flumazenil has been researched along with fg 7142 in 86 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 46 (53.49) | 18.7374 |
1990's | 33 (38.37) | 18.2507 |
2000's | 7 (8.14) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Järvinen, A; Männistö, PT; Rägo, L | 1 |
Galpern, WR; Lumpkin, M; Miller, LG; Pritchard, GA | 1 |
Agmo, A; Fernández, H | 1 |
Falk, JL; Lau, CE; Tang, M; Vigorito, M | 1 |
Allen, M; Cook, JM; Griffiths, RR; Sannerud, CA | 1 |
Little, HJ | 1 |
Franklin, SR; Tang, AH | 1 |
Elsworth, JD; Ida, Y; Roth, RH | 1 |
Devi, K; Hrishikeshavan, HJ; Munonyedi, S; Shanbhogue, R | 1 |
Morse, WH; Teeple, ES; Wettstein, JG | 1 |
Bradberry, CW; Lory, JD; Roth, RH | 1 |
Fernández-Guasti, A; Roldán-Roldán, G; Saldívar, A | 1 |
Fillenz, M; Zetterström, T | 1 |
Koob, GF; Schreiber, JF; Weinger, MB | 1 |
Di Scala, G; Rohmer, JG; Sandner, G | 1 |
Kulkarni, SK; Sharma, AC | 1 |
Blier, P; de Montigny, C; Lista, A | 1 |
Greenblatt, DJ; Heller, J; Lumpkin, M; Miller, LG; Shader, RI; Weill, CL | 1 |
Deutsch, SI; Huntzinger, JA; Mastropaolo, J; Novitzki, MR; Rosse, RB | 1 |
Dragunow, M | 1 |
Becker, HC | 1 |
Mehta, AK; Ticku, MK | 1 |
Donnerer, J | 1 |
Fillenz, M; Pei, Q; Zetterström, T | 1 |
Wettstein, JG | 1 |
Becker, HC; Hale, RL | 1 |
Bodnoff, SR; Meaney, MJ; Quirion, R; Suranyi-Cadotte, BE | 1 |
Arora, PK; Petitto, JM; Skolnick, P | 1 |
Haraguchi, M; Sadeghi, KG; Samson, HH; Tolliver, GA | 1 |
Cooper, SJ; Estall, LB | 1 |
Green, S; Hodges, H | 1 |
Biggio, G; Corda, MG; Fernández, A; Giorgi, O | 1 |
Allen, MS; Cook, JM; Ginter, H; Hagen, TJ; Jackson, B; Skolnick, P; Trullas, R | 1 |
Moody, EJ; Skolnick, P | 1 |
Cole, BJ; Koob, GF | 1 |
File, SE; Pellow, S | 4 |
Dubroeucq, MC; Gauthier, A; Guérémy, C; Le Fur, G; Mizoule, J; Renault, C; Uzan, A | 1 |
Braestrup, C; Petersen, EN; Scheel-Krüger, J | 1 |
Caporali, MG; Gatta, F; Lucantoni, D; Massotti, M; Mele, L | 1 |
Bamonte, F; Guzzon, V; Marzanatti, M; Monopoli, A; Ongini, E | 1 |
Barber, DJ; Cooper, SJ; Gilbert, DB; Moores, WR | 1 |
Biggio, G; Corda, MG; Gatta, F; Giorgi, O | 1 |
Beck, CH; Cooper, SJ | 1 |
Lister, RG; Nutt, DJ | 1 |
Jensen, LH; Petersen, EN | 1 |
Little, HJ; Nutt, DJ; Stanford, SC; Taylor, SC | 1 |
Dingemanse, J; File, SE; Friedman, HL; Greenblatt, DJ | 1 |
Braestrup, C; Koob, GF; Thatcher Britton, K | 1 |
Randall, JI; Rodgers, RJ | 1 |
Ableitner, A; Herz, A | 1 |
Jones, GH; Mittleman, G; Robbins, TW | 1 |
Britton, KT; Koob, GF; Lee, G | 1 |
Costello, MJ; Nutt, DJ | 1 |
Little, HJ; Nutt, DJ; Sellars, N; Taylor, SC | 1 |
Glushankov, PG; Skrebitskiĭ, VG; Vorob'ev, VS | 1 |
Fillenz, M; Fung, SC | 1 |
Little, HJ; Nutt, DJ; Taylor, SC | 1 |
Nutt, D | 1 |
Ongini, E | 1 |
Crawley, JN; Paul, SM; Skolnick, P | 1 |
Corda, MG; Costa, E; Guidotti, A | 1 |
Braestrup, C; Honoré, T; Jensen, LH; Nielsen, M; Petersen, EN | 1 |
Barzaghi, C; Marzanatti, M; Ongini, E | 1 |
De Aguiar, JC; Graeff, FG; Guimarães, FS; Russo, AS | 1 |
Belachew, S; Kettenmann, H; Lefebvre, PP; Leprince, P; Malgrange, B; Moonen, G; Rigo, JM; Rogister, B | 1 |
Laurie, DJ; Pratt, JA | 1 |
Alastra, AJ; Cohen, C; Goldberg, SR; Marley, RJ; Sannerud, CA; Serdikoff, SL | 1 |
Maier, SF; Short, KR | 1 |
Arnsten, AF; Goldman-Rakic, PS; Murphy, BL; Roth, RH | 1 |
Auta, J; Faust, WB; Lambert, P; Moerschbaecher, JM; Winsauer, PJ | 1 |
Matsumoto, K; Ojima, K; Watanabe, H | 1 |
Kohno, SI; Matsumoto, K; Ojima, K; Watanabe, H | 1 |
Jordan, S; Kramer, GL; Petty, F; Wu, J; Zukas, PK | 1 |
Kulkarni, SK; Reddy, DS | 1 |
Gobert, J; Klitgaard, H; Matagne, A; Wülfert, E | 1 |
Adamec, RE | 3 |
Forman, SA; Rüsch, D | 1 |
Cottone, P; Sabino, V; Steardo, L; Zorrilla, EP | 1 |
Halliday, DM; Marsden, CA; Mason, R; Stevenson, CW | 1 |
Ishii, S; Ito, T; Kurumaji, A; Nishikawa, T | 1 |
2 review(s) available for flumazenil and fg 7142
Article | Year |
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The benzodiazepines: anxiolytic and withdrawal effects.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Carbolines; Diazepam; Disease Models, Animal; Ethanol; Flumazenil; Humans; Rats; Receptors, GABA-A; Substance Withdrawal Syndrome; Verapamil | 1991 |
Behavioural pharmacology of food, water and salt intake in relation to drug actions at benzodiazepine receptors.
Topics: Animals; Anti-Anxiety Agents; Appetite; Appetite Depressants; Benzodiazepines; Benzodiazepinones; Carbolines; Chlordiazepoxide; Chlorides; Choice Behavior; Diazepam; Drinking Behavior; Feeding Behavior; Flumazenil; Food Deprivation; Food Preferences; gamma-Aminobutyric Acid; Ion Channels; Midazolam; Picrotoxin; Punishment; Pyrazoles; Receptors, GABA-A; Satiation; Sodium Chloride; Species Specificity | 1985 |
84 other study(ies) available for flumazenil and fg 7142
Article | Year |
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Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Effects of central and peripheral type benzodiazepine ligands on thyrotropin and prolactin secretion.
Topics: Animals; Benzodiazepinones; Carbolines; Clonazepam; Cold Temperature; Diazepam; Flumazenil; Hypothalamo-Hypophyseal System; Isoquinolines; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Secretory Rate; Thyrotropin; Thyrotropin-Releasing Hormone | 1992 |
Chronic benzodiazepine administration. VIII. Receptor upregulation produced by chronic exposure to the inverse agonist FG-7142.
Topics: Animals; Appetite Depressants; Benzodiazepines; Binding Sites; Carbolines; Flumazenil; Injections, Intravenous; Male; Mice; Motor Activity; Receptors, GABA-A; Up-Regulation | 1991 |
Benzodiazepine receptor ligands and sexual behavior in the male rat: the role of GABAergic mechanisms.
Topics: Animals; Bicuculline; Carbolines; Chlordiazepoxide; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Male; Motor Activity; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal | 1991 |
Midazolam withdrawal and discriminative motor control: effects of FG 7142 and Ro 15-1788.
Topics: Animals; Brain Chemistry; Carbolines; Discrimination, Psychological; Dose-Response Relationship, Drug; Drinking Behavior; Flumazenil; GABA-A Receptor Antagonists; Male; Midazolam; Rats; Reinforcement Schedule; Substance Withdrawal Syndrome; Substance-Related Disorders | 1991 |
Behavioral effects of benzodiazepine ligands in non-dependent, diazepam-dependent and diazepam-withdrawn baboons.
Topics: Animals; Behavior, Animal; Benzodiazepines; Carbolines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Ligands; Male; Midazolam; Papio; Receptors, GABA-A; Social Behavior; Substance Withdrawal Syndrome; Substance-Related Disorders | 1991 |
The discriminative stimulus effects of diazepam in rats at two training doses.
Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Male; Morphine; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Triazolam | 1991 |
Anxiogenic beta-carboline FG 7142 produces activation of noradrenergic neurons in specific brain regions of rats.
Topics: Animals; Brain Chemistry; Carbolines; Clonidine; Flumazenil; Male; Methoxyhydroxyphenylglycol; Neurons; Norepinephrine; Rats; Rats, Inbred Strains; Sympathetic Nervous System | 1991 |
Behavioral neurobiology of inverse agonist FG 7142 induced anxiety syndrome in rats.
Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Avoidance Learning; Carbolines; Diazepam; Exploratory Behavior; Flumazenil; Grooming; Male; Motor Activity; Rats; Rats, Inbred Strains; Stereotyped Behavior | 1990 |
Respiratory effects of benzodiazepine-related drugs in awake rhesus monkeys.
Topics: Administration, Inhalation; Alprazolam; Animals; Anti-Anxiety Agents; Appetite Depressants; Benzodiazepines; Buspirone; Carbolines; Carbon Dioxide; Drug Therapy, Combination; Female; Flumazenil; Lorazepam; Macaca mulatta; Male; Pentobarbital; Plethysmography; Pyrazoles; Respiration | 1990 |
The anxiogenic beta-carboline FG 7142 selectively increases dopamine release in rat prefrontal cortex as measured by microdialysis.
Topics: Animals; Anxiety; Benzodiazepines; Carbolines; Corpus Striatum; Dialysis; Dopamine; Flumazenil; Frontal Lobe; Male; Rats; Rats, Inbred Strains | 1991 |
Pharmacological manipulation of anxiety and male rat sexual behavior.
Topics: Animals; Anxiety; Carbolines; Copulation; Diazepam; Flumazenil; Male; Psychomotor Performance; Rats; Rats, Inbred Strains | 1990 |
Local administration of flurazepam has different effects on dopamine release in striatum and nucleus accumbens: a microdialysis study.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Carbolines; Corpus Striatum; Dialysis; Dopamine; Flumazenil; Flurazepam; In Vitro Techniques; Male; Nucleus Accumbens; Picrotoxin; Rats; Rats, Inbred Strains; Septal Nuclei | 1990 |
Effects of two benzodiazepine inverse agonists, RO 15-4513 and FG 7142, on recovery from pentobarbital and halothane anesthesia in the rat.
Topics: Anesthesia Recovery Period; Animals; Azides; Benzodiazepines; Carbolines; Flumazenil; Halothane; Male; Pentobarbital; Random Allocation; Rats; Rats, Inbred Strains; Reflex | 1990 |
Behavioral analysis of the effects of benzodiazepine receptor ligands in the conditioned burying paradigm.
Topics: Animals; Arousal; Benzodiazepinones; Brain; Carbolines; Conditioning, Classical; Diazepam; Dose-Response Relationship, Drug; Electroshock; Fear; Flumazenil; Grooming; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereotyped Behavior | 1990 |
Evidence for GABA-BZ receptor modulation in short-term memory passive avoidance task paradigm in mice.
Topics: Animals; Avoidance Learning; Carbolines; Electroshock; Female; Flumazenil; gamma-Aminobutyric Acid; Male; Memory, Short-Term; Mice; Physostigmine; Receptors, GABA-A; Scopolamine | 1990 |
Benzodiazepine receptors modulate 5-hydroxytryptamine neurotransmission in the rat hippocampus: in vivo electrophysiological evidence.
Topics: Animals; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Hippocampus; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synaptic Transmission | 1990 |
Augmentation of GABAA receptor function by chronic exposure to GABA-neutral and GABA-negative benzodiazepine ligands in cultured cortical neurons.
Topics: Animals; Appetite Depressants; Binding Sites; Carbolines; Chick Embryo; Chlorides; Culture Techniques; Flumazenil; Muscimol; Neurons; Ouabain; Receptors, GABA-A | 1990 |
Profound stress-induced alterations in flurazepam's antiseizure efficacy can be attenuated.
Topics: Animals; Carbolines; Clonazepam; Cold Temperature; Diazepam; Dose-Response Relationship, Drug; Electroshock; Flumazenil; Flurazepam; Male; Mice; Mice, Inbred Strains; Midazolam; Seizures; Stress, Psychological | 1990 |
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines | 1990 |
Effects of the imidazobenzodiazepine RO15-4513 on the stimulant and depressant actions of ethanol on spontaneous locomotor activity.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Chlorides; Ethanol; Flumazenil; Ion Channels; Male; Mice; Mice, Inbred C3H; Motor Activity; Receptors, GABA-A | 1988 |
Ethanol potentiation of GABAergic transmission in cultured spinal cord neurons involves gamma-aminobutyric acidA-gated chloride channels.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Cells, Cultured; Chlorine; Ethanol; Female; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Mice; Mice, Inbred C57BL; Neurons; Radioisotopes; Spinal Cord | 1988 |
Evidence for an excitatory action of the benzodiazepine receptor inverse agonist FG 7142 on C-fibre afferents.
Topics: Adrenocorticotropic Hormone; Animals; Carbolines; Female; Flumazenil; In Vitro Techniques; Male; Nerve Fibers; Neurons, Afferent; Rats; Receptors, GABA-A; Spinal Cord; Substance P | 1989 |
Both systemic and local administration of benzodiazepine agonists inhibit the in vivo release of 5-HT from ventral hippocampus.
Topics: Animals; Benzodiazepines; Carbolines; Chromatography, High Pressure Liquid; Dialysis; Diazepam; Flumazenil; Flurazepam; Hippocampus; Hydroxyindoleacetic Acid; Ion Channels; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin | 1989 |
Behavioral studies with the beta-carboline FG 7142 combined with related drugs in monkeys.
Topics: Animals; Appetite Depressants; Behavior, Animal; Benzodiazepines; Carbolines; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Lorazepam; Male; Pyrazoles; Reinforcement Schedule; Saimiri | 1989 |
Ethanol-induced locomotor stimulation in C57BL/6 mice following RO15-4513 administration.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Ethanol; Flumazenil; Male; Mice; Mice, Inbred C57BL; Motor Activity | 1989 |
Role of the central benzodiazepine receptor system in behavioral habituation to novelty.
Topics: Animals; Carbolines; Diazepam; Exploratory Behavior; Flumazenil; Habituation, Psychophysiologic; Male; Rats; Reaction Time; Receptors, GABA-A | 1989 |
Suppression of natural killer cell activity by FG 7142, a benzodiazepine receptor "inverse agonist".
Topics: Animals; Carbolines; Cytotoxicity Tests, Immunologic; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Antagonists; Killer Cells, Natural; Male; Mice; Receptors, GABA-A | 1989 |
Antagonism of ethanol-reinforced behavior by the benzodiazepine inverse agonists Ro15-4513 and FG 7142: relation to sucrose reinforcement.
Topics: Animals; Azides; Behavior, Animal; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Flumazenil; Male; Rats; Receptors, GABA-A; Reinforcement, Psychology; Self Administration; Sucrose | 1989 |
Are the effects of benzodiazepines on discrimination and punishment dissociable?
Topics: Amygdala; Animals; Behavior, Animal; Benzodiazepines; Carbolines; Chlordiazepoxide; Discrimination, Psychological; Ethanolamines; Flumazenil; gamma-Aminobutyric Acid; Midazolam; Punishment; Pyrazoles; Rats; Receptors, GABA-A | 1987 |
The abstinence syndrome in diazepam-dependent cats is precipitated by Ro 15-1788 and Ro 15-4513 but not by the benzodiazepine receptor antagonist ZK 93426.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Cats; Diazepam; Flumazenil; Receptors, GABA-A; Substance Withdrawal Syndrome | 1988 |
3-Ethoxy-beta-carboline: a high affinity benzodiazepine receptor ligand with partial inverse agonist properties.
Topics: Animals; Binding, Competitive; Brain; Carbolines; Cerebellum; Cerebral Cortex; Convulsants; Drug Synergism; Flumazenil; Hippocampus; In Vitro Techniques; Ligands; Peptic Ulcer; Rats; Receptors, GABA-A; Seizures; Solubility; Stress, Psychological | 1988 |
The imidazobenzodiazepine Ro 15-4513 antagonizes methoxyflurane anesthesia.
Topics: Anesthesia, General; Animals; Azides; Benzodiazepines; Carbolines; Flumazenil; Male; Methoxyflurane; Mice; Receptors, GABA-A; Sleep | 1988 |
Propranolol antagonizes the enhanced conditioned fear produced by corticotropin releasing factor.
Topics: Animals; Anxiety; Carbolines; Conditioning, Psychological; Corticotropin-Releasing Hormone; Fear; Flumazenil; Locus Coeruleus; Male; Motor Activity; Propranolol; Rats; Receptors, Adrenergic, beta; Receptors, Serotonin; Stereoisomerism | 1988 |
Anxiolytic and anxiogenic drug effects on exploratory activity in an elevated plus-maze: a novel test of anxiety in the rat.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Convulsants; Exploratory Behavior; Flumazenil; Male; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats | 1986 |
Opposite effects of two ligands for peripheral type benzodiazepine binding sites, PK 11195 and RO5-4864, in a conflict situation in the rat.
Topics: Animals; Benzodiazepinones; Carbolines; Conditioning, Operant; Conflict, Psychological; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Flumazenil; Isoquinolines; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Evidence that the anticonflict effect of midazolam in amygdala is mediated by the specific benzodiazepine receptors.
Topics: Amygdala; Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Conflict, Psychological; Flumazenil; Male; Midazolam; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Supraspinal convulsions induced by inverse benzodiazepine agonists in rabbits.
Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electroencephalography; Flumazenil; Male; Pyrazoles; Rabbits; Receptors, GABA-A; Seizures | 1985 |
A beta-carboline antagonizes benzodiazepine actions but does not precipitate the abstinence syndrome in cats.
Topics: Animals; Behavior, Animal; Benzodiazepinones; Brain; Carbolines; Cats; Diazepam; Electroencephalography; Flumazenil; Humans; Indoles; Receptors, GABA-A; Substance Withdrawal Syndrome | 1985 |
Benzodiazepine receptor ligands and the consumption of a highly palatable diet in non-deprived male rats.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Drug Interactions; Feeding Behavior; Flumazenil; Ligands; Male; Midazolam; Pyrazoles; Rats; Receptors, GABA-A | 1985 |
The effects of putative anxiogenic compounds (FG 7142, CGS 8216 and Ro 15-1788) on the rat corticosterone response.
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Corticosterone; Flumazenil; Male; Pyrazoles; Rats; Receptors, GABA-A; Stress, Psychological | 1985 |
Long-lasting proconflict effect induced by chronic administration of the beta-carboline derivative FG 7142.
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Conflict, Psychological; Disease Models, Animal; Drinking Behavior; Drug Administration Schedule; Flumazenil; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Time Factors | 1985 |
beta-Carboline FG 7142-reduced aggression in male rats: reversed by the benzodiazepine receptor antagonist, Ro15-1788.
Topics: Aggression; Analysis of Variance; Animals; Avoidance Learning; Benzodiazepinones; Carbolines; Chlordiazepoxide; Flumazenil; Male; Motor Activity; Rats; Receptors, GABA-A | 1986 |
Mice and rats are sensitized to the proconvulsant action of a benzodiazepine-receptor inverse agonist (FG 7142) following a single dose of lorazepam.
Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Drug Interactions; Flumazenil; Injections, Intraperitoneal; Lorazepam; Mice; Rats; Receptors, GABA-A; Species Specificity; Time Factors | 1986 |
Chronic treatment with lorazepam and FG 7142 may change the effects of benzodiazepine receptor agonists, antagonists and inverse agonists by different mechanisms.
Topics: Animals; Carbolines; Drug Interactions; Drug Tolerance; Female; Flumazenil; Lorazepam; Mice; Pentylenetetrazole; Receptors, GABA-A | 1987 |
A single dose of FG 7142 causes long-term increases in mouse cortical beta-adrenoceptors.
Topics: Animals; Appetite Depressants; Carbolines; Cerebral Cortex; Dihydroalprenolol; Flumazenil; Male; Mice; Receptors, Adrenergic, beta | 1987 |
Chronic treatment with Ro 15-1788 distinguishes between its benzodiazepine antagonist, agonist and inverse agonist properties.
Topics: Animals; Behavior, Animal; Benzodiazepinones; Brain Chemistry; Carbolines; Drug Interactions; Drug Tolerance; Exploratory Behavior; Flumazenil; Lorazepam; Male; Rats; Social Behavior | 1986 |
The effects of FG 7142 and RO 15-1788 on the release of punished responding produced by chlordiazepoxide and ethanol in the rat.
Topics: Animals; Carbolines; Chlordiazepoxide; Conditioning, Operant; Conflict, Psychological; Electroshock; Ethanol; Flumazenil; Male; Punishment; Rats; Rats, Inbred Strains | 1986 |
Benzodiazepine ligands, nociception and 'defeat' analgesia in male mice.
Topics: Analgesia; Animals; Appetite Depressants; Benzodiazepines; Carbolines; Chlordiazepoxide; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Nociceptors; Pyrazoles | 1987 |
Changes in local cerebral glucose utilization induced by the beta-carbolines FG 7142 and DMCM reveal brain structures involved in the control of anxiety and seizure activity.
Topics: Animals; Anxiety; Autoradiography; Brain; Carbolines; Convulsants; Deoxyglucose; Flumazenil; Glucose; Male; Rats; Rats, Inbred Strains; Seizures | 1987 |
Effects of diazepam, FG 7142, and RO 15-1788 on schedule-induced polydipsia and the temporal control of behavior.
Topics: Animals; Appetite Depressants; Carbolines; Diazepam; Drinking Behavior; Flumazenil; Male; Motor Activity; Rats | 1988 |
Corticotropin releasing factor and amphetamine exaggerate partial agonist properties of benzodiazepine antagonist Ro 15-1788 in the conflict test.
Topics: Amphetamine; Animals; Behavior, Animal; Carbolines; Chlordiazepoxide; Conflict, Psychological; Corticotropin-Releasing Hormone; Drug Interactions; Flumazenil; Male; Motor Activity; Rats; Rats, Inbred Strains | 1988 |
Rapid induction of lorazepam dependence and reversal with flumazenil.
Topics: Animals; Carbolines; Flumazenil; Lorazepam; Male; Mice; Mice, Inbred Strains; Seizures; Substance-Related Disorders | 1988 |
A benzodiazepine agonist and contragonist have hypothermic effects in rodents.
Topics: Animals; Benzodiazepinones; Body Temperature; Carbolines; Convulsants; Flumazenil; Flurazepam; Hypothermia; Indoles; Male; Mice; Mice, Inbred Strains; Motor Activity; Rats; Rats, Inbred Strains | 1985 |
Chlordiazepoxide enhances the anxiogenic action of CGS 8216 in the social interaction test: evidence for benzodiazepine withdrawal?
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Chlordiazepoxide; Flumazenil; Humans; Male; Pyrazoles; Rats; Social Behavior; Species Specificity; Substance Withdrawal Syndrome | 1985 |
[Effect of the beta-carboline derivative FG 7142 on inhibition in hippocampal sections].
Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electric Stimulation; Evoked Potentials; Flumazenil; Hippocampus; Neural Inhibition; Neurons; Rats; Rats, Inbred Strains | 1985 |
Multiple effects of drugs acting on benzodiazepine receptors.
Topics: Animals; Benzodiazepinones; Calcium; Carbolines; Chlordiazepoxide; Drug Interactions; Flumazenil; gamma-Aminobutyric Acid; Male; Norepinephrine; Potassium; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1984 |
Acute and chronic effects of the benzodiazepine receptor ligand FG 7142: proconvulsant properties and kindling.
Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Flumazenil; Indoles; Kindling, Neurologic; Male; Mice; Mice, Inbred Strains; Receptors, GABA-A | 1984 |
Pharmacological and behavioural studies of benzodiazepine antagonists and contragonists.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepinones; Carbolines; Conditioning, Operant; Conflict, Psychological; Flumazenil; Ganglia, Spinal; Hippocampus; Male; Rats; Seizures; Social Behavior | 1983 |
Behavioral and EEG effects of benzodiazepines and their antagonists in the cat.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Carbolines; Cats; Diazepam; Electroencephalography; Flumazenil | 1983 |
Absence of intrinsic antagonist actions of benzodiazepine antagonists on an exploratory model of anxiety in the mouse.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Carbolines; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Humans; Male; Mice; Pyrazoles | 1984 |
Involvement of GABA in the facilitation of punishment suppressed behavior induced by beta-carbolines in rat.
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Conditioning, Operant; Diazepam; Drug Interactions; Flumazenil; gamma-Aminobutyric Acid; Humans; Indoles; Models, Psychological; Punishment; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Ligands for benzodiazepine receptors with positive and negative efficacy.
Topics: Animals; Benzodiazepinones; Carbolines; Flumazenil; Humans; Ligands; Radioligand Assay; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Intrinsic and antagonistic effects of beta-carboline FG 7142 on behavioral and EEG actions of benzodiazepines and pentobarbital in cats.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Carbolines; Cats; Diazepam; Drug Interactions; Electroencephalography; Flumazenil; Indoles; Male; Pentobarbital | 1983 |
The anxiogenic action of FG 7142 in the social interaction test is reversed by chlordiazepoxide and Ro 15-1788 but not by CGS 8216.
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Chlordiazepoxide; Convulsants; Flumazenil; Humans; Indoles; Male; Motor Activity; Pyrazoles; Rats; Social Behavior | 1984 |
Role of benzodiazepine receptors located in the dorsal periaqueductal grey of rats in anxiety.
Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anticonvulsants; Anxiety; Appetite Depressants; Carbolines; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Male; Microinjections; Midazolam; Periaqueductal Gray; Rats; Rats, Wistar; Receptors, GABA-A | 1993 |
Astroglia-released factor shows similar effects as benzodiazepine inverse agonists.
Topics: Animals; Animals, Newborn; Appetite Depressants; Astrocytes; Benzodiazepines; Biological Factors; Brain; Carbolines; Cells, Cultured; Cerebellum; Cerebral Cortex; Culture Media, Conditioned; Dose-Response Relationship, Drug; Embryo, Mammalian; Flumazenil; gamma-Aminobutyric Acid; Ganglia, Spinal; Glutamic Acid; Hippocampus; Membrane Potentials; Molecular Weight; Neurons; PC12 Cells; Rats; Receptors, GABA-A | 1994 |
Flumazenil induces localised increases in glucose utilization during diazepam withdrawal in rats.
Topics: Animals; Autoradiography; Brain Chemistry; Carbolines; Densitometry; Deoxyglucose; Diazepam; Flumazenil; Glucose; Male; Rats; Substance Withdrawal Syndrome | 1993 |
Tolerance to the behavioral effects of chlordiazepoxide: pharmacological and biochemical selectivity.
Topics: Amphetamine; Animals; Behavior, Animal; Caffeine; Carbolines; Chlordiazepoxide; Chlorides; Chlorine; Dose-Response Relationship, Drug; Drug Tolerance; Flumazenil; gamma-Aminobutyric Acid; Male; Midazolam; Morphine; Pentobarbital; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sensitivity and Specificity; Stimulation, Chemical | 1993 |
Stressor controllability, social interaction, and benzodiazepine systems.
Topics: Animals; Anxiety; Carbolines; Chlordiazepoxide; Dose-Response Relationship, Drug; Electroshock; Flumazenil; Interpersonal Relations; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stress, Psychological | 1993 |
Increased dopamine turnover in the prefrontal cortex impairs spatial working memory performance in rats and monkeys.
Topics: Analysis of Variance; Animals; Benzazepines; Carbolines; Clozapine; Dopamine; Dopamine Antagonists; Female; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Haloperidol; Macaca mulatta; Male; Maze Learning; Memory; Motor Activity; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Space Perception; Stress, Psychological | 1996 |
Effects of negative allosteric modulators of gamma-aminobutyric acidA receptors on complex behavioral processes in monkeys.
Topics: Allosteric Regulation; Alprazolam; Animals; Carbolines; Conditioning, Psychological; Discrimination Learning; Dose-Response Relationship, Drug; Erythrocebus patas; Female; Flumazenil; Receptors, GABA-A | 1997 |
Flumazenil reverses the decrease in the hypnotic activity of pentobarbital by social isolation stress: are endogenous benzodiazepine receptor ligands involved?
Topics: Animals; Carbolines; Chlorides; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Hypnotics and Sedatives; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred Strains; Pentobarbital; Receptors, GABA-A; Sleep; Social Isolation; Stress, Psychological; Synaptosomes | 1997 |
Flumazenil but not FG7142 reverses the decrease in pentobarbital sleep caused by activation of central noradrenergic systems in mice.
Topics: Animals; Appetite Depressants; Carbolines; Cerebral Ventricles; Flumazenil; Injections, Intravenous; Injections, Intraventricular; Male; Methoxamine; Mice; Mice, Inbred Strains; Pentobarbital; Sleep; Yohimbine | 1997 |
Benzodiazepine prevention of swim stress-induced sensitization of cortical biogenic amines: an in vivo microdialysis study.
Topics: Animals; Anti-Anxiety Agents; Biogenic Amines; Carbolines; Diazepam; Drug Evaluation, Preclinical; Flumazenil; GABA Agonists; GABA Antagonists; Male; Microdialysis; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Stress, Physiological; Swimming | 1997 |
Reversal of benzodiazepine inverse agonist FG 7142-induced anxiety syndrome by neurosteroids in mice.
Topics: Animals; Anxiety; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; Isoquinolines; Male; Maze Learning; Mice; Mice, Inbred BALB C; Motor Activity; Progesterone; Receptors, GABA-A; Steroids | 1997 |
Evidence for a unique profile of levetiracetam in rodent models of seizures and epilepsy.
Topics: Amygdala; Animals; Anticonvulsants; Behavior, Animal; Carbolines; Convulsants; Diazepam; Disease Models, Animal; Electroconvulsive Therapy; Epilepsy; Excitatory Amino Acid Agonists; Flumazenil; GABA-A Receptor Antagonists; Kindling, Neurologic; Levetiracetam; Male; Mice; Pentylenetetrazole; Piracetam; Rats; Rats, Sprague-Dawley; Seizures | 1998 |
Evidence that NMDA-dependent limbic neural plasticity in the right hemisphere mediates pharmacological stressor (FG-7142)-induced lasting increases in anxiety-like behavior: study 3--the effects on amygdala efferent physiology of block of NMDA receptors p
Topics: Amygdala; Animals; Anxiety; Behavior, Animal; Carbolines; Cats; Electrodes, Implanted; Evoked Potentials; Flumazenil; Functional Laterality; GABA Antagonists; GABA Modulators; Limbic System; Long-Term Potentiation; Male; N-Methylaspartate; Neuronal Plasticity; Neurons, Efferent; Receptors, N-Methyl-D-Aspartate; Vocalization, Animal | 1998 |
Evidence that long-lasting potentiation in limbic circuits mediating defensive behaviour in the right hemisphere underlies pharmacological stressor (FG-7142) induced lasting increases in anxiety-like behaviour: role of benzodiazepine receptors.
Topics: Aggression; Animals; Anxiety; Behavior, Animal; Carbolines; Catheterization; Cats; Flumazenil; Functional Laterality; GABA Agonists; GABA Modulators; Jugular Veins; Limbic System; Male; Predatory Behavior; Rats; Receptors, GABA-A; Stress, Psychological; Vocalization, Animal | 2000 |
Evidence that long-lasting potentiation of amygdala efferents in the right hemisphere underlies pharmacological stressor (FG-7142) induced lasting increases in anxiety-like behaviour: role of GABA tone in initiation of brain and behavioural changes.
Topics: Aggression; Amygdala; Animals; Anticonvulsants; Anxiety; Behavior, Animal; Brain Chemistry; Carbolines; Cats; Efferent Pathways; Flumazenil; Functional Laterality; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Hypothalamus, Middle; Male; Predatory Behavior; Rats; Receptors, GABA-A; Stress, Psychological; Vigabatrin; Vocalization, Animal | 2000 |
Classic benzodiazepines modulate the open-close equilibrium in alpha1beta2gamma2L gamma-aminobutyric acid type A receptors.
Topics: Algorithms; Animals; Benzodiazepines; Binding Sites; Carbolines; Cattle; Electrophysiology; Flumazenil; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Ligands; Midazolam; Oocytes; Patch-Clamp Techniques; Plasmids; Xenopus laevis | 2005 |
FG 7142 specifically reduces meal size and the rate and regularity of sustained feeding in female rats: evidence that benzodiazepine inverse agonists reduce food palatability.
Topics: Animals; Anorexia; Anxiety Disorders; Appetite; Appetite Depressants; Appetite Regulation; Brain; Carbolines; Circadian Rhythm; Dose-Response Relationship, Drug; Feeding Behavior; Female; Flumazenil; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Rats; Rats, Wistar; Receptors, GABA-A; Stress, Psychological | 2007 |
Systemic administration of the benzodiazepine receptor partial inverse agonist FG-7142 disrupts corticolimbic network interactions.
Topics: Amygdala; Animals; Carbolines; Cortical Synchronization; Dose-Response Relationship, Drug; Electrophysiology; Flumazenil; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; Male; Microelectrodes; Neural Pathways; Neurons; Prefrontal Cortex; Rats | 2007 |
Effects of FG7142 and immobilization stress on the gene expression in the neocortex of mice.
Topics: Animals; Anti-Inflammatory Agents; Carbolines; Corticosterone; Flumazenil; GABA Antagonists; GABA Modulators; Gene Expression; Male; Mice; Mice, Inbred C57BL; Neocortex; Oligonucleotide Array Sequence Analysis; Restraint, Physical; Reverse Transcriptase Polymerase Chain Reaction; RNA; Stress, Psychological | 2008 |