoholism; Animals; Ataxia; Behavior, Animal; Brain; Carbolines; Chlorides; Drug Administration Schedule; Drug Tolerance; Ethanol; Flumazenil; Hypothermia; Male; Mice; Mice, Inbred ICR; Neurons; Receptors, GABA-A

1991
Effects of chlordiazepoxide, flumazenil and DMCM on plasma catecholamine and corticosterone concentrations in rats.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 38, Issue:1

    Topics: Animals; Carbolines; Catecholamines; Chlordiazepoxide; Corticosterone; Epinephrine; Flumazenil; Injections, Intraperitoneal; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A

1991
Benzodiazepine agonist and inverse agonist actions on GABAA receptor-operated chloride channels. I. Acute effects of ethanol.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:2

    Topics: Animals; Benzodiazepines; Brain; Carbolines; Chloride Channels; Chlorides; Convulsants; Ethanol; Flumazenil; Flunitrazepam; Injections, Intraperitoneal; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Tritium

1990
The benzodiazepine receptor inverse agonist DMCM decreases serotonergic transmission in rat hippocampus: an in vivo electrophysiological study.
    Synapse (New York, N.Y.), 1990, Volume: 6, Issue:2

    Topics: Animals; Carbolines; Diazepam; Electrophysiology; Flumazenil; Hippocampus; Neural Pathways; Pargyline; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synaptic Transmission

1990
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines

1990
Chloride channel modulation through the benzodiazepine recognition site.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Bicuculline; Carbolines; Cells, Cultured; Chlorides; Convulsants; Flumazenil; Flunitrazepam; Ion Channels; Neurons; Receptors, GABA-A

1988
Responses of substantia nigra pars reticulata neurons to benzodiazepine ligands after acute and prolonged diazepam exposure. I. Modulation of gamma-aminobutyric acid sensitivity.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:2

    Topics: Animals; Carbolines; Diazepam; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Ligands; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1989
Responses of substantia nigra pars reticulata neurons to benzodiazepine ligands after acute and prolonged diazepam exposure. II. Modulation of firing rate.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:2

    Topics: Animals; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1989
Heterogeneity of gamma-aminobutyric acid/benzodiazepine/beta-carboline receptor complex in rat spinal cord.
    Journal of neurochemistry, 1988, Volume: 50, Issue:4

    Topics: Animals; Bicuculline; Binding, Competitive; Carbolines; Cerebellum; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Receptors, GABA-A; Spinal Cord; Synaptic Membranes

1988
Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.
    Journal of neurochemistry, 1988, Volume: 51, Issue:5

    Topics: Animals; Benzodiazepines; Carbolines; Cerebral Cortex; Diazepam; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Monoamine Oxidase Inhibitors; Pargyline; Pyrazoles; Pyridazines; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin

1988
The imidazobenzodiazepine Ro 15-4513 antagonizes methoxyflurane anesthesia.
    Life sciences, 1988, Volume: 43, Issue:16

    Topics: Anesthesia, General; Animals; Azides; Benzodiazepines; Carbolines; Flumazenil; Male; Methoxyflurane; Mice; Receptors, GABA-A; Sleep

1988
Discriminative stimulus properties of CGS 9896: interactions within the GABA/benzodiazepine receptor complex.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:2

    Topics: Animals; Carbolines; Chlordiazepoxide; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Male; Pentobarbital; Pentylenetetrazole; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
ZK 91296, an anticonvulsant beta-carboline which lacks muscle relaxant properties.
    European journal of pharmacology, 1985, Apr-16, Volume: 110, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Electromyography; Electroshock; Flumazenil; Indoles; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle Relaxants, Central; Muscle Tonus; Phenobarbital; Rats; Rats, Inbred Strains

1985
Modulation of neurotransmitter action: control of the gamma-aminobutyric acid response through the benzodiazepine receptor.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1985, Volume: 5, Issue:9

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Chick Embryo; Electric Conductivity; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Neurotransmitter Agents; Picrotoxin; Pyridazines; Receptors, GABA-A

1985
Benzodiazepine receptor ligands and the consumption of a highly palatable diet in non-deprived male rats.
    Psychopharmacology, 1985, Volume: 86, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Drug Interactions; Feeding Behavior; Flumazenil; Ligands; Male; Midazolam; Pyrazoles; Rats; Receptors, GABA-A

1985
Protection against the lethal effects of pentobarbital in mice by a benzodiazepine receptor inverse agonist, 6,7-dimethoxy-4-ethyl-3-carbomethoxy-beta-carboline.
    The Journal of clinical investigation, 1987, Volume: 79, Issue:2

    Topics: Animals; Carbolines; Flumazenil; Male; Mice; Mice, Inbred Strains; Pentobarbital; Receptors, GABA-A

1987
Chronic treatment with lorazepam and FG 7142 may change the effects of benzodiazepine receptor agonists, antagonists and inverse agonists by different mechanisms.
    European journal of pharmacology, 1987, Jan-20, Volume: 133, Issue:3

    Topics: Animals; Carbolines; Drug Interactions; Drug Tolerance; Female; Flumazenil; Lorazepam; Mice; Pentylenetetrazole; Receptors, GABA-A

1987
Benzodiazepine receptors studied in living primates by positron emission tomography: inverse agonist interactions.
    European journal of pharmacology, 1987, Jun-19, Volume: 138, Issue:2

    Topics: Animals; Binding, Competitive; Carbolines; Cerebral Cortex; Convulsants; Dose-Response Relationship, Drug; Electroencephalography; Flumazenil; Male; Papio; Receptors, GABA-A; Tomography, Emission-Computed

1987
Modulation of gamma-aminobutyric acid-mediated inhibitory synaptic currents in dissociated cortical cell cultures.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:23

    Topics: Animals; Bicuculline; Carbolines; Cells, Cultured; Cerebral Cortex; Electric Conductivity; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Potentials; Neural Inhibition; Rats; Synapses

1986
Benzodiazepine ligands, nociception and 'defeat' analgesia in male mice.
    Psychopharmacology, 1987, Volume: 91, Issue:3

    Topics: Analgesia; Animals; Appetite Depressants; Benzodiazepines; Carbolines; Chlordiazepoxide; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Nociceptors; Pyrazoles

1987
Changes in local cerebral glucose utilization induced by the beta-carbolines FG 7142 and DMCM reveal brain structures involved in the control of anxiety and seizure activity.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:4

    Topics: Animals; Anxiety; Autoradiography; Brain; Carbolines; Convulsants; Deoxyglucose; Flumazenil; Glucose; Male; Rats; Rats, Inbred Strains; Seizures

1987
A benzodiazepine agonist and contragonist have hypothermic effects in rodents.
    Neuropharmacology, 1985, Volume: 24, Issue:1

    Topics: Animals; Benzodiazepinones; Body Temperature; Carbolines; Convulsants; Flumazenil; Flurazepam; Hypothermia; Indoles; Male; Mice; Mice, Inbred Strains; Motor Activity; Rats; Rats, Inbred Strains

1985
Evaluation of the beta-carboline ZK 93 426 as a benzodiazepine receptor antagonist.
    Psychopharmacology, 1984, Volume: 83, Issue:3

    Topics: Animals; Anticonvulsants; Ataxia; Benzodiazepinones; Binding, Competitive; Carbolines; Diazepam; Discrimination, Psychological; Drinking; Exploratory Behavior; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Mice; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Sleep

1984
Differential modulation of etazolate or pentobarbital enhanced [3H] muscimol binding by benzodiazepine agonists and inverse agonists.
    Brain research, 1983, Dec-05, Volume: 280, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Etazolate; Flumazenil; Flunitrazepam; Kinetics; Muscimol; Nicotinic Acids; Oxazoles; Pentobarbital; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Increase of cyclic GMP in cerebellum by methyl-6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate (DMCM).
    Brain research, 1983, Aug-29, Volume: 273, Issue:2

    Topics: Animals; Benzodiazepinones; Carbolines; Cerebellar Cortex; Cyclic GMP; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Indoles; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Stimulation, Chemical

1983
beta-Carbolines activate neurons in the substantia nigra pars reticulata: an effect reversed by diazepam and Ro15-1788.
    European journal of pharmacology, 1983, Dec-09, Volume: 96, Issue:1-2

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Drug Interactions; Flumazenil; Indoles; Injections, Intravenous; Male; Rats; Rats, Inbred Strains; Substantia Nigra; Synaptic Transmission

1983
Effect of agonists, inverse agonists, and antagonists of benzodiazepine receptors on the firing rate of substantia nigra pars reticulata neurons.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electrophysiology; Flumazenil; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra

1983
Ligands for benzodiazepine receptors with positive and negative efficacy.
    Biochemical pharmacology, 1984, Mar-15, Volume: 33, Issue:6

    Topics: Animals; Benzodiazepinones; Carbolines; Flumazenil; Humans; Ligands; Radioligand Assay; Receptors, Cell Surface; Receptors, GABA-A

1984
Interaction of beta-carboline inverse agonists for the benzodiazepine site with another site on GABAA receptors.
    British journal of pharmacology, 1995, Volume: 114, Issue:5

    Topics: Barbiturates; Carbolines; Cell Line; Chloride Channels; Convulsants; Flumazenil; GABA Antagonists; GABA-A Receptor Agonists; Humans; Kidney; Patch-Clamp Techniques; Plasmids; Receptors, GABA-A; Steroids

1995
Discriminative stimulus properties of the benzodiazepine receptor inverse agonist methyl-6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate (DMCM).
    Psychopharmacology, 1994, Volume: 113, Issue:3-4

    Topics: Animals; Carbolines; Convulsants; Discrimination, Psychological; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Generalization, Stimulus; Male; Rats; Rats, Sprague-Dawley; Saccharin; Taste

1994
Benzodiazepine antagonists reduce epileptiform discharges in rat hippocampal slices.
    Epilepsia, 1996, Volume: 37, Issue:10

    Topics: Animals; Carbolines; Convulsants; Disease Models, Animal; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Leucine; Epilepsy; Flumazenil; Hippocampus; Kindling, Neurologic; Male; Rats; Rats, Wistar; Receptors, GABA-A; Structure-Activity Relationship; Synaptic Transmission

1996
Azirino[1, 2-d][1, 4]benzodiazepine derivatives and related 1,4-benzodiazepines as anticonvulsant agents in DBA/2 mice.
    General pharmacology, 1996, Volume: 27, Issue:7

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Benzodiazepines; Binding, Competitive; Carbolines; Cell Membrane; Cerebellum; Cerebral Cortex; Chemical Phenomena; Chemistry, Physical; Convulsants; Flumazenil; GABA Modulators; Male; Mice; Mice, Inbred DBA; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1996
Modulation of long-term potentiation in CA1 region of mouse hippocampal brain slices by GABAA receptor benzodiazepine site ligands.
    Neuropharmacology, 1997, Volume: 36, Issue:6

    Topics: Animals; Carbolines; Convulsants; Dizocilpine Maleate; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Mice; Quinolones; Receptors, GABA-A

1997
Anticonvulsant activity of azirino[1,2-d][1,4]benzodiazepines and related 1,4-benzodiazepines in mice.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:1

    Topics: Animals; Anticonvulsants; Benzodiazepines; Carbolines; Cell Line; Convulsants; Flumazenil; GABA Modulators; Male; Membranes; Mice; Mice, Inbred DBA; Movement; Pentylenetetrazole; Radioligand Assay; Receptors, GABA-A; Seizures

1997
Central benzodiazepine involvement in clonidine cardiovascular actions.
    Canadian journal of physiology and pharmacology, 1999, Volume: 77, Issue:11

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Atropine Derivatives; Blood Pressure; Carbolines; Cardiovascular Agents; Clonidine; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Heart Rate; Infusions, Intravenous; Injections, Intraventricular; Male; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, GABA-A; Stereotaxic Techniques; Time Factors; Yohimbine

1999
Reduction of pentylenetetrazol-induced convulsions by the octadecaneuropeptide ODN.
    Peptides, 1999, Volume: 20, Issue:12

    Topics: Acoustic Stimulation; Amino Acid Sequence; Animals; Carbolines; Convulsants; Diazepam Binding Inhibitor; Electric Stimulation; Flumazenil; Injections, Intraventricular; Male; Mice; Mice, Inbred DBA; Molecular Sequence Data; Neuropeptides; Pentylenetetrazole; Peptide Fragments; Receptors, GABA-A; Seizures

1999
Enhanced ultrasonic vocalization and Fos protein expression following ethanol withdrawal: effects of flumazenil.
    Psychopharmacology, 2000, Volume: 152, Issue:2

    Topics: Animals; Carbolines; Ethanol; Flumazenil; Male; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Substance Withdrawal Syndrome; Vocalization, Animal

2000
The octadecaneuropeptide ODN stimulates neurosteroid biosynthesis through activation of central-type benzodiazepine receptors.
    Journal of neurochemistry, 2001, Volume: 76, Issue:1

    Topics: 17-alpha-Hydroxypregnenolone; 17-alpha-Hydroxyprogesterone; 3-Hydroxysteroid Dehydrogenases; Animals; Carbolines; Chromatography, High Pressure Liquid; Dehydroepiandrosterone; Diazepam Binding Inhibitor; Dihydrotestosterone; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hydroxysteroids; Hypothalamus; Immunohistochemistry; In Vitro Techniques; Ligands; Male; Neuroglia; Neurons; Neuropeptides; Peptide Fragments; Pregnenolone; Progesterone; Rana ridibunda; Receptors, GABA-A

2001
Influence of benzodiazepine binding site ligands on fear-conditioned contextual memory.
    European journal of pharmacology, 2001, Aug-24, Volume: 426, Issue:1-2

    Topics: Animals; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; Conditioning, Psychological; Convulsants; Fear; Flumazenil; GABA Antagonists; GABA Modulators; Imidazoles; Ligands; Male; Memory; Mice; Mice, Inbred C57BL; Motor Activity; N-Methylscopolamine; Piperazines; Quinolines; Receptors, GABA-A; Scopolamine; Silanes; Tritium

2001
Bidirectional effects of benzodiazepine binding site ligands in the elevated plus-maze: differential antagonism by flumazenil and beta-CCt.
    Pharmacology, biochemistry, and behavior, 2004, Volume: 79, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding Sites; Carbolines; Drug Interactions; Flumazenil; GABA Modulators; Ligands; Male; Maze Learning; Mice; Midazolam; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Zolpidem

2004
Bidirectional effects of benzodiazepine binding site ligands on active avoidance acquisition and retention: differential antagonism by flumazenil and beta-CCt.
    Psychopharmacology, 2005, Volume: 180, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Benzodiazepines; Binding Sites; Carbolines; Convulsants; Dose-Response Relationship, Drug; Flumazenil; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; Habituation, Psychophysiologic; Injections, Intraperitoneal; Ligands; Male; Midazolam; Motor Activity; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Retention, Psychology; Zolpidem

2005
Negative GABA(A) modulators attenuate the discriminative stimulus effects of benzodiazepines and the neuroactive steroid pregnanolone in rhesus monkeys.
    Psychopharmacology, 2005, Volume: 181, Issue:4

    Topics: Animals; Benzodiazepines; Carbolines; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Female; Flumazenil; Macaca mulatta; Male; Midazolam; Pregnanolone; Receptors, GABA-A; Serotonin Antagonists; Serotonin Receptor Agonists

2005
A high-throughput functional assay for characterization of gamma-aminobutyric acid(A) channel modulators using cryopreserved transiently transfected cells.
    Assay and drug development technologies, 2008, Volume: 6, Issue:6

    Topics: Carbolines; Cell Culture Techniques; Cell Line; Cell Membrane; Cryopreservation; Diazepam; DNA; Dose-Response Relationship, Drug; Drug Discovery; Flumazenil; Flunitrazepam; Fluorescent Dyes; Fluorobenzenes; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Receptors, GABA-A; Reproducibility of Results; Spectrometry, Fluorescence; Transfection; Triazoles; Tritium

2008
Similar anxiolytic-like effects following intra-amygdala infusions of benzodiazepine receptor agonist and antagonist: evidence for the release of an endogenous benzodiazepine inverse agonist in mice exposed to elevated plus-maze test.
    Brain research, 2009, Apr-24, Volume: 1267

    Topics: Amygdala; Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Carbolines; Catheterization; Exploratory Behavior; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Maze Learning; Mice; Microinjections; Midazolam; Motor Activity

2009