flumazenil and diazepam

flumazenil has been researched along with diazepam in 733 studies

Research

Studies (733)

TimeframeStudies, this research(%)All Research%
pre-1990262 (35.74)18.7374
1990's266 (36.29)18.2507
2000's140 (19.10)29.6817
2010's53 (7.23)24.3611
2020's12 (1.64)2.80

Authors

AuthorsStudies
Bianucci, AM; Da Settimo, A; Da Settimo, F; Giannaccini, G; Lucacchini, A; Martini, C; Primofiore, G1
Cecchi, L; Colotta, V; Filacchioni, G; Giannaccini, G; Lucacchini, A; Martini, C; Melani, F1
Baker, R; Engelstoff, M; Herbert, R; Knight, A; MacLeod, A; Merchant, K; Moseley, J; Saunders, J; Swain, CJ; Watjen, F1
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Barone, D; Gallico, L; Luzzani, F; Tarzia, G; Toja, E1
Lüddens, H; Wieland, HA1
de Costa, BR; Dominguez, C; Gu, ZQ; Rice, KC; Skolnick, P; Wong, G1
Basile, AS; Fryer, RI; Gu, ZQ; Rios, R; Skolnick, P; Zhang, P1
Catarzi, D; Cecchi, L; Colotta, V; Costagli, C; Filacchioni, G; Galli, A; Varano, F1
Da Settimo, A; Da Settimo, F; Gesi, M; Giannaccini, G; Greco, G; Lucacchini, A; Marini, AM; Martini, C; Novellino, E; Primofiore, G1
Aiello, PM; Bruni, F; Ciciani, G; Costa, B; Costanzo, A; Guerrini, G; Ipponi, A; Lucacchini, A; Martini, C; Selleri, S1
Dekermendjian, K; Kahnberg, P; Liljefors, T; Nielsen, M; Sterner, O; Witt, MR1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Da Settimo, F; Gesi, M; Greco, G; La Motta, C; Marini, AM; Martini, C; Novellino, E; Primofiore, G; Taliani, S; Trincavelli, L1
Topliss, JG; Yoshida, F1
Besnard, F; Bruni, F; Ciciani, G; Costa, B; Costagli, C; Costanzo, A; Guerrini, G; Malmberg-Aiello, P; Martini, C; Selleri, S1
Kuribara, H; Maruyama, Y; Weintraub, ST; Yoshihama, T1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Besnard, F; Cosimelli, B; Costa, B; Da Settimo, F; Greco, G; Martini, C; Montali, M; Novellino, E; Primofiore, G; Salerno, S; Taliani, S1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Besnard, F; Cosimelli, B; Da Settimo, F; Ehlardo, M; Greco, G; La Motta, C; Marini, AM; Martini, C; Montali, M; Novellino, E; Primofiore, G; Sala, A; Simorini, F; Taliani, S1
Besnard, F; Calderone, V; Cosimelli, B; Da Settimo, F; Greco, G; La Motta, C; Marini, AM; Martini, C; Montali, M; Novellino, E; Patrizi, MP; Primofiore, G; Sergianni, V; Simorini, F; Taliani, S1
Bruni, F; Cambi, G; Ciciani, G; Costanzo, A; Ghelardini, C; Guerrini, G; Martini, C; Melani, F; Montali, M; Norcini, M; Selleri, S1
Lombardo, F; Obach, RS; Waters, NJ1
Clayton, T; Cook, J; DeLorey, TM; Furtmüller, R; Halliwell, RF; Harris, D; Huck, S; Sahbaie, P; Sieghart, W1
Anzini, M; Betti, L; Braile, C; Cappelli, A; Ghelardini, C; Giannaccini, G; Giorgi, G; Ian Fryer, R; Limongelli, V; Lucacchini, A; Makovec, F; Marinelli, L; Norcini, M; Novellino, E; Valenti, S; Vomero, S1
Ahman, M; Holmén, AG; Wan, H1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Bruni, F; Cambi, G; Ciciani, G; Costanzo, A; Ghelardini, C; Guarino, C; Guerrini, G; Martini, C; Melani, F; Montali, M; Norcini, M; Selleri, S1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Bruni, F; Ciattini, S; Ciciani, G; Costanzo, A; Daniele, S; Ghelardini, C; Guarino, C; Guerrini, G; Martini, C; Melani, F; Montali, M; Norcini, M; Selleri, S1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Alcaro, S; Anzini, M; Betti, L; Biggio, G; Braile, C; Cappelli, A; Daniele, S; Di Cesare Mannelli, L; Ghelardini, C; Giannaccini, G; Giorgi, G; Limongelli, V; Lucacchini, A; Marinelli, L; Martini, C; Mascia, MP; Novellino, E; Ortuso, F; Valenti, S; Vomero, S1
Bagal, SK; Brown, AD; Cox, PJ; Omoto, K; Owen, RM; Pryde, DC; Sidders, B; Skerratt, SE; Stevens, EB; Storer, RI; Swain, NA1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Anzini, M; Betti, L; Biggio, G; Braile, C; Cappelli, A; Castriconi, F; Di Capua, A; Di Cesare Mannelli, L; Frosini, M; Ghelardini, C; Giannaccini, G; Giorgi, G; Giuliani, G; Grisci, G; Lucacchini, A; Mascia, MP; Paolino, M; Ricci, L; Valenti, S; Vomero, S1
Anzini, M; Brogi, S; Cappelli, A; Chemi, G; Di Capua, A; Di Cesare Mannelli, L; Garofalo, A; Ghelardini, C; Giorgi, G; Grande, F; Matucci, R; Paolino, M; Reale, A1
Davies, MF; Loew, GH; Maguire, PA; Villar, HO1
Facklam, M; Haefely, WE; Schoch, P1
Bonetti, EP; Facklam, M; Haefely, WE; Jenck, F; Martin, JR; Moreau, JL; Schoch, P1
Arakawa, K; Benson, KT; Goto, H; Yokoyama, M1
Järvinen, A; Männistö, PT; Rägo, L1
Inano, S1
Dudley, MW; Kane, JM; Kehne, JH; Miller, JA; Sorensen, SM1
Coale, A; Friedhoff, AJ; Gruen, RJ; Moghaddam, B1
Fukuda, N; Wada, T4
McNamara, RK; Skelton, RW2
Hönack, D; Löscher, W2
Hirose, A; Kumasaka, Y; Nakamura, M; Shimizu, H; Tanaka, H1
Barlin, GB; Davies, LP; Ireland, SJ; Ngu, MM1
Bernasconi, R; Leonhardt, T; Martin, P; Portet, C; Schmutz, M; Steulet, AF1
Gröger, P; Kettler, D; Kolenda, H; Michaelis, HC; Steinwachs, M; Sydow, M1
Brain, PF; Kurishingal, H; Restall, CJ1
Gallagher, LV; Greene, SA; Keegan, RD; Moore, MP1
Almog, S; Ezra, D; Mordel, A; Tirosh, M; Winkler, E1
Boone, MS; Emmett-Oglesby, MW; Pugh, SL1
Sim, MK; Tsoi, WF1
Ator, NA; Griffiths, RR2
File, SE; Hitchcott, PK; Zharkovsky, A1
Gallaher, EJ; Phillips, TJ1
Tietz, EI1
Mori, K; Murayama, T; Ogawa, T; Shindo, K; Shingu, K; Tamai, S; Tomoda, K1
Hart, YM; Meinardi, H; Nutt, DJ; Sander, JW; Shorvon, SD2
Basile, AS; Harrison, PM; Hughes, RD; Jones, EA; Murata, Y; Pannell, L; Skolnick, P; Williams, R1
Backus, KH; Pflimlin, P; Trube, G1
Agmo, A; Fernández, H1
al-Tikriti, MS; Baldwin, RM; Innis, RB; Johnson, EW; Laruelle, MA; Malison, RT; Seibyl, JP; Sybirska, EH; Zimmermann, RC; Zoghbi, SS1
Bottlaender, M; Brouillet, E; Chavoix, C; Dodd, RH; Fournier, D; Hantraye, P; Khalili-Varasteh, M; Mazière, M1
Allen, M; Cook, JM; Griffiths, RR; Sannerud, CA1
Bitran, D; Ison, JR; Kellogg, CK; Sullivan, AT1
Engel, JA; Söderpalm, B1
Little, HJ1
Engel, JA; Hulthe, P; Johannessen, K; Söderpalm, B; Svensson, L1
Inoue, Y; Ohno, M; Shibata, S; Teshima, K; Tominaga, K; Ueki, S; Ushio, M; Watanabe, S; Yamamoto, T1
Franklin, SR; Tang, AH1
Blasquez, C; Braquet, P; Delbende, C; Jégou, S; Tranchand Bunel, D; Vaudry, H1
Franklin, SR; Himes, CS; Ho, PM; Tang, AH1
Dickey, KM; Martin, WR; Sloan, JW; Wala, E1
Hernández, J1
Kaneyuki, H; Mizuki, Y; Tanaka, M; Tsuda, A; Yamada, M; Yokoo, H; Yoshida, M1
Coates, W; Evans, TC; Harchelroad, F; Isaacs, M; Jehle, D1
De Meo, F; De Meo, M; Fellico, C; Ferone, A; Gaeta, N1
Consiglio, F; De Lisio, C; Finelli, B; Iannotti, M; Pace, MC; Passavanti, MB1
Suzuki, H1
Blakeman, DP; Im, WB1
Basile, AS1
Simon, A1
Flemström, G; Jedstedt, G; Säfsten, B1
Andersen, B; Forrest, M; Gjørup, I; Vilien, M1
Nagatani, T; Yamamoto, T1
Cruccu, G; Fabbri, A; Ferracuti, S; Leardi, MG; Manfredi, M1
Bing, LH; Matsumoto, K; Ohta, H; Satoh, T; Watanabe, H1
Martin, WR; Sloan, JW; Wala, EP3
De Luca, C; De Medici, D; Massotti, M1
Devi, K; Hrishikeshavan, HJ; Munonyedi, S; Shanbhogue, R1
Doenicke, A; Greim, M; Juhl, G; Rampf, U; Suttmann, H1
Biggio, G; Carcangiu, G; Concas, A; Mereu, G; Passino, N1
Budhram, P; Deacon, RM; Gardner, CR; Thomson, TA1
Izquierdo, I; Medina, JH; Pereira, ME1
File, SE; Hitchcott, PK1
Hicks, TP; Oka, JI1
Borsini, F; D'Aranno, V; Lecci, A; Mancinelli, A; Meli, A; Stasi, MA; Volterra, G1
Kucharik, RF; Lucki, I1
Elgoyhen, AB; Kazanietz, MG1
McCloy, RF; Pearson, RC1
Blanchard, JC; Boireau, A; Doble, A; Dubedat, P; Laduron, PM1
Hole, K; Rosland, JH1
Chernilas, J; Geller, E; Halpern, P; Miller, HB; Niv, D1
Isaac, PA; Okell, RW; Piggott, SE; Roberts, B; Robinson, JO; Rosen, M; Sanders, LD1
Kadiwar, RM; Pillay, R1
Knudsen, J; Nielsen, M1
Bauerle, LM; DeNoble, VJ; Jones, KW; Schaeffer, CL1
Fernández-Guasti, A; Roldán-Roldán, G; Saldívar, A1
Chapouthier, G; Dodd, RH; Raffalli-Sebille, MJ; Venault, P1
Coenen, AM; Nutt, DJ; Peeters, BW; Titulaer, MN; Van Rijn, CM; Vossen, JM1
Ida, Y; Nishimura, H; Tanaka, M1
McNamara, RK; Whishaw, IQ1
Bogdanov, NN; Molodavkin, GM; Voronina, TA1
Amaki, Y; Hajiri, H; Kaneko, M; Kobayashi, K; Kumagai, M; Shudo, Y1
Briley, M; Lerner-Natoli, M; Rondouin, G; Stenger, A1
Ceckler, T; Guillet, R; Kellogg, C; Miranda, R1
Nagatani, T; Sugihara, T; Takao, K; Ueki, S; Yamamoto, T1
Di Scala, G; Rohmer, JG; Sandner, G1
Blier, P; de Montigny, C; Lista, A2
Corda, MG; Fratta, W; Orlandi, M1
Giros, B; Llorens-Cortes, C; Quach, TT; Schwartz, JC; Van Amsterdam, JG1
Deutsch, SI; Huntzinger, JA; Mastropaolo, J; Novitzki, MR; Rosse, RB1
Dragunow, M1
Myers, RD; Paez, X1
Baartmans, MG; Kopp, EF; Oudesluys-Murphy, AM1
Lopez, A; Rebollo, J1
Hashida, T; Katoh, H; Kawamoto, T; Mishima, S; Mori, K; Murakawa, M; Sasai, S; Urabe, N; Yamaoka, H1
Amaki, Y; Horiguchi, T; Kobayashi, K; Takinami, M1
Doi, M; Ikeda, K1
Hashemi, FS; Niles, LP1
Fuccaro, P; Mantero, L; Mazzarello, MR; Roccatagliata, DC; Sburlati, E1
Hill, JL; Insel, TR; Mayor, RB1
Crespi, F; Keane, PE1
Haefely, W1
Hernández, J; Pérez, D; Ruiz, F1
Adler-Graschinsky, E; Elgoyhen, B1
Fillenz, M; Pei, Q; Zetterström, T1
Jensen, S; Kirkegaard, L; Knudsen, EB; Knudsen, L; Kruse, A1
Mora, CT; Torjman, M; White, PF1
Bursztein, S1
Block, RI; Dembo, JB; Ghoneim, MM1
Koot, M; Van Duin, CT; Van Miert, AS1
Belknap, JK; Crabbe, JC; Laursen, SE1
Kovács, I; Maksay, G; Simonyi, M1
Ida, Y; Nishimura, H; Tanaka, M; Tsuda, A1
Cherniack, NS; Deal, EC; Haxhiu, MA; van Lunteren, E1
Ida, Y; Shirao, I; Sueyoshi, K; Tanaka, M; Tsuda, A1
Andersen, P; Christiansen, C; Jarnvig, IL; Jørgensen, B; Skielboe, M; Weber, M1
Gallager, DW; Heninger, C; Hernandez, TD; Wilson, MA1
Gallager, DW; Wilson, MA2
Bodnoff, SR; Meaney, MJ; Quirion, R; Suranyi-Cadotte, BE1
Bachy, A; Cordeau, LR; Croizat, BP; Gros, F; Keane, PE; Larcher, JC; Le Marquer, FJ; Vayssiere, JL1
Innes, DG; Kavaliers, M2
Canonaco, M; McEwen, BS; O'Connor, LH; Pfaff, DW1
Hernandez, TD; Jones, GH; Schallert, T1
Harary, N; Kellogg, C1
Lüddens, H; Pritchett, DB; Seeburg, PH1
Albertson, TE; Joy, RM1
Barth, TM; Bowery, NG; Moratalla, R1
Kellogg, CK; Miranda, RC; Wagner, JP1
Kaneto, H; Takahashi, M; Tokuyama, S1
Appel, M; Bron, HN; Hooymans, PM; Janknegt, R1
Gavish, M; Katz, Y1
Fassbender, CP; Hönack, D; Löscher, W1
Antelman, SM; Edwards, DJ; Knopf, S; Kocan, D1
Bizière, K; Fournier, M; Keane, P; Santucci, V; Worms, P1
Garamvölgyi, G; Hamar, O; Kálmán, A1
Costall, B; Jones, BJ; Kelly, ME; Naylor, RJ; Oakley, NR; Onaivi, ES; Tyers, MB1
Cooper, SJ; Estall, LB1
Crabbe, JC; Gallaher, EJ; Gionet, SE; Hollister, LE1
Dan'ura, T; Ishibashi, S; Kurokawa, T; Yamashita, A; Yanagiuchi, H1
Randall, JI; Rodgers, RJ3
Cox, DH; Guidotti, A; Santi, MR1
Hanada, S; Hashimoto, S; Tanaka, C; Taniyama, K1
Nagatani, T; Sugihara, T; Ueki, S; Yamamoto, T1
Biggio, G; Corda, MG; Fernández, A; Giorgi, O1
Jensen, S; Kirkegaard, L; Knudsen, L1
Dunton, AW; Hendler, J; McGrath, J; Pitman, V; Schwam, E; Siegel, J1
Dan'ura, T; Ishibashi, S; Kurokawa, T; Une, Y; Yamashita, A1
Arbilla, S; Langer, SZ; Lista, A1
Brown, CL; Dodd, RH; Potier, MC; Prado de Carvalho, L; Rossier, J1
Hawkins, M; Pravica, M; Radulovacki, M1
Blanchard, JC; Boireau, A; Dubédat, P; Farges, G; Laduron, PM; Martel, M1
Kuga, T; Moroi, K; Takashi, K1
De Medici, D; Gatta, F; Longo, VG; Massotti, M1
Marczynski, TJ; Urbancic, M1
Mehta, AK; Mhatre, M; Ticku, MK1
Lister, RG1
Bonetti, EP; Burkard, WP; Gabl, M; Hunkeler, W; Lorez, HP; Martin, JR; Moehler, H; Osterrieder, W; Pieri, L; Polc, P1
Chiu, TH; Rosenberg, HC3
Hofer, P; Scollo-Lavizzari, G1
Griffiths, RR; Lamb, RJ2
Kubota, K; Matsuda, I; Matsuoka, Y; Sugaya, K; Terawaki, Y1
Klockgether, T; Schwarz, M; Sontag, KH; Turski, L1
Le Bihan, C; Simon, P; Soubrié, P; Thiébot, MH1
Ellis, S; Foltin, RW; Schuster, CR1
Spealman, RD2
Spealman, RD; Wettstein, JG2
Barrett, JE; Mansbach, RS; Skolnick, P; Weissman, BA; Witkin, JM1
Ueki, S; Yamamoto, T1
Crul, JF; Driessen, JJ; van der Pol, F; van Egmond, J1
Albertson, TE; Foulke, GE1
O'Brien, DP; White, FJ1
Biziere, K; Keane, PE; Morre, M; Simiand, J1
Davis, M; Gallager, DW1
O'Regan, MH; Phillis, JW1
Concas, A; Morelli, M; Obata, T; Serra, M; Yamamura, HI1
Elsasser, S; Ritz, R; Schwander, J1
De Deyn, PP; Macdonald, RL2
Benkert, O; Heuser, I; Wetzel, H1
Fillenz, M; Fung, SC1
Biggio, G; Concas, A; Corda, MG; Crisponi, G; Nurchi, V; Serra, M1
Böke-Kuhn, K; Danneberg, PB; Hommer, D; Kuhn, FJ; Lehr, E; Paul, SM; Skolnick, P; Weber, KH1
Kempner, ES; Paul, SM; Schwartz, RD; Skolnick, P; Thomas, JW1
Capek, R; Davies, MF; Esplin, B1
Moura, D; Soares-da-Silva, P1
Consolo, S; Forloni, G; Garattini, S; Kolasa, K; Ladinsky, H1
Caporali, MG; Gatta, F; Lucantoni, D; Massotti, M; Mele, L1
Romstedt, K1
Dingledine, R; King, GL; Knox, JJ1
Bamonte, F; Guzzon, V; Marzanatti, M; Monopoli, A; Ongini, E1
Paul, SM; Reed, GF; Skolnick, P1
Biggio, G; Concas, A; Corda, MG1
Abraham, CJ; De Blas, AL; Haney, SA; Park, D; Rayner, CA; Sangameswaran, L1
Cole, R; De Vellis, J; Noble, EP; Syapin, PJ1
Fares, F; Gavish, M1
Bourn, WM; Garrett, RL1
Ehrin, E; Eriksson, L; Farde, L; Hedström, CG; Litton, JE; Mindus, P; Persson, A; Sedvall, G1
Ida, Y; Nagasaki, N; Tanaka, M; Tsuda, A; Tsujimaru, S1
Agarwal, AK; Gulati, A; Kumar, P; Sethi, BB; Sethi, N; Trivedi, JK1
Meiners, BA; Salama, AI1
Adinoff, B; Linnoila, M; Majchrowicz, E; Martin, PR1
Barrett, JE; Cook, JM; Larscheid, P; Witkin, JM1
Hicks, TP; Jang, EK; Oka, JI1
Bryere, P; Naquet, R; Valin, A1
Biggio, G; Corda, MG1
Ayhan, IH; Palaoğlu, O2
Glowa, JR; Paul, SM; Skolnick, P1
Kulkarni, SK; Kunchandy, J1
Astier, H; Roussel, JP; Tapia-Arancibia, L1
Biziere, K; Bourguignon, JJ; Chambon, JP; Heaulme, M; Perio, A; Tebib, S; Wermuth, CG1
Biggio, G; Carcangiu, P; Corda, MG; Giorgi, O; Mereu, G1
Bender, AS; Hertz, L1
Barksdale, CM; Kalin, NH; Shelton, SE1
Goldstein, JM; Malick, JB; Sutton, EB1
Ciuffi, M; Franchi-Micheli, S; Luzzi, S; Rosi, E; Spagnesi, S; Zilletti, L1
Gwee, MC; Wong, PT; Yoong, YL1
Chiba, S; Haruta, K; Homma, N; Iwatsuki, K; Yamagishi, F1
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K1
Ferrario, P; Hafner, B; Mantegazza, P; Tammiso, R; Zambotti, F; Zonta, N1
Michenfelder, JD; Milde, JH; Roald, OK; Steen, PA1
Martin, WR; McNicholas, LF2
Dhawan, BN; Gulati, A; Singh, HK; Srimal, RC1
Katzman, NJ; Shannon, HE1
Biziere, K; Calassi, R; Chambon, JP; Heaulme, M; Perio, A1
Sanger, DJ1
Albertson, TE; Walby, WF1
Teo, WL; Wong, PT1
Jensen, S; Kirkegaard, L; Knudsen, L; Kruse, A1
Gallager, DW; Heninger, G; Heninger, K1
Eison, MS1
Levin, ED; Liebeskind, JC; Morgan, MM1
Dodgson, MS; Emhjellen, S; Skeie, B; Steen, PA; Wickstrøm, E1
Crawford, RD; Johnson, DD; Pedder, SC; Tuchek, JM; Wilcox, R1
Iwasawa, H; Naito, H; Tonoue, T1
Engel, J; Hård, E1
Idemudia, SO; Lal, H; Mathis, DA1
Jones, GH; Mittleman, G; Robbins, TW1
Lanore, JJ; Manfredi, R; Sockeel, F; Tannières, ML; Vourc'h, G1
Kanto, J; Klotz, U1
Martin, WR; McNicholas, LF; Sloan, JW; Wala, E1
Kataoka, Y; Kumakura, K; Ohara-Imaizumi, M; Ueki, S1
Kunert-Radek, J; Pawlikowski, M; Radek, A; Stepien, H1
Pacilli, P; Sicignano, A; Spinelli, P1
Chiu, TH; Rosenberg, HC; Yu, O1
Cagiano, R; Cuomo, V; De Salvia, MA; Maselli, MA; Racagni, G; Renna, G1
Malick, JB; Patel, JB; Rinarelli, CA1
Aitken, DH; Bodnoff, SR; Meaney, MJ; Quirion, R; Suranyi-Cadotte, B1
Gelb, AW; Ume, EO1
Kawasaki, K; Matsushita, A; Satoh, M; Takagi, H1
Kavaliers, M1
Hernández, J; Ribeiro, JA; Ruiz, F1
Hiltunen, AJ; Järbe, TU1
Emmett-Oglesby, MW; Harris, CM; Idemudia, SO; Lal, H; Mathis, DA1
Fenerty, JP; Finkelstein, MF; Galloway, MP; Grant, SJ; Mayor, R; Redmond, DE; Roth, RH1
Longo, VG; Sagratella, S1
Klockgether, T; Pardowitz, I; Schwarz, M; Sontag, KH; Turski, L1
Glushankov, PG; Skrebitskiĭ, VG; Vorob'ev, VS1
Ableitner, A; Herz, A; Wüster, M1
Caccia, S; Ceci, A; Garattini, S; Masturzo, P; Mennini, T; Salmona, M1
Barone, D; Colombo, G; Glasser, A; Luzzani, F; Mennini, T1
Belin, C; Carriot, T; Dubroeucq, MC; Guérémy, C; Le Fur, G; Mestre, M; Renault, C; Uzan, A1
Braestrup, C; Honoré, T; Jensen, LH; Kehr, W; Petersen, EN; Schmiechen, R; Schneider, H; Seidelmann, D; Stephens, DN1
Kawasaki, K; Kodama, M; Matsushita, A1
Morin, AM1
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Curley, MD; Ferrigno, M; Lovrincevic, MM; Lundgren, CE; Wylegala, J1
Gangisetty, O; Reddy, DS1
Acher, F; Brański, P; Pałucha-Poniewiera, A; Pilc, A; Stachowicz, K; Wierońska, JM1
Antkowiak, B; Drexler, B; Hentschke, H; Zinser, S1
Beyer, C; Emadi, F; Hadjiakhoondi, A; Sharifzadeh, M; Yassa, N1
Cardenas, R; Quintero, L; Suarez-Roca, H1
Chebib, M; Gavande, N; Hanrahan, JR; Johnston, GA; Karim, N; Wellendorph, P1
Cook, JM; Divljaković, J; Milić, M; Rallapalli, S; Savić, MM; Timić, T; van Linn, ML1
Costa, JP; de Almeida, AA; de Carvalho, RB; de Freitas, RM; de Sousa, DP1
Baldisserotto, B; Barros, FM; Bürger, ME; Caron, BO; Heinzmann, BM; Heldwein, CG; Mallmann, CA; Reckziegel, P; Schmidt, D; Silva, LL1
Chen, CR; Huang, ZL; Luo, YJ; Qu, WM; Urade, Y; Zhou, XZ1
Prather, JF1
Cook, JM; Groenink, L; Hansen, HH; Mirza, NR; Nielsen, EØ; Olivier, B; van Oorschot, R; Vinkers, CH1
Furuya, H; Inoue, S; Iwata, M; Kawaguchi, M1
Cook, JM; Divljaković, J; Milić, M; Namjoshi, OA; Savić, MM; Timić, T; Tiruveedhula, VV1
Brito, GA; Cavalheiro, EA; da Costa, MA; da Cruz, GM; da Graça Naffah-Mazzacoratti, M; de Andrade, GM; de Barros Viana, GS; Felipe, CF; Leal, LK; Menezes, ML; Scorza, FA; Tavares, AF1
Cho, S; Han, D; Jin, YH; Jin, Z; Kim, IH; Kim, S1
Farbood, Y; Mansouri, MT; Mashak, A; Naghizadeh, B; Sarkaki, A; Soltani, M1
de Almeida, AA; de Carvalho, RB; de Freitas, RM; de Sousa, DP; Silva, OA1
Cho, NC; Cho, S; Han, JK; Huang, ZL; Jin, YH; Kim, J; Kim, JS; Kim, S; Pae, AN; Shimizu, M; Takata, Y; Urade, Y; Yang, H; Yoon, M1
Baldisserotto, B; Bürger, ME; Flores, ÉM; Gai, EZ; Heinzmann, BM; Heldwein, CG; Parodi, TV; Roman, C; Silva, Lde L1
Gruca, P; Lason-Tyburkiewicz, M; Litwa, E; Papp, M; Willner, P1
Asadi-Shekaari, M; Eslami, A; Joukar, S; Kalantaripour, T1
Bäckström, T; Helström, L; Möller, AT; Nyberg, S; Söndergaard, HP1
Baur, R; Maldifassi, MC; Middendorp, SJ; Sigel, E1
Banks, ML; Shelton, KL; Tracy, ME1
Baldisserotto, B; Bürger, ME; Garlet, QI; Gressler, LT; Heinzmann, BM; Pires, LC; Silva, DT; Spall, S1
Bonnefoi, F; Bouillot, C; Liger, F; Zimmer, L1
Chen, SL; Liu, XG; Wei, XH; Zang, Y; Zheng, WH1
Djordjević, S; Jović-Stosić, J; Kilibarda, V; Perković-Vukcević, N; Segrt, Z1
Djordjević, S; Ercegović, GV; Segrt, Z; Stosić, JJ; Vukcević, NP1
Absalom, NL; Chebib, M; Christensen, ET; Chua, HC; Hartiadi, LY; Hoestgaard-Jensen, K; Jensen, AA; Ramzan, I1
Beckman, D; Blaha, CD; Boschen, SL; Da Cunha, C; Ferreira, ST; Fiorenza, AM; Gomez-A, A; Lee, K; Sugi, AH1
Fernández-Guasti, A; González-Trujano, ME; Hernandez-Leon, A1
Deng, S; Ding, J; Fan, HR; Ge, WH; Huang, C; Li, F; Li, WG; Liu, YM; Xu, TL; Zhu, T1
Erfanparast, A; Henareh-Chareh, F; Tamaddonfard, E1
Brodnik, ZD; España, RA; Oleson, EB; Pultorak, KJ; Rakowski, DR; Sambells, AT; Schelp, SA1
Barbosa-Filho, JM; Chaves, EMC; Dantas, LP; Honório-Júnior, JER; Lúcio, ASSC; Monteiro, VS; Nonato, DTT; Patrocínio, MCA; Sousa, CNS; Vasconcelos, SMM; Viana, GSB1
Christian, CA; Courtney, CD1
Chen, JG; Deng, Q; Gao, SQ; Hu, ZL; Liu, WH; Long, LH; Lu, JJ; Nie, TL; Shen, ZC; Wang, F; Wu, PF; Xia, ZX; Yao, XP; Zhang, SQ; Zheng, HL1
Das, N; Ganeshpurkar, A; Gupta, SK; Krishnamurthy, S; Kumar, D; Singh, R; Singh, SK1
Clodfelder-Miller, B; McNaught, J; Nelson, DE; Ness, TJ; Su, X1
Gharpure, A; Hibbs, RE; Howard, RJ; Kim, JJ; Lindahl, E; Noviello, CM; Teng, J; Walsh, RM; Zhu, S; Zhuang, Y1
Marjanović, DS; Nikolic, K; Perdih, A; Stevanovic, S; Trailović, SM; Zdravković, N1
Amundarain, MJ; Caffarena, ER; Costabel, MD1
Acquas, E; Bassareo, V; Cottiglia, F; Kasture, SB; Maccioni, E; Maccioni, R; Sanna, E; Talani, G1
Esumi, S; Izushi, Y; Kitamura, Y; Matsumoto, D; Noda, Y; Sendo, T; Ushio, S; Wada, Y1
Behzad, S; Faizi, M; Jahani, R; Saffariha, M; Toufan Tabrizi, N1
Cao, Y; Lian, J; Ma, Y; Muheyati, A; Su, R; Wang, N; Yu, G; Yuan, S; Zhang, S1
Basso-Hulse, G; Bennett, KS; Gallo, AT; Hulse, GK; MacDonald, T1
Basso-Hulse, G; Gallo, AT; Hulse, GK; MacDonald, T1
Ahmed, T; Al-Khafaji, K; Araújo, IM; Bappi, MH; Coutinho, HDM; de Andrade, EM; Hanif, MA; Hossain, R; Islam, MS; Islam, MT; Khan, RA; Kowalska, G; Kowalski, R; Rahaman, MM; Sarkar, C1

Reviews

17 review(s) available for flumazenil and diazepam

ArticleYear
Ion channels as therapeutic targets: a drug discovery perspective.
    Journal of medicinal chemistry, 2013, Feb-14, Volume: 56, Issue:3

    Topics: Drug Discovery; Humans; Ion Channels; Models, Molecular; Phylogeny

2013
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
The benzodiazepines: anxiolytic and withdrawal effects.
    Neuropeptides, 1991, Volume: 19 Suppl

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Carbolines; Diazepam; Disease Models, Animal; Ethanol; Flumazenil; Humans; Rats; Receptors, GABA-A; Substance Withdrawal Syndrome; Verapamil

1991
Behavioural pharmacology of food, water and salt intake in relation to drug actions at benzodiazepine receptors.
    Neuroscience and biobehavioral reviews, 1985,Spring, Volume: 9, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Appetite; Appetite Depressants; Benzodiazepines; Benzodiazepinones; Carbolines; Chlordiazepoxide; Chlorides; Choice Behavior; Diazepam; Drinking Behavior; Feeding Behavior; Flumazenil; Food Deprivation; Food Preferences; gamma-Aminobutyric Acid; Ion Channels; Midazolam; Picrotoxin; Punishment; Pyrazoles; Receptors, GABA-A; Satiation; Sodium Chloride; Species Specificity

1985
Flumazenil: US clinical pharmacology studies.
    European journal of anaesthesiology. Supplement, 1988, Volume: 2

    Topics: Adult; Diazepam; Double-Blind Method; Drug Interactions; Female; Flumazenil; Humans; Lorazepam; Male; Memory; Receptors, GABA-A; Triazolam

1988
Time course for development of benzodiazepine tolerance and physical dependence.
    Neuroscience and biobehavioral reviews, 1985,Spring, Volume: 9, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Drug Tolerance; Flumazenil; Flurazepam; Humans; Hypnotics and Sedatives; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1985
The role of adenosine in the central actions of the benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1988, Volume: 12, Issue:4

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Arousal; Benzodiazepinones; Brain; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Neural Inhibition; Neurons; Purkinje Cells; Rats; Receptors, GABA-A

1988
[Drug activation of GABAergic transmission in the central nervous system: benzodiazepines and GABAergic agonists].
    Acta medica portuguesa, 1985, Volume: 6, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Chemical Phenomena; Chemistry; Cyclic GMP; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Humans; Receptors, GABA-A; Synaptic Transmission; Valproic Acid

1985
Pharmacokinetics and clinical use of flumazenil (Ro 15-1788).
    Clinical pharmacokinetics, 1988, Volume: 14, Issue:1

    Topics: Anesthesia; Benzodiazepines; Diazepam; Flumazenil; Humans; Injections, Intravenous; Poisoning

1988
Adenosine's role in the central actions of the benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1984, Volume: 8, Issue:4-6

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Brain; Cats; Cell Line; Cerebral Cortex; Diazepam; Flumazenil; Rats; Synaptosomes; Thioinosine

1984
The neuropharmacology of various diazepam antagonists.
    Neuropharmacology, 1983, Volume: 22, Issue:12B

    Topics: Animals; Benzodiazepinones; Caffeine; Carbolines; Diazepam; Flumazenil; Humans; Physostigmine; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A; Theophylline

1983
Antagonists to the benzodiazepines.
    British dental journal, 1984, Dec-08, Volume: 157, Issue:11

    Topics: Anesthesia, Dental; Benzodiazepines; Benzodiazepinones; Diazepam; Flumazenil; Humans

1984
Benzodiazepines for intravenous conscious sedation: agonists and antagonists.
    Compendium (Newtown, Pa.), 1993, Volume: 14, Issue:8

    Topics: Anesthesia, Dental; Benzodiazepines; Conscious Sedation; Diazepam; Flumazenil; Humans; Injections, Intravenous; Lorazepam; Midazolam

1993
Comparing drugs for short-term sedation.
    Contemporary internal medicine, 1994, Volume: 6, Issue:12

    Topics: Anesthesia; Benzodiazepines; Conscious Sedation; Diazepam; Flumazenil; Humans; Lorazepam; Midazolam; Pain; Propofol

1994
[Parenteral use of benzodiazepines in dentistry in order to reduce stress in adult patients].
    Oral surgery, oral diagnosis : OSD, 1996, Volume: 7

    Topics: Adult; Anesthetics; Antidotes; Conscious Sedation; Dental Care; Diazepam; Flumazenil; Humans; Midazolam; Middle Aged; Monitoring, Physiologic; Oximetry; Premedication; Stress, Psychological

1996
Sedation and analgesia for gastrointestinal endoscopy during pregnancy.
    Gastrointestinal endoscopy clinics of North America, 2006, Volume: 16, Issue:1

    Topics: Analgesia; Analgesics, Opioid; Cholangiopancreatography, Endoscopic Retrograde; Conscious Sedation; Diazepam; Endoscopy, Gastrointestinal; Female; Fentanyl; Fetus; Flumazenil; Humans; Hypnotics and Sedatives; Ketamine; Lidocaine; Meperidine; Naloxone; Pregnancy; Propofol; Risk Assessment; Triage

2006
Midazolam and other benzodiazepines.
    Handbook of experimental pharmacology, 2008, Issue:182

    Topics: Anesthetics, Intravenous; Animals; Benzodiazepines; Biotransformation; Central Nervous System; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Humans; Lorazepam; Midazolam; Molecular Structure; Receptors, GABA-A; Structure-Activity Relationship

2008

Trials

38 trial(s) available for flumazenil and diazepam

ArticleYear
The effect of intravenous flumazenil on interictal electroencephalographic epileptic activity: results of a placebo-controlled study.
    Journal of neurology, neurosurgery, and psychiatry, 1991, Volume: 54, Issue:4

    Topics: Adult; Anticonvulsants; Brain; Diazepam; Dose-Response Relationship, Drug; Drug Therapy, Combination; Electroencephalography; Epilepsies, Partial; Epilepsy; Epilepsy, Temporal Lobe; Evoked Potentials; Female; Flumazenil; Humans; Infusions, Intravenous; Male; Middle Aged; Receptors, GABA-A; Single-Blind Method

1991
[The sequence chlorodimethyldiazepam/anexate in the pharmacologic hypnosis of patients undergoing peripheral anesthesia in orthopedics and traumatology].
    Minerva anestesiologica, 1991, Volume: 57, Issue:9

    Topics: Aged; Anesthesia, Local; Diazepam; Double-Blind Method; Female; Flumazenil; Humans; Hypnosis, Anesthetic; Male; Middle Aged; Orthopedics; Wounds and Injuries

1991
The effect of the benzodiazepine antagonist flumazenil on the sequels of diazepam given before upper gastrointestinal endoscopy. A double-blind randomized trial.
    Scandinavian journal of gastroenterology, 1991, Volume: 26, Issue:7

    Topics: Adult; Aged; Analysis of Variance; Conscious Sedation; Diazepam; Double-Blind Method; Endoscopy, Digestive System; Female; Flumazenil; Humans; Male; Middle Aged; Psychomotor Performance; Time Factors

1991
Nociceptive quality of the orbicularis oculi reflexes as evaluated by distinct opiate- and benzodiazepine-induced changes in man.
    Brain research, 1991, Aug-16, Volume: 556, Issue:2

    Topics: Adult; Blinking; Diazepam; Electric Stimulation; Electromyography; Fentanyl; Flumazenil; Humans; Naloxone; Nociceptors; Placebos

1991
[Beta activation following the intravenous administration of benzodiazepines and the specific antagonist flumazenil (Ro 15-1788)].
    EEG-EMG Zeitschrift fur Elektroenzephalographie, Elektromyographie und verwandte Gebiete, 1990, Volume: 21, Issue:1

    Topics: Adult; Anti-Anxiety Agents; Benzodiazepines; Beta Rhythm; Diazepam; Dose-Response Relationship, Drug; Electroencephalography; Flumazenil; Flunitrazepam; Humans; Injections, Intravenous; Lorazepam; Male; Midazolam; Prospective Studies; Randomized Controlled Trials as Topic; Stimulation, Chemical

1990
Reversal of benzodiazepine sedation with the antagonist flumazenil.
    British journal of anaesthesia, 1991, Volume: 66, Issue:4

    Topics: Adolescent; Adult; Aged; Ambulatory Care; Anesthesia Recovery Period; Anesthesia, Intravenous; Benzodiazepines; Cognition; Diazepam; Double-Blind Method; Female; Flumazenil; Gastroscopy; Headache; Humans; Male; Memory; Midazolam; Middle Aged; Psychomotor Performance

1991
Flumazenil used for antagonizing the central effects of midazolam and diazepam in outpatients.
    Acta anaesthesiologica Scandinavica, 1989, Volume: 33, Issue:1

    Topics: Adult; Aged; Ambulatory Care; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Flumazenil; Gastroscopy; Humans; Male; Midazolam; Middle Aged; Random Allocation

1989
Time course of antagonism of sedative and amnesic effects of diazepam by flumazenil.
    Anesthesiology, 1989, Volume: 70, Issue:6

    Topics: Adult; Arousal; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Flumazenil; Humans; Male; Memory; Molar, Third; Random Allocation; Time Factors; Tooth, Impacted

1989
Antagonism of diazepam sedation by flumazenil.
    British journal of anaesthesia, 1989, Volume: 63, Issue:5

    Topics: Aged; Aged, 80 and over; Alfentanil; Anesthesia, General; Carbon Dioxide; Diazepam; Double-Blind Method; Flumazenil; Humans; Middle Aged; Nitrous Oxide; Oxygen; Randomized Controlled Trials as Topic; Wakefulness

1989
Fentanyl-midazolam-flumazenil anesthesia for induced abortion.
    International journal of gynaecology and obstetrics: the official organ of the International Federation of Gynaecology and Obstetrics, 1989, Volume: 30, Issue:1

    Topics: Abortion, Induced; Adolescent; Adult; Ambulatory Care Facilities; Anesthesia Recovery Period; Diazepam; Drug Therapy, Combination; Female; Fentanyl; Flumazenil; Humans; Ketamine; Meperidine; Midazolam; Pain Measurement; Pregnancy; Random Allocation

1989
Flumazenil used in the antagonizing of diazepam and midazolam sedation in out-patients undergoing gastroscopy.
    European journal of anaesthesiology. Supplement, 1988, Volume: 2

    Topics: Adolescent; Adult; Aged; Diazepam; Double-Blind Method; Flumazenil; Gastroscopy; Humans; Midazolam; Middle Aged; Outpatients; Random Allocation; Receptors, GABA-A; Sleep

1988
Flumazenil: US clinical pharmacology studies.
    European journal of anaesthesiology. Supplement, 1988, Volume: 2

    Topics: Adult; Diazepam; Double-Blind Method; Drug Interactions; Female; Flumazenil; Humans; Lorazepam; Male; Memory; Receptors, GABA-A; Triazolam

1988
Benzodiazepine antagonist Ro 15-1788. Antagonism of diazepam sedation in outpatients undergoing gastroscopy.
    Anaesthesia, 1986, Volume: 41, Issue:12

    Topics: Adolescent; Adult; Aged; Amnesia; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; Flumazenil; Gastroscopy; Humans; Hypnotics and Sedatives; Male; Middle Aged; Time Factors

1986
Antagonism of diazepam-induced sedative effects by Ro15-1788 in patients after surgery under lumbar epidural block. A double-blind placebo-controlled investigation of efficacy and safety.
    Acta anaesthesiologica Scandinavica, 1987, Volume: 31, Issue:7

    Topics: Adult; Aged; Amnesia; Anesthesia, Epidural; Clinical Trials as Topic; Diazepam; Double-Blind Method; Emotions; Female; Flumazenil; Humans; Hypnotics and Sedatives; Male; Middle Aged; Psychomotor Performance; Random Allocation

1987
[Clinical evaluation of flumazenil (Anexate) on the recovery parameters following the administration of 3 benzodiazepines (flunitrazepam, midazolam or diazepam].
    Cahiers d'anesthesiologie, 1987, Volume: 35, Issue:8

    Topics: Adult; Aged; Analgesics; Anesthesia Recovery Period; Anesthesia, General; Benzodiazepines; Diazepam; Drug Evaluation; Female; Flumazenil; Flunitrazepam; Humans; Male; Midazolam; Middle Aged; Postoperative Period; Prospective Studies; Random Allocation; Respiration

1987
Clinical use of flumazenil (Ro 15-1788) after endoscopic procedures.
    Endoscopy, 1988, Volume: 20, Issue:2

    Topics: Adult; Aged; Clinical Trials as Topic; Diazepam; Double-Blind Method; Endoscopy; Female; Flumazenil; Humans; Male; Middle Aged; Random Allocation

1988
Ro 15-1788 antagonizes the effects of diazepam in man without affecting its bioavailability.
    British journal of anaesthesia, 1983, Volume: 55, Issue:4

    Topics: Adolescent; Adult; Benzodiazepines; Benzodiazepinones; Biological Availability; Clinical Trials as Topic; Diazepam; Double-Blind Method; Flumazenil; Humans; Learning; Male; Memory; Psychomotor Performance; Random Allocation; Time Factors

1983
RO 15-1788 antagonises the central effects of diazepam in man without altering diazepam bioavailability.
    British journal of clinical pharmacology, 1982, Volume: 14, Issue:5

    Topics: Adult; Benzodiazepinones; Biological Availability; Diazepam; Double-Blind Method; Emotions; Flumazenil; Humans; Male; Psychomotor Performance

1982
[The effect of flumazenil in reversing midazolam, flunitrazepam or diazepam].
    Masui. The Japanese journal of anesthesiology, 1995, Volume: 44, Issue:6

    Topics: Adolescent; Adult; Anesthesia Recovery Period; Anesthesia, Epidural; Anesthesia, Spinal; Diazepam; Female; Flumazenil; Flunitrazepam; Hemodynamics; Humans; Male; Midazolam; Middle Aged; Respiration

1995
Differential acute psychomotor and cognitive effects of diazepam on long-term benzodiazepine users.
    International clinical psychopharmacology, 1994, Volume: 9, Issue:3

    Topics: Adult; Anxiety Disorders; Cognition; Depressive Disorder; Diazepam; Dose-Response Relationship, Drug; Double-Blind Method; Drug Tolerance; Female; Flumazenil; Humans; Injections, Intravenous; Long-Term Care; Male; Mental Recall; Middle Aged; Neuropsychological Tests; Personality Inventory; Psychomotor Performance; Receptors, GABA-A; Substance Withdrawal Syndrome; Substance-Related Disorders

1994
Dissociation of benzodiazepine-induced amnesia from sedation by flumazenil pretreatment.
    Psychopharmacology, 1993, Volume: 112, Issue:4

    Topics: Adult; Amnesia; Attention; Cross-Over Studies; Diazepam; Double-Blind Method; Flumazenil; Humans; Hypnotics and Sedatives; Male; Memory, Short-Term; Mental Recall

1993
The effect of intravenously administered diazepam, midazolam and flumazenil on the sensitivity of upper airway reflexes.
    Anaesthesia, 1994, Volume: 49, Issue:2

    Topics: Adult; Ammonia; Diazepam; Double-Blind Method; Flumazenil; Gagging; Humans; Injections, Intravenous; Male; Midazolam; Reaction Time; Time Factors

1994
Ability of flumazenil, butorphanol, and naloxone to reverse the anesthetic effects of oxymorphone-diazepam in dogs.
    Journal of the American Veterinary Medical Association, 1996, Aug-15, Volume: 209, Issue:4

    Topics: Adjuvants, Anesthesia; Anesthetics, Combined; Animals; Butorphanol; Cross-Over Studies; Diazepam; Dogs; Drug Combinations; Female; Flumazenil; Male; Naloxone; Narcotic Antagonists; Oxymorphone; Time Factors

1996
Flumazenil reversal of psychomotor impairment due to midazolam or diazepam for conscious sedation for upper endoscopy.
    Gastrointestinal endoscopy, 1996, Volume: 44, Issue:4

    Topics: Adult; Aged; Aged, 80 and over; Akathisia, Drug-Induced; Anesthetics, Intravenous; Antidotes; Chi-Square Distribution; Conscious Sedation; Diazepam; Duodenoscopy; Esophagoscopy; Female; Flumazenil; Gastroscopy; Humans; Male; Midazolam; Middle Aged; Treatment Outcome

1996
Flumazenil reversal of conscious sedation induced with intravenous fentanyl and diazepam.
    Anesthesia progress, 1995, Volume: 42, Issue:1

    Topics: Adult; Analysis of Variance; Anesthesia Recovery Period; Anesthesia, Dental; Anesthetics, Intravenous; Conscious Sedation; Diazepam; Double-Blind Method; Female; Fentanyl; Flumazenil; GABA Antagonists; Humans; Hypnotics and Sedatives; Male; Middle Aged

1995
A placebo controlled study of flumazenil in bronchoscopic procedures.
    British journal of clinical pharmacology, 1997, Volume: 43, Issue:1

    Topics: Adolescent; Aged; Anti-Anxiety Agents; Antidotes; Bronchoscopy; Conscious Sedation; Diazepam; Double-Blind Method; Female; Flumazenil; Hemodynamics; Humans; Injections, Intravenous; Male; Middle Aged; Psychomotor Performance

1997
Benzodiazepine mediated antagonism of opioid analgesia.
    Pain, 1997, Volume: 71, Issue:1

    Topics: Adult; Analgesics, Non-Narcotic; Analgesics, Opioid; Anti-Anxiety Agents; Diazepam; Double-Blind Method; Drug Synergism; Female; Flumazenil; GABA Modulators; Humans; Ibuprofen; Injections, Intravenous; Male; Molar, Third; Morphine; Pain Measurement; Pain, Postoperative; Premedication; Receptors, GABA-A; Tooth Extraction

1997
Midazolam versus diazepam in lipid emulsion as conscious sedation for colonoscopy with or without reversal of sedation with flumazenil.
    Gastrointestinal endoscopy, 1998, Volume: 47, Issue:1

    Topics: Adolescent; Adult; Analysis of Variance; Anesthetics, Combined; Anesthetics, Intravenous; Antidotes; Colonoscopy; Conscious Sedation; Diazepam; Double-Blind Method; Fat Emulsions, Intravenous; Female; Flumazenil; Humans; Logistic Models; Male; Midazolam; Middle Aged; Pain; Pain Measurement; Patient Satisfaction

1998
Stressful reactions and panic attacks induced by flumazenil in chronic benzodiazepine users.
    Journal of psychopharmacology (Oxford, England), 1998, Volume: 12, Issue:2

    Topics: Adult; Anti-Anxiety Agents; Arousal; Diazepam; Double-Blind Method; Female; Flumazenil; GABA Modulators; Humans; Infusions, Intravenous; Male; Middle Aged; Panic; Panic Disorder; Substance-Related Disorders

1998
Flumazenil in children after esophagogastroduodenoscopy.
    The American journal of gastroenterology, 1999, Volume: 94, Issue:7

    Topics: Adolescent; Analgesics, Opioid; Anesthesia Recovery Period; Benzodiazepines; Child; Conscious Sedation; Diazepam; Double-Blind Method; Endoscopy, Gastrointestinal; Esophagoscopy; Female; Flumazenil; Humans; Hypnotics and Sedatives; Male; Meperidine; Prospective Studies

1999
Short-term effects of intravenous benzodiazepines on autonomic neurocardiac regulation in humans: a comparison between midazolam, diazepam, and lorazepam.
    Critical care medicine, 2002, Volume: 30, Issue:5

    Topics: Adult; Autonomic Nervous System; Benzodiazepines; Diazepam; Female; Flumazenil; Heart; Heart Rate; Humans; Injections, Intravenous; Lorazepam; Male; Midazolam; Middle Aged; Preanesthetic Medication; Prospective Studies

2002
Flumazenil-precipitated withdrawal in healthy volunteers following repeated diazepam exposure.
    Psychopharmacology, 2005, Volume: 178, Issue:2-3

    Topics: Administration, Oral; Adult; Blood Pressure; Diazepam; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Flumazenil; GABA Modulators; Humans; Hypnotics and Sedatives; Injections, Intravenous; Male; Skin Temperature; Substance Withdrawal Syndrome; Substance-Related Disorders

2005
Diazepam-induced disruption of classically-conditioned fear-potentiation of late-latency auditory evoked potentials is prevented by flumazenil given before, but not after, CS/US pairing.
    Journal of psychopharmacology (Oxford, England), 2007, Volume: 21, Issue:1

    Topics: Adult; Anti-Anxiety Agents; Association Learning; Conditioning, Classical; Diazepam; Double-Blind Method; Drug Administration Schedule; Electroshock; Evoked Potentials, Auditory; Evoked Potentials, Somatosensory; Fear; Flumazenil; GABA Antagonists; Humans; Male; Photic Stimulation; Reaction Time; Receptors, GABA-A; Reference Values; Reflex, Startle; Time Factors

2007
Clinical evaluation of intranasal benzodiazepines, alpha-agonists and their antagonists in canaries.
    Veterinary anaesthesia and analgesia, 2006, Volume: 33, Issue:3

    Topics: Administration, Intranasal; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anesthesia; Animals; Behavior, Animal; Benzodiazepines; Canaries; Diazepam; Drug Therapy, Combination; Female; Flumazenil; Hypnotics and Sedatives; Imidazoles; Male; Midazolam; Prospective Studies; Xylazine; Yohimbine

2006
Extending submarine crew survival by reducing CO2 production with quickly reversible sedation.
    Aviation, space, and environmental medicine, 2010, Volume: 81, Issue:6

    Topics: Acceleration; Adult; Analysis of Variance; Antidotes; Carbon Dioxide; Cognition; Diazepam; Flumazenil; GABA Modulators; Health Status Indicators; Humans; Hypnotics and Sedatives; Male; Oxygen Consumption; Respiration; Submarine Medicine; Time Factors; Young Adult

2010
Rapid and reliable sedation induced by diazepam and antagonized by flumazenil in zebra finches (Taeniopygia guttata).
    Journal of avian medicine and surgery, 2012, Volume: 26, Issue:2

    Topics: Anesthesia Recovery Period; Animals; Antidotes; Consciousness; Diazepam; Dose-Response Relationship, Drug; Female; Finches; Flumazenil; Hypnotics and Sedatives; Male

2012
A double-blind randomised crossover trial of low-dose flumazenil for benzodiazepine withdrawal: A proof of concept.
    Drug and alcohol dependence, 2022, 07-01, Volume: 236

    Topics: Benzodiazepines; Cross-Over Studies; Diazepam; Double-Blind Method; Flumazenil; GABA-A Receptor Antagonists; Humans; Inactivation, Metabolic; Pilot Projects; Receptors, GABA-A; Substance Withdrawal Syndrome

2022
Outcomes of patients treated with low-dose flumazenil for benzodiazepine detoxification: A description of 26 participants.
    Drug and alcohol dependence, 2022, 08-01, Volume: 237

    Topics: Benzodiazepines; Diazepam; Flumazenil; Humans; Substance Withdrawal Syndrome

2022

Other Studies

679 other study(ies) available for flumazenil and diazepam

ArticleYear
Benzodiazepine receptor affinity and interaction of some N-(indol-3-ylglyoxylyl)amine derivatives.
    Journal of medicinal chemistry, 1992, Jun-12, Volume: 35, Issue:12

    Topics: Animals; Anticonvulsants; Binding, Competitive; Cattle; Cell Membrane; Cerebral Cortex; Convulsants; Dopamine; Flunitrazepam; Indoles; Mice; Molecular Structure; Receptors, GABA-A; Structure-Activity Relationship; Tryptamines; Tyramine

1992
Tricyclic heteroaromatic systems. [1]benzopyranopyrrol-4-ones and [1]benzopyrano-1,2,3-triazol-4-ones as benzodiazepine receptor ligands. Synthesis and structure-activity relationships.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:9

    Topics: Animals; Azoles; Benzopyrans; Cattle; Chemical Phenomena; Chemistry; Dibenzazepines; Ligands; Pyrroles; Receptors, GABA-A; Structure-Activity Relationship

1990
Novel benzodiazepine receptor partial agonists: oxadiazolylimidazobenzodiazepines.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:10

    Topics: Animals; Benzodiazepines; Cell Membrane; Cerebral Cortex; Models, Molecular; Molecular Conformation; Molecular Structure; Oxadiazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship; X-Ray Diffraction

1989
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Benzodiazepine receptor binding and anticonflict activity in a series of 3,6-disubstituted pyridazino[4,3-c]isoquinolines devoid of anticonvulsant properties.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:9

    Topics: Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Conflict, Psychological; Diazepam; Isoquinolines; Male; Mice; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Structure-Activity Relationship

1985
Four amino acid exchanges convert a diazepam-insensitive, inverse agonist-preferring GABAA receptor into a diazepam-preferring GABAA receptor.
    Journal of medicinal chemistry, 1994, Dec-23, Volume: 37, Issue:26

    Topics: Amino Acid Sequence; Azides; Base Sequence; Benzodiazepines; Binding Sites; Diazepam; GABA Agonists; Humans; Molecular Sequence Data; Mutation; Receptors, GABA-A; Structure-Activity Relationship

1994
Synthesis and evaluation of imidazo[1,5-a][1,4]benzodiazepine esters with high affinities and selectivities at "diazepam-insensitive" benzodiazepine receptors.
    Journal of medicinal chemistry, 1993, Apr-16, Volume: 36, Issue:8

    Topics: Animals; Benzodiazepines; Binding Sites; Brain; Esters; Imidazoles; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1993
Structure-activity relationship studies at the benzodiazepine receptor (BZR): a comparison of the substitutent effects of pyrazoloquinolinone analogs.
    Journal of medicinal chemistry, 1993, May-28, Volume: 36, Issue:11

    Topics: Animals; Brain; In Vitro Techniques; Pyrazoles; Quinolones; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Solubility; Structure-Activity Relationship

1993
Synthesis and binding activity of some pyrazolo[1,5-c]quinazolines as tools to verify an optional binding site of a benzodiazepine receptor ligand.
    Journal of medicinal chemistry, 1996, Jul-19, Volume: 39, Issue:15

    Topics: Animals; Binding Sites; Flunitrazepam; Hydrogen Bonding; Male; Pyrazoles; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Structure-Activity Relationship; Tritium

1996
N'-Phenylindol-3-ylglyoxylohydrazide derivatives: synthesis, structure-activity relationships, molecular modeling studies, and pharmacological action on brain benzodiazepine receptors.
    Journal of medicinal chemistry, 1998, Sep-24, Volume: 41, Issue:20

    Topics: Animals; Anticonvulsants; Binding, Competitive; Brain; Cattle; Cerebral Cortex; Convulsants; Diazepam; Flumazenil; GABA Modulators; Glyoxylates; Hydrazines; In Vitro Techniques; Indoles; Ligands; Mice; Models, Molecular; Molecular Conformation; Receptors, GABA-A; Seizures; Structure-Activity Relationship

1998
Benzodiazepine receptor ligands. 4. Synthesis and pharmacological evaluation of 3-heteroaryl-8-chloropyrazolo[5,1-c][1,2,4] benzotriazine 5-oxides.
    Journal of medicinal chemistry, 1999, Jun-17, Volume: 42, Issue:12

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Cattle; Cerebral Cortex; Cyclic N-Oxides; In Vitro Techniques; Ligands; Male; Mice; Muscle Relaxants, Central; Radioligand Assay; Receptors, GABA-A; Triazines

1999
Structure-activity relationships and molecular modeling analysis of flavonoids binding to the benzodiazepine site of the rat brain GABA(A) receptor complex.
    Journal of medicinal chemistry, 1999, Oct-21, Volume: 42, Issue:21

    Topics: Animals; Binding Sites; Brain; Flavonoids; In Vitro Techniques; Male; Models, Molecular; Molecular Conformation; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Reproducibility of Results; Structure-Activity Relationship

1999
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: tricyclic heteroaromatic derivatives as a new class of benzodiazepine receptor ligands.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Anticonvulsants; Benzimidazoles; Brain; Cattle; Convulsants; Diazepam; Flumazenil; GABA Modulators; In Vitro Techniques; Ligands; Membranes; Mice; Models, Molecular; Radioligand Assay; Receptors, GABA-A

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Benzodiazepine receptor ligands. 7. Synthesis and pharmacological evaluation of new 3-esters of the 8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide. 3-(2-Thienylmethoxycarbonyl) derivative: an anxioselective agent in rodents.
    Journal of medicinal chemistry, 2002, Dec-19, Volume: 45, Issue:26

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Avoidance Learning; Cell Line; Cerebral Cortex; Cyclic N-Oxides; Drug Interactions; Ethanol; Exploratory Behavior; GABA Agents; Heterocyclic Compounds, 3-Ring; Humans; In Vitro Techniques; Ligands; Memory; Mice; Motor Skills; Neuromuscular Agents; Rats; Receptors, GABA-A; Seizures; Sleep; Structure-Activity Relationship; Triazines

2002
An anxiolytic-like effect of Ginkgo biloba extract and its constituent, ginkgolide-A, in mice.
    Journal of natural products, 2003, Volume: 66, Issue:10

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Caffeine; Cyclopentanes; Diazepam; Diterpenes; Dose-Response Relationship, Drug; Furans; Ginkgo biloba; Ginkgolides; Lactones; Male; Maze Learning; Mice; Mice, Inbred Strains; Molecular Structure; Motor Activity; Phenobarbital; Plant Extracts; Plants, Medicinal; Sleep

2003
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
High affinity central benzodiazepine receptor ligands: synthesis and biological evaluation of a series of phenyltriazolobenzotriazindione derivatives.
    Journal of medicinal chemistry, 2005, Apr-21, Volume: 48, Issue:8

    Topics: Animals; Binding, Competitive; Brain; Cattle; Cell Line; Chlorides; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Humans; In Vitro Techniques; Models, Molecular; Protein Isoforms; Radioligand Assay; Rats; Recombinant Proteins; Structure-Activity Relationship; Triazines; Triazoles

2005
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Refinement of the benzodiazepine receptor site topology by structure-activity relationships of new N-(heteroarylmethyl)indol-3-ylglyoxylamides.
    Journal of medicinal chemistry, 2006, Apr-20, Volume: 49, Issue:8

    Topics: Amides; Animals; Binding Sites; Binding, Competitive; Cell Line; GABA-A Receptor Antagonists; Humans; Hydrogen Bonding; Indoles; Ligands; Molecular Structure; Rats; Stereoisomerism; Structure-Activity Relationship

2006
Novel N-substituted indol-3-ylglyoxylamides probing the LDi and L1/L2 lipophilic regions of the benzodiazepine receptor site in search for subtype-selective ligands.
    Journal of medicinal chemistry, 2007, Apr-05, Volume: 50, Issue:7

    Topics: Amides; Animals; Cattle; Cell Line; Cerebral Cortex; GABA-A Receptor Agonists; Glyoxylates; Hypnotics and Sedatives; In Vitro Techniques; Indoles; Ligands; Male; Mice; Mice, Inbred BALB C; Molecular Conformation; Motor Activity; Radioligand Assay; Rats; Structure-Activity Relationship

2007
Novel 3-aroylpyrazolo[5,1-c][1,2,4]benzotriazine 5-oxides 8-substituted, ligands at GABAA/benzodiazepine receptor complex: synthesis, pharmacological and molecular modeling studies.
    Bioorganic & medicinal chemistry, 2008, Apr-15, Volume: 16, Issue:8

    Topics: Animals; Anxiety; Behavior, Animal; Ethanol; Ligands; Male; Memory; Models, Molecular; Molecular Structure; Oxides; Pyrazoles; Rats; Receptors, GABA-A; Seizures; Sleep; Structure-Activity Relationship; Time Factors; Triazines

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.
    Journal of medicinal chemistry, 2008, Jul-10, Volume: 51, Issue:13

    Topics: Animals; Behavior, Animal; Benzodiazepines; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Databases, Factual; Electrophysiology; Female; Ligands; Male; Memory; Mice; Models, Molecular; Molecular Structure; Oocytes; Protein Isoforms; Protein Subunits; Quantitative Structure-Activity Relationship; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis

2008
Ethyl 8-fluoro-6-(3-nitrophenyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate as novel, highly potent, and safe antianxiety agent.
    Journal of medicinal chemistry, 2008, Aug-14, Volume: 51, Issue:15

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding Sites; Brain; Cattle; Computer Simulation; Crystallography, X-Ray; gamma-Aminobutyric Acid; Humans; Hydrogen Bonding; Imidazoles; Mice; Models, Molecular; Molecular Structure; Pentylenetetrazole; Seizures; Structure-Activity Relationship

2008
Relationship between brain tissue partitioning and microemulsion retention factors of CNS drugs.
    Journal of medicinal chemistry, 2009, Mar-26, Volume: 52, Issue:6

    Topics: Brain; Central Nervous System; Chromatography, Liquid; Emulsions; Mass Spectrometry

2009
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Synthesis, in vivo evaluation, and molecular modeling studies of new pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide derivatives. Identification of a bifunctional hydrogen bond area related to the inverse agonism.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Cattle; Drug Inverse Agonism; GABA-A Receptor Agonists; Hydrogen Bonding; Male; Mice; Models, Molecular; Motor Activity; Rats; Rats, Wistar; Receptors, GABA-A; Structure-Activity Relationship; Triazines

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
New fluoro derivatives of the pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide system: evaluation of fluorine binding properties in the benzodiazepine site on γ-aminobutyrric acid type A (GABA(A)) receptor. Design, synthesis, biological, and molecular modeling
    Journal of medicinal chemistry, 2010, Nov-11, Volume: 53, Issue:21

    Topics: Animals; Anti-Anxiety Agents; Binding Sites; Cattle; Cerebral Cortex; Crystallography, X-Ray; Drug Design; Drug Inverse Agonism; In Vitro Techniques; Male; Mice; Models, Molecular; Molecular Structure; Pyrazoles; Radioligand Assay; Rats; Rats, Wistar; Receptors, GABA-A; Structure-Activity Relationship; Triazines

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
New insight into the central benzodiazepine receptor-ligand interactions: design, synthesis, biological evaluation, and molecular modeling of 3-substituted 6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and related compounds.
    Journal of medicinal chemistry, 2011, Aug-25, Volume: 54, Issue:16

    Topics: Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Cattle; Cerebral Cortex; Chlorides; Flumazenil; HEK293 Cells; Humans; Ligands; Male; Mice; Models, Molecular; Molecular Structure; Motor Activity; Protein Structure, Tertiary; Protein Subunits; Radioligand Assay; Receptors, GABA-A; Synaptosomes; Tritium; Xenopus laevis

2011
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Design, Synthesis, and Biological Evaluation of Imidazo[1,5-a]quinoline as Highly Potent Ligands of Central Benzodiazepine Receptors.
    Journal of medicinal chemistry, 2016, Apr-14, Volume: 59, Issue:7

    Topics: Amnesia; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Binding Sites; Brain; Cattle; Drug Design; Humans; Ischemia; Ligands; Male; Mice; Models, Molecular; Neuroprotective Agents; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Structure-Activity Relationship; Synaptosomes

2016
Design, synthesis and biological evaluation of 7-substituted 4-phenyl-6H-imidazo[1,5-a]thieno[3,2-f] [1,4]diazepines as safe anxiolytic agents.
    European journal of medicinal chemistry, 2020, Aug-15, Volume: 200

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Binding Sites; Drug Design; Locomotion; Memory Disorders; Mice; Molecular Docking Simulation; Rats; Receptors, GABA-A

2020
Evidence for more than two central benzodiazepine receptors in rat spinal cord.
    European journal of pharmacology, 1992, Apr-07, Volume: 214, Issue:1

    Topics: Animals; Binding, Competitive; Diazepam; Flumazenil; Flunitrazepam; Rats; Receptors, GABA-A; RNA, Messenger; Spinal Cord

1992
Relationship between benzodiazepine receptor occupancy and potentiation of gamma-aminobutyric acid-stimulated chloride flux in vitro of four ligands of differing intrinsic efficacies.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Animals; Benzodiazepinones; Cell Membrane; Cerebral Cortex; Chlorides; Diazepam; Drug Synergism; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Rats; Receptors, GABA-A; Triazolam

1992
Relationship between benzodiazepine receptor occupancy and functional effects in vivo of four ligands of differing intrinsic efficacies.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Administration, Oral; Animals; Benzodiazepinones; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Male; Mice; Mice, Inbred DBA; Motor Activity; Receptors, GABA-A; Seizures; Triazolam

1992
Effects of flumazenil on intravenous lidocaine-induced convulsions and anticonvulsant property of diazepam in rats.
    Anesthesia and analgesia, 1992, Volume: 75, Issue:1

    Topics: Animals; Anticonvulsants; Bicarbonates; Blood Pressure; Carbon Dioxide; Convulsants; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Heart Rate; Hydrogen-Ion Concentration; Infusions, Intravenous; Lidocaine; Male; Oxygen; Partial Pressure; Rats; Rats, Inbred Strains; Seizures

1992
Effects of central and peripheral type benzodiazepine ligands on thyrotropin and prolactin secretion.
    Neuropeptides, 1992, Volume: 21, Issue:3

    Topics: Animals; Benzodiazepinones; Carbolines; Clonazepam; Cold Temperature; Diazepam; Flumazenil; Hypothalamo-Hypophyseal System; Isoquinolines; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Secretory Rate; Thyrotropin; Thyrotropin-Releasing Hormone

1992
[Effects of agonists and antagonists of benzodiazepine, GABA and NMDA receptors, on caffeine-induced seizures in mice].
    Yakubutsu, seishin, kodo = Japanese journal of psychopharmacology, 1992, Volume: 12, Issue:4

    Topics: Animals; Baclofen; Benzodiazepines; Caffeine; Diazepam; Dizocilpine Maleate; Flumazenil; Male; Mice; Muscimol; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Receptors, Purinergic; Seizures

1992
MDL 26,479: a potential cognition enhancer with benzodiazepine inverse agonist-like properties.
    British journal of pharmacology, 1992, Volume: 107, Issue:1

    Topics: Animals; Behavior, Animal; Benzodiazepines; Binding Sites; Carbolines; Cognition; Convulsants; Diazepam; Flumazenil; Hemicholinium 3; Hippocampus; In Vitro Techniques; Male; Mice; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Triazoles

1992
Tonic inhibition of striatal dopamine transmission: effects of benzodiazepine and GABAA receptor antagonists on extracellular dopamine levels.
    Brain research, 1992, Dec-18, Volume: 599, Issue:1

    Topics: Animals; Corpus Striatum; Dialysis; Diazepam; Dopamine; Dose-Response Relationship, Drug; Extracellular Space; Flumazenil; GABA-A Receptor Antagonists; Male; Pyridazines; Rats; Rats, Sprague-Dawley; Synaptic Transmission

1992
Effect of a new anxiolytic, DN-2327, on learning and memory in rats.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Buspirone; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Isoindoles; Learning; Male; Memory; Naphthyridines; Rats; Rats, Inbred Strains; Spiro Compounds

1992
Like diazepam, CL 218,872, a selective ligand for the benzodiazepine omega 1 receptor subtype, impairs place learning in the Morris water maze.
    Psychopharmacology, 1992, Volume: 107, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Flumazenil; Learning; Male; Memory; Motor Activity; Pyridazines; Rats; Receptors, GABA-A

1992
Withdrawal precipitation by benzodiazepine receptor antagonists in dogs chronically treated with diazepam or the novel anxiolytic and anticonvulsant beta-carboline abecarnil.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Carbolines; Diazepam; Dogs; Female; Flumazenil; GABA-A Receptor Antagonists; Oxazepam; Substance Withdrawal Syndrome

1992
Anticonflict action of tandospirone in a modified Geller-Seifter conflict test in rats.
    Japanese journal of pharmacology, 1992, Volume: 58, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Behavior, Animal; Conditioning, Operant; Conflict, Psychological; Diazepam; Electroshock; Flumazenil; Isoindoles; Male; Piperazines; Pyrimidines; Rats; Rats, Inbred Strains; Tetrahydronaphthalenes

1992
Substituted imidazo[1,2-b]pyridazines. New compounds with activity at central and peripheral benzodiazepine receptors.
    Biochemical pharmacology, 1992, Oct-20, Volume: 44, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Mice; Prosencephalon; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1992
Effects of benzodiazepine receptor ligands with different intrinsic activities on seizures induced by inhibition of GAD.
    Epilepsy research. Supplement, 1992, Volume: 8

    Topics: Animals; Anti-Anxiety Agents; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hippocampus; Isoniazid; Male; Mice; Mice, Inbred Strains; Pyrazoles; Reaction Time; Receptors, GABA-A; Seizures

1992
[Extreme duration of action of diazepam as a cause of respiratory insufficiency in a female geriatric patient].
    Anasthesiologie, Intensivmedizin, Notfallmedizin, Schmerztherapie : AINS, 1992, Volume: 27, Issue:2

    Topics: Aged; Diazepam; Female; Flumazenil; Humans; Postoperative Complications; Respiratory Insufficiency; Time Factors; Unconsciousness

1992
Benzodiazepine-induced changes in biomembrane fluidity.
    Biochemical Society transactions, 1992, Volume: 20, Issue:2

    Topics: Chlordiazepoxide; Diazepam; Egg Yolk; Flumazenil; Lipid Bilayers; Liposomes; Membrane Fluidity; Models, Biological; Phosphatidylcholines; Spectrometry, Fluorescence

1992
Pharmacological dissociation between the spatial learning deficits produced by morphine and diazepam.
    Psychopharmacology, 1992, Volume: 108, Issue:1-2

    Topics: Animals; Cues; Diazepam; Flumazenil; Learning; Male; Morphine; Naloxone; Rats; Space Perception

1992
Quantitative electroencephalography for measurement of central nervous system responses to diazepam and the benzodiazepine antagonist, flumazenil, in isoflurane-anaesthetized dogs.
    Journal of veterinary pharmacology and therapeutics, 1992, Volume: 15, Issue:3

    Topics: Anesthesia, Inhalation; Animals; Brain; Diazepam; Dogs; Electroencephalography; Female; Flumazenil; Hemodynamics; Isoflurane

1992
Seizures after flumazenil administration in a case of combined benzodiazepine and tricyclic antidepressant overdose.
    Critical care medicine, 1992, Volume: 20, Issue:12

    Topics: Adult; Clonazepam; Diazepam; Drug Overdose; Epilepsy, Tonic-Clonic; Female; Flumazenil; Humans; Imipramine; Poisoning

1992
Tolerance, cross-tolerance and withdrawal in rats made dependent on diazepam.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: Animals; Chlordiazepoxide; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Drug Tolerance; Flumazenil; Male; Midazolam; Pentylenetetrazole; Rats; Substance Withdrawal Syndrome; Substance-Related Disorders

1992
The effects of centrally acting drugs on the EEG correlates of meditation.
    Biofeedback and self-regulation, 1992, Volume: 17, Issue:3

    Topics: Adult; Computers; Diazepam; Electroencephalography; Flumazenil; Humans; Male; Naloxone; Relaxation Therapy

1992
Oral self-administration of triazolam, diazepam and ethanol in the baboon: drug reinforcement and benzodiazepine physical dependence.
    Psychopharmacology, 1992, Volume: 108, Issue:3

    Topics: Animals; Conditioning, Operant; Diazepam; Drinking Behavior; Ethanol; Flumazenil; Food; Half-Life; Male; Papio; Reinforcement Schedule; Reward; Self Administration; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1992
Effects of nitrendipine, chlordiazepoxide, flumazenil and baclofen on the increased anxiety resulting from alcohol withdrawal.
    Progress in neuro-psychopharmacology & biological psychiatry, 1992, Volume: 16, Issue:1

    Topics: Animals; Anxiety; Baclofen; Chlordiazepoxide; Diazepam; Ethanol; Flumazenil; Interpersonal Relations; Male; Nitrendipine; Rats; Substance Withdrawal Syndrome; Tremor

1992
Locomotor responses to benzodiazepines, barbiturates and ethanol in diazepam-sensitive (DS) and -resistant (DR) mice.
    Psychopharmacology, 1992, Volume: 107, Issue:1

    Topics: Analysis of Variance; Animals; Diazepam; Dose-Response Relationship, Drug; Ethanol; Female; Flumazenil; Flunitrazepam; Male; Mice; Motor Activity; Pentobarbital; Phenobarbital

1992
Repeated anticonvulsant testing: contingent tolerance to diazepam and clobazam in kindled rats.
    Epilepsy research, 1992, Volume: 11, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Clobazam; Diazepam; Drug Tolerance; Flumazenil; Kindling, Neurologic; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Seizures

1992
Flumazenil does not antagonize halothane, thiamylal or propofol anaesthesia in rats.
    British journal of anaesthesia, 1992, Volume: 69, Issue:1

    Topics: Anesthesia, Inhalation; Anesthesia, Intravenous; Animals; Behavior, Animal; Diazepam; Drug Interactions; Electroencephalography; Flumazenil; Halothane; Male; Propofol; Rats; Rats, Inbred Strains; Sleep; Thiamylal

1992
Elevated brain concentrations of 1,4-benzodiazepines in fulminant hepatic failure.
    The New England journal of medicine, 1991, Aug-15, Volume: 325, Issue:7

    Topics: Adult; Aged; Benzodiazepines; Brain Chemistry; Chromatography; Diazepam; Flumazenil; Frontal Lobe; gamma-Aminobutyric Acid; Hepatic Encephalopathy; Humans; Mass Spectrometry; Middle Aged; Nordazepam; Receptors, GABA-A; Synaptic Transmission

1991
Action of diazepam on the voltage-dependent Na+ current. Comparison with the effects of phenytoin, carbamazepine, lidocaine and flumazenil.
    Brain research, 1991, May-10, Volume: 548, Issue:1-2

    Topics: Action Potentials; Animals; Carbamazepine; Cell Line; Cells, Cultured; Diazepam; Embryo, Mammalian; Flumazenil; Kinetics; Lidocaine; Mice; Neuroblastoma; Neurons; Phenytoin; Sodium Channels; Spinal Cord

1991
Benzodiazepine receptor ligands and sexual behavior in the male rat: the role of GABAergic mechanisms.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 38, Issue:4

    Topics: Animals; Bicuculline; Carbolines; Chlordiazepoxide; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Male; Motor Activity; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sexual Behavior, Animal

1991
SPECT imaging of the benzodiazepine receptor: feasibility of in vivo potency measurements from stepwise displacement curves.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1991, Volume: 32, Issue:9

    Topics: Alprazolam; Animals; Benzodiazepines; Brain; Brain Chemistry; Clonazepam; Diazepam; Female; Flumazenil; Injections, Intravenous; Macaca mulatta; Male; Papio; Receptors, GABA-A; Tomography, Emission-Computed, Single-Photon

1991
In vivo bidirectional modulatory effect of benzodiazepine receptor ligands on GABAergic transmission evaluated by positron emission tomography in non-human primates.
    Brain research, 1991, Aug-23, Volume: 557, Issue:1-2

    Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Carbolines; Cerebral Cortex; Diazepam; Electroencephalography; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Papio; Pentylenetetrazole; Receptors, GABA-A; Seizures; Synaptic Transmission; Tomography, Emission-Computed

1991
Behavioral effects of benzodiazepine ligands in non-dependent, diazepam-dependent and diazepam-withdrawn baboons.
    European journal of pharmacology, 1991, Sep-17, Volume: 202, Issue:2

    Topics: Animals; Behavior, Animal; Benzodiazepines; Carbolines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Ligands; Male; Midazolam; Papio; Receptors, GABA-A; Social Behavior; Substance Withdrawal Syndrome; Substance-Related Disorders

1991
Modulation of noise-potentiated acoustic startle via the benzodiazepine--gamma-aminobutyric acid receptor complex.
    Behavioral neuroscience, 1991, Volume: 105, Issue:5

    Topics: Acoustic Stimulation; Animals; Auditory Perception; Benzodiazepinones; Brain; Convulsants; Diazepam; Flumazenil; GABA-A Receptor Antagonists; Male; Neurons; Rats; Receptors, GABA-A; Reflex, Startle

1991
Flumazenil as an anti-epileptic agent.
    Lancet (London, England), 1991, Mar-23, Volume: 337, Issue:8743

    Topics: Diazepam; Drug Evaluation; Epilepsy; Flumazenil; Humans; Time Factors

1991
Pharmacologic profile of a new anxiolytic, DN-2327: effect of Ro15-1788 and interaction with diazepam in rodents.
    Psychopharmacology, 1991, Volume: 103, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Isoindoles; Male; Mice; Mice, Inbred ICR; Muscle Relaxation; Naphthyridines; Pentobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Spiro Compounds

1991
Involvement of the GABAA/benzodiazepine chloride ionophore receptor complex in the 5,7-DHT Induced anticonflict effect.
    Life sciences, 1991, Volume: 49, Issue:2

    Topics: 5,7-Dihydroxytryptamine; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Bicuculline; Diazepam; Drinking Behavior; Electroshock; Flumazenil; Hippocampus; Injections, Intraventricular; Limbic System; Male; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin

1991
Evidence for a role for dopamine in the diazepam locomotor stimulating effect.
    Psychopharmacology, 1991, Volume: 104, Issue:1

    Topics: alpha-Methyltyrosine; Animals; Benzazepines; Diazepam; Dopamine; Flumazenil; Haloperidol; Male; Methyltyrosines; Mice; Motor Activity; Spiperone; Stimulation, Chemical; Tyrosine 3-Monooxygenase

1991
[Behavioral pharmacological and electroencephalographic effects of the 5-HT1A partial agonist ipsapirone].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1991, Volume: 98, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Buspirone; Diazepam; Drug Synergism; Electroencephalography; Flumazenil; Male; Mice; Motor Activity; Pyrimidines; Rabbits; Rats; Rats, Inbred Strains; Serotonin

1991
The discriminative stimulus effects of diazepam in rats at two training doses.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Male; Morphine; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Triazolam

1991
Central-type benzodiazepines inhibit release of alpha-melanocyte-stimulating hormone from the rat hypothalamus.
    Neuroscience, 1991, Volume: 42, Issue:2

    Topics: Animals; Anti-Anxiety Agents; beta-Endorphin; Clonazepam; Diazepam; Flumazenil; GABA Antagonists; Hypothalamus; In Vitro Techniques; Male; Melanocyte-Stimulating Hormones; Perfusion; Pituitary Gland; Potassium Chloride; Pro-Opiomelanocortin; Pyridazines; Radioimmunoassay; Rats; Rats, Inbred Strains

1991
Behavioral effects of U-78875, a quinoxalinone anxiolytic with potent benzodiazepine antagonist activity.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Behavior, Animal; Diazepam; Electroencephalography; Flumazenil; Injections, Intraperitoneal; Male; Motor Activity; Oxadiazoles; Quinoxalines; Rats; Rats, Inbred F344

1991
Chronic administration of and dependence on halazepam, diazepam, and nordiazepam in the dog.
    Drug and alcohol dependence, 1991, Volume: 28, Issue:3

    Topics: Administration, Oral; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Dogs; Dose-Response Relationship, Drug; Flumazenil; Neurologic Examination; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders

1991
Effects of DN-2327, a new anxiolytic, diazepam and buspirone on exploratory activity of the rat in an elevated plus-maze.
    Psychopharmacology, 1991, Volume: 104, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Buspirone; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Exploratory Behavior; Flumazenil; Isoindoles; Male; Naphthyridines; Pentylenetetrazole; Rats; Rats, Inbred Strains; Spiro Compounds; Yohimbine

1991
The negative inotropic effect of diazepam in rat right ventricular strips.
    The Journal of pharmacy and pharmacology, 1991, Volume: 43, Issue:12

    Topics: Animals; Depression, Chemical; Diazepam; Electric Stimulation; Female; Flumazenil; Heart Ventricles; In Vitro Techniques; Isoquinolines; Male; Myocardial Contraction; Rats; Rats, Inbred Strains; Receptors, GABA-A

1991
Psychological stress increases dopamine turnover selectively in mesoprefrontal dopamine neurons of rats: reversal by diazepam.
    Brain research, 1991, Aug-23, Volume: 557, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Catecholamines; Corticosterone; Diazepam; Dopamine; Electroshock; Flumazenil; Frontal Lobe; Homovanillic Acid; Indoles; Male; Nerve Endings; Neurons; Rats; Rats, Inbred Strains; Stress, Psychological; Tegmentum Mesencephali

1991
Flumazenil for the reversal of refractory benzodiazepine-induced shock.
    Journal of toxicology. Clinical toxicology, 1991, Volume: 29, Issue:4

    Topics: Aged; Cardiovascular System; Central Nervous System; Diazepam; Female; Flumazenil; Humans; Respiration; Shock

1991
[The use of flumazenil to antagonize the effect of diazepam after bronchoscopy].
    Minerva anestesiologica, 1991, Volume: 57, Issue:9

    Topics: Adult; Bronchoscopy; Diazepam; Female; Flumazenil; Humans; Male; Middle Aged

1991
Effects of a benzodiazepine antagonist, Ro 15-1788, on hippocampal field potentials in freely moving rats.
    The Tohoku journal of experimental medicine, 1991, Volume: 165, Issue:4

    Topics: Animals; Depression, Chemical; Diazepam; Evoked Potentials; Flumazenil; Hippocampus; Male; Rats; Rats, Inbred Strains

1991
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
    Molecular pharmacology, 1991, Volume: 39, Issue:3

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes

1991
The contribution of endogenous benzodiazepine receptor ligands to the pathogenesis of hepatic encephalopathy.
    Synapse (New York, N.Y.), 1991, Volume: 7, Issue:2

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chromatography, High Pressure Liquid; Diazepam; Flumazenil; Hepatic Encephalopathy; Kinetics; Ligands; Male; Mass Spectrometry; Muscimol; Peripheral Nerves; Rabbits; Radioligand Assay; Receptors, GABA-A; Sulfur Radioisotopes

1991
[Accidental diazepam overdose in a 12-month-old infant. Therapy using flumazenil].
    Anasthesiologie, Intensivmedizin, Notfallmedizin, Schmerztherapie : AINS, 1991, Volume: 26, Issue:3

    Topics: Accidents; Diazepam; Flumazenil; Humans; Infant

1991
Effects of diazepam and Ro 15-1788 on duodenal bicarbonate secretion in the rat.
    Gastroenterology, 1991, Volume: 101, Issue:4

    Topics: Animals; Bicarbonates; Diazepam; Duodenum; Flumazenil; Intestinal Mucosa; Intestinal Secretions; Male; Rana catesbeiana; Rats; Rats, Inbred Strains; Stimulation, Chemical; Trimipramine; Vagus Nerve

1991
Antagonism by propyl-beta-carboline-3-carboxylate of passive avoidance impairment induced by diazepam.
    European journal of pharmacology, 1991, May-30, Volume: 198, Issue:1

    Topics: Animals; Avoidance Learning; Carbolines; Convulsants; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Learning; Male; Memory; Mice; Mice, Inbred Strains

1991
Effects of forced shaking stress at low temperature on pentobarbital-induced sleeping in mice.
    General pharmacology, 1991, Volume: 22, Issue:4

    Topics: Animals; Cold Temperature; Diazepam; Drug Resistance; Flumazenil; Male; Mice; Naloxone; Nociceptors; Pentobarbital; Sleep; Stress, Physiological

1991
A comparison of the physical dependence inducing properties of flunitrazepam and diazepam.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:2

    Topics: Animals; Biotransformation; Blood Proteins; Brain Chemistry; Diazepam; Dogs; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Protein Binding; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1991
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
    Psychopharmacology, 1990, Volume: 102, Issue:4

    Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem

1990
Behavioral neurobiology of inverse agonist FG 7142 induced anxiety syndrome in rats.
    Progress in neuro-psychopharmacology & biological psychiatry, 1990, Volume: 14, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Avoidance Learning; Carbolines; Diazepam; Exploratory Behavior; Flumazenil; Grooming; Male; Motor Activity; Rats; Rats, Inbred Strains; Stereotyped Behavior

1990
Reduction of reticulata neuronal activity by zolpidem and alpidem, two imidazopyridines with high affinity for type I benzodiazepine receptors.
    European journal of pharmacology, 1990, Apr-25, Volume: 179, Issue:3

    Topics: Action Potentials; Animals; Anti-Anxiety Agents; Diazepam; Flumazenil; Hypnotics and Sedatives; Imidazoles; Male; Neurons; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reticular Formation; Zolpidem

1990
Differential interactions of Ro 15-4513 with benzodiazepines, ethanol and pentobarbital.
    European journal of pharmacology, 1990, May-16, Volume: 180, Issue:2-3

    Topics: Anesthesia; Animals; Anti-Anxiety Agents; Azides; Behavior, Animal; Benzodiazepines; Diazepam; Drug Interactions; Ethanol; Female; Flumazenil; Male; Muscle Contraction; Muscles; Pentobarbital; Rats; Rats, Inbred Strains; Urethane; Vocalization, Animal

1990
Benzodiazepine receptor ligand influences on acquisition: suggestion of an endogenous modulatory mechanism mediated by benzodiazepine receptors.
    Behavioral and neural biology, 1990, Volume: 54, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Arousal; Avoidance Learning; Benzodiazepinones; Brain; Carbolines; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Flumazenil; Habituation, Psychophysiologic; Memory; Mental Recall; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Retention, Psychology

1990
A theory of benzodiazepine dependence that can explain whether flumazenil will enhance or reverse the phenomena.
    Psychopharmacology, 1990, Volume: 101, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Flumazenil; Male; Rats; Substance Withdrawal Syndrome; Substance-Related Disorders

1990
Benzodiazepines and synaptic processing in the spatial domain within the cat's primary somatosensory cortex.
    Canadian journal of physiology and pharmacology, 1990, Volume: 68, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Bicuculline; Cats; Diazepam; Electric Stimulation; Electrophysiology; Female; Flumazenil; Fluphenazine; gamma-Aminobutyric Acid; Male; Midazolam; Physical Stimulation; Somatosensory Cortex; Space Perception; Synapses

1990
Effect of serotoninergic drugs on stress-induced hyperthermia (SIH) in mice.
    Journal of neural transmission. General section, 1990, Volume: 82, Issue:3

    Topics: 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Body Temperature Regulation; Buspirone; Diazepam; Ergolines; Fenclonine; Fever; Flumazenil; Imidazoles; Male; Mice; Ondansetron; Piperazines; Piperidines; Ritanserin; Serotonin; Serotonin Antagonists; Stress, Psychological; Tetrahydronaphthalenes

1990
Increased sensitivity to benzodiazepine antagonists in rats following chronic treatment with a low dose of diazepam.
    Psychopharmacology, 1990, Volume: 102, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Food; Male; Pyrazoles; Rats; Rats, Inbred Strains; Reinforcement Schedule; Reinforcement, Psychology

1990
Relaxant effect of benzodiazepines on uterine rings isolated from estrogen-treated rats.
    European journal of pharmacology, 1990, Aug-28, Volume: 185, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Bicuculline; Clonazepam; Convulsants; Diazepam; Estradiol; Estrogens; Female; Flumazenil; In Vitro Techniques; Isoquinolines; Muscle, Smooth; Potassium Chloride; Propranolol; Rats; Rats, Inbred Strains; Uterine Contraction

1990
Which agent and how to deliver it? A review of benzodiazepine sedation and its reversal in endoscopy.
    Scandinavian journal of gastroenterology. Supplement, 1990, Volume: 179

    Topics: Analgesics, Opioid; Anti-Anxiety Agents; Conscious Sedation; Diazepam; Endoscopy, Gastrointestinal; Flumazenil; Humans; Midazolam

1990
Preferential decrease in dopamine utilization in prefrontal cortex by zopiclone, diazepam and zolpidem in unstressed rats.
    The Journal of pharmacy and pharmacology, 1990, Volume: 42, Issue:8

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Azabicyclo Compounds; Cerebral Cortex; Corpus Striatum; Diazepam; Dopamine; Flumazenil; Male; Piperazines; Pyridines; Rats; Rats, Inbred Strains; Stress, Physiological; Zolpidem

1990
Benzodiazepine-induced antagonism of opioid antinociception may be abolished by spinalization or blockade of the benzodiazepine receptor.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:3

    Topics: Analgesics; Animals; Anti-Anxiety Agents; Diazepam; Flumazenil; Male; Mice; Midazolam; Morphine; Narcotics; Nordazepam; Psychomotor Performance; Reaction Time; Receptors, GABA-A; Receptors, Opioid; Skin Temperature; Spinal Cord

1990
Cardiorespiratory effects of antagonism of diazepam sedation with flumazenil in patients with cardiac disease.
    Anesthesia and analgesia, 1991, Volume: 72, Issue:2

    Topics: Aged; Cardiac Catheterization; Coronary Angiography; Coronary Disease; Diazepam; Female; Flumazenil; Heart; Heart Diseases; Heart Valve Diseases; Hemodynamics; Humans; Hypnotics and Sedatives; Male; Middle Aged; Respiratory System

1991
Flumazenil therapy in benzodiazepine self-poisoning.
    Irish medical journal, 1991, Volume: 84, Issue:1

    Topics: Adult; Diazepam; Female; Flumazenil; Humans; Lorazepam; Middle Aged; Poisoning

1991
Flumazenil and hypoxic ventilatory response.
    Anesthesia and analgesia, 1990, Volume: 70, Issue:1

    Topics: Diazepam; Flumazenil; Humans; Hypoxia; Respiration

1990
Diazepam-binding inhibitor: a neuropeptide and/or an acyl-CoA ester binding protein?
    The Biochemical journal, 1990, Feb-01, Volume: 265, Issue:3

    Topics: Acyl Coenzyme A; Adrenal Cortex; Amino Acid Sequence; Animals; Benzodiazepinones; Brain; Carboxylic Acids; Carrier Proteins; Cattle; Diazepam; Diazepam Binding Inhibitor; Esters; Flumazenil; Liver; Molecular Sequence Data; Nerve Tissue Proteins; Neuropeptides; Peptide Fragments; Rats

1990
3-((+-)-2-carboxypiperazin-4-yl)propyl-1-phosphonic acid (CPP) and phencyclidine produce a deficit of passive avoidance retention in rats.
    European journal of pharmacology, 1990, Jan-10, Volume: 175, Issue:2

    Topics: Animals; Anticonvulsants; Avoidance Learning; Behavior, Animal; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Latency Period, Psychological; Male; Phencyclidine; Piperazines; Rats; Rats, Inbred Strains

1990
Pharmacological manipulation of anxiety and male rat sexual behavior.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 35, Issue:1

    Topics: Animals; Anxiety; Carbolines; Copulation; Diazepam; Flumazenil; Male; Psychomotor Performance; Rats; Rats, Inbred Strains

1990
Methyl beta-carboline-3-carboxylate enhances performance in a multiple-trial learning task in mice.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 35, Issue:2

    Topics: Animals; Benzodiazepines; Carbolines; Diazepam; Drug Synergism; Flumazenil; Learning; Male; Mice; Retention, Psychology

1990
Diazepam and Ro 15-1788 increase absence epilepsy in WAG/Rij rats chronically exposed to diazepam.
    European journal of pharmacology, 1990, Mar-13, Volume: 178, Issue:1

    Topics: Animals; Diazepam; Electroencephalography; Epilepsy; Flumazenil; Hypnotics and Sedatives; Male; Rats; Rats, Inbred Strains

1990
Enhancing effects of Ro 15-1788 on straw-climbing behavior as measured with the straw-suspension method: reversal by diazepam.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:1

    Topics: Animals; Anxiety; Diazepam; Drug Interactions; Flumazenil; Male; Motor Activity; Rats; Rats, Inbred Strains

1990
Blockade of hoarding in rats by diazepam: an analysis of the anxiety and object value hypotheses of hoarding.
    Psychopharmacology, 1990, Volume: 101, Issue:2

    Topics: Animals; Anxiety; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Eating; Female; Flumazenil; Food Deprivation; Learning; Male; Rats

1990
[Buspirone: correlation of its anxiolytic and electroencephalographic effects].
    Biulleten' eksperimental'noi biologii i meditsiny, 1990, Volume: 109, Issue:3

    Topics: Animals; Buspirone; Diazepam; Dose-Response Relationship, Drug; Electroencephalography; Flumazenil; Fourier Analysis; Male; Rats; Somatosensory Cortex; Time Factors

1990
[The effect of RO15-1788 on the interaction between pancuronium and diazepam].
    Masui. The Japanese journal of anesthesiology, 1990, Volume: 39, Issue:6

    Topics: Animals; Diazepam; Drug Interactions; Flumazenil; Male; Neuromuscular Junction; Pancuronium; Rats; Rats, Inbred Strains

1990
Anticonvulsive properties of F1933 (dulozafone) on kindled seizures in the rat.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: Acetanilides; Amygdala; Animals; Anticonvulsants; Diazepam; Electric Stimulation; Flumazenil; Kindling, Neurologic; Male; Rats; Rats, Inbred Strains; Seizures

1990
Early developmental exposure to benzodiazepine ligands alters brain 31P-NMR spectra in young adult rats.
    Brain research, 1990, Jan-01, Volume: 506, Issue:1

    Topics: Animals; Brain; Diazepam; Female; Flumazenil; Hydrogen-Ion Concentration; Magnetic Resonance Spectroscopy; Phosphocreatine; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Receptors, GABA-A

1990
beta-CCM inhibits muricide induced by olfactory bulbectomy in rats.
    Japanese journal of pharmacology, 1990, Volume: 52, Issue:3

    Topics: Aggression; Animals; Brain; Carbolines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Injections, Intravenous; Male; Mice; Motor Activity; Muscle Relaxants, Central; Olfactory Bulb; Phenoxybenzamine; Postural Balance; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Behavioral analysis of the effects of benzodiazepine receptor ligands in the conditioned burying paradigm.
    Behavioural brain research, 1990, Apr-16, Volume: 38, Issue:1

    Topics: Animals; Arousal; Benzodiazepinones; Brain; Carbolines; Conditioning, Classical; Diazepam; Dose-Response Relationship, Drug; Electroshock; Fear; Flumazenil; Grooming; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stereotyped Behavior

1990
Benzodiazepine receptors modulate 5-hydroxytryptamine neurotransmission in the rat hippocampus: in vivo electrophysiological evidence.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: Animals; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Hippocampus; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synaptic Transmission

1990
Proconflict effect of ACTH1-24: interaction with benzodiazepines.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:3

    Topics: Adrenocorticotropic Hormone; alpha-MSH; Animals; Anxiety; Conflict, Psychological; Cosyntropin; Diazepam; Electroshock; Flumazenil; Injections, Intraventricular; Male; Peptide Fragments; Rats; Rats, Inbred Strains; Stress, Physiological

1990
Enkephalin biosynthesis and release in mouse striatum are inhibited by GABA receptor stimulation: compared changes in preproenkephalin mRNA and Tyr-Gly-Gly levels.
    Brain research. Molecular brain research, 1990, Volume: 8, Issue:3

    Topics: Aminooxyacetic Acid; Animals; Corpus Striatum; Diazepam; Enkephalins; Flumazenil; Kinetics; Leucine; Male; Mice; Muscimol; Oligopeptides; Protein Precursors; Receptors, GABA-A; RNA, Messenger

1990
The benzodiazepine receptor inverse agonist DMCM decreases serotonergic transmission in rat hippocampus: an in vivo electrophysiological study.
    Synapse (New York, N.Y.), 1990, Volume: 6, Issue:2

    Topics: Animals; Carbolines; Diazepam; Electrophysiology; Flumazenil; Hippocampus; Neural Pathways; Pargyline; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin; Synaptic Transmission

1990
Profound stress-induced alterations in flurazepam's antiseizure efficacy can be attenuated.
    Brain research, 1990, Jun-18, Volume: 520, Issue:1-2

    Topics: Animals; Carbolines; Clonazepam; Cold Temperature; Diazepam; Dose-Response Relationship, Drug; Electroshock; Flumazenil; Flurazepam; Male; Mice; Mice, Inbred Strains; Midazolam; Seizures; Stress, Psychological

1990
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines

1990
Differential actions of RO 15-1788 and diazepam on poikilothermia, motor impairment and sleep produced by ethanol.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Animals; Body Temperature; Body Temperature Regulation; Diazepam; Drug Interactions; Ethanol; Flumazenil; Injections, Intraperitoneal; Male; Psychomotor Performance; Rats; Rats, Inbred Strains; Sleep

1990
[The risks of diazepam in newborn infants].
    Nederlands tijdschrift voor geneeskunde, 1990, Oct-27, Volume: 134, Issue:43

    Topics: Diazepam; Flumazenil; Humans; Infant, Newborn; Respiratory Insufficiency

1990
Benzodiazepine withdrawal syndrome after a benzodiazepine antagonist.
    Critical care medicine, 1990, Volume: 18, Issue:12

    Topics: Adolescent; Akathisia, Drug-Induced; Diazepam; Drug Overdose; Flumazenil; Humans; Injections, Intravenous; Intubation, Gastrointestinal; Lorazepam; Male; Psychomotor Agitation; Substance Withdrawal Syndrome; Therapeutic Irrigation; Thiopental

1990
[Antagonism of diazepam-induced sedative effects by flumazenil in patients after surgery under lumbar spinal or epidural anesthesia].
    Masui. The Japanese journal of anesthesiology, 1990, Volume: 39, Issue:9

    Topics: Adult; Aged; Anesthesia Recovery Period; Anesthesia, Epidural; Anesthesia, Spinal; Diazepam; Female; Flumazenil; Humans; Male; Middle Aged

1990
[EEG analysis of the effectiveness of the benzodiazepine antagonist RO 15-1788 after diazepam sedation].
    Masui. The Japanese journal of anesthesiology, 1990, Volume: 39, Issue:9

    Topics: Adult; Diazepam; Electroencephalography; Evaluation Studies as Topic; Flumazenil; Humans; Male

1990
[Clinical investigation of flumazenil in reversing the respiratory effects of diazepam].
    Masui. The Japanese journal of anesthesiology, 1990, Volume: 39, Issue:10

    Topics: Aged; Diazepam; Female; Flumazenil; Humans; Male; Middle Aged; Respiration

1990
Pharmacological inhibition of forskolin-stimulated adenylate cyclase activity in rat brain by melatonin, its analogs, and diazepam.
    Biochemical pharmacology, 1990, Dec-15, Volume: 40, Issue:12

    Topics: Adenylyl Cyclases; Animals; Benzodiazepinones; Brain; Brain Mapping; Cell Membrane; Colforsin; Corpus Striatum; Diazepam; Dose-Response Relationship, Drug; Enzyme Activation; Flumazenil; In Vitro Techniques; Male; Melatonin; Rats; Rats, Inbred Strains

1990
[Flumazenil: possible suppression of the antipsychotic effect of diazepam in anesthesia with ketamine].
    Minerva anestesiologica, 1990, Volume: 56, Issue:9

    Topics: Adult; Diazepam; Female; Flumazenil; Humans; Ketamine; Male; Middle Aged; Random Allocation

1990
Rat pup ultrasonic isolation calls: possible mediation by the benzodiazepine receptor complex.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:5

    Topics: Animals; Benzodiazepinones; Chlorides; Diazepam; Flumazenil; Ion Channels; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sex Factors; Temperature; Vocalization, Animal

1986
The effect of diazepam and Ro 15-1788 on extracellular ascorbic acid, DOPAC and 5-HIAA in the striatum of anaesthetized and conscious freely moving rats, as measured by differential pulse voltammetry.
    Neuroscience research, 1987, Volume: 4, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Ascorbic Acid; Corpus Striatum; Diazepam; Electrochemistry; Extracellular Space; Flumazenil; Hydroxyindoleacetic Acid; Male; Rats; Rats, Inbred Strains

1987
Partial agonists of the benzodiazepine receptor: from animal data to results in patients.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Affinity Labels; Allosteric Site; Animals; Azides; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Chlorides; Clonazepam; Diazepam; Drug Interactions; Ethanol; Flumazenil; Flurazepam; Humans; Ion Channels; Ligands; Models, Neurological; Neurons; Receptors, GABA-A

1988
The effect of diazepam on ventricular automaticity induced by a local injury. Evidence of involvement of "peripheral type" benzodiazepine receptors.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Diazepam; Diltiazem; Dose-Response Relationship, Drug; Female; Flumazenil; Heart Ventricles; Isoquinolines; Male; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Ventricular Function

1989
Diminution by benzodiazepines of the chronotropic responses to noradrenaline in rat isolated atria.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Colforsin; Cyclic AMP; Diazepam; Female; Flumazenil; Heart; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains

1989
Both systemic and local administration of benzodiazepine agonists inhibit the in vivo release of 5-HT from ventral hippocampus.
    Neuropharmacology, 1989, Volume: 28, Issue:10

    Topics: Animals; Benzodiazepines; Carbolines; Chromatography, High Pressure Liquid; Dialysis; Diazepam; Flumazenil; Flurazepam; Hippocampus; Hydroxyindoleacetic Acid; Ion Channels; Male; Muscimol; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin

1989
Effects of diazepam and flumazenil on sedation and hypoxic ventilatory response.
    Anesthesia and analgesia, 1989, Volume: 68, Issue:4

    Topics: Adult; Brain; Diazepam; Flumazenil; Humans; Hypnotics and Sedatives; Hypoxia; Respiration

1989
Sedation and reversal of sedation in intensive care.
    Acta anaesthesiologica Belgica, 1989, Volume: 40, Issue:1

    Topics: Adolescent; Adult; Aged; Anesthesia Recovery Period; Blood Pressure; Carbon Dioxide; Diazepam; Female; Flumazenil; Heart Rate; Humans; Male; Midazolam; Middle Aged; Postoperative Period; Preanesthetic Medication; Respiration

1989
Appetite-modulating drugs in dwarf goats, with special emphasis on benzodiazepine-induced hyperphagia and its antagonism by flumazenil and RO 15-3505.
    Journal of veterinary pharmacology and therapeutics, 1989, Volume: 12, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Appetite Regulation; Azepines; Benzodiazepines; Benzodiazepinones; Body Weight; Diazepam; Female; Flumazenil; Goats; Hyperphagia; Ivermectin; Male; Midazolam; Time Factors

1989
Ethanol and diazepam withdrawal convulsions are extensively codetermined in WSP and WSR mice.
    Life sciences, 1989, Volume: 44, Issue:26

    Topics: Animals; Diazepam; Ethanol; Flumazenil; Mice; Mice, Inbred Strains; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1989
Inhibition of high-affinity synaptosomal uptake of gamma-aminobutyric acid by a bicyclo-heptane derivative.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:3

    Topics: Animals; Anticonvulsants; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Camphanes; Carbolines; Cerebral Cortex; Diazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Synaptic Membranes; Synaptosomes

1989
Opposite effects of diazepam and beta-CCE on immobility and straw-climbing behavior of rats in a modified forced-swim test.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:1

    Topics: Animals; Carbolines; Diazepam; Flumazenil; Male; Motor Activity; Rats; Rats, Inbred Strains; Stress, Psychological; Swimming

1989
Benzodiazepines acting on ventral surface of medulla cause airway dilation.
    The American journal of physiology, 1989, Volume: 257, Issue:4 Pt 2

    Topics: Animals; Atropine; Blood Pressure; Cats; Diazepam; Female; Flumazenil; Lung; Male; Medulla Oblongata; Midazolam; Muscle Relaxation; Muscle, Smooth; Phrenic Nerve; Trachea

1989
Blockade by diazepam of conditioned fear-induced activation of rat mesoprefrontal dopamine neurons.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Brain Chemistry; Conditioning, Psychological; Corticosterone; Diazepam; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Fear; Flumazenil; Male; Rats; Rats, Inbred Strains; Stress, Psychological

1989
Relationship of agonist efficacy to changes in GABA sensitivity and anticonvulsant tolerance following chronic benzodiazepine ligand exposure.
    European journal of pharmacology, 1989, Nov-07, Volume: 170, Issue:3

    Topics: Animals; Anticonvulsants; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Bicuculline; Brain Chemistry; Diazepam; Drug Tolerance; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Male; Raphe Nuclei; Rats; Rats, Inbred Strains; Seizures

1989
Responses of substantia nigra pars reticulata neurons to benzodiazepine ligands after acute and prolonged diazepam exposure. I. Modulation of gamma-aminobutyric acid sensitivity.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:2

    Topics: Animals; Carbolines; Diazepam; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Ligands; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1989
Responses of substantia nigra pars reticulata neurons to benzodiazepine ligands after acute and prolonged diazepam exposure. II. Modulation of firing rate.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:2

    Topics: Animals; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1989
Role of the central benzodiazepine receptor system in behavioral habituation to novelty.
    Behavioral neuroscience, 1989, Volume: 103, Issue:1

    Topics: Animals; Carbolines; Diazepam; Exploratory Behavior; Flumazenil; Habituation, Psychophysiologic; Male; Rats; Reaction Time; Receptors, GABA-A

1989
Effects of peripheral benzodiazepines upon the O2 consumption of neuroblastoma cells.
    European journal of pharmacology, 1989, Feb-28, Volume: 161, Issue:2-3

    Topics: Animals; Benzodiazepines; Cells, Cultured; Clonazepam; Clone Cells; Diazepam; Flumazenil; Isoquinolines; Mice; Mitochondria; Neuroblastoma; Oxygen Consumption; Receptors, GABA-A

1989
Population differences in benzodiazepine sensitive male scent-induced analgesia in the deer mouse, Peromyscus maniculatus.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:3

    Topics: Analgesia; Animals; Central Nervous System; Diazepam; Flumazenil; Male; Mice; Naloxone; Olfactory Pathways; Peromyscus; Receptors, GABA-A; Receptors, Opioid

1989
GABA[A] receptor level changes in female hamster forebrain following in vivo estrogen progesterone and benzodiazepine treatment: a quantitative autoradiography analysis.
    Experimental brain research, 1989, Volume: 75, Issue:3

    Topics: Animals; Autoradiography; Benzodiazepines; Cricetinae; Diazepam; Estradiol; Female; Flumazenil; Frontal Lobe; Muscimol; Ovariectomy; Progesterone; Receptors, GABA-A

1989
Co-administration of Ro 15-1788 prevents diazepam-induced retardation of recovery of function.
    Brain research, 1989, May-15, Volume: 487, Issue:1

    Topics: Animals; Diazepam; Flumazenil; Functional Laterality; Male; Rats; Receptors, GABA-A; Somatosensory Cortex; Time Factors

1989
The relationship of benzodiazepine binding sites to the norepinephrine projection in the hypothalamus of the adult rat.
    Brain research, 1989, Jul-17, Volume: 492, Issue:1-2

    Topics: Animals; Diazepam; Flumazenil; Flunitrazepam; Hypothalamus; Norepinephrine; Rats; Receptors, GABA-A

1989
Type I and type II GABAA-benzodiazepine receptors produced in transfected cells.
    Science (New York, N.Y.), 1989, Sep-22, Volume: 245, Issue:4924

    Topics: Cell Line; Diazepam; Flumazenil; Flunitrazepam; Humans; Molecular Weight; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Transfection

1989
Modification of evoked hippocampal dentate inhibition by diazepam and three antagonists in urethane-anesthetized rats.
    Experimental neurology, 1989, Volume: 106, Issue:2

    Topics: Anesthesia; Animals; Diazepam; Evoked Potentials; Flumazenil; gamma-Aminobutyric Acid; Hippocampus; Isoquinolines; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synapses; Urethane

1989
Benzodiazepine receptor autoradiography in corpus striatum of rat after large frontal cortex lesions and chronic treatment with diazepam.
    Neuropharmacology, 1989, Volume: 28, Issue:9

    Topics: Animals; Autoradiography; Behavior, Animal; Cerebral Cortex; Corpus Striatum; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Male; Nucleus Accumbens; Rats; Receptors, GABA-A; Time Factors

1989
Early developmental exposure to benzodiazepine ligands alters brain levels of thiobarbituric acid-reactive products in young adult rats.
    Neurochemical research, 1989, Volume: 14, Issue:11

    Topics: Animals; Benzodiazepines; Brain; Clonazepam; Diazepam; Female; Flumazenil; Gestational Age; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Receptors, GABA-A; Thiobarbiturates

1989
Blockade of the development of analgesic tolerance to morphine by psychological stress through benzodiazepine receptor mediated mechanism.
    Japanese journal of pharmacology, 1989, Volume: 51, Issue:3

    Topics: Analgesia; Animals; Carbolines; Diazepam; Drug Tolerance; Flumazenil; Male; Mice; Morphine; Receptors, GABA-A; Stress, Psychological

1989
Efficacy of flumazenil in COPD patient with therapeutic diazepam levels.
    Lancet (London, England), 1989, Feb-18, Volume: 1, Issue:8634

    Topics: Aged; Diazepam; Drug Evaluation; Flumazenil; Humans; Lung Diseases, Obstructive; Male; Nordazepam

1989
Aminophylline reversal of diazepam intoxication.
    Lancet (London, England), 1989, Apr-22, Volume: 1, Issue:8643

    Topics: Aminophylline; Diazepam; Flumazenil; Half-Life; Humans; Male; Respiratory Insufficiency

1989
Physical dependence on diazepam in the dog: precipitation of different abstinence syndromes by the benzodiazepine receptor antagonists Ro 15-1788 and ZK 93426.
    British journal of pharmacology, 1989, Volume: 97, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Carbolines; Diazepam; Dogs; Female; Flumazenil; Nordazepam; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1989
Anticonvulsant and other effects of diazepam grow with time after a single treatment.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Anticonvulsants; Antipsychotic Agents; Blepharoptosis; Brain Chemistry; Catalepsy; Diazepam; Dopamine; Drug Interactions; Flumazenil; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Stress, Psychological; Time Factors

1989
Cerebral-activating (EEG) properties of two inverse agonists and of an antagonist at the benzodiazepine receptor in the rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Central Nervous System Stimulants; Chlorpromazine; Diazepam; Electroencephalography; Flumazenil; Imipramine; Male; Pentobarbital; Pyrazoles; Pyridazines; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
The effects of ondansetron (GR38032F) in rats and mice treated subchronically with diazepam.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 34, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Buspirone; Darkness; Diazepam; Flumazenil; Imidazoles; Light; Male; Mice; Mice, Inbred Strains; Ondansetron; Rats; Rats, Inbred Strains; Serotonin Antagonists; Social Behavior; Substance Withdrawal Syndrome; Time Factors

1989
Mouse lines selected for genetic differences in diazepam sensitivity.
    Psychopharmacology, 1987, Volume: 93, Issue:1

    Topics: Animals; Brain; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Mice; Mice, Inbred Strains; Motor Skills; Receptors, GABA-A; Selection, Genetic

1987
Inhibition of rat brain adenylate cyclase activity by benzodiazepine through the effects on Gi and catalytic proteins.
    Life sciences, 1988, Volume: 42, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Aluminum; Aluminum Chloride; Aluminum Compounds; Animals; Benzodiazepines; Brain; Chlorides; Diazepam; Flumazenil; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes

1988
Are the analgesic effects of social defeat mediated by benzodiazepine receptors?
    Physiology & behavior, 1987, Volume: 41, Issue:3

    Topics: Analgesia; Animals; Behavior, Animal; Carbolines; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Pyrazoles; Receptors, GABA-A; Social Behavior

1987
Heterogeneity of gamma-aminobutyric acid/benzodiazepine/beta-carboline receptor complex in rat spinal cord.
    Journal of neurochemistry, 1988, Volume: 50, Issue:4

    Topics: Animals; Bicuculline; Binding, Competitive; Carbolines; Cerebellum; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Male; Muscimol; Rats; Receptors, GABA-A; Spinal Cord; Synaptic Membranes

1988
Benzodiazepines and barbiturate potentiate the pre- and postsynaptic gamma-aminobutyric acid (GABA)A receptor-mediated response in the enteric nervous system of guinea pig small intestine.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Acetylcholine; Animals; Barbiturates; Benzodiazepines; Clonazepam; Diazepam; Female; Flumazenil; Guinea Pigs; Intestine, Small; Male; Muscimol; Pentobarbital; Potassium; Receptors, GABA-A

1988
Male scent-induced analgesia in the deer mouse, Peromyscus maniculatus: involvement of benzodiazepine systems.
    Physiology & behavior, 1988, Volume: 42, Issue:2

    Topics: Aggression; Analgesia; Animals; Diazepam; Female; Flumazenil; Male; Naloxone; Nociceptors; Peromyscus; Receptors, GABA-A; Smell

1988
The effect of agonists at the GABA-benzodiazepine-receptor-complex on the proconflict effect induced by beta-CCM and pentetrazol in rats.
    Japanese journal of pharmacology, 1988, Volume: 46, Issue:3

    Topics: Aminooxyacetic Acid; Animals; Azabicyclo Compounds; Carbolines; Conflict, Psychological; Convulsants; Diazepam; Flumazenil; Hypnotics and Sedatives; Male; Pentylenetetrazole; Phenobarbital; Piperazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
The abstinence syndrome in diazepam-dependent cats is precipitated by Ro 15-1788 and Ro 15-4513 but not by the benzodiazepine receptor antagonist ZK 93426.
    Neuroscience letters, 1988, May-26, Volume: 88, Issue:2

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Cats; Diazepam; Flumazenil; Receptors, GABA-A; Substance Withdrawal Syndrome

1988
Involvement of the inhibitory GTP-binding regulatory protein and a low-affinity benzodiazepine receptor in the inhibitory effect of diazepam on rat brain adenylate cyclase system.
    Japanese journal of pharmacology, 1988, Volume: 47, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Brain; Bromides; Diazepam; Flumazenil; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes

1988
Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.
    Journal of neurochemistry, 1988, Volume: 51, Issue:5

    Topics: Animals; Benzodiazepines; Carbolines; Cerebral Cortex; Diazepam; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Monoamine Oxidase Inhibitors; Pargyline; Pyrazoles; Pyridazines; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin

1988
In vivo binding of (3H)Ro 15-1788 in mice: comparison with the in vivo binding of (3H)flunitrazepam.
    Life sciences, 1988, Volume: 43, Issue:16

    Topics: Animals; Brain; Cerebellum; Cerebral Cortex; Diazepam; Flumazenil; Flunitrazepam; Hippocampus; Male; Mice; Receptors, GABA-A

1988
Chronic administration of diazepam downregulates adenosine receptors in the rat brain.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:2

    Topics: Animals; Brain; Diazepam; Flumazenil; Flunitrazepam; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Purinergic

1988
In vivo determination of the profile of benzodiazepine ligands by comparing the inhibition of 3H-Ro 15-1788 binding to the modulation of cGMP levels in mouse cerebellum.
    Biochemical pharmacology, 1988, Oct-01, Volume: 37, Issue:19

    Topics: Animals; Cerebellum; Cyclic GMP; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Ligands; Male; Mice; Naphthyridines; Piperazines; Receptors, GABA-A; Sulfur Compounds; Tritium

1988
Involvement of GABAergic systems and benzodiazepine receptors in the jumping behavior induced by harmine and apomorphine in rats.
    Japanese journal of pharmacology, 1988, Volume: 47, Issue:4

    Topics: Alkaloids; Animals; Apomorphine; Brain; Diazepam; Flumazenil; Harmine; Hydroxydopamines; Male; Motor Activity; Muscimol; Oxidopamine; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Effects of drugs on the electrical activity of the red nucleus in the rabbit. Activation of benzodiazepine and barbiturate receptors.
    Annali dell'Istituto superiore di sanita, 1988, Volume: 24, Issue:3

    Topics: Animals; Bicuculline; Carbolines; Diazepam; Drug Interactions; Electroencephalography; Flumazenil; Muscle Relaxation; Pentobarbital; Pyridazines; Rabbits; Receptors, GABA-A; Receptors, Neurotransmitter; Red Nucleus

1988
Animal models of chronic anxiety and "fearlessness".
    Brain research bulletin, 1988, Volume: 21, Issue:3

    Topics: Animals; Anxiety; Brain; Cats; Diazepam; Disease Models, Animal; Fear; Female; Flumazenil; Flunitrazepam; Male; Pregnancy; Prenatal Exposure Delayed Effects; Receptors, GABA-A

1988
Chronic ethanol administration increases the binding of the benzodiazepine inverse agonist and alcohol antagonist [3H]RO15-4513 in rat brain.
    European journal of pharmacology, 1988, Aug-09, Volume: 153, Issue:1

    Topics: Acoustic Stimulation; Animals; Azides; Benzodiazepines; Body Temperature; Brain Chemistry; Diazepam; Ethanol; Flumazenil; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1988
Partial reversal of ethanol-induced reductions in exploration by two benzodiazepine antagonists (flumazenil and ZK 93426).
    Brain research bulletin, 1988, Volume: 21, Issue:5

    Topics: Animals; Carbolines; Diazepam; Dose-Response Relationship, Drug; Ethanol; Exploratory Behavior; Flumazenil; Male; Mice; Receptors, GABA-A

1988
Ro 15-4513: partial inverse agonism at the BZR and interaction with ethanol.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:3

    Topics: Animals; Azides; Behavior, Animal; Benzodiazepines; Brain; Brain Chemistry; Cats; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Ethanol; Flumazenil; Meta-Analysis as Topic; Mice; Phenobarbital; Rats; Receptors, GABA-A

1988
Benzodiazepine antagonist Ro 15-1788 in self-poisoning. Diagnostic and therapeutic use.
    Archives of internal medicine, 1985, Volume: 145, Issue:4

    Topics: Adult; Aged; Anti-Anxiety Agents; Antidotes; Benzodiazepinones; Coma; Diazepam; Electroencephalography; Female; Flumazenil; Flunitrazepam; Humans; Male; Middle Aged; Naloxone; Suicide, Attempted

1985
Effects of repeated RO 15-1788 administration in benzodiazepine-dependent baboons.
    European journal of pharmacology, 1985, Apr-02, Volume: 110, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Convulsants; Diazepam; Drug Tolerance; Flumazenil; Humans; Male; Papio; Posture; Substance Withdrawal Syndrome; Substance-Related Disorders; Tremor; Triazolam; Vomiting

1985
Reversal of antinociceptive effect of cholecystokinin by benzodiazepines and a benzodiazepine antagonist, Ro 15-1788.
    Japanese journal of pharmacology, 1985, Volume: 37, Issue:1

    Topics: Analgesics; Animals; Anti-Anxiety Agents; Benzodiazepinones; Chlordiazepoxide; Cholecystokinin; Diazepam; Flumazenil; Flurazepam; Male; Mice; Morphine; Naloxone; Pain; Sensory Thresholds; Time Factors

1985
ZK 91296, an anticonvulsant beta-carboline which lacks muscle relaxant properties.
    European journal of pharmacology, 1985, Apr-16, Volume: 110, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Electromyography; Electroshock; Flumazenil; Indoles; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle Relaxants, Central; Muscle Tonus; Phenobarbital; Rats; Rats, Inbred Strains

1985
Benzodiazepines reduce the tolerance to reward delay in rats.
    Psychopharmacology, 1985, Volume: 86, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Choice Behavior; Diazepam; Flumazenil; Male; Piperidines; Rats; Rats, Inbred Strains; Reward; Serotonin Antagonists; Synaptic Transmission; Zimeldine

1985
Specific antagonism by RO 15-1788 of benzodiazepine-induced increases in food intake in rhesus monkeys.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Bromazepam; Convulsants; Diazepam; Dose-Response Relationship, Drug; Feeding Behavior; Female; Flumazenil; Macaca mulatta; Male; Pentobarbital

1985
Disruption of schedule-controlled behavior by Ro 15-1788 one day after acute treatment with benzodiazepines.
    Psychopharmacology, 1986, Volume: 88, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Chlordiazepoxide; Conditioning, Operant; Convulsants; Diazepam; Flumazenil; Male; Nordazepam; Reinforcement Schedule; Saimiri

1986
Behavioral effects of zopiclone, CL 218,872 and diazepam in squirrel monkeys: antagonism by Ro 15-1788 and CGS 8216.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepinones; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Piperazines; Pyrazoles; Pyridazines; Saimiri

1986
Behavioral studies with anxiolytic drugs. III. Antipunishment actions of buspirone in the pigeon do not involve benzodiazepine receptor mechanisms.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Buspirone; Chlordiazepoxide; Columbidae; Diazepam; Flumazenil; Flunitrazepam; Punishment; Pyrimidines; Receptors, GABA-A

1986
A new method for screening anxiolytic drugs in rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 26, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Azabicyclo Compounds; Diazepam; Drug Evaluation, Preclinical; Flumazenil; Male; Models, Psychological; Piperazines; Rats; Rats, Inbred WKY

1987
Effects of two benzodiazepines and a benzodiazepine antagonist on neuromuscular blockade in the anaesthetized cat.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 286, Issue:1

    Topics: Animals; Blood Pressure; Cats; Diazepam; Drug Interactions; Drug Synergism; Female; Flumazenil; Male; Midazolam; Neuromuscular Blocking Agents; Neuromuscular Junction; Pancuronium; Sciatic Nerve; Vecuronium Bromide

1987
Interactions of aminophylline and three benzodiazepine compounds with amygdala-kindled seizures in rats.
    Experimental neurology, 1987, Volume: 97, Issue:3

    Topics: Aminophylline; Amygdala; Animals; Anti-Anxiety Agents; Diazepam; Drug Interactions; Flumazenil; Kindling, Neurologic; Male; Pyrazoles; Rats; Rats, Inbred Strains; Seizures

1987
Inhibition of non-dopamine cells in the ventral tegmental area by benzodiazepines: relationship to A10 dopamine cell activity.
    European journal of pharmacology, 1987, Oct-27, Volume: 142, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Flumazenil; Haloperidol; Iontophoresis; Male; Rats; Rats, Inbred Strains; Receptors, Dopamine; Tegmentum Mesencephali

1987
Tetrazepam: a benzodiazepine which dissociates sedation from other benzodiazepine activities. I. Psychopharmacological profile in rodents.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Diazepam; Feeding Behavior; Flumazenil; Male; Mice; Motor Activity; Pentylenetetrazole; Rats; Seizures

1988
Continuous slow release of low levels of diazepam produces tolerance to its depressant and anxiolytic effects on the startle reflex.
    European journal of pharmacology, 1988, May-20, Volume: 150, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Brain; Conditioning, Operant; Depression, Chemical; Diazepam; Drug Implants; Drug Tolerance; Flumazenil; Male; Rats; Rats, Inbred Strains; Reflex, Startle

1988
Modulation of GABA-stimulated chloride influx into membrane vesicles from rat cerebral cortex by benzodiazepines and nonbenzodiazepines.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Anti-Anxiety Agents; Cell Membrane; Cerebral Cortex; Chlorides; Clonazepam; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Inbred Strains

1988
Controlled sedation in ventilated intensive care patients.
    Resuscitation, 1988, Volume: 16 Suppl

    Topics: Adult; Aged; Anti-Anxiety Agents; Coma; Critical Care; Diazepam; Female; Flumazenil; Humans; Injections, Intravenous; Male; Middle Aged; Respiration, Artificial

1988
Effects of non-sedative anxiolytic drugs on responses to GABA and on diazepam-induced enhancement of these responses on mouse neurones in cell culture.
    British journal of pharmacology, 1988, Volume: 95, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Buspirone; Carbolines; Cells, Cultured; Convulsants; Diazepam; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Mice; Neurons; Pyrazoles; Quinolines; Spinal Cord

1988
Benzodiazepines for catatonic symptoms, stupor, and mutism.
    Pharmacopsychiatry, 1988, Volume: 21, Issue:6

    Topics: Anti-Anxiety Agents; Benzodiazepines; Catatonia; Depressive Disorder; Diazepam; Female; Flumazenil; Humans; Lorazepam; Mutism

1988
Discriminative-stimulus effects of midazolam in squirrel monkeys: comparison with other drugs and antagonism by Ro 15-1788.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Azabicyclo Compounds; Barbital; Benzodiazepines; Benzodiazepinones; Buspirone; Caffeine; Chlordiazepoxide; Cinanserin; Clozapine; Conditioning, Operant; Cyproheptadine; Diazepam; Diphenhydramine; Discrimination Learning; Electroshock; Flumazenil; Male; Midazolam; Muscimol; Nordazepam; Pentobarbital; Piperazines; Pyridazines; Pyrimidines; Saimiri; Tripelennamine

1985
Effects of guanyl nucleotides on [3H]flunitrazepam binding to rat hippocampal synaptic membranes: equilibrium binding and dissociation kinetics.
    Journal of neurochemistry, 1985, Volume: 44, Issue:1

    Topics: Adenosine Triphosphate; Animals; Benzodiazepinones; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Hippocampus; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes

1985
Changes in the characteristics of low affinity GABA binding sites elicited by Ro15-1788.
    Life sciences, 1985, Jan-28, Volume: 36, Issue:4

    Topics: Animals; Benzodiazepinones; Carbolines; Cerebral Cortex; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Handling, Psychological; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Pharmacological and neurochemical properties of 1,4-diazepines with two annelated heterocycles ('hetrazepines').
    European journal of pharmacology, 1985, Feb-12, Volume: 109, Issue:1

    Topics: Action Potentials; Aggression; Animals; Anticonvulsants; Azepines; Behavior, Animal; Benzodiazepinones; Brain Chemistry; Carbolines; Cerebral Cortex; Conflict, Psychological; Diazepam; Flumazenil; Heterocyclic Compounds; Humans; Hypnotics and Sedatives; Male; Mice; Motor Activity; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sleep; Social Isolation; Wakefulness

1985
Radiation inactivation studies of the benzodiazepine/gamma-aminobutyric acid/chloride ionophore receptor complex.
    Journal of neurochemistry, 1985, Volume: 45, Issue:1

    Topics: Animals; Barbiturates; Benzodiazepines; Benzodiazepinones; Binding Sites; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Flumazenil; Flunitrazepam; Ionophores; Male; Molecular Weight; Muscimol; Picrotoxin; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
The effects of benzodiazepines on spinal homosynaptic depression.
    Neuropharmacology, 1985, Volume: 24, Issue:4

    Topics: Animals; Benzodiazepinones; Cats; Clonazepam; Diazepam; Female; Flumazenil; Male; Receptors, GABA-A; Reflex, Monosynaptic; Reflex, Stretch; Spinal Nerve Roots; Synapses

1985
Blockade of the diazepam-induced increase in rat striatal acetylcholine content by the specific benzodiazepine antagonists ethyl-beta-carboline-3-carboxylate and Ro 15-1788.
    Brain research, 1985, Jun-17, Volume: 336, Issue:2

    Topics: Acetylcholine; Animals; Benzodiazepines; Benzodiazepinones; Brain Chemistry; Carbolines; Corpus Striatum; Diazepam; Female; Flumazenil; Indoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Supraspinal convulsions induced by inverse benzodiazepine agonists in rabbits.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 234, Issue:1

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electroencephalography; Flumazenil; Male; Pyrazoles; Rabbits; Receptors, GABA-A; Seizures

1985
Benzodiazepines inhibit human platelet activation: comparison of the mechanism of antiplatelet actions of flurazepam and diazepam.
    Thrombosis research, 1985, May-15, Volume: 38, Issue:4

    Topics: Adenosine Diphosphate; Arachidonic Acid; Arachidonic Acids; Benzodiazepinones; Blood Platelets; Collagen; Cyclic AMP; Cyclic GMP; Diazepam; Epinephrine; Flumazenil; Flurazepam; Humans; Malondialdehyde; Platelet Aggregation; Prostaglandin Endoperoxides, Synthetic; Serotonin; Thrombin; Type C Phospholipases

1985
Reduction of inhibition by a benzodiazepine antagonist, Ro15-1788, in the rat hippocampal slice.
    Neuroscience, 1985, Volume: 15, Issue:2

    Topics: Animals; Benzodiazepinones; Chlordiazepoxide; Diazepam; Electric Conductivity; Evoked Potentials; Flumazenil; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Neural Inhibition; Rats; Synaptic Transmission

1985
A beta-carboline antagonizes benzodiazepine actions but does not precipitate the abstinence syndrome in cats.
    Psychopharmacology, 1985, Volume: 86, Issue:1-2

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Brain; Carbolines; Cats; Diazepam; Electroencephalography; Flumazenil; Humans; Indoles; Receptors, GABA-A; Substance Withdrawal Syndrome

1985
Benzodiazepine-receptor mediated inhibition of isolation-induced aggression in mice.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:1

    Topics: Aggression; Animals; Benzodiazepinones; Carbolines; Diazepam; Flumazenil; Humans; Indoles; Male; Mice; Receptors, GABA-A; Social Isolation

1985
Involvement of benzodiazepine recognition sites in the foot shock-induced decrease of low affinity GABA receptors in the rat cerebral cortex.
    Brain research, 1985, Aug-19, Volume: 341, Issue:1

    Topics: Animals; Benzodiazepinones; Cerebral Cortex; Diazepam; Electroshock; Flumazenil; Foot; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Monoclonal antibodies to benzodiazepines.
    Journal of neurochemistry, 1985, Volume: 45, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Antibodies, Monoclonal; Benzodiazepines; Benzodiazepinones; Diazepam; Flumazenil; Flunitrazepam; Flurazepam; Mice; Mice, Inbred BALB C; Receptors, GABA-A; Structure-Activity Relationship

1985
Benzodiazepine binding characteristics of embryonic rat brain neurons grown in culture.
    Journal of neurochemistry, 1985, Volume: 45, Issue:6

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cells, Cultured; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Neurons; Pyridazines; Rats; Receptors, GABA-A

1985
Solubilization of peripheral benzodiazepine-binding sites from rat kidney.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1985, Volume: 5, Issue:11

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Carbolines; Chlordiazepoxide; Clonazepam; Diazepam; Digitonin; Flumazenil; Flurazepam; Guanidine; Guanidines; Hot Temperature; Isoquinolines; Kidney; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Solubility; Time Factors; Urea

1985
Convulsant component of a depressant benzodiazepine.
    Life sciences, 1985, Nov-18, Volume: 37, Issue:20

    Topics: Animals; Benzodiazepinones; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Pentylenetetrazole; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1985
Imaging of [11C]-labelled Ro 15-1788 binding to benzodiazepine receptors in the human brain by positron emission tomography.
    Journal of psychiatric research, 1985, Volume: 19, Issue:4

    Topics: Adult; Animals; Benzodiazepinones; Brain; Cerebral Cortex; Diazepam; Flumazenil; Humans; Kinetics; Macaca fascicularis; Male; Mental Disorders; Middle Aged; Receptors, GABA-A; Tomography, Emission-Computed

1985
Attenuating effect of diazepam on stress-induced increases in noradrenaline turnover in specific brain regions of rats: antagonism by Ro 15-1788.
    Life sciences, 1985, Dec-30, Volume: 37, Issue:26

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Brain; Diazepam; Flumazenil; Male; Methoxyhydroxyphenylglycol; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Restraint, Physical; Stress, Physiological; Tissue Distribution

1985
Antianxiety effect of cannabis: involvement of central benzodiazepine receptors.
    Biological psychiatry, 1986, Volume: 21, Issue:1

    Topics: Adult; Aggression; Animals; Anxiety; Benzodiazepinones; Cannabinoids; Diazepam; Dronabinol; Electroshock; Female; Flumazenil; Frontal Lobe; Humans; Male; Mice; Mice, Inbred Strains; Middle Aged; Receptors, GABA-A; Tritium

1986
Enhancement of GABA binding by the benzodiazepine partial agonist CGS9896.
    European journal of pharmacology, 1985, Dec-10, Volume: 119, Issue:1-2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Calcium Chloride; Diazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Magnesium; Pyrazoles; Pyridazines; Rats; Receptors, GABA-A

1985
The benzodiazepine antagonist Ro 15-1788 does not antagonize the ethanol withdrawal syndrome.
    Biological psychiatry, 1986, Volume: 21, Issue:7

    Topics: Animals; Arousal; Benzodiazepinones; Brain; Diazepam; Drug Therapy, Combination; Ethanol; Flumazenil; Male; Motor Skills; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substance Withdrawal Syndrome

1986
Differential antagonism of diazepam-induced loss of the righting response.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:4

    Topics: Animals; Benzodiazepinones; Carbolines; Columbidae; Diazepam; Flumazenil; Inosine; Male; Pentobarbital; Posture; Receptors, GABA-A; Reflex; Saimiri

1986
Benzodiazepine receptor involvement in the control of receptive field size and responsiveness in primary somatosensory cortex.
    Brain research, 1986, Jun-18, Volume: 376, Issue:1

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Cats; Diazepam; Female; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Male; Midazolam; Neurons; Receptors, GABA-A; Sensory Thresholds; Somatosensory Cortex; Touch

1986
Convulsant effect of Ro 5-4864, a peripheral type benzodiazepine, on the baboon (Papio papio).
    Neuroscience letters, 1986, May-15, Volume: 66, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Isoquinolines; Papio; Receptors, GABA-A; Seizures

1986
Proconflict effect of GABA receptor complex antagonists. Reversal by diazepam.
    Neuropharmacology, 1986, Volume: 25, Issue:5

    Topics: Animals; Benzodiazepinones; Bicuculline; Conflict, Psychological; Diazepam; Flumazenil; Male; Pentylenetetrazole; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
The possible role of benzodiazepine receptors in morphine analgesia.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:1

    Topics: Animals; Benzodiazepinones; Diazepam; Drug Interactions; Flumazenil; Male; Mice; Morphine; Pain; Receptors, GABA-A

1986
Effects of beta-carboline-3-carboxylic acid ethyl ester on suppressed and non-suppressed responding in the rhesus monkey.
    European journal of pharmacology, 1986, Sep-23, Volume: 129, Issue:1-2

    Topics: Adrenocorticotropic Hormone; Animals; Blood Pressure; Carbolines; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Heart Rate; Macaca mulatta; Male; Punishment; Reinforcement Schedule

1986
Apparent pA2 estimation of benzodiazepine receptor antagonists.
    Methods and findings in experimental and clinical pharmacology, 1986, Volume: 8, Issue:9

    Topics: Animals; Diazepam; Drug Interactions; Female; Flumazenil; Male; Pentylenetetrazole; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1986
Benzodiazepines inhibit thyrotropin (TSH)-releasing hormone-induced TSH and growth hormone release from perifused rat pituitaries.
    Endocrinology, 1986, Volume: 119, Issue:6

    Topics: Animals; Benzodiazepines; Bicuculline; Diazepam; Flumazenil; Growth Hormone; Growth Hormone-Releasing Hormone; In Vitro Techniques; Isoquinolines; Male; Picrotoxin; Pituitary Gland, Anterior; Rats; Receptors, GABA-A; Secretory Rate; Thyrotropin; Thyrotropin-Releasing Hormone

1986
The possible modulation of morphine analgesia by the supramolecular GABA receptor complex.
    Psychopharmacology, 1986, Volume: 90, Issue:2

    Topics: Analgesics; Animals; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Mice; Morphine; Picrotoxin; Receptors, GABA-A

1986
A 7-phenyl substituted triazolopyridazine has inverse agonist activity at the benzodiazepine receptor site.
    British journal of pharmacology, 1987, Volume: 90, Issue:1

    Topics: Animals; Binding, Competitive; Brain; Conditioning, Operant; Convulsants; Diazepam; Female; Flumazenil; Flunitrazepam; In Vitro Techniques; Male; Mice; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship

1987
The beta-carboline ZK 93423 inhibits reticulata neurons: an effect reversed by benzodiazepine antagonists.
    Life sciences, 1987, Apr-06, Volume: 40, Issue:14

    Topics: Action Potentials; Animals; Carbolines; Diazepam; Flumazenil; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Substantia Nigra

1987
Dissimilarities between benzodiazepine-binding sites and adenosine uptake sites in astrocytes and neurons in primary cultures.
    Journal of neuroscience research, 1987, Volume: 17, Issue:2

    Topics: Adenosine; Animals; Astrocytes; Benzodiazepines; Binding Sites; Cells, Cultured; Diazepam; Flumazenil; Isoquinolines; Neurons; Pyrazoles; Receptors, GABA-A

1987
Separation distress in infant rhesus monkeys: effects of diazepam and Ro 15-1788.
    Brain research, 1987, Apr-07, Volume: 408, Issue:1-2

    Topics: Adrenocorticotropic Hormone; Animals; Animals, Newborn; Anxiety, Separation; Behavior, Animal; Diazepam; Female; Flumazenil; Hydrocortisone; Macaca mulatta; Male; Maternal Deprivation; Vocalization, Animal

1987
CGS 9896 and ZK 91296, but not CGS 8216 and RO 15-1788, are pure benzodiazepine receptor antagonists on mouse neurons in culture.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:1

    Topics: Animals; Brain; Carbolines; Cells, Cultured; Diazepam; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Mice; Neurons; Pyrazoles; Receptors, GABA-A; Spinal Cord

1987
Interactions of Ro 15-1788, CGS 8216 and diazepam on head-turning in rats.
    Life sciences, 1986, Feb-03, Volume: 38, Issue:5

    Topics: Animals; Benzodiazepinones; Diazepam; Drug Interactions; Electric Stimulation; Flumazenil; Head; Male; Movement; Muscimol; Pyrazoles; Rats; Rats, Inbred Strains

1986
Diazepam potentiates GABA-contraction in guinea-pig ileum.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 279, Issue:1

    Topics: Animals; Baclofen; Benzodiazepinones; Carbolines; Diazepam; Drug Synergism; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth

1986
Acute tolerance to diazepam induced by benzodiazepines.
    Clinical and experimental pharmacology & physiology, 1986, Volume: 13, Issue:1

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Flumazenil; Lorazepam; Male; Mice; Sleep

1986
Effects of diazepam on pancreatic exocrine secretion in the dog.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 280, Issue:2

    Topics: Animals; Benzodiazepinones; Bicarbonates; Diazepam; Dogs; Female; Flumazenil; Male; Pancreas; Pancreatic Juice; Proteins; Regional Blood Flow; Secretin

1986
Diazepam-induced decrease in histamine turnover in mouse brain.
    European journal of pharmacology, 1986, May-27, Volume: 124, Issue:3

    Topics: Animals; Benzodiazepinones; Brain; Diazepam; Drug Interactions; Flumazenil; Histamine; Male; Methylhistamines; Mice; Muscimol; Pargyline

1986
Reversal of the effect of centrally-administered diazepam on morphine antinociception by specific (Ro 15-1788 and Ro 15-3505) and non-specific (bicuculline and caffeine) benzodiazepine antagonists.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:1

    Topics: Animals; Benzodiazepinones; Bicuculline; Caffeine; Diazepam; Flumazenil; Injections, Intraventricular; Male; Morphine; Pain; Rats; Rats, Inbred Strains

1986
Reversal of the cerebral effects of diazepam in the dog by the benzodiazepine antagonist Ro15-1788.
    Acta anaesthesiologica Scandinavica, 1986, Volume: 30, Issue:4

    Topics: Anesthesia; Animals; Benzodiazepinones; Brain; Cerebrovascular Circulation; Diazepam; Dogs; Electroencephalography; Female; Flumazenil; Male; Nitrous Oxide; Oxygen

1986
Benzodiazepine antagonist, CGS-8216, in diazepam- or pentobarbital-dependent and non-dependent rats.
    Drug and alcohol dependence, 1986, Volume: 17, Issue:4

    Topics: Animals; Arousal; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Pentobarbital; Pyrazoles; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Substance-Related Disorders

1986
Effect of RO 15-1788 on diazepam, GABA & pentobarbitone induced EEG changes in rabbits.
    The Indian journal of medical research, 1986, Volume: 83

    Topics: Animals; Cerebral Cortex; Diazepam; Electroencephalography; Electromyography; Female; Flumazenil; gamma-Aminobutyric Acid; Male; Pentobarbital; Rabbits

1986
CGS 8216: agonist and diazepam-antagonist effects in rodents.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:1

    Topics: Animals; Ataxia; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Male; Mice; Pentylenetetrazole; Pyrazoles; Rats; Rats, Inbred F344; Reinforcement, Psychology

1986
Evaluation of two anticonvulsant amino-pyridazine derivatives in the conflict test in rats.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2

    Topics: Animals; Anticonvulsants; Conflict, Psychological; Diazepam; Flumazenil; Meprobamate; Mice; Papio; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Valproic Acid

1986
Investigation of the actions of the benzodiazepine antagonists Ro 15-1788 and CGS 8216 using the schedule-controlled behavior of rats.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:3

    Topics: Animals; Anxiety; Behavior, Animal; Benzodiazepines; Diazepam; Drug Interactions; Flumazenil; Male; Pyrazoles; Pyridines; Rats; Rats, Inbred Strains; Zolpidem

1986
Effects of the benzodiazepine antagonists RO 15-1788, CGS-8216 and PK-11195 on amygdaloid kindled seizures and the anticonvulsant efficacy of diazepam.
    Neuropharmacology, 1986, Volume: 25, Issue:11

    Topics: Amygdala; Animals; Diazepam; Flumazenil; Isoquinolines; Kindling, Neurologic; Male; Pyrazoles; Rats; Rats, Inbred Strains

1986
Diazepam-sensitive specific binding of phenytoin in rat brain.
    Journal of receptor research, 1986, Volume: 6, Issue:3-4

    Topics: Animals; Benzodiazepinones; Binding Sites; Cell Membrane; Cerebral Cortex; Clonazepam; Diazepam; Flumazenil; Male; Phenytoin; Rats; Rats, Inbred Strains

1986
Periodic benzodiazepine antagonist administration prevents benzodiazepine withdrawal symptoms in primates.
    European journal of pharmacology, 1986, Dec-02, Volume: 132, Issue:1

    Topics: Animals; Behavior, Animal; Body Weight; Diazepam; Drug Administration Schedule; Flumazenil; Macaca mulatta; Substance Withdrawal Syndrome

1986
Benzodiazepine ligands, nociception and 'defeat' analgesia in male mice.
    Psychopharmacology, 1987, Volume: 91, Issue:3

    Topics: Analgesia; Animals; Appetite Depressants; Benzodiazepines; Carbolines; Chlordiazepoxide; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Nociceptors; Pyrazoles

1987
Lack of withdrawal signs of dependence following cessation of treatment or Ro-15,1788 administration to rats chronically treated with buspirone.
    Neuropsychobiology, 1986, Volume: 16, Issue:1

    Topics: Animals; Body Weight; Buspirone; Diazepam; Flumazenil; Food Deprivation; Male; Pyrimidines; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome

1986
Characterization of the analgesic effects of the benzodiazepine antagonist, Ro 15-1788.
    Brain research, 1987, Jul-14, Volume: 415, Issue:2

    Topics: Analgesics; Animals; Diazepam; Flumazenil; Male; Naloxone; Rats; Rats, Inbred Strains

1987
Social conflict analgesia: inhibition of early non-opioid component by diazepam or flumazepil fails to affect appearance of late opioid component.
    Brain research bulletin, 1987, Volume: 19, Issue:1

    Topics: Aggression; Animals; Appetitive Behavior; Conflict, Psychological; Diazepam; Endorphins; Flumazenil; Male; Mice; Mice, Inbred DBA; Pain; Predatory Behavior; Reaction Time

1987
Benzodiazepine antagonist Ro 15-1788 (flumazepil) attenuates the anticonvulsant activity of diazepam in epileptic fowl.
    Brain research, 1987, Oct-20, Volume: 424, Issue:1

    Topics: Animals; Chickens; Diazepam; Epilepsy; Female; Flumazenil; Male; Poultry Diseases

1987
Diazepam and endorphin independently inhibit ultrasonic distress calls in rats.
    European journal of pharmacology, 1987, Oct-06, Volume: 142, Issue:1

    Topics: Animals; Convulsants; Depression, Chemical; Diazepam; Endorphins; Flumazenil; Injections, Subcutaneous; Male; Pyrazoles; Rats; Rats, Inbred Strains; Ultrasonics; Vocalization, Animal

1987
Effects of Ro 15-1788 and CGS 8216 in diazepam-dependent baboons.
    European journal of pharmacology, 1987, Nov-10, Volume: 143, Issue:2

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Papio; Pyrazoles; Substance Withdrawal Syndrome; Substance-Related Disorders

1987
Effects of diazepam, ethanol and Ro 15-1788 on ultrasonic vocalization, locomotor activity and body righting in the neonatal rat.
    Alcohol and alcoholism (Oxford, Oxfordshire). Supplement, 1987, Volume: 1

    Topics: Animals; Animals, Newborn; Diazepam; Dose-Response Relationship, Drug; Ethanol; Flumazenil; Motor Activity; Posture; Rats; Rats, Inbred Strains; Reflex; Ultrasonics; Vocalization, Animal

1987
Enhancement of a diazepam withdrawal symptom by bicuculline and yohimbine.
    Neuropharmacology, 1987, Volume: 26, Issue:12

    Topics: Animals; Bicuculline; Diazepam; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; Male; Rats; Substance Withdrawal Syndrome; Yohimbine

1987
Effects of diazepam, FG 7142, and RO 15-1788 on schedule-induced polydipsia and the temporal control of behavior.
    Psychopharmacology, 1988, Volume: 94, Issue:1

    Topics: Animals; Appetite Depressants; Carbolines; Diazepam; Drinking Behavior; Flumazenil; Male; Motor Activity; Rats

1988
Precipitation of abstinence in nordiazepam- and diazepam-dependent dogs.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Analysis of Variance; Animals; Diazepam; Dogs; Flumazenil; Nordazepam; Oxazepam; Pyrazoles; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1988
Stimulatory action of gamma-aminobutyric acid on catecholamine secretion from bovine adrenal chromaffin cells measured by a real-time monitoring system.
    Journal of neurochemistry, 1988, Volume: 50, Issue:6

    Topics: Adrenal Glands; Animals; Catecholamines; Cattle; Chromaffin System; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Magnesium; Nifedipine

1988
Inhibition of cell proliferation of human gliomas by benzodiazepines in vitro.
    Acta neurologica Scandinavica, 1988, Volume: 77, Issue:3

    Topics: Astrocytoma; Benzodiazepines; Benzodiazepinones; Cell Division; Clonazepam; Diazepam; Female; Flumazenil; Glioma; Humans; Male; Middle Aged; Thymidine; Tumor Cells, Cultured

1988
Treatment of severe chloroquine poisoning.
    The New England journal of medicine, 1988, Jul-07, Volume: 319, Issue:1

    Topics: Animals; Chloroquine; Diazepam; Epinephrine; Flumazenil; Gastric Lavage; Humans; Respiration, Artificial

1988
Modulation of GABA-gated chloride ion flux in rat brain by acute and chronic benzodiazepine administration.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1

    Topics: Animals; Benzodiazepines; Brain; Chlorides; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains

1988
Ultrasonic vocalization in response to unavoidable aversive stimuli in rats: effects of benzodiazepines.
    Life sciences, 1988, Volume: 43, Issue:6

    Topics: Alprazolam; Animals; Benzodiazepines; Desipramine; Diazepam; Electroshock; Flumazenil; Haloperidol; Male; Rats; Rats, Inbred Strains; Ultrasonics; Vocalization, Animal

1988
Distinctive behavioral effects of the pyrazoloquinoline CGS 8216 in squirrel monkeys.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:4

    Topics: Animals; Behavior, Animal; Benzodiazepines; Clonidine; Diazepam; Flumazenil; Male; Pyrazoles; Saimiri

1988
A simple and rapid method of inducing physical dependence with benzodiazepines in mice.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:4

    Topics: Animals; Benzodiazepines; Diazepam; Flumazenil; Injections, Intraperitoneal; Male; Mice; Mice, Inbred Strains; Substance Withdrawal Syndrome; Substance-Related Disorders

1988
The effects of chronic antidepressant treatment in an animal model of anxiety.
    Psychopharmacology, 1988, Volume: 95, Issue:3

    Topics: Amitriptyline; Animals; Antidepressive Agents; Anxiety; Desipramine; Diazepam; Disease Models, Animal; Flumazenil; Male; Rats; Time Factors

1988
Reversal of iatrogenic diazepam overdose with flumazenil.
    Clinical pharmacy, 1988, Volume: 7, Issue:8

    Topics: Aged; Coma; Diazepam; Flumazenil; Humans; Intensive Care Units; Male

1988
The lateral vestibular nucleus is a site for the depressant action of benzodiazepines on the crossed extensor reflex.
    Brain research, 1988, Oct-04, Volume: 461, Issue:2

    Topics: Action Potentials; Animals; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flurazepam; Male; Microinjections; Neural Inhibition; Posture; Rats; Rats, Inbred Strains; Reflex; Vestibular Nuclei

1988
Brief exposure to a natural predator, the short-tailed weasel, induces benzodiazepine-sensitive analgesia in white-footed mice.
    Physiology & behavior, 1988, Volume: 43, Issue:2

    Topics: Analgesia; Animals; Appetitive Behavior; Diazepam; Flumazenil; Handling, Psychological; Hot Temperature; Male; Naloxone; Pain; Peromyscus; Predatory Behavior; Rabbits; Reference Values; Rodentia

1988
Theophylline antagonizes the effect of diazepam on ventricular automaticity.
    European journal of pharmacology, 1988, Oct-18, Volume: 155, Issue:3

    Topics: Adenosine; Animals; Diazepam; Female; Flumazenil; Heart Rate; Heart Ventricles; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Theophylline; Ventricular Function

1988
Effects of Ro 15-4513, alone or in combination with ethanol, Ro 15-1788, diazepam, and pentobarbital on instrumental behaviors of rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:3

    Topics: Animals; Azides; Behavior, Animal; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Female; Flumazenil; Pentobarbital; Rats; Rats, Inbred Strains; Time Factors

1988
Withdrawal from diazepam substitutes for the discriminative stimulus properties of pentylenetetrazol.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:3

    Topics: Animals; Diazepam; Discrimination Learning; Disease Models, Animal; Flumazenil; Male; Pentylenetetrazole; Rats; Substance Withdrawal Syndrome; Substance-Related Disorders

1988
Blood pressure response to Ro15-1788, a benzodiazepine antagonist.
    Life sciences, 1985, Feb-25, Volume: 36, Issue:8

    Topics: Animals; Benzodiazepinones; Blood Pressure; Cats; Convulsants; Diazepam; Drug Tolerance; Flumazenil; Flurazepam; Heart Rate; Humans; Substance-Related Disorders

1985
Precipitated diazepam withdrawal elevates noradrenergic metabolism in primate brain.
    European journal of pharmacology, 1985, Jan-02, Volume: 107, Issue:2

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Brain; Chlorocebus aethiops; Diazepam; Female; Flumazenil; Humans; Male; Methoxyhydroxyphenylglycol; Narcotics; Norepinephrine; Substance Withdrawal Syndrome

1985
An EEG investigation on the role of cerebello-rubral system in the effects of diazepam and pentobarbital.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A

    Topics: Animals; Benzodiazepinones; Cerebellum; Diazepam; Electroencephalography; Female; Flumazenil; Male; Pentobarbital; Pentylenetetrazole; Picrotoxin; Rabbits; Red Nucleus

1985
Evaluation of the muscle relaxant properties of a novel beta-carboline, ZK 93423 in rats and cats.
    British journal of pharmacology, 1985, Volume: 86, Issue:2

    Topics: Animals; Benzodiazepinones; Carbolines; Cats; Decerebrate State; Diazepam; Electromyography; Evoked Potentials; Female; Flumazenil; Male; Muscle Relaxants, Central; Neurons, Afferent; Rats; Rats, Mutant Strains; Reflex; Species Specificity; Time Factors

1985
[Effect of the beta-carboline derivative FG 7142 on inhibition in hippocampal sections].
    Biulleten' eksperimental'noi biologii i meditsiny, 1985, Volume: 100, Issue:12

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electric Stimulation; Evoked Potentials; Flumazenil; Hippocampus; Neural Inhibition; Neurons; Rats; Rats, Inbred Strains

1985
Specific changes in local cerebral glucose utilization in the rat brain induced by acute and chronic diazepam.
    Brain research, 1985, Dec-16, Volume: 359, Issue:1-2

    Topics: Animals; Benzodiazepinones; Brain; Diazepam; Flumazenil; Glucose; Male; Rats; Rats, Inbred Strains; Time Factors

1985
Diazepam increases membrane fluidity of rat hippocampus synaptosomes.
    FEBS letters, 1984, Jul-23, Volume: 173, Issue:1

    Topics: Animals; Benzodiazepinones; Cerebellum; Diazepam; Flumazenil; Hippocampus; Male; Membrane Fluidity; Rats; Receptors, Cell Surface; Receptors, GABA-A; Synaptosomes

1984
In vitro interaction of premazepam with benzodiazepine receptors in rat brain regions.
    Life sciences, 1984, Jul-23, Volume: 35, Issue:4

    Topics: Animals; Azepines; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Brain; Cerebellum; Convulsants; Diazepam; Flumazenil; Flunitrazepam; Kinetics; Male; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Synaptosomes; Thermodynamics

1984
Electrophysiological and pharmacological characterization of peripheral benzodiazepine receptors in a guinea pig heart preparation.
    Life sciences, 1984, Aug-27, Volume: 35, Issue:9

    Topics: Action Potentials; Animals; Benzodiazepinones; Clonazepam; Convulsants; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Flumazenil; Guinea Pigs; Heart; In Vitro Techniques; Isoquinolines; Myocardial Contraction; Myocardium; Receptors, Cell Surface; Receptors, GABA-A

1984
Evaluation of the beta-carboline ZK 93 426 as a benzodiazepine receptor antagonist.
    Psychopharmacology, 1984, Volume: 83, Issue:3

    Topics: Animals; Anticonvulsants; Ataxia; Benzodiazepinones; Binding, Competitive; Carbolines; Diazepam; Discrimination, Psychological; Drinking; Exploratory Behavior; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Mice; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Sleep

1984
An imidazodiazepine derivative, Ro 15-1788, behaves as a weak partial agonist in the crossed extensor reflex.
    European journal of pharmacology, 1984, Jun-15, Volume: 102, Issue:1

    Topics: Animals; Benzodiazepinones; Carbolines; Chlorpromazine; Diazepam; Flumazenil; Male; Phenobarbital; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reflex

1984
Beta-carboline kindling of the benzodiazepine receptor.
    Brain research, 1984, Oct-29, Volume: 321, Issue:1

    Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Flumazenil; Indoles; Kindling, Neurologic; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Pharmacological evidence that PK 8165 behaves as a partial agonist of brain type benzodiazepine receptors.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 271, Issue:2

    Topics: Aggression; Animals; Anticonvulsants; Benzodiazepinones; Conflict, Psychological; Diazepam; Drinking; Flumazenil; Humans; Male; Mice; Mice, Inbred Strains; Phenobarbital; Quinolines; Receptors, GABA-A; Reflex

1984
The benzodiazepine receptor and sleep.
    Psychiatric developments, 1984,Autumn, Volume: 2, Issue:3

    Topics: Animals; Barbiturates; Benzodiazepines; Benzodiazepinones; Calcium; Carbolines; Diazepam; Flumazenil; Flurazepam; Humans; Motor Activity; Nifedipine; Phenobarbital; Pyrazoles; Rats; Receptors, GABA-A; Sleep; Synaptosomes

1984
Benzodiazepine agonist-type activity of raubasine, a rauwolfia serpentina alkaloid.
    European journal of pharmacology, 1984, Nov-13, Volume: 106, Issue:2

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Binding, Competitive; Brain; Diazepam; Flumazenil; Flurazepam; In Vitro Techniques; Kinetics; Male; Mice; Rats; Receptors, GABA-A; Secologanin Tryptamine Alkaloids; Yohimbine

1984
Benzodiazepine binding sites in human pineal gland.
    European journal of pharmacology, 1984, Nov-13, Volume: 106, Issue:2

    Topics: Adolescent; Adult; Aged; Animals; Benzodiazepinones; Binding, Competitive; Cerebral Cortex; Child; Child, Preschool; Clonazepam; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Infant; Kinetics; Male; Middle Aged; Pineal Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Scopolamine-induced locomotor stimulation in mice: effect of diazepam and a benzodiazepine antagonist.
    Psychopharmacology, 1982, Volume: 77, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Flumazenil; Male; Mice; Mice, Inbred BALB C; Motor Activity; Scopolamine

1982
Comparison of the kinetics of [3H]diazepam and [3H]flunitrazepam binding to cortical synaptosomal membranes.
    Journal of neurochemistry, 1982, Volume: 39, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Cerebral Cortex; Diazepam; Filtration; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Male; Pentobarbital; Rats; Rats, Inbred Strains; Sodium Chloride; Synaptic Membranes

1982
RO 15-1788 selectively reverses antagonism of pentylenetetrazol-induced discriminative stimuli by benzodiazepines but not by barbiturates.
    Life sciences, 1982, Dec-27, Volume: 31, Issue:26

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Barbiturates; Benzodiazepines; Benzodiazepinones; Diazepam; Flumazenil; Male; Pentobarbital; Pentylenetetrazole; Rats; Stimulation, Chemical

1982
Lorazepam and pentobarbital drug discrimination in baboons: cross-drug generalization and interaction with Ro 15-1788.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 226, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Generalization, Response; Lorazepam; Male; Papio; Pentobarbital

1983
Benzodiazepine selectively antagonize kainate-induced activation in the rat hippocampus.
    European journal of pharmacology, 1983, Sep-16, Volume: 93, Issue:1-2

    Topics: Acetylcholine; Animals; Anti-Anxiety Agents; Benzodiazepinones; Chlorpromazine; Diazepam; Flumazenil; Glutamates; Hippocampus; Injections, Intravenous; Iontophoresis; Kainic Acid; Lorazepam; Male; Phenobarbital; Pyramidal Tracts; Pyrrolidines; Rats; Rats, Inbred Strains

1983
Benzodiazepine receptor ligands with opposing pharmacologic actions.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Flumazenil; Flunitrazepam; Kinetics; Ligands; Membranes; Models, Psychological; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Temperature

1983
Behavioral and EEG effects of benzodiazepines and their antagonists in the cat.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Carbolines; Cats; Diazepam; Electroencephalography; Flumazenil

1983
Anxiolytic-like properties of fominoben.
    European journal of pharmacology, 1984, Jan-27, Volume: 97, Issue:3-4

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Diazepam; Flumazenil; Male; Mice; Mice, Inbred C57BL; Morpholines

1984
Benzodiazepine Ro 15-1788: electrophysiological evidence for partial agonist activity.
    Neuroscience letters, 1983, Dec-30, Volume: 43, Issue:2-3

    Topics: Animals; Benzodiazepinones; Culture Techniques; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Ganglia, Spinal; Glutamates; Glutamic Acid; Membrane Potentials; Mice; Neurons; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord; Synaptic Transmission

1983
Benzodiazepine receptor antagonists reverse the effect of diazepam on plasma corticosterone in stressed rats.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:2

    Topics: Animals; Benzodiazepinones; Corticosterone; Diazepam; Flumazenil; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Stress, Physiological

1984
Differential effects of the benzodiazepine antagonist Ro 15-1788 after "general anaesthetic" doses of benzodiazepines in mice.
    British journal of anaesthesia, 1984, Volume: 56, Issue:10

    Topics: Anesthesia, General; Anesthetics; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Convulsants; Diazepam; Flumazenil; Flurazepam; Male; Mice; Mice, Inbred Strains; Midazolam; Reflex

1984
The effects of GABA and benzodiazepine receptor antagonists on the anti-conflict actions of diazepam or ethanol.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Bicuculline; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Ethanol; Flumazenil; Male; Picrotoxin; Punishment; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Self-injection of diazepam in naive rats: effects of dose, schedule and blockade of different receptors.
    Psychopharmacology, 1984, Volume: 84, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Bicuculline; Diazepam; Dose-Response Relationship, Drug; Extinction, Psychological; Flumazenil; Haloperidol; Male; Naloxone; Rats; Receptors, Drug; Reinforcement Schedule; Self Administration

1984
Comparison of five preanesthetic medicaments in thiopental-anesthetized cats: antagonism by selected compounds.
    American journal of veterinary research, 1984, Volume: 45, Issue:11

    Topics: 4-Aminopyridine; Acepromazine; Aminopyridines; Anesthesia, General; Animals; Arousal; Benzodiazepinones; Cats; Central Nervous System Stimulants; Convulsants; Diazepam; Drug Antagonism; Female; Flumazenil; Ketamine; Male; Meperidine; Naloxone; Pentobarbital; Preanesthetic Medication; Sodium Chloride; Xylazine; Yohimbine

1984
Modification of seizures elicited by the benzodiazepine Ro 5-3663--a comparison with picrotoxin.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:12

    Topics: Animals; Benzodiazepinones; Chemical Phenomena; Chemistry; Convulsants; Diazepam; Drug Synergism; Flumazenil; Male; Mice; Picrotoxin; Pyrazoles; Quinolines; Seizures

1984
Benzodiazepine antagonist Ro 15-1788: binding characteristics and interaction with drug-induced changes in dopamine turnover and cerebellar cGMP levels.
    Journal of neurochemistry, 1981, Volume: 37, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Brain; Cerebellum; Cerebral Cortex; Cyclic GMP; Diazepam; Dopamine; Flumazenil; Flunitrazepam; Kinetics; Mice; Receptors, Drug; Receptors, GABA-A

1981
Reversal of the antiaversive and anticonvulsant actions of diazepam, but not of progabide, by a selective antagonist of benzodiazepine receptors.
    European journal of pharmacology, 1981, Oct-15, Volume: 75, Issue:1

    Topics: Animals; Anxiety; Benzodiazepinones; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Humans; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures

1981
Caerulein and cholecystokinin octapeptide (CCK-8): sedative and anticonvulsive effects in mice unaffected by the benzodiazepine antagonist Ro 15-1788.
    Neuroscience letters, 1982, Mar-05, Volume: 28, Issue:3

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Blepharoptosis; Body Temperature; Ceruletide; Cholecystokinin; Diazepam; Flumazenil; Harmine; Hypnotics and Sedatives; Male; Mice; Peptide Fragments; Seizures; Sincalide

1982
Benzodiazepine antagonists abolish electrophysiological effects of sodium valproate in the rat.
    Life sciences, 1982, May-10, Volume: 30, Issue:19

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Diazepam; Evoked Potentials, Visual; Female; Flumazenil; gamma-Aminobutyric Acid; Immobilization; Kinetics; Male; Rats; Receptors, Drug; Receptors, GABA-A; Valproic Acid

1982
Precipitated withdrawal by a benzodiazepine receptor antagonist (Ro 15-1788) after 7 days of diazepam.
    Science (New York, N.Y.), 1982, Sep-17, Volume: 217, Issue:4565

    Topics: Animals; Benzodiazepinones; Diazepam; Flumazenil; Humans; Male; Papio; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Substance Withdrawal Syndrome; Time Factors

1982
Anxiogenic and non-anxiogenic benzodiazepine antagonists.
    Nature, 1983, Jan-06, Volume: 301, Issue:5895

    Topics: Animals; Anxiety; Benzodiazepines; Benzodiazepinones; Carbolines; Diazepam; Flumazenil; Food Deprivation; Humans; Indoles; Mice; Receptors, Cell Surface; Receptors, GABA-A

1983
Using Ro 15-1788 to investigate the benzodiazepine receptor in vivo: studies on the anticonvulsant and sedative effect of melatonin and the convulsant effect of the benzodiazepine Ro 05-3663.
    Psychopharmacology, 1982, Volume: 78, Issue:3

    Topics: Animals; Arousal; Benzodiazepinones; Brain; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Male; Melatonin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1982
Purines interact with 'central' but not 'peripheral' benzodiazepine binding sites.
    Neuroscience letters, 1982, Dec-23, Volume: 34, Issue:1

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Diazepam; Flumazenil; Purines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Synaptosomes

1982
Is the muscle relaxant effect of diazepam in spastic mutant rats mediated through GABA-independent benzodiazepine receptors?
    Neuroscience letters, 1983, Apr-11, Volume: 36, Issue:2

    Topics: Animals; Benzodiazepinones; Bicuculline; Diazepam; Electromyography; Female; Flumazenil; Male; Muscle Contraction; Muscle Relaxation; Picrotoxin; Rats; Rats, Mutant Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
Contrasting effects of ethyl beta-carboline-3-carboxylate (beta CCE) and diazepam on cerebellar cyclic GMP content and antagonism of both effects by Ro 15-1788, a specific benzodiazepine receptor blocker.
    European journal of pharmacology, 1983, May-20, Volume: 90, Issue:1

    Topics: Animals; Benzodiazepinones; Carbolines; Cerebellum; Cyclic GMP; Diazepam; Flumazenil; In Vitro Techniques; Indoles; Isoniazid; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
Is Ro15-1788 a partial agonist at benzodiazepine receptors?
    European journal of pharmacology, 1983, Jun-03, Volume: 90, Issue:2-3

    Topics: Animals; Benzodiazepinones; Bicuculline; Convulsants; Diazepam; Flumazenil; Male; Mice; Mice, Inbred C3H; Phenobarbital; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A

1983
Increase of cyclic GMP in cerebellum by methyl-6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate (DMCM).
    Brain research, 1983, Aug-29, Volume: 273, Issue:2

    Topics: Animals; Benzodiazepinones; Carbolines; Cerebellar Cortex; Cyclic GMP; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Indoles; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Stimulation, Chemical

1983
Diazepam receptor in frog muscle fibres.
    Acta physiologica Scandinavica, 1983, Volume: 118, Issue:1

    Topics: Animals; Anura; Benzodiazepinones; Diazepam; Flumazenil; Muscle Contraction; Receptors, Cell Surface; Receptors, GABA-A

1983
Diazepam, pentobarbital and D-etomidate produced increases in bicuculline seizure threshold; selective antagonism by RO15-1788, picrotoxin and (+/-)-DMBB.
    European journal of pharmacology, 1983, Oct-28, Volume: 94, Issue:3-4

    Topics: Animals; Barbiturates; Benzodiazepinones; Bicuculline; Diazepam; Etomidate; Flumazenil; Imidazoles; Male; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1983
beta-Carbolines activate neurons in the substantia nigra pars reticulata: an effect reversed by diazepam and Ro15-1788.
    European journal of pharmacology, 1983, Dec-09, Volume: 96, Issue:1-2

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Drug Interactions; Flumazenil; Indoles; Injections, Intravenous; Male; Rats; Rats, Inbred Strains; Substantia Nigra; Synaptic Transmission

1983
Evidence for distinct benzodiazepine receptors for anticonvulsant and sedative actions: implications for the treatment of temporal lobe epilepsy.
    Progress in neuro-psychopharmacology & biological psychiatry, 1983, Volume: 7, Issue:4-6

    Topics: Amygdala; Animals; Anticonvulsants; Benzodiazepinones; Diazepam; Epilepsy, Temporal Lobe; Flumazenil; Kindling, Neurologic; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
The benzodiazepine agonist diazepam inhibits basal and secretagogue-stimulated prolactin release in vitro.
    Brain research, 1984, Jan-23, Volume: 291, Issue:2

    Topics: Animals; Benzodiazepinones; Calcimycin; Cells, Cultured; Cyclic AMP; Diazepam; Drug Interactions; Female; Flumazenil; In Vitro Techniques; Male; Muscimol; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Thyrotropin

1984
The action of stress, beta-carbolines, diazepam, and Ro 15-1788 on GABA receptors in the rat brain.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Benzodiazepinones; Brain; Brain Chemistry; Carbolines; Diazepam; Electroshock; Flumazenil; Handling, Psychological; Humans; Indoles; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Stress, Psychological; Synaptic Transmission

1983
Involvement of GABA in the facilitation of punishment suppressed behavior induced by beta-carbolines in rat.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Conditioning, Operant; Diazepam; Drug Interactions; Flumazenil; gamma-Aminobutyric Acid; Humans; Indoles; Models, Psychological; Punishment; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Benzodiazepines receptor binding in vivo: pharmacokinetic and pharmacological significance.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Adrenal Glands; Animals; Benzodiazepinones; Brain; Carbolines; Corticosterone; Diazepam; Flumazenil; Flunitrazepam; Kinetics; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Effect of agonists, inverse agonists, and antagonists of benzodiazepine receptors on the firing rate of substantia nigra pars reticulata neurons.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electrophysiology; Flumazenil; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra

1983
On the convulsant action of Ro 5-4864 and the existence of a micromolar benzodiazepine binding site in rat brain.
    Psychopharmacology, 1984, Volume: 82, Issue:3

    Topics: Animals; Benzodiazepinones; Binding Sites; Brain; Convulsants; Diazepam; Electroshock; Flumazenil; Male; Mice; Pentylenetetrazole; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1984
Changes in benzodiazepine receptors by acute stress: different effect of chronic diazepam or RO 15-1788 treatment.
    European journal of pharmacology, 1983, Dec-23, Volume: 96, Issue:3-4

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Cerebral Cortex; Diazepam; Female; Flumazenil; Flunitrazepam; Hippocampus; Male; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Stress, Physiological

1983
A benzodiazepine antagonist action of CL 218,872.
    Life sciences, 1984, May-28, Volume: 34, Issue:22

    Topics: Animals; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Convulsants; Diazepam; Flumazenil; Male; Mice; Mice, Inbred C57BL; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1984
Ro 15-1788 and beta-CCE selectively eliminate diazepam-induced feeding in the rabbit.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 20, Issue:5

    Topics: Animals; Benzodiazepinones; Carbolines; Chlorpromazine; Cyproheptadine; Diazepam; Eating; Flumazenil; Indoles; Rabbits; Receptors, Cell Surface; Receptors, GABA-A; Water Deprivation

1984
Benzodiazepine inhibition of adenosine uptake is not prevented by benzodiazepine antagonists.
    European journal of pharmacology, 1983, Jan-28, Volume: 87, Issue:1

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Flumazenil; Flurazepam; Hexobendine; In Vitro Techniques; Pyrazoles; Rats; Rats, Inbred Strains; Synaptosomes; Temperature

1983
Inhibition of cold-induced TSH release by benzodiazepines.
    Brain research, 1983, Apr-18, Volume: 265, Issue:2

    Topics: Animals; Benzodiazepinones; Clonazepam; Cold Temperature; Depression, Chemical; Diazepam; Drug Interactions; Flumazenil; Male; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Thyrotropin; Thyrotropin-Releasing Hormone

1983
Diazepam-induced release of behavior in an extinction procedure: its reversal by Ro 15-1788.
    European journal of pharmacology, 1983, Mar-18, Volume: 88, Issue:1

    Topics: Amnesia; Animals; Behavior, Animal; Benzodiazepinones; Diazepam; Drinking; Extinction, Psychological; Flumazenil; Humans; Punishment; Rats

1983
Convulsions induced by submaximal dose of pentylenetetrazol in mice are antagonized by the benzodiazepine antagonist Ro 15-1788.
    Life sciences, 1983, May-30, Volume: 32, Issue:22

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Flumazenil; Male; Mice; Pentylenetetrazole; Seizures

1983
Selective effects of diltiazem, a benzothiazepine calcium channel blocker, and diazepam, and other benzodiazepines on the Na+/Ca2+ exchange carrier system of heart and brain mitochondria.
    Life sciences, 1983, Jun-20, Volume: 32, Issue:25

    Topics: Animals; Benzazepines; Benzodiazepines; Benzodiazepinones; Brain; Calcium; Carrier Proteins; Clonazepam; Diazepam; Diltiazem; Flumazenil; Mitochondria; Mitochondria, Heart; Rabbits; Rats; Sodium; Sodium-Calcium Exchanger

1983
Reversal of the muscle relaxant effect of diazepam but not of progabide by a specific benzodiazepine antagonist: Ro 15-1788.
    European journal of pharmacology, 1983, May-20, Volume: 90, Issue:1

    Topics: Animals; Benzodiazepinones; Diazepam; Female; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Male; Muscle Contraction; Muscle Relaxants, Central; Rats; Rats, Inbred Strains; Time Factors

1983
Diazepam, pentobarbital, and methaqualone effects on several behaviors in the rat and antagonism by Ro 15-1788.
    NIDA research monograph, 1983, Volume: 43

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Diazepam; Female; Flumazenil; Methaqualone; Pentobarbital; Postural Balance; Rats; Rats, Inbred Strains

1983
A benzodiazepine antagonist is an anticonvulsant in an animal model for limbic epilepsy.
    Brain research, 1983, Jul-04, Volume: 270, Issue:2

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Diazepam; Drug Interactions; Flumazenil; Kindling, Neurologic; Male; Rats; Seizures

1983
Anxiogenic aspects of diazepam withdrawal can be detected in animals.
    European journal of pharmacology, 1983, Aug-19, Volume: 92, Issue:1-2

    Topics: Animals; Anxiety; Benzodiazepinones; Diazepam; Discrimination Learning; Flumazenil; Humans; Male; Pentobarbital; Pentylenetetrazole; Rats; Substance Withdrawal Syndrome

1983
Diazepam antagonizes GABA- and muscimol-induced changes of acetylcholine release in slices of guinea-pig cerebral cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:1

    Topics: Acetylcholine; Animals; Benzodiazepinones; Cerebral Cortex; Diazepam; Flumazenil; GABA Antagonists; Guinea Pigs; In Vitro Techniques; Muscimol; Oxazoles

1983
Studies on [3H]diazepam and [3H]ethyl-beta-carboline carboxylate binding to rat brain in vivo. I. Regional variations in displacement.
    Journal of neurochemistry, 1983, Volume: 41, Issue:6

    Topics: Animals; Benzodiazepinones; Brain; Carbolines; Convulsants; Diazepam; Flumazenil; Flurazepam; Indoles; Male; Rats; Rats, Inbred Strains; Tissue Distribution

1983
Inhibition of adenosine accumulation by a CNS benzodiazepine antagonist (Ro 15-1788) and a peripheral benzodiazepine receptor ligand (Ro 05-4864).
    Neuroscience letters, 1983, Oct-31, Volume: 41, Issue:1-2

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Central Nervous System; Diazepam; Flumazenil; Flurazepam; Hexobendine; Male; Rats; Synaptosomes; Time Factors

1983
Reversal of the muscle relaxant effect of diazepam by the specific benzodiazepine antagonist Ro 15-1788: an electromyographic study in morphine model of muscular rigidity in rats.
    Life sciences, 1983, Volume: 33 Suppl 1

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Diazepam; Drug Antagonism; Flumazenil; Male; Morphine; Muscle Contraction; Muscle Relaxation; Rats; Rats, Inbred Strains

1983
Mechanism of potentiation by diazepam of adenosine response.
    Life sciences, 1984, Jan-02, Volume: 34, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Animals; Benzodiazepinones; Cecum; Diazepam; Dipyridamole; Dose-Response Relationship, Drug; Drug Synergism; Female; Flumazenil; Hypoxanthine; Hypoxanthines; Inosine; Male; Rats; Rats, Inbred Strains

1984
[Prolonged coma caused by diazepam sedation in ventilated patients. Diagnostic and therapeutic use of the benzodiazepine antagonist Ro 15-1788].
    Deutsche medizinische Wochenschrift (1946), 1984, Mar-02, Volume: 109, Issue:9

    Topics: Aged; Benzodiazepinones; Coma; Convulsants; Diazepam; Electroencephalography; Female; Flumazenil; Humans; Male; Middle Aged; Respiration, Artificial

1984
Intrinsic and antagonistic effects of beta-carboline FG 7142 on behavioral and EEG actions of benzodiazepines and pentobarbital in cats.
    European journal of pharmacology, 1983, Nov-11, Volume: 95, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Carbolines; Cats; Diazepam; Drug Interactions; Electroencephalography; Flumazenil; Indoles; Male; Pentobarbital

1983
Antagonism of caffeine-induced seizures in mice by Ro15-1788.
    European journal of pharmacology, 1984, Jan-27, Volume: 97, Issue:3-4

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Caffeine; Diazepam; Female; Flumazenil; Mice; Receptors, Drug; Seizures

1984
Diazepam blocks fear-enhanced startle elicited electrically from the brainstem.
    Physiology & behavior, 1984, Volume: 32, Issue:2

    Topics: Animals; Benzodiazepinones; Cochlea; Conditioning, Classical; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Fear; Flumazenil; Male; Rats; Rats, Inbred Strains; Reflex, Startle

1984
Evidence against the involvement of serotonergic neurons in the anti-punishment activity of diazepam in the rat.
    Psychopharmacology, 1984, Volume: 82, Issue:4

    Topics: 5,7-Dihydroxytryptamine; Animals; Benzodiazepinones; Conditioning, Operant; Diazepam; Dihydroxytryptamines; Electroshock; Flumazenil; Injections; Male; Neurons; Punishment; Raphe Nuclei; Rats; Rats, Inbred Strains; Reinforcement Schedule; Serotonin; Substantia Nigra

1984
Precipitated diazepam withdrawal in baboons: effects of dose and duration of diazepam exposure.
    European journal of pharmacology, 1984, Apr-20, Volume: 100, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Humans; Male; Papio; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1984
Effects of a benzodiazepine antagonist on the diazepam-induced electrical brain activity modifications.
    Neuropsychobiology, 1984, Volume: 11, Issue:1

    Topics: Adult; Benzodiazepinones; Brain; Diazepam; Electroencephalography; Evoked Potentials, Auditory; Flumazenil; Humans

1984
Anticonvulsant and antipunishment effects of toluene.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:2

    Topics: Animals; Benzodiazepinones; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Male; Mice; Pentylenetetrazole; Punishment; Rats; Seizures; Time Factors; Toluene; Xylenes

1984
Biphasic effects of Ro 15-1788 on spontaneous petit mal-like seizures in rats.
    European journal of pharmacology, 1984, Jul-13, Volume: 102, Issue:2

    Topics: Animals; Anticonvulsants; Benzodiazepinones; Convulsants; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electroencephalography; Epilepsy, Absence; Flumazenil; Male; Rats; Rats, Inbred Strains

1984
CGS 8216, Ro 15-1788 and methyl-beta-carboline-3-carboxylate, but not EMD 41717 antagonize the muscle relaxant effect of diazepam in genetically spastic rats.
    Life sciences, 1984, Oct-01, Volume: 35, Issue:14

    Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Electromyography; Female; Flumazenil; Imidazoles; Kinetics; Male; Muscle Contraction; Muscle Relaxation; Muscle Spasticity; Pyrazoles; Rats; Rats, Mutant Strains

1984
Bioassay of subjective effects associated with benzodiazepine withdrawal in animals: a novel direction in dependence research.
    NIDA research monograph, 1984, Volume: 49

    Topics: Animals; Benzodiazepinones; Biological Assay; Clonidine; Conditioning, Operant; Diazepam; Discrimination Learning; Flumazenil; Generalization, Stimulus; Humans; Male; Pentobarbital; Pentylenetetrazole; Rats; Substance Withdrawal Syndrome; Substance-Related Disorders

1984
The effects of RO15-1788, alone and in combination with diazepam, on ethanol-induced loss of righting reflex in rats.
    NIDA research monograph, 1984, Volume: 49

    Topics: Animals; Benzodiazepinones; Diazepam; Drug Synergism; Ethanol; Flumazenil; Motor Skills; Rats; Reflex

1984
Characterization of convulsions induced by methyl beta-carboline-3-carboxylate in mice.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electroencephalography; Flumazenil; Hypnotics and Sedatives; Indoles; Male; Mice; Pentylenetetrazole; Postural Balance; Time Factors

1984
Use of the specific benzodiazepine antagonist, Ro 15-1788, in studies of physiological dependence on benzodiazepines.
    Experientia, 1982, Jul-15, Volume: 38, Issue:7

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Cats; Diazepam; Female; Flumazenil; Humans; Lorazepam; Male; Mice; Rats; Saimiri; Substance Withdrawal Syndrome; Substance-Related Disorders; Triazolam

1982
Effects of benzodiazepines on single unit activity in the substantia nigra pars reticulata.
    Life sciences, 1982, Sep-06, Volume: 31, Issue:10

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Bicuculline; Caffeine; Diazepam; Dose-Response Relationship, Drug; Electric Conductivity; Flumazenil; Flurazepam; Male; Neurons; Picrotoxin; Rats; Rats, Inbred Strains; Substantia Nigra; Theophylline

1982
The effect of a benzodiazepine antagonist, RO15-1788, in diazepam dependent rats.
    Life sciences, 1982, Aug-23, Volume: 31, Issue:8

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Humans; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Substance-Related Disorders

1982
Modification of the anticonvulsant efficacy of diazepam by Ro-15-1788 in the kindled amygdaloid seizure model.
    Life sciences, 1982, Oct-11, Volume: 31, Issue:15

    Topics: Amygdala; Animals; Anticonvulsants; Benzodiazepinones; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Electric Stimulation; Flumazenil; Kindling, Neurologic; Male; Rats; Rats, Inbred Strains; Seizures

1982
Blockade of 3-carbomethoxy-beta-carboline induced seizures by diazepam and the benzodiazepine antagonists, Ro 15-1788 and CGS 8216.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:3

    Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Harmaline; Indoles; Male; Mice; Pyrazoles; Seizures; Tremor

1982
Ro 15-1788 antagonizes the discriminative stimulus effects of diazepam in rats but not similar effects of pentobarbital.
    Life sciences, 1982, Nov-08, Volume: 31, Issue:19

    Topics: Animals; Benzodiazepinones; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Kinetics; Male; Pentobarbital; Rats; Rats, Inbred F344

1982
Methyl-beta-carboline-induced convulsions are antagonized by Ro 15-1788 and by propyl-beta-carboline.
    European journal of pharmacology, 1982, Nov-05, Volume: 85, Issue:1

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Flumazenil; Indoles; Papio; Photosensitivity Disorders; Seizures; Time Factors

1982
Reversal of the anticonvulsant effects of diazepam on amygdaloid-kindled seizures by a specific benzodiazepine antagonist: RO 15-1788.
    European journal of pharmacology, 1982, Dec-17, Volume: 86, Issue:1

    Topics: Amygdala; Animals; Anticonvulsants; Benzodiazepinones; Diazepam; Electroencephalography; Flumazenil; Kindling, Neurologic; Male; Rats; Rats, Inbred Strains

1982
Benzodiazepines influence melatonin secretion of the pineal organ of the trout in vitro.
    Journal of pineal research, 1994, Volume: 17, Issue:2

    Topics: 5-Methoxytryptamine; Animals; Benzodiazepines; Calcium; Clonazepam; Culture Media; Dark Adaptation; Diazepam; Flumazenil; Hydroxyindoleacetic Acid; In Vitro Techniques; Indoles; Isoquinolines; Light; Magnesium; Melatonin; Oncorhynchus mykiss; Pineal Gland

1994
Effect of diazepam on cortical 5-HT release and behaviour in the guinea-pig on exposure to the elevated plus maze.
    Psychopharmacology, 1993, Volume: 110, Issue:4

    Topics: Animals; Anxiety; Behavior, Animal; Diazepam; Exploratory Behavior; Extracellular Space; Female; Flumazenil; Guinea Pigs; Hydroxyindoleacetic Acid; Microdialysis; Prefrontal Cortex; Serotonin

1993
Role of GABAergic systems in the development of morphine tolerance in formalin-treated mice.
    Japanese journal of pharmacology, 1995, Volume: 68, Issue:2

    Topics: Analgesics, Opioid; Animals; Baclofen; Bicuculline; Diazepam; Drug Tolerance; Flumazenil; Formaldehyde; GABA Agonists; GABA Antagonists; Male; Mice; Mice, Inbred Strains; Morphine; Muscimol; Pain; Pain Measurement; Receptors, GABA

1995
Involvement of benzodiazepine/GABA-A receptor complex in ethanol-induced state-dependent learning in rats.
    Brain research, 1995, Jul-17, Volume: 686, Issue:1

    Topics: Animals; Avoidance Learning; Azides; Benzodiazepines; Bicuculline; Diazepam; Ethanol; Evaluation Studies as Topic; Flumazenil; Male; Muscimol; Picrotoxin; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A

1995
Flunitrazepam and nordiazepam slowly released from silastic capsules induce physical dependence in rat.
    Drug and alcohol dependence, 1995, Volume: 39, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Antidotes; Biological Availability; Delayed-Action Preparations; Diazepam; Drug Implants; Female; Flumazenil; Flunitrazepam; Nordazepam; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Substance-Related Disorders

1995
Stereospecific transduction of behavioral effects via diazepam-insensitive GABAA receptors.
    European journal of pharmacology, 1995, May-24, Volume: 278, Issue:3

    Topics: Animals; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Columbidae; Diazepam; Discrimination Learning; Flumazenil; GABA Modulators; Imidazoles; Male; Midazolam; Oxadiazoles; Radioligand Assay; Receptors, GABA-A; Sensitivity and Specificity; Stereoisomerism

1995
Precipitated withdrawal in squirrel monkeys after repeated daily oral administration of alprazolam, diazepam, flunitrazepam or oxazepam.
    Psychopharmacology, 1995, Volume: 118, Issue:3

    Topics: Administration, Oral; Alprazolam; Animals; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drug Tolerance; Female; Flumazenil; Flunitrazepam; Male; Muscle Relaxation; Oxazepam; Saimiri; Sleep; Substance Withdrawal Syndrome; Substance-Related Disorders; Tremor

1995
Effects of intravenous anesthetics on phosphatidylinositol turnover in rat cerebral cortical prisms.
    Anesthesia and analgesia, 1994, Volume: 79, Issue:2

    Topics: Anesthetics, Intravenous; Animals; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Droperidol; Fentanyl; Flumazenil; Inositol Phosphates; Ketamine; Male; Naloxone; Norepinephrine; Phosphatidylinositols; Prazosin; Rats; Rats, Wistar; Thiamylal

1994
Oral flumazenil in the treatment of epilepsy.
    The Annals of pharmacotherapy, 1995, Volume: 29, Issue:5

    Topics: Administration, Oral; Clinical Trials as Topic; Diazepam; Drug Therapy, Combination; Epilepsy; Epilepsy, Generalized; Flumazenil; Humans; Randomized Controlled Trials as Topic; Single-Blind Method

1995
Benzodiazepine agonists reverse the effects of noise exposure on central benzodiazepine receptors and cardiac responsiveness.
    Life sciences, 1995, Volume: 57, Issue:11

    Topics: Animals; Brain; Clonazepam; Diazepam; Flumazenil; Imidazoles; Male; Myocardium; Noise; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, GABA-A; Stress, Psychological

1995
Gastrointestinal effects of diazepam-withdrawal are linked to activation of central cholecystokinin-ergic pathways in rats.
    The Journal of pharmacy and pharmacology, 1994, Volume: 46, Issue:10

    Topics: Animals; Benzodiazepinones; Brain; Cholecystokinin; Devazepide; Diazepam; Flumazenil; Gastrointestinal Motility; Gastrointestinal Transit; Male; Phenylurea Compounds; Rats; Rats, Wistar; Receptors, Cholecystokinin; Substance Withdrawal Syndrome

1994
The effects of drugs acting at GABA-benzodiazepine-barbiturate receptor complex on the behaviour of sleep-deprived mice.
    Pharmacology & toxicology, 1995, Volume: 76, Issue:1

    Topics: Analysis of Variance; Animals; Azides; Behavior, Animal; Benzodiazepines; Convulsants; Diazepam; Flumazenil; Male; Mice; Receptors, GABA-A; Sleep Deprivation

1995
Paradoxical reactions to diazepam.
    Gastrointestinal endoscopy, 1995, Volume: 41, Issue:2

    Topics: Conscious Sedation; Diazepam; Flumazenil; Humans; Psychomotor Agitation

1995
Different location of benzodiazepine sites involved in gut and behavioral effects of benzodiazepine withdrawal in rats.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Capsaicin; Diazepam; Digestive System; Flumazenil; Gastric Emptying; Injections, Intraventricular; Male; Rats; Rats, Wistar; Receptors, GABA-A; Substance Withdrawal Syndrome

1994
Diazepam attenuates hyperexcitability and mechanical hypersensitivity of dorsal horn convergent neurones during reperfusion of the rat's tail following ischaemia.
    Brain research, 1994, Oct-03, Volume: 659, Issue:1-2

    Topics: Animals; Diazepam; Electrophysiology; Flumazenil; Ischemia; Male; Naloxone; Neurons; Physical Stimulation; Rats; Rats, Sprague-Dawley; Reperfusion; Spinal Cord; Tail

1994
Discriminative stimulus properties of a new anxiolytic, DN-2327, in rats.
    Psychopharmacology, 1993, Volume: 110, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Buspirone; Cues; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; Generalization, Stimulus; Isoindoles; Male; Naphthyridines; Pentobarbital; Pentylenetetrazole; Rats; Rats, Wistar; Spiro Compounds

1993
Benzodiazepine receptor mediation of the anxiolytic-like effect of (-)-nicotine in mice.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Diazepam; Flumazenil; Male; Mecamylamine; Mice; Nicotine; Receptors, GABA-A; Receptors, Nicotinic

1994
Corticosterone increases severity of acute withdrawal from ethanol, pentobarbital, and diazepam in mice.
    Psychopharmacology, 1994, Volume: 115, Issue:1-2

    Topics: Animals; Behavior, Animal; Corticosterone; Diazepam; Ethanol; Female; Flumazenil; Handling, Psychological; Mice; Mice, Inbred Strains; Pentobarbital; Seizures; Substance Withdrawal Syndrome

1994
Role of benzodiazepine receptors located in the dorsal periaqueductal grey of rats in anxiety.
    Psychopharmacology, 1993, Volume: 110, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anticonvulsants; Anxiety; Appetite Depressants; Carbolines; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Male; Microinjections; Midazolam; Periaqueductal Gray; Rats; Rats, Wistar; Receptors, GABA-A

1993
Diazepam and gepirone selectively attenuate either 20-32 or 32-64 kHz ultrasonic vocalizations during aggressive encounters.
    Psychopharmacology, 1993, Volume: 112, Issue:1

    Topics: Aggression; Animals; Anti-Anxiety Agents; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Male; Motor Activity; Pain Measurement; Pyrimidines; Rats; Vocalization, Animal

1993
Differential profile of the CCKB receptor antagonist CI-988 and diazepam in the four-plate test.
    Psychopharmacology, 1993, Volume: 112, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Electroshock; Exploratory Behavior; Flumazenil; Indoles; Male; Meglumine; Mice; Ondansetron; Receptors, Cholecystokinin

1993
Effects of the non-NMDA antagonists NBQX and the 2,3-benzodiazepine GYKI 52466 on different seizure types in mice: comparison with diazepam and interactions with flumazenil.
    British journal of pharmacology, 1994, Volume: 113, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Excitatory Amino Acid Antagonists; Flumazenil; Male; Mice; Muscle Relaxants, Central; Pentylenetetrazole; Quinoxalines; Receptors, AMPA; Reflex; Seizures; Synaptic Transmission

1994
Different functional effect of Ro 15-4513 and Ro 19-4603 on synaptic responses of Purkinje cells in the rat cerebellar slice.
    Brain research, 1994, Dec-05, Volume: 665, Issue:2

    Topics: Animals; Azepines; Azides; Benzodiazepines; Cerebellum; Diazepam; Electrophysiology; Flumazenil; In Vitro Techniques; Male; Neural Inhibition; Purkinje Cells; Rats; Rats, Wistar; Receptors, GABA-A; Synapses

1994
Gender differences in diazepam withdrawal syndrome in mice.
    Pharmacology & toxicology, 1994, Volume: 75, Issue:6

    Topics: Animals; Body Weight; Castration; Diazepam; Disease Models, Animal; Estrogens; Female; Flumazenil; Injections, Intraperitoneal; Male; Mice; Seizures; Sex Characteristics; Substance Withdrawal Syndrome; Testosterone

1994
Repeated treatment with alpidem, a new anxiolytic, does not induce tolerance or physical dependence.
    Neuropharmacology, 1993, Volume: 32, Issue:9

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Bicuculline; Carbolines; Convulsants; Diazepam; Drug Tolerance; Flumazenil; Imidazoles; Isoniazid; Male; Mice; Pentylenetetrazole; Pyridines; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
A system for testing the development and reversal of anticonvulsant tolerance to benzodiazepines in mice.
    Epilepsy research, 1993, Volume: 16, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Carbolines; Diazepam; Drug Tolerance; Flumazenil; Flunitrazepam; Infusion Pumps, Implantable; Infusions, Parenteral; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Seizures; Solvents; Time Factors

1993
Anxiolytic activity of melatonin in mice: involvement of benzodiazepine receptors.
    Research communications in chemical pathology and pharmacology, 1993, Volume: 82, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Choice Behavior; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Melatonin; Mice; Motor Activity; Receptors, GABA-A

1993
Duodenal bicarbonate secretion and mucosal protection. Neurohumoral influence and transport mechanisms.
    Acta physiologica Scandinavica. Supplementum, 1993, Volume: 613

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antiporters; Bicarbonates; Biological Transport; Carbachol; Carrier Proteins; Catechol O-Methyltransferase Inhibitors; Catechols; Chloride-Bicarbonate Antiporters; Cyclic AMP; Cytophotometry; Diazepam; Dopamine; Dopamine Agents; Duodenum; Ergolines; Flumazenil; Gastric Mucosa; Intestinal Mucosa; Male; Microvilli; Pentanones; Phentolamine; Pirenzepine; Quinpirole; Radioimmunoassay; Rana catesbeiana; Rats; Rats, Sprague-Dawley; Sodium-Bicarbonate Symporters; Sodium-Hydrogen Exchangers; Ulcer

1993
Possible anxiolytic effects of chrysin, a central benzodiazepine receptor ligand isolated from Passiflora coerulea.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Exploratory Behavior; Flavonoids; Flumazenil; Male; Mice; Mice, Inbred Strains; Motor Activity; Plants, Medicinal; Receptors, GABA-A

1994
Dehydroepiandrosterone is an anxiolytic in mice on the plus maze.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; Diazepam; Ethanol; Flumazenil; Male; Mice; Mice, Inbred C57BL; Motor Activity; Pentylenetetrazole; Receptors, GABA

1994
F 2692: flumazenil-reversible anxiolytic effects but inactive on [3H]-Ro 15-4513 binding.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:1

    Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding, Competitive; Carbolines; Cerebellum; Diazepam; Flumazenil; GABA-A Receptor Antagonists; In Vitro Techniques; Interpersonal Relations; Male; Membranes; Motor Activity; Pyridazines; Rats; Receptors, GABA-A

1994
Involvement of pain associated anxiety in the development of morphine tolerance in formalin treated mice.
    Japanese journal of pharmacology, 1994, Volume: 65, Issue:4

    Topics: Animals; Anxiety; Aspirin; Diazepam; Drug Tolerance; Flumazenil; Formaldehyde; Indomethacin; Inflammation; Male; Mice; Morphine; Pain; Pain Threshold; Receptors, GABA-A

1994
Differential effects of abecarnil on basal release of acetylcholine and dopamine in the rat brain.
    European journal of pharmacology, 1994, Aug-11, Volume: 261, Issue:1-2

    Topics: Acetylcholine; Animals; Anti-Anxiety Agents; Brain; Carbolines; Diazepam; Dopamine; Flumazenil; GABA-A Receptor Agonists; Hippocampus; Male; Microdialysis; Neurons; Prefrontal Cortex; Rats; Rats, Sprague-Dawley

1994
Ejaculation induced changes in escape latency in the hot plate test: pharmacological analysis of anxiolytic versus analgesic effect.
    Behavioural brain research, 1994, Feb-28, Volume: 60, Issue:2

    Topics: Animals; Arousal; Copulation; Diazepam; Ejaculation; Escape Reaction; Female; Flumazenil; Habituation, Psychophysiologic; Male; Morphine; Naloxone; Pain Threshold; Rats; Rats, Wistar; Reaction Time; Thermosensing; Vocalization, Animal

1994
The benzodiazepine receptor antagonist flumazenil increases acetylcholine release in rat hippocampus.
    Brain research, 1994, May-30, Volume: 647, Issue:1

    Topics: Acetylcholine; Animals; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Antagonists; Hippocampus; Injections; Injections, Intraperitoneal; Male; Microdialysis; Rats; Rats, Sprague-Dawley; Septum Pellucidum

1994
Seizure after reversal of benzodiazepine treatment with flumazenil: a report of two cases.
    Zhonghua yi xue za zhi = Chinese medical journal; Free China ed, 1994, Volume: 53, Issue:6

    Topics: Aged; Diazepam; Female; Flumazenil; Humans; Male; Middle Aged; Receptors, GABA; Seizures

1994
Melatonin as an anxiolytic in rats: time dependence and interaction with the central GABAergic system.
    European journal of pharmacology, 1993, Jun-24, Volume: 237, Issue:2-3

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Behavior, Animal; Brain; Circadian Rhythm; Diazepam; Dose-Response Relationship, Drug; Drug Administration Schedule; Flumazenil; gamma-Aminobutyric Acid; Male; Melatonin; Rats; Rats, Wistar

1993
Flumazenil as a diagnostic tool in the differential diagnosis of coma in a critically ill patient.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1994, Volume: 41, Issue:1

    Topics: Aged; Bacterial Infections; Coma; Critical Illness; Diagnosis, Differential; Diazepam; Flumazenil; Hepatic Encephalopathy; Humans; Lorazepam; Male; Midazolam

1994
Flumazenil induces localised increases in glucose utilization during diazepam withdrawal in rats.
    Brain research, 1993, Dec-24, Volume: 631, Issue:2

    Topics: Animals; Autoradiography; Brain Chemistry; Carbolines; Densitometry; Deoxyglucose; Diazepam; Flumazenil; Glucose; Male; Rats; Substance Withdrawal Syndrome

1993
Flumazenil induces seizures and death in mixed cocaine-diazepam intoxications.
    Annals of emergency medicine, 1994, Volume: 23, Issue:3

    Topics: Animals; Cocaine; Diazepam; Electroencephalography; Flumazenil; Male; Rats; Rats, Sprague-Dawley; Seizures

1994
[A pregnant woman with convulsion treated with diazepam which was reversed with flumazenil just prior to cesarean section].
    Masui. The Japanese journal of anesthesiology, 1994, Volume: 43, Issue:4

    Topics: Adult; Anesthesia, General; Anesthesia, Obstetrical; Cesarean Section; Diazepam; Eclampsia; Emergencies; Female; Flumazenil; Humans; Injections, Intravenous; Pregnancy

1994
[The effect of flumazenil administration on acute cocaine intoxication of rats].
    Arukoru kenkyu to yakubutsu izon = Japanese journal of alcohol studies & drug dependence, 1994, Volume: 29, Issue:2

    Topics: Acute Disease; Animals; Cocaine; Diazepam; Flumazenil; Male; Poisoning; Rats; Rats, Wistar

1994
Propofol activates GABAA receptor-chloride ionophore complex in dissociated hippocampal pyramidal neurons of the rat.
    Anesthesiology, 1993, Volume: 79, Issue:4

    Topics: Animals; Central Nervous System; Chloride Channels; Chlorides; Diazepam; Flumazenil; Hippocampus; Kinetics; Membrane Potentials; Neurons; Propofol; Pyramidal Tracts; Rats; Rats, Wistar; Receptors, GABA

1993
Pentobarbital, diazepam, and ethanol abolish the interphase diminution of pain in the formalin test: evidence for pain modulation by GABAA receptors.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 46, Issue:3

    Topics: Analgesics; Animals; Chloride Channels; Diazepam; Ethanol; Flumazenil; Formaldehyde; Male; Pain Measurement; Pentobarbital; Picrotoxin; Rats; Receptors, GABA-A

1993
Precipitated abstinence in the diazepam-dependent rat.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 46, Issue:3

    Topics: Animals; Behavior, Animal; Brain; Diazepam; Drug Implants; Epilepsy, Tonic-Clonic; Female; Flumazenil; Microdialysis; Particle Size; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
Effects of benzodiazepine agonist, antagonist and inverse agonist on ethanol-induced changes in beta-endorphin levels in specific rat brain regions.
    Pharmacology, 1993, Volume: 47, Issue:6

    Topics: Affinity Labels; Animals; Azides; Benzodiazepines; beta-Endorphin; Brain Chemistry; Cerebral Cortex; Diazepam; Ethanol; Flumazenil; Hippocampus; Hypothalamus; Male; Rats; Rats, Sprague-Dawley

1993
Attenuation of reperfusion hyperalgesia in the rat by systemic administration of benzodiazepines.
    British journal of pharmacology, 1993, Volume: 110, Issue:3

    Topics: Animals; Behavior, Animal; Benzodiazepines; Chlordiazepoxide; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Hyperalgesia; Ischemia; Male; Motor Activity; Naloxone; Pain Measurement; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Reperfusion Injury; Tail

1993
In vitro inhibition of cellular immune responses by benzodiazepines and PK 11195. Effects on mitogen- and alloantigen-driven lymphocyte proliferation and on IL-1, IL-2 synthesis and IL-2 receptor expression.
    Immunopharmacology and immunotoxicology, 1993, Volume: 15, Issue:5

    Topics: Animals; B-Lymphocytes; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Female; Flumazenil; Immunity, Cellular; In Vitro Techniques; Interleukin-1; Interleukin-2; Isoquinolines; Lymphocyte Activation; Male; Mice; Mice, Inbred A; Mice, Inbred C57BL; Neuroimmunomodulation; Receptors, GABA-A; T-Lymphocytes

1993
Flumazenil reverses diazepam-induced neonatal apnoea and hypotonia.
    European journal of pediatrics, 1993, Volume: 152, Issue:5

    Topics: Apnea; Diazepam; Flumazenil; Humans; Infant, Newborn; Male; Muscle Hypotonia

1993
Functional integrity of benzodiazepine receptors of the geniculo-striate visual pathways in Creutzfeldt-Jakob disease. A pharmacological evoked potential study.
    Journal of neurology, 1993, Volume: 240, Issue:1

    Topics: Creutzfeldt-Jakob Syndrome; Diazepam; Evoked Potentials, Visual; Flumazenil; Humans; Male; Middle Aged; Reaction Time; Receptors, GABA-A; Visual Cortex

1993
Interaction between benzodiazepine and GABA-A receptors in state-dependent learning.
    Life sciences, 1993, Volume: 52, Issue:24

    Topics: Animals; Avoidance Learning; Baclofen; Bicuculline; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Muscimol; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-A; Reference Values

1993
Imidazenil: a new partial positive allosteric modulator of gamma-aminobutyric acid (GABA) action at GABAA receptors.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Benzodiazepinones; Chloride Channels; Conflict, Psychological; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Membrane Proteins; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reflex; Seizures

1993
Transduction of a discriminative stimulus through a diazepam-insensitive gamma-aminobutyric acidA receptor.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: Animals; Columbidae; Diazepam; Discrimination Learning; Flumazenil; gamma-Aminobutyric Acid; Male; Receptors, GABA-A

1993
Inhibitory effect of diazepam on the activity of the hypothalamic-pituitary-adrenal axis in female rats.
    Journal of neural transmission. General section, 1993, Volume: 92, Issue:2-3

    Topics: Adrenocorticotropic Hormone; Animals; Bicuculline; Corticosterone; Depression, Chemical; Diazepam; Female; Flumazenil; GABA-A Receptor Antagonists; Hypothalamo-Hypophyseal System; Isoquinolines; Picrotoxin; Pituitary-Adrenal System; Rats; Receptors, GABA-A

1993
Potentiation of gamma-aminobutyric acid type A receptor-mediated synaptic currents by pentobarbital and diazepam in immature hippocampal CA1 neurons.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Diazepam; Drug Synergism; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Neurons; Pentobarbital; Rats; Rats, Wistar; Receptors, GABA-A; Synapses

1993
Inhibition of hippocampal acetylcholine release by benzodiazepines: antagonism by flumazenil.
    European journal of pharmacology, 1993, Jul-06, Volume: 238, Issue:1

    Topics: Acetylcholine; Analysis of Variance; Animals; Diazepam; Drug Interactions; Flumazenil; Hippocampus; Male; Midazolam; Rats; Rats, Sprague-Dawley

1993
Pharmacokinetics of nordiazepam in physical dependence and precipitated abstinence in dogs.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:4

    Topics: Administration, Oral; Animals; Blood Proteins; Diazepam; Dogs; Female; Flumazenil; Hydrolysis; Injections, Intravenous; Nordazepam; Oxazepam; Protein Binding; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
Reversal of fetal benzodiazepine intoxication using flumazenil.
    British journal of obstetrics and gynaecology, 1993, Volume: 100, Issue:2

    Topics: Adult; Cardiotocography; Diazepam; Drug Overdose; Female; Fetal Diseases; Flumazenil; Gastric Lavage; Humans; Pregnancy

1993
Effect of the chronic dose of diazepam on the intensity and characteristics of the precipitated abstinence syndrome in the dog.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:3

    Topics: Animals; Diazepam; Dogs; Dose-Response Relationship, Drug; Female; Flumazenil; Substance Withdrawal Syndrome

1993
The relative efficacy of antidotes.
    Journal of toxicology. Clinical toxicology, 1995, Volume: 33, Issue:6

    Topics: Antidotes; Atropine; Chelating Agents; Diazepam; Flumazenil; Humans; Naloxone; Poisoning

1995
Enhancement of acetylcholine release by flumazenil in the hippocampus of rats chronically treated with diazepam but not with imidazenil or abecarnil.
    Psychopharmacology, 1995, Volume: 121, Issue:2

    Topics: Acetylcholine; Animals; Anticonvulsants; Benzodiazepines; Carbolines; Diazepam; Flumazenil; GABA Modulators; Hippocampus; Imidazoles; Male; Microdialysis; Rats; Rats, Sprague-Dawley; Time Factors

1995
Blockade of morphine-induced place preference by diazepam in mice.
    European journal of pharmacology, 1995, Jul-14, Volume: 280, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Chromatography, High Pressure Liquid; Conditioning, Psychological; Diazepam; Dopamine; Drug Interactions; Flumazenil; GABA Modulators; Homovanillic Acid; Injections, Intraperitoneal; Male; Mice; Morphine; Narcotic Antagonists

1995
[The effect of diazepam and flumazenil on pulsatile secretion of prolactin and LH in women].
    Ceska gynekologie, 1996, Volume: 61, Issue:1

    Topics: Adult; Diazepam; Female; Flumazenil; GABA Modulators; Humans; Luteinizing Hormone; Menstrual Cycle; Prolactin

1996
Long-term intravenous and oral flumazenil treatment of acute diazepam overdose in an older patient.
    Journal of the American Geriatrics Society, 1996, Volume: 44, Issue:6

    Topics: Administration, Oral; Aged; Antidotes; Coma; Diazepam; Female; Flumazenil; Glasgow Coma Scale; Humans; Infusions, Intravenous

1996
Lack of anticonvulsant tolerance and benzodiazepine receptor down regulation with imidazenil in rats.
    British journal of pharmacology, 1996, Volume: 117, Issue:4

    Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Diazepam; Down-Regulation; Drug Tolerance; Flumazenil; GABA Modulators; Imidazoles; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Tritium

1996
Diazepam increases melatonin secretion of photosensitive pineal organs of trout in the photopic and mesopic range of illumination.
    Neuroscience letters, 1996, Mar-22, Volume: 207, Issue:1

    Topics: Animals; Diazepam; Flumazenil; GABA Modulators; In Vitro Techniques; Light; Melatonin; Pineal Gland; Trout

1996
Effects of several benzodiazepines, alone and in combination with flumazenil, in rhesus monkeys trained to discriminate pentobarbital from saline.
    Psychopharmacology, 1995, Volume: 122, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Chlordiazepoxide; Conditioning, Operant; Diazepam; Discrimination Learning; Drug Interactions; Flumazenil; GABA-A Receptor Antagonists; Macaca mulatta

1995
Vigabatrin modulates benzodiazepine receptor activity in vivo: a positron emission tomography study in baboon.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:3

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flumazenil; gamma-Aminobutyric Acid; Linear Models; Male; Papio; Radioligand Assay; Receptors, GABA-A; Tomography, Emission-Computed; Vigabatrin

1996
Reciprocal effects of chronic diazepam and melatonin on brain melatonin and benzodiazepine binding sites.
    Journal of pineal research, 1996, Volume: 20, Issue:2

    Topics: Animals; Body Weight; Brain; Cerebral Cortex; Diazepam; Flumazenil; Flunitrazepam; Kinetics; Male; Medulla Oblongata; Melatonin; Pons; Rats; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Receptors, Melatonin

1996
Effects of diazepam, baclofen and thiopental on the silent period evoked by transcranial magnetic stimulation in humans.
    Experimental brain research, 1996, Volume: 109, Issue:3

    Topics: Adult; Baclofen; Diazepam; Electric Stimulation; Evoked Potentials; Flumazenil; GABA Agonists; GABA Modulators; Humans; Middle Aged; Motor Cortex; Neural Inhibition; Thiopental; Transcranial Magnetic Stimulation

1996
Anticonvulsant profile of the imidazoquinazolines NNC 14-0185 and NNC 14-0189 in rats and mice.
    European journal of pharmacology, 1996, Jul-11, Volume: 308, Issue:1

    Topics: Acoustic Stimulation; Amygdala; Animals; Anticonvulsants; Bicuculline; Carbolines; Clonazepam; Diazepam; Electroshock; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Kindling, Neurologic; Male; Mice; Mice, Inbred DBA; Mice, Inbred Strains; Pentylenetetrazole; Quinazolines; Rats; Rats, Wistar; Seizures

1996
Effects of benzodiazepine receptor ligands on isolated rat superior cervical ganglia neurons.
    Pharmacology, 1996, Volume: 52, Issue:6

    Topics: Age Factors; Animals; Animals, Newborn; Anti-Anxiety Agents; Diazepam; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Ligands; Neurons; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Superior Cervical Ganglion

1996
Functional preservation of benzodiazepine receptors of the primary somatosensory cortex in Creutzfeldt-Jakob disease: a pharmacologic-evoked potential study.
    Clinical neuropharmacology, 1996, Volume: 19, Issue:1

    Topics: Aged; Creutzfeldt-Jakob Syndrome; Diazepam; Electroencephalography; Evoked Potentials, Somatosensory; Fatal Outcome; Female; Flumazenil; GABA Modulators; Humans; Median Nerve; Receptors, GABA-A; Somatosensory Cortex

1996
Flumazenil, diazepam, nordiazepam and oxazepam interactions on plasma protein binding.
    Pharmacological research, 1995, Volume: 32, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Biotransformation; Blood Proteins; Diazepam; Dogs; Drug Interactions; Flumazenil; In Vitro Techniques; Nordazepam; Oxazepam; Protein Binding

1995
PK 11195 blockade of benzodiazepine-induced inhibition of forskolin-stimulated adenylate cyclase activity in the striatum.
    British journal of pharmacology, 1996, Volume: 119, Issue:2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Benzodiazepines; Benzodiazepinones; Colforsin; Corpus Striatum; Diazepam; Drug Interactions; Flumazenil; GABA-A Receptor Antagonists; Guanosine Triphosphate; Indoles; Isoquinolines; Kinetics; Male; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Stimulation, Chemical; Virulence Factors, Bordetella

1996
The possible involvement of GABAA systems in the antinarcotic effect of majonoside-R2, a major constituent of Vietnamese ginseng, in mice.
    Japanese journal of pharmacology, 1996, Volume: 71, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Analgesics, Opioid; Analysis of Variance; Animals; Convulsants; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Ginsenosides; Male; Mice; Morphine; Pain Measurement; Picrotoxin; Pyrrolidines; Saponins

1996
Effect of inhalation of chamomile oil vapour on plasma ACTH level in ovariectomized-rat under restriction stress.
    Biological & pharmaceutical bulletin, 1996, Volume: 19, Issue:9

    Topics: Administration, Inhalation; Adrenocorticotropic Hormone; Animals; Anti-Anxiety Agents; Diazepam; Female; Flumazenil; GABA Modulators; Hypnotics and Sedatives; Ovariectomy; Plant Oils; Plants, Medicinal; Rats; Rats, Wistar; Restraint, Physical; Stress, Psychological

1996
Diazepam physical dependence and withdrawal in rats is associated with alteration in GABAA receptor function.
    Life sciences, 1996, Volume: 59, Issue:19

    Topics: Animals; Benzodiazepines; Cerebral Cortex; Chloride Channels; Chlorides; Diazepam; Flumazenil; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred F344; Receptors, GABA-A; Substance Withdrawal Syndrome; Substance-Related Disorders

1996
Pharmacology of the human gamma-aminobutyric acidA receptor alpha 4 subunit expressed in Xenopus laevis oocytes.
    Molecular pharmacology, 1996, Volume: 50, Issue:5

    Topics: Animals; Benzodiazepines; Binding Sites; Diazepam; Electrophysiology; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; Humans; Macromolecular Substances; Pentobarbital; Receptors, GABA-A; Sensitivity and Specificity; Xenopus laevis

1996
Intraseptal flumazenil enhances, while diazepam binding inhibitor impairs, performance in a working memory task.
    Neurobiology of learning and memory, 1996, Volume: 66, Issue:3

    Topics: Animals; Diazepam; Flumazenil; Male; Maze Learning; Memory; Rats; Rats, Sprague-Dawley; Septal Nuclei; Task Performance and Analysis

1996
Characterisation of the furanocoumarin phellopterin as a rat brain benzodiazepine receptor partial agonist in vitro.
    Neuroscience letters, 1996, Nov-29, Volume: 219, Issue:3

    Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds, Heterocyclic; Coumarins; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; In Vitro Techniques; Male; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A

1996
Role of GABA-A and mitochondrial diazepam binding inhibitor receptors in the anti-stress activity of neurosteroids in mice.
    Psychopharmacology, 1996, Volume: 128, Issue:3

    Topics: Analysis of Variance; Animals; Ascorbic Acid; Behavior, Animal; Binding Sites; Cerebellum; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Antagonists; GABA Modulators; Isoquinolines; Male; Mice; Mitochondria; Motor Activity; Pain Measurement; Picrotoxin; Progesterone; Receptors, GABA-A; RNA; Stress, Psychological; Triazolam

1996
Progesterone modulation of diazepam withdrawal syndrome in mice.
    Pharmacology & toxicology, 1996, Volume: 79, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Estradiol; Estrus; Female; Flumazenil; GABA Modulators; Mice; Progesterone; Substance Withdrawal Syndrome

1996
Intrathecally administered flumazenil and PK 11195 precipitate abstinence syndrome in freely moving diazepam dependent rats.
    Drug and alcohol dependence, 1996, Dec-11, Volume: 43, Issue:3

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Electrodes, Implanted; Electroencephalography; Female; Flumazenil; GABA-A Receptor Antagonists; Injections, Spinal; Isoquinolines; Rats; Rats, Sprague-Dawley; Tremor

1996
Flumazenil reverses the decrease in the hypnotic activity of pentobarbital by social isolation stress: are endogenous benzodiazepine receptor ligands involved?
    Brain research, 1997, Jan-16, Volume: 745, Issue:1-2

    Topics: Animals; Carbolines; Chlorides; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Hypnotics and Sedatives; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred Strains; Pentobarbital; Receptors, GABA-A; Sleep; Social Isolation; Stress, Psychological; Synaptosomes

1997
In vivo modulation of benzodiazepine receptor function after inhibition of endogenous gamma-aminobutyyric acid synthesis.
    European journal of pharmacology, 1997, Feb-19, Volume: 321, Issue:1

    Topics: Allylglycine; Animals; Binding, Competitive; Brain; Convulsants; Diazepam; Electroencephalography; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Ligands; Male; Papio; Pentylenetetrazole; Tomography, Emission-Computed

1997
Stimulatory effect of diazepam on gastric acid secretion in the continuously perfused stomach in rats under urethane anesthesia.
    Research communications in molecular pathology and pharmacology, 1997, Volume: 95, Issue:2

    Topics: 3-Mercaptopropionic Acid; Analysis of Variance; Anesthetics, Intravenous; Animals; Atropine; Diazepam; Flumazenil; GABA Agents; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; Gastric Acid; Gastric Mucosa; Hexamethonium; Isoquinolines; Male; Parasympatholytics; Pentylenetetrazole; Picrotoxin; Pylorus; Rats; Rats, Wistar; Receptors, GABA; Urethane; Vagotomy

1997
Benzodiazepine receptor distribution and diazepam binding in schizophrenia: an exploratory study.
    Psychiatry research, 1997, Feb-07, Volume: 68, Issue:2-3

    Topics: Adult; Benzodiazepines; Binding Sites; Chronic Disease; Diazepam; Flumazenil; Frontal Lobe; Growth Hormone; Humans; Hydrocortisone; Occipital Lobe; Receptors, GABA-A; Schizophrenia; Temporal Lobe; Tomography, Emission-Computed, Single-Photon

1997
Sex differences in bicuculline-induced convulsions: interaction with stress and ligands of benzodiazepine binding sites.
    Brain research, 1997, Mar-28, Volume: 752, Issue:1-2

    Topics: Animals; Benzodiazepines; Bicuculline; Binding Sites; Cold Temperature; Diazepam; Differential Threshold; Dose-Response Relationship, Drug; Female; Flumazenil; Handling, Psychological; Ligands; Male; Rats; Rats, Wistar; Seizures; Sex Characteristics; Stress, Physiological; Swimming

1997
Subtle changes in residue 77 of the gamma subunit of alpha1beta2gamma2 GABAA receptors drastically alter the affinity for ligands of the benzodiazepine binding site.
    The Journal of biological chemistry, 1997, May-02, Volume: 272, Issue:18

    Topics: Animals; Benzodiazepines; Binding Sites; Cell Line; Diazepam; Female; Flumazenil; Humans; Kinetics; Macromolecular Substances; Mutagenesis, Site-Directed; Oocytes; Phenylalanine; Point Mutation; Pyridines; Radioligand Assay; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection; Xenopus laevis; Zolpidem

1997
Antianxiety profile of ondansetron, a selective 5-HT3 antagonist, in a novel animal model.
    Methods and findings in experimental and clinical pharmacology, 1997, Volume: 19, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Conflict, Psychological; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Female; Flumazenil; GABA Modulators; Male; Mice; Mice, Inbred BALB C; Ondansetron; Serotonin Antagonists

1997
Enhancement by flumazenil of dopamine release in the nucleus accumbens of rats repeatedly exposed to diazepam or imidazenil.
    Psychopharmacology, 1997, Volume: 131, Issue:1

    Topics: Animals; Benzodiazepines; Diazepam; Dopamine; Drug Synergism; Flumazenil; GABA Modulators; Imidazoles; Male; Nucleus Accumbens; Rats; Rats, Sprague-Dawley

1997
Hippocampal GABA(A) channel conductance increased by diazepam.
    Nature, 1997, Jul-03, Volume: 388, Issue:6637

    Topics: Animals; Cells, Cultured; Diazepam; Dose-Response Relationship, Drug; Electric Conductivity; Flumazenil; GABA Modulators; Hippocampus; Neurons; Rats; Receptors, GABA-A

1997
GABA(A) receptors containing the alpha4-subunit: prevalence, distribution, pharmacology, and subunit architecture in situ.
    Journal of neurochemistry, 1997, Volume: 69, Issue:2

    Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Brain; Cell Membrane; Cerebellum; Diazepam; Flumazenil; Immunohistochemistry; Immunosorbent Techniques; Macromolecular Substances; Male; Muscimol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Recombinant Proteins

1997
Benzodiazepine prevention of swim stress-induced sensitization of cortical biogenic amines: an in vivo microdialysis study.
    Neurochemical research, 1997, Volume: 22, Issue:9

    Topics: Animals; Anti-Anxiety Agents; Biogenic Amines; Carbolines; Diazepam; Drug Evaluation, Preclinical; Flumazenil; GABA Agonists; GABA Antagonists; Male; Microdialysis; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Stress, Physiological; Swimming

1997
Non-GABAergic effects of midazolam, diazepam and flumazenil on voltage-dependent ion currents in NG108-15 cells.
    Neuroreport, 1997, Jul-28, Volume: 8, Issue:11

    Topics: Animals; Calcium Channels; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Glioma; Hybrid Cells; Ion Channels; Membrane Potentials; Midazolam; Neuroblastoma; Patch-Clamp Techniques; Potassium Channels; Receptors, GABA-A; Sodium Channels

1997
Dorsal raphe and substantia nigra response to flumazenil in diazepam-dependent rats.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:1

    Topics: Animals; Diazepam; Electroencephalography; Electrophysiology; Female; Flumazenil; GABA Modulators; Microinjections; Prefrontal Cortex; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Substance-Related Disorders; Substantia Nigra

1997
Mechanism of the negative inotropic effect of midazolam and diazepam in cultured foetal mouse cardiac myocytes.
    European journal of anaesthesiology, 1997, Volume: 14, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Calcium; Calcium Channel Agonists; Cells, Cultured; Depression, Chemical; Diazepam; Female; Fetal Heart; Flumazenil; GABA-A Receptor Antagonists; Heart Rate, Fetal; Hypnotics and Sedatives; Mice; Mice, Inbred ICR; Midazolam; Pregnancy; Ryanodine; Sarcoplasmic Reticulum

1997
A fatality due to moclobemide.
    Journal of forensic sciences, 1997, Volume: 42, Issue:5

    Topics: Antidepressive Agents; Benzamides; Diazepam; Fatal Outcome; Female; Flumazenil; Humans; Liver; Middle Aged; Moclobemide; Nordazepam; Trifluoperazine

1997
Influence of anxiolytic drugs on the effects of specific serotonin reuptake inhibitors in the forced swimming test in mice.
    Journal of psychopharmacology (Oxford, England), 1997, Volume: 11, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents; Diazepam; Drug Interactions; Flumazenil; Fluoxetine; GABA Modulators; Male; Mice; Motor Activity; Selective Serotonin Reuptake Inhibitors

1997
125I-iomazenil binding shows stress- and/or diazepam-induced reductions in mouse brain: supporting data for 123I-iomazenil SPECT study of anxiety disorders.
    Annals of nuclear medicine, 1997, Volume: 11, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Autoradiography; Brain; Diazepam; Flumazenil; Iodine Radioisotopes; Male; Mice; Mice, Inbred ICR; Stress, Physiological; Tomography, Emission-Computed, Single-Photon

1997
The direct effects of diazepam and midazolam on myocardial depression in cultured rat ventricular myocytes.
    Anesthesia and analgesia, 1997, Volume: 85, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Cells, Cultured; Depression, Chemical; Diazepam; Flumazenil; Heart; Heart Rate; Midazolam; Rats

1997
Comparison of abstinence syndromes precipitated by flumazenil and PK 11195 in female diazepam-dependent rats.
    Psychopharmacology, 1997, Volume: 133, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Central Nervous System; Diazepam; Dose-Response Relationship, Drug; Drug Implants; Female; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Isoquinolines; Male; Peripheral Nervous System; Rats; Rats, Sprague-Dawley; Seizures; Sex Characteristics; Substance Withdrawal Syndrome; Substance-Related Disorders

1997
Use of inhalational and intravenous sedation in dentistry.
    International dental journal, 1997, Volume: 47, Issue:1

    Topics: Accidents; Anesthesia, Dental; Anesthesia, Inhalation; Anesthesia, Intravenous; Anesthesia, Local; Anesthetics, Inhalation; Anesthetics, Intravenous; Anti-Anxiety Agents; Antidotes; Cause of Death; Computers; Conscious Sedation; Dental Care; Diazepam; Drug Overdose; Emergencies; Flumazenil; GABA Modulators; Humans; Hypnotics and Sedatives; Iatrogenic Disease; Infusion Pumps; Isoflurane; Midazolam; Nitrous Oxide; Oxygen; Practice Guidelines as Topic; Propofol; United Kingdom

1997
Interaction between alpha-MSH and gabaergic agents upon striatal cAMP levels: an in vitro model.
    Peptides, 1998, Volume: 19, Issue:2

    Topics: alpha-MSH; Animals; Baclofen; Benzazepines; Corpus Striatum; Cyclic AMP; Diazepam; Drug Interactions; Flumazenil; GABA Agents; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Male; Models, Neurological; Rats; Rats, Wistar; Receptors, Dopamine D1

1998
Neonatal flumazenil therapy reverses maternal diazepam.
    Acta paediatrica (Oslo, Norway : 1992), 1998, Volume: 87, Issue:2

    Topics: Adult; Anticonvulsants; Antidotes; Apnea; Chromatography, High Pressure Liquid; Diazepam; Eclampsia; Emergency Treatment; Female; Flumazenil; Humans; Infant, Newborn; Male; Maternal-Fetal Exchange; Pregnancy

1998
The anxiolytic effect of gamma-hydroxybutyrate in the elevated plus maze is reversed by the benzodiazepine receptor antagonist, flumazenil.
    European journal of pharmacology, 1998, Jan-19, Volume: 342, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Benzocycloheptenes; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Male; Motor Activity; Naloxone; Narcotic Antagonists; Rats; Sodium Oxybate

1998
The effect of chronic benzodiazepines exposure on body weight in rats.
    Pharmacological research, 1998, Volume: 37, Issue:3

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Flunitrazepam; GABA Modulators; Male; Nordazepam; Oxazepam; Rats; Rats, Sprague-Dawley; Sex Factors; Time Factors; Weight Gain

1998
Modification of the anxiolytic action of 5-HT1A compounds by GABA-benzodiazepine agents in rats.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 60, Issue:1

    Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Anxiety; Bicuculline; Buspirone; Diazepam; Drug Interactions; Flumazenil; GABA Agonists; Male; Psychomotor Performance; Pyrimidines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1

1998
Evidence of GABAergic modulation in melatonin-induced short-term memory deficits and food consumption.
    Methods and findings in experimental and clinical pharmacology, 1998, Volume: 20, Issue:4

    Topics: Animals; Antioxidants; Diazepam; Eating; Female; Flumazenil; GABA Modulators; Latency Period, Psychological; Male; Maze Learning; Melatonin; Memory Disorders; Memory, Short-Term; Mice; Muscarinic Antagonists; Rats; Rats, Wistar; Receptors, GABA; Scopolamine; Triazolam

1998
The octadecaneuropeptide ODN induces anxiety in rodents: possible involvement of a shorter biologically active fragment.
    Peptides, 1998, Volume: 19, Issue:5

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Diazepam Binding Inhibitor; Discrimination Learning; Exploratory Behavior; Flumazenil; Injections, Intraventricular; Male; Maze Learning; Mice; Mice, Inbred Strains; Molecular Sequence Data; Neuropeptides; Peptide Fragments; Rats; Rats, Sprague-Dawley; Reaction Time

1998
Oral midazolam: pediatric conscious sedation.
    Compendium of continuing education in dentistry (Jamesburg, N.J. : 1995), 1998, Volume: 19, Issue:6

    Topics: Administration, Oral; Anesthesia, Dental; Child; Child, Preschool; Conscious Sedation; Dental Anxiety; Dental Care for Children; Diazepam; Flumazenil; GABA Modulators; Humans; Hypnotics and Sedatives; Midazolam

1998
Diazepam-treated female rats: flumazenil- and PK 11195-induced withdrawal in the hippocampus CA1.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 61, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Dose-Response Relationship, Drug; Electroencephalography; Female; Flumazenil; GABA Modulators; Hippocampus; Isoquinolines; Microinjections; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome

1998
Behavioural pharmacological characteristics of honokiol, an anxiolytic agent present in extracts of Magnolia bark, evaluated by an elevated plus-maze test in mice.
    The Journal of pharmacy and pharmacology, 1998, Volume: 50, Issue:7

    Topics: Administration, Oral; Animals; Anti-Anxiety Agents; Bicuculline; Biphenyl Compounds; Caffeine; Central Nervous System Depressants; Central Nervous System Stimulants; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Antagonists; GABA Modulators; Injections, Subcutaneous; Lignans; Male; Maze Learning; Mice; Mice, Inbred BALB C; Motor Activity; Tetragastrin; Therapeutic Equivalency

1998
Evidence for a unique profile of levetiracetam in rodent models of seizures and epilepsy.
    European journal of pharmacology, 1998, Jul-24, Volume: 353, Issue:2-3

    Topics: Amygdala; Animals; Anticonvulsants; Behavior, Animal; Carbolines; Convulsants; Diazepam; Disease Models, Animal; Electroconvulsive Therapy; Epilepsy; Excitatory Amino Acid Agonists; Flumazenil; GABA-A Receptor Antagonists; Kindling, Neurologic; Levetiracetam; Male; Mice; Pentylenetetrazole; Piracetam; Rats; Rats, Sprague-Dawley; Seizures

1998
Plasma and CSF benzodiazepine receptor ligand concentrations in cirrhotic patients with hepatic encephalopathy: relationship to severity of encephalopathy and to pharmaceutical benzodiazepine intake.
    Metabolic brain disease, 1998, Volume: 13, Issue:3

    Topics: Animals; Benzodiazepines; Binding, Competitive; Cell Fractionation; Cerebellum; Chronic Disease; Clonazepam; Diazepam; Flumazenil; GABA Modulators; Hepatic Encephalopathy; Humans; Isoquinolines; Liver Cirrhosis; Oxazepam; Radioligand Assay; Rats; Receptors, GABA-A; Tritium

1998
[Characteristics of human lymphocyte benzodiazepine receptors].
    Biulleten' eksperimental'noi biologii i meditsiny, 1998, Volume: 126, Issue:10

    Topics: Adult; Baclofen; Benzodiazepinones; Binding, Competitive; Diazepam; Flumazenil; GABA Agonists; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Ligands; Lymphocytes; Male; Receptors, GABA-A

1998
Inhibitory regulation of amylase release in rat parotid acinar cells by benzodiazepine receptors.
    European journal of pharmacology, 1998, Oct-23, Volume: 359, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amylases; Animals; Atropine; Benzodiazepinones; Carbachol; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoproterenol; Male; Muscarinic Agonists; Muscarinic Antagonists; Parotid Gland; Propranolol; Rats; Rats, Wistar; Receptors, GABA-A

1998
Effect of benzodiazepines and neurosteroids on ammonia-induced swelling in cultured astrocytes.
    Journal of neuroscience research, 1998, Dec-01, Volume: 54, Issue:5

    Topics: Ammonia; Astrocytes; Atrial Natriuretic Factor; Benzodiazepines; Benzodiazepinones; Brain Edema; Cell Size; Clonazepam; Dehydroepiandrosterone Sulfate; Desoxycorticosterone; Diazepam; Diazepam Binding Inhibitor; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoquinolines; Nerve Tissue Proteins; Neuropeptides; Peptide Fragments; Pregnanolone; Pregnenolone; Protoporphyrins; Receptors, GABA-A; Steroids; Up-Regulation

1998
Inhibitory effects of diazepam and midazolam on Ca2+ and K+ channels in canine tracheal smooth muscle cells.
    Anesthesiology, 1999, Volume: 90, Issue:1

    Topics: Anesthetics, Intravenous; Animals; Calcium Channel Blockers; Calcium Channels; Diazepam; Dogs; Electrophysiology; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; In Vitro Techniques; Isoquinolines; Midazolam; Muscle, Smooth; Patch-Clamp Techniques; Potassium Channel Blockers; Trachea

1999
Cardiac effects of benzodiazepine receptor agonists and antagonists in the isolated rat heart: a comparative study.
    Life sciences, 1998, Volume: 63, Issue:16

    Topics: Animals; Benzodiazepines; Cardiac Output; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Heart; In Vitro Techniques; Isoquinolines; Myocardial Contraction; Perfusion; Pyridines; Rats; Receptors, GABA-A; Zolpidem

1998
The effects of flumazenil on two way active avoidance and locomotor activity in diazepam-treated rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 1999, Volume: 9, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Injections, Intraperitoneal; Male; Motor Activity; Rats; Rats, Wistar; Time Factors

1999
Behavioral effects of diazepam in the murine plus-maze: flumazenil antagonism of enhanced head dipping but not the disinhibition of open-arm avoidance.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 62, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Avoidance Learning; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; GABA Modulators; Grooming; Male; Mice; Mice, Inbred DBA; Motor Activity

1999
Lack of sex differences in anxiety behaviors during precipitated benzodiazepine withdrawal in rats.
    Physiology & behavior, 1999, Volume: 66, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Corticosterone; Diazepam; Estradiol; Female; Flumazenil; GABA Modulators; Male; Progesterone; Radioligand Assay; Rats; Rats, Long-Evans; Sex Characteristics; Substance Withdrawal Syndrome

1999
Neurotransmitter modulation of glucocorticoid receptor mRNA levels in the rat hippocampus.
    Neuroendocrinology, 1999, Volume: 69, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Blotting, Northern; Diazepam; Dizocilpine Maleate; Down-Regulation; Excitatory Amino Acid Antagonists; Flumazenil; GABA Modulators; Hippocampus; Injections, Intraperitoneal; Male; Neurotransmitter Agents; Propranolol; Rats; Rats, Wistar; Receptors, Glucocorticoid; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Stress, Psychological

1999
Diazepam reduces action potential duration in guinea-pig papillary muscle by a cAMP-dependent mechanism.
    Life sciences, 1999, Volume: 64, Issue:25

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Action Potentials; Animals; Carbachol; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Diazepam; Enzyme Inhibitors; Flumazenil; gamma-Aminobutyric Acid; Guinea Pigs; In Vitro Techniques; Papillary Muscles; Thionucleotides

1999
Modification of the effect of diazepam on the propofol-induced loss of the righting reflex in mice by diabetes.
    Brain research, 1999, Jul-03, Volume: 833, Issue:2

    Topics: Anesthetics, Intravenous; Animals; Diabetes Mellitus, Experimental; Diazepam; Flumazenil; GABA Modulators; Injections, Intravenous; Male; Mice; Mice, Inbred ICR; Posture; Propofol; Receptors, GABA-A; Reflex

1999
Abecarnil enhances recovery from diazepam tolerance.
    Neuropharmacology, 1999, Volume: 38, Issue:9

    Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Carbolines; Cell Membrane; Cerebral Cortex; Clonazepam; Diazepam; Drug Interactions; Drug Tolerance; Flumazenil; Imidazoles; Ligands; Male; Mice; Receptors, GABA-A; Seizures; Tritium

1999
Discriminative stimulus effects of ethyl-beta-carboline-3-carboxylate at two training doses in rats.
    Psychopharmacology, 1999, Volume: 145, Issue:3

    Topics: Animals; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1999
Anticonflict effects of plant-derived essential oils.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 64, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Conflict, Psychological; Diazepam; Drug Interactions; Electroshock; Flumazenil; GABA Modulators; Male; Mice; Mice, Inbred ICR; Oils, Volatile

1999
New evidence that the pharmacological effects of benzodiazepine receptor ligands can be associated with activities at different BZ (omega) receptor subtypes.
    Psychopharmacology, 1999, Volume: 146, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Benzodiazepines; Binding, Competitive; Carbolines; Diazepam; Flumazenil; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Ligands; Male; Mice; Mice, Inbred BALB C; Motor Activity; Muscle Relaxants, Central; Patch-Clamp Techniques; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zolpidem

1999
Discriminative stimulus effects of flumazenil in untreated and in diazepam-treated rhesus monkeys.
    Psychopharmacology, 1999, Volume: 146, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Macaca mulatta; Male; Receptors, GABA-A

1999
Substantia nigra: the involvement of central and peripheral benzodiazepine receptors in physical dependence on diazepam as evidenced by behavioral and EEG effects.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 64, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Antineoplastic Agents; Behavior, Animal; Central Nervous System; Diazepam; Dose-Response Relationship, Drug; Drug Implants; Electrodes, Implanted; Electroencephalography; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Isoquinolines; Male; Peripheral Nervous System; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Substance Withdrawal Syndrome; Substance-Related Disorders; Substantia Nigra; Weight Gain

1999
Precipitated withdrawal in the substantia nigra in diazepam-dependent female rats.
    Pharmacology, biochemistry, and behavior, 1999, Volume: 64, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Electroencephalography; Female; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Isoquinolines; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Substance-Related Disorders; Substantia Nigra

1999
Central benzodiazepine involvement in clonidine cardiovascular actions.
    Canadian journal of physiology and pharmacology, 1999, Volume: 77, Issue:11

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Atropine Derivatives; Blood Pressure; Carbolines; Cardiovascular Agents; Clonidine; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Heart Rate; Infusions, Intravenous; Injections, Intraventricular; Male; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, GABA-A; Stereotaxic Techniques; Time Factors; Yohimbine

1999
Gabaergic-benzodiazepine system is involved in the crotoxin-induced anxiogenic effect.
    Pharmacology, biochemistry, and behavior, 2000, Jan-01, Volume: 65, Issue:1

    Topics: Animals; Anxiety; Behavior, Animal; Crotoxin; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Motor Activity; Rats; Rats, Wistar; Receptors, GABA-A

2000
The allocentric place discrimination task is selectively and highly dependent on the central muscarinic system in rats.
    Pharmacology, biochemistry, and behavior, 2000, Jan-01, Volume: 65, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Diazepam; Discrimination Learning; Dizocilpine Maleate; Flumazenil; Male; Mecamylamine; Ondansetron; Rats; Rats, Inbred F344; Receptors, Muscarinic; Scopolamine; Swimming

2000
The role of the benzodiazepine-GABA system in the memory processes of the day-old chick.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 65, Issue:2

    Topics: Animals; Animals, Newborn; Bicuculline; Chickens; Diazepam; Discrimination, Psychological; Flumazenil; GABA Antagonists; GABA Modulators; Male; Memory; Receptors, GABA-A; Reinforcement, Psychology

2000
Differential sensitivity to Zolpidem of IPSPs activated by morphologically identified CA1 interneurons in slices of rat hippocampus.
    The European journal of neuroscience, 2000, Volume: 12, Issue:2

    Topics: Animals; Diazepam; Evoked Potentials; Flumazenil; GABA Agonists; GABA Modulators; Hippocampus; Interneurons; Male; Presynaptic Terminals; Pyramidal Cells; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zolpidem

2000
Effect of chronic (-)-nicotine treatment on rat cerebral benzodiazepine receptors.
    Nuclear medicine and biology, 2000, Volume: 27, Issue:1

    Topics: Animals; Anticonvulsants; Cerebral Cortex; Diazepam; Flumazenil; Iodine Radioisotopes; Male; Nicotine; Nicotinic Agonists; Radionuclide Imaging; Rats; Rats, Wistar; Receptors, GABA-A; Tissue Distribution

2000
Acute opioid but not benzodiazepine dependence in rats responding for intracranial self-stimulation.
    Psychopharmacology, 2000, Volume: 148, Issue:3

    Topics: Animals; Benzodiazepines; Brain; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Morphine; Naltrexone; Opioid-Related Disorders; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Self Stimulation; Substance-Related Disorders

2000
Sedative but not anxiolytic properties of benzodiazepines are mediated by the GABA(A) receptor alpha1 subtype.
    Nature neuroscience, 2000, Volume: 3, Issue:6

    Topics: Allosteric Site; Animals; Anti-Anxiety Agents; Anticonvulsants; Azides; Benzodiazepines; Binding, Competitive; Brain; Cell Line; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Fluorobenzenes; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Ligands; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Motor Activity; Patch-Clamp Techniques; Receptors, GABA-A; Reflex, Startle; Triazoles

2000
Hypnotic, anticonvulsant and muscle relaxant effects of Rubus brasiliensis. Involvement of GABA(A)-system.
    Journal of ethnopharmacology, 2000, Volume: 70, Issue:3

    Topics: Animals; Anticonvulsants; Barbiturates; Brazil; Diazepam; Flumazenil; GABA Modulators; Hexanes; Hypnotics and Sedatives; Male; Mice; Muscle Relaxants, Central; Pentylenetetrazole; Plant Extracts; Plants, Medicinal; Receptors, GABA-A; Seizures

2000
Socio-psychological stress-induced antinociception in diabetic mice.
    Psychopharmacology, 2000, Volume: 149, Issue:4

    Topics: Animals; Anti-Bacterial Agents; Anticonvulsants; Carbolines; Convulsants; Diabetes Mellitus, Experimental; Diazepam; Flumazenil; GABA Modulators; Male; Mice; Mice, Inbred ICR; Pain Measurement; Streptozocin; Stress, Psychological

2000
Sex-specific effects of in utero manipulation of GABA(A) receptors on pre- and postnatal expression of BDNF in rats.
    Brain research. Developmental brain research, 2000, Jun-30, Volume: 121, Issue:2

    Topics: Animals; Brain-Derived Neurotrophic Factor; Cerebral Cortex; Diazepam; Female; Flumazenil; GABA Modulators; Gene Expression Regulation, Developmental; Hypothalamus; Male; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Long-Evans; Receptors, GABA-A; RNA, Messenger; Sex Characteristics

2000
Effect of flumazenil and diazepam on transient actions in defensive burying elicited by the social interaction experience in rats.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 66, Issue:2

    Topics: Animals; Behavior, Animal; Diazepam; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Rats; Rats, Wistar; Social Behavior; Time Factors

2000
Mice lacking the long splice variant of the gamma 2 subunit of the GABA(A) receptor are more sensitive to benzodiazepines.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 66, Issue:2

    Topics: Alternative Splicing; Animals; Azides; Benzodiazepines; Brain; Carbolines; Diazepam; Drug Resistance; Female; Flumazenil; GABA Modulators; Genetic Variation; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Midazolam; Pyridines; Receptors, GABA-A; Sleep; Zolpidem

2000
The influence of the benzodiazepine receptor antagonist flumazenil on the anxiolytic-like effects of CGP 37849 and ACPC in rats.
    Neuropharmacology, 2000, Jul-24, Volume: 39, Issue:10

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Amino Acids, Cyclic; Animals; Anti-Anxiety Agents; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drinking Behavior; Electroshock; Excitatory Amino Acid Antagonists; Flumazenil; GABA-A Receptor Antagonists; Male; Maze Learning; Rats; Rats, Wistar; Seizures

2000
Benzodiazepine-sensitive GABA(A) receptors limit the activity of the NMDA/NO/cyclic GMP pathway: a microdialysis study in the cerebellum of freely moving rats.
    Journal of neurochemistry, 2000, Volume: 75, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Bicuculline; Cerebellum; Cyclic GMP; Diazepam; Flumazenil; Infusions, Parenteral; Kinetics; Male; Microdialysis; Muscimol; N-Methylaspartate; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zolpidem

2000
Antagonism of the discriminative stimulus effects of positive gamma-aminobutyric acid(A) modulators in rhesus monkeys discriminating midazolam.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Diazepam; Discrimination Learning; Drug Antagonism; Female; Flumazenil; GABA Modulators; Macaca mulatta; Male; Midazolam; Receptors, GABA-A

2000
The pharmacodynamics of PK 11195 in diazepam-dependent male and female rats.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 66, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Antineoplastic Agents; Body Weight; Brain; Diazepam; Female; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Isoquinolines; Male; Rats; Rats, Sprague-Dawley; Seizures; Sex Characteristics; Substance Withdrawal Syndrome; Substance-Related Disorders

2000
Does dihydrohonokiol, a potent anxiolytic compound, result in the development of benzodiazepine-like side effects?
    The Journal of pharmacy and pharmacology, 2000, Volume: 52, Issue:8

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Biphenyl Compounds; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; GABA Modulators; Hexobarbital; Hypnotics and Sedatives; Learning; Male; Memory; Mice; Motor Activity; Sleep

2000
Benzodiazepines induce a conformational change in the region of the gamma-aminobutyric acid type A receptor alpha(1)-subunit M3 membrane-spanning segment.
    Molecular pharmacology, 2000, Volume: 58, Issue:5

    Topics: 4-Chloromercuribenzenesulfonate; Amino Acid Substitution; Animals; Benzodiazepines; Carbolines; Cysteine; Diazepam; Flumazenil; GABA Modulators; Membrane Proteins; Oocytes; Protein Conformation; Rats; Receptors, GABA-A; Xenopus laevis

2000
Flumazenil prevents diazepam-elicited anticonvulsant action and concomitant attenuation of glutamate overflow.
    European journal of pharmacology, 2000, Oct-27, Volume: 407, Issue:1-2

    Topics: Animals; Anticonvulsants; Convulsants; Diazepam; Flumazenil; GABA Modulators; Glutamic Acid; Male; Pilocarpine; Rats; Rats, Wistar; Receptors, GABA-A; Seizures

2000
Anticonflict effect of the glycineB receptor partial agonist, D-cycloserine, in rats. Pharmacological analysis.
    Psychopharmacology, 2000, Volume: 152, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Conflict, Psychological; Cycloserine; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Rats; Rats, Wistar; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate

2000
Benzodiazepines act on GABAA receptors via two distinct and separable mechanisms.
    Nature neuroscience, 2000, Volume: 3, Issue:12

    Topics: Animals; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Membrane Potentials; Mutation; Oocytes; Receptors, GABA-A; RNA, Messenger; Xenopus laevis; Zinc

2000
Diazepam-binding inhibitor-like activity in rat cerebrospinal fluid after stimulation by an aversive quinine taste.
    Chemical senses, 2000, Volume: 25, Issue:6

    Topics: Animals; Cerebrospinal Fluid; Diazepam; Drinking; Flumazenil; GABA-A Receptor Antagonists; Glutathione; Hydra; Male; Mice; Peptide Fragments; Pronase; Quinine; Rats; Rats, Wistar; Sucrose; Taste

2000
Behaviour of pigs given corticotrophin-releasing hormone in combination with flumazenil or diazepam.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 67, Issue:3

    Topics: Animals; Arousal; Corticotropin-Releasing Hormone; Diazepam; Flumazenil; GABA Modulators; Hormone Antagonists; Male; Motor Activity; Peptide Fragments; Receptors, GABA-A; Swine

2000
Evaluation of native GABA(A) receptors containing an alpha 5 subunit.
    European journal of pharmacology, 2001, Feb-09, Volume: 413, Issue:1

    Topics: Alkynes; Animals; Anti-Anxiety Agents; Anticonvulsants; Autoradiography; Benzodiazepines; Cerebellum; Clobazam; Clonazepam; Diazepam; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Hippocampus; Imidazoles; Male; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

2001
Massive dose of diazepam poisoning.
    The Journal of the Association of Physicians of India, 1998, Volume: 46, Issue:11

    Topics: Diazepam; Dose-Response Relationship, Drug; Drug Overdose; Flumazenil; Gastric Lavage; Humans; Infusions, Intravenous; Male; Metabolic Clearance Rate; Middle Aged

1998
[3H]Ro 15-1788 binding sites to brain membrane of the saltwater Mugil cephalus.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2001, Volume: 128, Issue:3

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Female; Fishes; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Imidazoles; Ionophores; Male; Pyridines; Receptors, GABA-A; Synaptosomes; Tritium; Zolpidem

2001
Negative inotropic effect of diazepam in isolated guinea pig heart.
    The Journal of veterinary medical science, 2001, Volume: 63, Issue:2

    Topics: Adjuvants, Anesthesia; Animals; Anti-Arrhythmia Agents; Calcium Channels; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Guinea Pigs; Heart; In Vitro Techniques; Isoquinolines; Male; Membrane Potentials; Myocardial Contraction; Patch-Clamp Techniques; Verapamil

2001
Zolpidem, triazolam, and diazepam decrease distress vocalizations in mouse pups: differential antagonism by flumazenil and beta-Carboline-3-carboxylate-t-butyl ester (beta-CCt).
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 297, Issue:1

    Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Body Temperature; Carbolines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Antagonists; Mice; Pyridines; Receptors, GABA-A; Triazolam; Vocalization, Animal; Zolpidem

2001
Effects of diazepam and beta-CCM on working memory in mice: relationships with emotional reactivity.
    Pharmacology, biochemistry, and behavior, 2001, Volume: 68, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Carbolines; Convulsants; Diazepam; Emotions; Flumazenil; GABA Modulators; Male; Memory; Mice; Mice, Inbred BALB C; Time Factors

2001
Use of negatively reinforcing electrical brain stimulation to detect conventional and nonconventional anxiolytics as well as an anxiogenic drug.
    Pharmacology, biochemistry, and behavior, 2001, Volume: 68, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Brain; Buspirone; Carbolines; Convulsants; Diazepam; Electric Stimulation; Electrodes; Flumazenil; GABA Modulators; Male; Pentylenetetrazole; Rats; Rats, Long-Evans; Reinforcement, Psychology

2001
Mice performance on the staircase test following acute ethanol administration.
    Pharmacology, biochemistry, and behavior, 2001, Volume: 68, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Central Nervous System Depressants; Diazepam; Dose-Response Relationship, Drug; Ethanol; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Psychomotor Performance

2001
Effects of diazepam and flumazenil on minimum alveolar concentrations for dogs anesthetized with isoflurane or a combination of isoflurane and fentanyl.
    American journal of veterinary research, 2001, Volume: 62, Issue:4

    Topics: Adjuvants, Anesthesia; Anesthetics, Inhalation; Animals; Anti-Anxiety Agents; Blood Pressure; Body Temperature; Diazepam; Dogs; Drug Interactions; Female; Fentanyl; Flumazenil; GABA Modulators; Heart Rate; Isoflurane; Pulmonary Alveoli

2001
Diazepam poisoning with one-month monitoring of diazepam and nordiazepam blood levels.
    Veterinary and human toxicology, 2001, Volume: 43, Issue:3

    Topics: Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Flumazenil; Humans; Male; Middle Aged; Nordazepam; Poisoning; Suicide, Attempted; Treatment Outcome

2001
Modification of the effects of benzodiazepines on the exploratory behaviors of mice on a hole-board by diabetes.
    Japanese journal of pharmacology, 2001, Volume: 86, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Carbolines; Convulsants; Diabetes Mellitus, Experimental; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Injections, Intraperitoneal; Male; Mice; Mice, Inbred ICR

2001
Increase in expression of the GABA(A) receptor alpha(4) subunit gene induced by withdrawal of, but not by long-term treatment with, benzodiazepine full or partial agonists.
    Brain research. Molecular brain research, 2001, Aug-15, Volume: 92, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Cell Membrane; Cells, Cultured; Cerebellum; Chloride Channels; Chlorides; Diazepam; Drug Tolerance; Female; Flumazenil; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Imidazoles; Ion Transport; Membrane Potentials; Microinjections; Nerve Tissue Proteins; Neurons; Oocytes; Protein Subunits; Rats; Receptors, GABA-A; RNA, Messenger; Substance Withdrawal Syndrome; Substance-Related Disorders; Up-Regulation; Xenopus laevis

2001
Diazepam increases the hypothalamic-pituitary-adrenocortical (HPA) axis activity by a cyclic AMP-dependent mechanism.
    British journal of pharmacology, 2001, Volume: 133, Issue:8

    Topics: Adrenal Cortex; Adrenocorticotropic Hormone; Animals; Corticosterone; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Diazepam; Flumazenil; Hypothalamus; Isoquinolines; Male; Phosphodiesterase Inhibitors; Pituitary Gland; Rats; Rats, Sprague-Dawley; Rolipram; Sulfonamides

2001
Potency of positive gamma-aminobutyric acid(A) modulators to substitute for a midazolam discriminative stimulus in untreated monkeys does not predict potency to attenuate a flumazenil discriminative stimulus in diazepam-treated monkeys.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 298, Issue:3

    Topics: Animals; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Hypnotics and Sedatives; Macaca mulatta; Male; Midazolam; Receptors, GABA-A; Steroids

2001
Synergistic interaction of diazepam with 3',5'-cyclic adenosine monophosphate-elevating agents on rat aortic rings.
    European journal of pharmacology, 2001, Oct-05, Volume: 428, Issue:2

    Topics: Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Female; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; In Vitro Techniques; Isoproterenol; Isoquinolines; Male; Milrinone; Muscle Relaxants, Central; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Rats; Rats, Sprague-Dawley; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2001
Involvement of benzodiazepine binding sites in an antiaggressive effect by 5-HT(1A) receptor activation in isolated mice.
    European journal of pharmacology, 2001, Dec-07, Volume: 432, Issue:2-3

    Topics: Aggression; Animals; Behavior, Animal; Binding Sites; Diazepam; Dioxanes; Dioxoles; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Male; Mice; Piperazines; Pyridines; Receptors, GABA-A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Social Isolation

2001
Discriminative stimulus effects of benzodiazepine (BZ)(1) receptor-selective ligands in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 300, Issue:2

    Topics: Acetamides; Animals; Carbolines; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Ligands; Macaca mulatta; Midazolam; Pyridines; Pyrimidines; Receptors, GABA-A; Zolpidem

2002
[Parenteral sedation in oral surgical procedures].
    Oral surgery, oral diagnosis : OSD, 1996, Volume: 7

    Topics: Antidotes; Benzodiazepines; Conscious Sedation; Diazepam; Flumazenil; Humans; Hypoxia; Infusions, Parenteral; Midazolam; Monitoring, Physiologic; Oral Surgical Procedures; Oximetry

1996
Mechanism of alpha-subunit selectivity of benzodiazepine pharmacology at gamma-aminobutyric acid type A receptors.
    European journal of pharmacology, 2002, Feb-15, Volume: 437, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Cell Line; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Mutation; Oocytes; Protein Subunits; Pyridazines; Pyridines; Radioligand Assay; Receptors, GABA-A; Tritium; Xenopus laevis; Zolpidem

2002
Evaluation of immunomodulatory potential of Ocimum sanctum seed oil and its possible mechanism of action.
    Journal of ethnopharmacology, 2002, Volume: 80, Issue:1

    Topics: Adjuvants, Immunologic; Animals; Antibody Formation; Diazepam; Erythrocytes; Flumazenil; Foot; GABA Modulators; Immunity, Cellular; Inflammation; Male; Medicine, Ayurvedic; Mice; Ocimum basilicum; Plant Oils; Rats; Rats, Wistar; Restraint, Physical; Seeds; Sheep; Stress, Physiological

2002
Role of benzodiazepine-GABAA receptor complex in attenuation of U-50,488H-induced analgesia and inhibition of tolerance to its analgesia by ginseng total saponin in mice.
    Life sciences, 2002, Mar-01, Volume: 70, Issue:15

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Animals; Bicuculline; Diazepam; Dose-Response Relationship, Drug; Drug Antagonism; Drug Tolerance; Drugs, Chinese Herbal; Flumazenil; Ginsenosides; Injections, Intraperitoneal; Male; Mice; Pain; Pain Threshold; Panax; Picrotoxin; Receptors, GABA-A; Receptors, Opioid, kappa; Saponins; Tail

2002
GABA(A)-benzodiazepine receptor complex sensitivity in 5-HT(1A) receptor knockout mice on a 129/Sv background.
    European journal of pharmacology, 2002, Jun-28, Volume: 447, Issue:1

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Diazepam; Ethanol; Fever; Flumazenil; GABA Antagonists; Hypnotics and Sedatives; Male; Maze Learning; Mice; Mice, Knockout; Pentylenetetrazole; Phenobarbital; Receptors, GABA-A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reflex; Species Specificity; Stress, Physiological

2002
The anxiolytic action of mGlu2/3 receptor agonist, LY354740, in the fear-potentiated startle model in rats is mechanistically distinct from diazepam.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 73, Issue:2

    Topics: Acoustic Stimulation; Amino Acids; Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Diazepam; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fear; Flumazenil; GABA Modulators; Male; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reflex, Startle; Xanthenes

2002
Reversal of benzodiazepine-induced renal vasculature relaxation with flumazenil.
    European journal of pharmacology, 2002, Aug-02, Volume: 449, Issue:1-2

    Topics: Animals; Clonazepam; Diazepam; Flumazenil; GABA Modulators; Male; Muscle Relaxants, Central; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Rats; Rats, Wistar; Renal Circulation; Vasoconstrictor Agents

2002
Gaba-benzodiazepine receptor complex in brain oxidative metabolism regulation.
    Pharmacological research, 2002, Volume: 46, Issue:2

    Topics: Animals; Diazepam; Flumazenil; Frontal Lobe; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Male; Oxygen Consumption; Picrotoxin; Rats; Rats, Wistar

2002
Diazepam withdrawal-induced anxiety and place aversion in the rat: differential effects of two chronic diazepam treatment regimes.
    Behavioural pharmacology, 2002, Volume: 13, Issue:5-6

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Avoidance Learning; Conditioning, Operant; Diazepam; Flumazenil; GABA Modulators; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Rats; Rats, Long-Evans; Substance Withdrawal Syndrome

2002
Cardiorespiratory effects of medetomidine-butorphanol, medetomidine-butorphanol-diazepam, and medetomidine-butorphanol-ketamine in captive red wolves (Canis rufus).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2002, Volume: 33, Issue:2

    Topics: Adrenergic alpha-Antagonists; Anesthetics, Dissociative; Animals; Animals, Zoo; Blood Pressure; Body Temperature; Butorphanol; Diazepam; Drug Combinations; Female; Flumazenil; GABA Modulators; Heart Rate; Hypertension; Hypnotics and Sedatives; Imidazoles; Immobilization; Ketamine; Male; Medetomidine; Muscle Relaxation; Naloxone; Narcotic Antagonists; Narcotics; Respiration; Wolves

2002
Flumazenil in acute benzodiazepine overdose.
    The Journal of the Association of Physicians of India, 2002, Volume: 50

    Topics: Anti-Anxiety Agents; Antidotes; Diazepam; Female; Flumazenil; Humans; Middle Aged

2002
Flumazenil antagonizes respiratory depression caused by diazepam and induces expiratory excitation of hypoglossal nerve.
    Masui. The Japanese journal of anesthesiology, 2002, Volume: 51, Issue:10

    Topics: Anesthetics, Intravenous; Animals; Depression, Chemical; Diazepam; Flumazenil; Hypoglossal Nerve; Phrenic Nerve; Pulmonary Ventilation; Rabbits; Respiration

2002
Inhibitory effect of diazepam on muscarinic receptor-stimulated inositol 1,4,5-trisphosphate production in rat parotid acinar cells.
    British journal of pharmacology, 2002, Volume: 137, Issue:7

    Topics: Animals; Anticonvulsants; Calcium; Carbachol; Chlorides; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; GTP-Binding Proteins; Inositol 1,4,5-Trisphosphate; Isoquinolines; Male; Parotid Gland; Phenylephrine; Phosphoinositide Phospholipase C; Phosphoric Diester Hydrolases; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Muscarinic; Time Factors

2002
Stereoselective discriminative stimulus effects of zopiclone in rhesus monkeys.
    Psychopharmacology, 2003, Volume: 165, Issue:3

    Topics: Administration, Oral; Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Macaca mulatta; Male; Midazolam; Piperazines; Stereoisomerism; Substance Withdrawal Syndrome

2003
Effects of cholecystokinin tetrapeptide (CCK(4)) and of anxiolytic drugs on GABA outflow from the cerebral cortex of freely moving rats.
    Neurochemistry international, 2003, Volume: 42, Issue:1

    Topics: Adamantane; Animals; Anti-Anxiety Agents; Buspirone; Cerebral Cortex; Diazepam; Epidural Space; Female; Flumazenil; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Motor Activity; Muscle Relaxants, Central; Nerve Tissue Proteins; Phenylurea Compounds; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetragastrin

2003
Discriminative stimulus effects of positive GABAA modulators and other anxiolytics, sedatives, and anticonvulsants in untreated and diazepam-treated monkeys.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 304, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Hypnotics and Sedatives; Macaca mulatta; Male; Midazolam; Receptors, GABA-A; Steroids

2003
Effects of diazepam and flumazenil on food competition behavior in high- and low-aggression pigeons.
    Pharmacology, biochemistry, and behavior, 2003, Volume: 74, Issue:3

    Topics: Aggression; Animals; Columbidae; Competitive Behavior; Diazepam; Feeding Behavior; Female; Flumazenil

2003
Modulation of development of tolerance to anticonvulsant effect of diazepam by flumazenil.
    Indian journal of physiology and pharmacology, 2002, Volume: 46, Issue:4

    Topics: Animals; Anticonvulsants; Diazepam; Drug Tolerance; Female; Flumazenil; Male; Mice; Seizures

2002
Role of platelet activating factor in triazolobenzodiazepines-induced retrograde amnesia.
    Behavioural brain research, 2003, Jun-16, Volume: 142, Issue:1-2

    Topics: 1-Alkyl-2-acetylglycerophosphocholine Esterase; Amnesia, Anterograde; Amnesia, Retrograde; Animals; Anti-Anxiety Agents; Azepines; Diazepam; Diterpenes; Escape Reaction; Female; Flumazenil; Ginkgolides; Lactones; Learning; Male; Mice; Phospholipases A; Platelet Activating Factor; Platelet Membrane Glycoproteins; Reaction Time; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Receptors, GABA-A; Retention, Psychology; Triazolam

2003
Involvement of presynaptic 5-HT(1A) and benzodiazepine receptors in the anticonflict activity of 5-HT(1A) receptor antagonists.
    European journal of pharmacology, 2003, Jun-13, Volume: 471, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Conflict, Psychological; Diazepam; Drinking Behavior; Drug Combinations; Flumazenil; Hippocampus; Injections, Intraperitoneal; Injections, Subcutaneous; Male; p-Chloroamphetamine; Piperazines; Punishment; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptors, GABA-A; Receptors, Presynaptic; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Succinimides; Time Factors

2003
Semisynthetic preparation of amentoflavone: A negative modulator at GABA(A) receptors.
    Bioorganic & medicinal chemistry letters, 2003, Jul-21, Volume: 13, Issue:14

    Topics: Animals; Biflavonoids; Diazepam; Flowers; Flumazenil; GABA Antagonists; GABA Modulators; Ginkgo biloba; Humans; Hypericum; Magnetic Resonance Spectroscopy; Methylation; Oocytes; Patch-Clamp Techniques; Plant Leaves; Receptors, GABA-A; Recombinant Proteins; Xenopus laevis

2003
Physical dependence in baboons chronically treated with low and high doses of diazepam.
    Behavioural pharmacology, 2003, Volume: 14, Issue:4

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Papio; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

2003
Extracts of kava (Piper methysticum) induce acute anxiolytic-like behavioral changes in mice.
    Psychopharmacology, 2003, Volume: 170, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Injections, Intraperitoneal; Kava; Male; Maze Learning; Mice; Mice, Inbred BALB C; Motor Activity; Plant Extracts

2003
Flumazenil attenuates development of tolerance to diazepam after chronic treatment of mice with either isoflurane or diazepam.
    Anesthesia and analgesia, 2003, Volume: 97, Issue:4

    Topics: Anesthetics, Inhalation; Animals; Anti-Anxiety Agents; Behavior, Animal; Binding Sites; Diazepam; Drug Tolerance; Flumazenil; GABA Modulators; Isoflurane; Mice; Postural Balance; Receptors, GABA-A

2003
Anticonvulsant and antiepileptogenic effects of GABAA receptor ligands in pentylenetetrazole-kindled mice.
    Progress in neuro-psychopharmacology & biological psychiatry, 2004, Volume: 28, Issue:1

    Topics: Animals; Anticonvulsants; Bicuculline; Convulsants; Dehydroepiandrosterone Sulfate; Diazepam; Dose-Response Relationship, Drug; Epilepsy; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; Isoxazoles; Kindling, Neurologic; Ligands; Mice; Pentylenetetrazole; Pregnanediones; Receptors, GABA-A

2004
[How do diazepam and flumazenil influence respiratory control by the activities of both hypoglossal and phrenic nerves in rabbits?].
    Masui. The Japanese journal of anesthesiology, 2003, Volume: 52, Issue:12

    Topics: Action Potentials; Animals; Diazepam; Flumazenil; Hypoglossal Nerve; Phrenic Nerve; Rabbits; Receptors, GABA-A; Respiration

2003
Anticonvulsant effects of thymoquinone, the major constituent of Nigella sativa seeds, in mice.
    Phytomedicine : international journal of phytotherapy and phytopharmacology, 2004, Volume: 11, Issue:1

    Topics: Animals; Anticonvulsants; Benzoquinones; Diazepam; Electroshock; Flumazenil; GABA Modulators; Injections, Intraperitoneal; Male; Mice; Mice, Inbred BALB C; Motor Activity; Nigella sativa; Pentylenetetrazole; Phytotherapy; Plant Extracts; Seeds; Seizures

2004
Pharmacological plasticity of GABA(A) receptors at dentate gyrus synapses in a rat model of temporal lobe epilepsy.
    The Journal of physiology, 2004, Jun-01, Volume: 557, Issue:Pt 2

    Topics: Animals; Anticonvulsants; Dentate Gyrus; Diazepam; Disease Models, Animal; Electric Conductivity; Epilepsy, Temporal Lobe; Flumazenil; GABA Modulators; Lithium; Male; Neural Inhibition; Patch-Clamp Techniques; Pilocarpine; Pregnanolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Status Epilepticus; Synapses

2004
Benzodiazepine-sensitive GABA(A) receptors in the commissural subnucleus of the NTS are involved in the carotid chemoreceptor reflex in rats.
    Autonomic neuroscience : basic & clinical, 2004, Feb-27, Volume: 110, Issue:2

    Topics: Animals; Blood Pressure; Carotid Arteries; Chemoreceptor Cells; Diazepam; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Male; Phrenic Nerve; Rats; Rats, Wistar; Receptors, GABA-A; Reflex; Solitary Nucleus; Synaptic Transmission; Visceral Afferents

2004
Flumazenil-independent positive modulation of gamma-aminobutyric acid action by 6-methylflavone at human recombinant alpha1beta2gamma2L and alpha1beta2 GABAA receptors.
    European journal of pharmacology, 2004, Apr-26, Volume: 491, Issue:1

    Topics: Allosteric Regulation; Animals; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Female; Flavones; Flavonoids; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Gene Expression; Humans; Membrane Potentials; Microinjections; Molecular Structure; Oocytes; Protein Subunits; Receptors, GABA; Receptors, GABA-A; Recombinant Proteins; RNA; Xenopus laevis

2004
Anxiolytic-like effects of MTEP, a potent and selective mGlu5 receptor agonist does not involve GABA(A) signaling.
    Neuropharmacology, 2004, Volume: 47, Issue:3

    Topics: Animals; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drinking; Drinking Behavior; Drug Interactions; Electroshock; Exploratory Behavior; Flumazenil; GABA Modulators; Male; Maze Learning; Mice; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Sensory Thresholds; Signal Transduction; Thiazoles

2004
[Effect of flumazenil on hypoglossal and phrenic nerves activities in rabbits].
    Masui. The Japanese journal of anesthesiology, 2004, Volume: 53, Issue:7

    Topics: Action Potentials; Animals; Benzodiazepines; Diazepam; Flumazenil; Hypoglossal Nerve; Male; Phrenic Nerve; Rabbits; Respiration

2004
Chronic exposure of cells expressing recombinant GABAA receptors to benzodiazepine antagonist flumazenil enhances the maximum number of benzodiazepine binding sites.
    Life sciences, 2004, Dec-03, Volume: 76, Issue:3

    Topics: Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Cell Membrane; Diazepam; Dose-Response Relationship, Drug; Drug Combinations; Flumazenil; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Humans; Kidney; Ligands; Receptors, GABA-A; Recombinant Proteins; Tritium

2004
Acetylcholine in the accumbens is decreased by diazepam and increased by benzodiazepine withdrawal: a possible mechanism for dependency.
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Acetylcholine; Animals; Behavior, Animal; Benzodiazepines; Diazepam; Dopamine; Dose-Response Relationship, Drug; Extracellular Space; Flumazenil; Male; Maze Learning; Microdialysis; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Substance-Related Disorders

2005
Benzodiazepine effect of (125)I-iomazenil-benzodiazepine receptor binding and serum corticosterone level in a rat model.
    Nuclear medicine and biology, 2005, Volume: 32, Issue:1

    Topics: Animals; Brain; Corticosterone; Diazepam; Disease Models, Animal; Flumazenil; Male; Radionuclide Imaging; Radiopharmaceuticals; Rats; Rats, Wistar; Receptors, GABA-A; Statistics as Topic; Stress, Psychological; Tissue Distribution

2005
The anxiolytic-like effect of 5-HT1B receptor ligands in rats: a possible mechanism of action.
    The Journal of pharmacy and pharmacology, 2005, Volume: 57, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzamides; Conflict, Psychological; Diazepam; Disease Models, Animal; Drinking Behavior; Drug Administration Schedule; Electroshock; Flumazenil; Men; Neurons; Oxadiazoles; p-Chloroamphetamine; Piperazines; Poland; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Water

2005
Benzodiazepine system is involved in hyperalgesia in rats induced by the exposure to extremely low frequency magnetic fields.
    Archives of pharmacal research, 2005, Volume: 28, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Baclofen; Bicuculline; Diazepam; Electromagnetic Fields; Flumazenil; GABA Antagonists; GABA Modulators; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Hot Temperature; Hyperalgesia; Injections, Intraventricular; Male; Pain Measurement; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A

2005
Intracerebroventricular administration of thymoquinone, the major constituent of Nigella sativa seeds, suppresses epileptic seizures in rats.
    Medical science monitor : international medical journal of experimental and clinical research, 2005, Volume: 11, Issue:4

    Topics: Animals; Anticonvulsants; Benzoquinones; Convulsants; Diazepam; Epilepsy; Flumazenil; Injections, Intraventricular; Male; Nigella; Pentylenetetrazole; Phytotherapy; Rats; Rats, Wistar; Seeds; Seizures

2005
6-Methylflavanone, a more efficacious positive allosteric modulator of gamma-aminobutyric acid (GABA) action at human recombinant alpha2beta2gamma2L than at alpha1beta2gamma2L and alpha1beta2 GABA(A) receptors expressed in Xenopus oocytes.
    European journal of pharmacology, 2005, Apr-11, Volume: 512, Issue:2-3

    Topics: Allosteric Regulation; Animals; Diazepam; DNA, Recombinant; Dose-Response Relationship, Drug; Female; Flavanones; Flavones; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Gene Expression; Humans; Membrane Potentials; Microinjections; Oocytes; Protein Isoforms; Receptors, GABA-A; RNA; Xenopus laevis

2005
Characterization in rats of the anxiolytic potential of ELB139 [1-(4-chlorophenyl)-4-piperidin-1-yl-1,5-dihydro-imidazol-2-on], a new agonist at the benzodiazepine binding site of the GABAA receptor.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Binding Sites; Binding, Competitive; Conflict, Psychological; Diazepam; Drug Tolerance; Flumazenil; Flunitrazepam; GABA Agonists; GABA Modulators; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Imidazoles; Light; Male; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Rats; Rats, Wistar

2005
Design and synthesis of new 2-substituted-5-(2-benzylthiophenyl)-1,3,4-oxadiazoles as benzodiazepine receptor agonists.
    Bioorganic & medicinal chemistry letters, 2005, Jun-15, Volume: 15, Issue:12

    Topics: Animals; Anticonvulsants; Benzodiazepines; Convulsants; Diazepam; Drug Design; Electroshock; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Mice; Models, Molecular; Molecular Structure; Oxadiazoles; Pentylenetetrazole; Seizures; Structure-Activity Relationship

2005
Chronic treatment with flumazenil enhances binding sites for convulsants at recombinant alpha(1)beta(2)gamma(2S) GABA(A) receptors.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2005, Volume: 59, Issue:7

    Topics: Binding Sites; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Convulsants; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Humans; Receptors, GABA-A; Recombinant Proteins

2005
GABA(A) receptors mediate orexin-A induced stimulation of food intake.
    Neuropharmacology, 2006, Volume: 50, Issue:1

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Eating; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; GABA-A Receptor Antagonists; Hyperphagia; Injections, Intraventricular; Intracellular Signaling Peptides and Proteins; Male; Muscimol; Neuropeptides; Orexin Receptors; Orexins; Rats; Rats, Sprague-Dawley; Receptors, G-Protein-Coupled; Receptors, GABA-A; Receptors, Neuropeptide; Stimulation, Chemical

2006
Influence of adenosine receptor agonists on benzodiazepine withdrawal signs in mice.
    European journal of pharmacology, 2005, Oct-31, Volume: 523, Issue:1-3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Mice; Pentylenetetrazole; Phenethylamines; Purinergic Agonists; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Agonists; Seizures; Substance Withdrawal Syndrome; Temazepam

2005
Diazepam inhibits the induction and maintenance of LTP of C-fiber evoked field potentials in spinal dorsal horn of rats.
    Neuropharmacology, 2006, Volume: 50, Issue:2

    Topics: Animals; Diazepam; Electrophysiology; Evoked Potentials; Flumazenil; GABA Modulators; Hypnotics and Sedatives; Long-Term Potentiation; Male; Nerve Fibers, Unmyelinated; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Taurine

2006
Cardiotonic and sedative effects of Cecropia pachystachya Mart. (ambay) on isolated rat hearts and conscious mice.
    Journal of ethnopharmacology, 2006, Jun-15, Volume: 106, Issue:1

    Topics: Amphetamine; Animals; Argentina; Benzodiazepines; Cardiotonic Agents; Cardiovascular Agents; Cecropia Plant; Chromatography, High Pressure Liquid; Diazepam; Dopamine; Female; Flumazenil; Heart; Heart Rate; Hypnotics and Sedatives; Male; Mice; Plant Extracts; Rats; Rats, Wistar; Receptors, GABA-A

2006
Involvement of diazepam-insensitive benzodiazepine receptors in the suppression of DOI-induced head-twitch responses in diabetic mice.
    Psychopharmacology, 2006, Volume: 186, Issue:1

    Topics: Amphetamines; Animals; Azides; Behavior, Animal; Benzodiazepines; Bicuculline; Diabetes Mellitus, Experimental; Diazepam; Flumazenil; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Mice; Mice, Inbred ICR; Receptors, GABA-A; Serotonin Receptor Agonists

2006
Effects of drugs acting on the GABA-benzodiazepine receptor complex on flurothyl-induced seizures in Mongolian gerbils.
    European journal of pharmacology, 2006, May-01, Volume: 536, Issue:3

    Topics: Amino Acids; Animals; Anticonvulsants; Brain; Convulsants; Diazepam; Ethanol; Flumazenil; Flurothyl; GABA Antagonists; GABA-A Receptor Antagonists; Gerbillinae; Male; Picrotoxin; Receptors, GABA-A; Seizures; Valproic Acid

2006
Protective effect of BR-16A, a polyherbal preparation against social isolation stress: possible GABAergic mechanism.
    Phytotherapy research : PTR, 2006, Volume: 20, Issue:7

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Female; Flumazenil; GABA Agonists; gamma-Aminobutyric Acid; Male; Mice; Motor Activity; Pain; Pentobarbital; Phytotherapy; Plant Extracts; Social Isolation; Stress, Psychological

2006
Efficacy and the discriminative stimulus effects of negative GABAA modulators, or inverse agonists, in diazepam-treated rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 2006, Volume: 318, Issue:2

    Topics: Animals; Azides; Benzodiazepines; Conditioning, Operant; Cues; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Agonists; GABA Modulators; Hypnotics and Sedatives; Macaca mulatta; Male; Pentobarbital; Pregnanolone; Receptors, GABA-A

2006
Enhanced sucrose pellet consumption induced by benzodiazepine-type drugs in squirrel monkeys: role of GABAA receptor subtypes.
    Psychopharmacology, 2006, Volume: 187, Issue:3

    Topics: Alprazolam; Animals; Benzodiazepines; Diazepam; Flumazenil; Male; Pyridines; Receptors, GABA-A; Saimiri; Sucrose; Zolpidem

2006
GABAA receptor regulation of voluntary ethanol drinking requires PKCepsilon.
    Synapse (New York, N.Y.), 2006, Volume: 60, Issue:6

    Topics: Alcohol Drinking; Animals; Diazepam; Flumazenil; GABA Agonists; GABA Modulators; Hypnotics and Sedatives; Mice; Mice, Knockout; Motor Activity; Protein Kinase C-epsilon; Pyridines; Receptors, GABA-A; Zolpidem

2006
Effects of genetic background and null mutation of 5-HT1A receptors on basal and stress-induced body temperature: modulation by serotonergic and GABAA-ergic drugs.
    European journal of pharmacology, 2006, Nov-21, Volume: 550, Issue:1-3

    Topics: Animals; Body Temperature; Body Temperature Regulation; Buspirone; Diazepam; Fever; Flumazenil; Fluorobenzenes; GABA Agonists; GABA Modulators; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Pyridines; Receptor, Serotonin, 5-HT1A; Receptors, GABA-A; Serotonin; Serotonin Agents; Serotonin Receptor Agonists; Stress, Psychological; Triazoles; Zolpidem

2006
Felbamate is a subunit selective modulator of recombinant gamma-aminobutyric acid type A receptors expressed in Xenopus oocytes.
    European journal of pharmacology, 2006, Dec-15, Volume: 552, Issue:1-3

    Topics: Animals; Cells, Cultured; Cerebellum; Diazepam; DNA, Recombinant; Felbamate; Female; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Gene Expression; Humans; Membrane Potentials; Oocytes; Patch-Clamp Techniques; Phenylcarbamates; Plasmids; Propylene Glycols; Protein Subunits; Receptors, GABA-A; Xenopus laevis

2006
Anti-anxiety effects of Apocynum venetum L. in the elevated plus maze test.
    Journal of ethnopharmacology, 2007, Apr-04, Volume: 110, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Apocynum; Behavior, Animal; Buspirone; Diazepam; Disease Models, Animal; Ethanol; Flumazenil; GABA Modulators; Male; Maze Learning; Mice; Mice, Inbred C57BL; Piperazines; Plant Extracts; Plants, Medicinal; Pyridines; Receptors, GABA; Serotonin Antagonists

2007
Effects of diazepam on 125I-iomazenil-benzodiazepine receptor binding and epileptic seizures in the El mouse.
    Annals of nuclear medicine, 2006, Volume: 20, Issue:8

    Topics: Animals; Anticonvulsants; Autoradiography; Brain; Diazepam; Disease Models, Animal; Epilepsy; Flumazenil; Iodine Radioisotopes; Mice; Protein Binding; Receptors, GABA-A; Seizures; Time Factors

2006
A possible mechanism for anxiolytic and antidepressant effects of alpha- and beta-amyrin from Protium heptaphyllum (Aubl.) March.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 85, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Antidepressive Agents, Tricyclic; Behavior, Animal; Burseraceae; Diazepam; Flumazenil; GABA Modulators; Hypnotics and Sedatives; Imipramine; Mice; Oleanolic Acid; Plant Preparations; Reserpine

2006
Pharmacological analysis of the effects of benzodiazepines on punished schedule-induced polydipsia in rats.
    Behavioural pharmacology, 2007, Volume: 18, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Chlordiazepoxide; Diazepam; Dose-Response Relationship, Drug; Drinking; Electroshock; Fear; Flumazenil; Food Deprivation; GABA Modulators; Imidazoles; Male; Oxazepam; Punishment; Pyrimidines; Rats; Rats, Wistar; Receptors, GABA-A; Reinforcement Schedule

2007
Changes in relative potency among positive GABA(A) receptor modulators upon discontinuation of chronic benzodiazepine treatment in rhesus monkeys.
    Psychopharmacology, 2007, Volume: 192, Issue:1

    Topics: Animals; Behavior, Animal; Benzodiazepines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Lorazepam; Macaca mulatta; Male; Midazolam; Pentobarbital; Pregnanediones; Pregnanolone; Receptors, GABA-A; Substance Withdrawal Syndrome

2007
Neuroprotection afforded by diazepam against oxygen/glucose deprivation-induced injury in rat cortical brain slices.
    European journal of pharmacology, 2007, Apr-30, Volume: 561, Issue:1-3

    Topics: Animals; Brain Ischemia; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Glucose; Hypoxia, Brain; Male; Neurons; Neuroprotective Agents; Oxygen; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

2007
Allosteric uncoupling and up-regulation of benzodiazepine and GABA recognition sites following chronic diazepam treatment of HEK 293 cells stably transfected with alpha1beta2gamma2S subunits of GABA (A) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:3

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Cell Line; Diazepam; Flumazenil; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Muscimol; Picrotoxin; Protein Subunits; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A; Receptors, GABA-B; Transfection; Up-Regulation

2007
Anxiolytic-like effects of sinapic acid in mice.
    Life sciences, 2007, Jun-27, Volume: 81, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Bicuculline; Cerebral Cortex; Chloride Channels; Coumaric Acids; Diazepam; Electrophysiology; Flumazenil; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Motor Activity; Muscle Relaxation; Muscle, Smooth; Neurons; Neurotransmitter Agents; Piperazines; Postural Balance; Pyridines; Serotonin Antagonists

2007
Anticonvulsant effects of aerial parts of Passiflora incarnata extract in mice: involvement of benzodiazepine and opioid receptors.
    BMC complementary and alternative medicine, 2007, Aug-08, Volume: 7

    Topics: Animals; Anticonvulsants; Antidotes; Convulsants; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Epilepsy, Absence; Flumazenil; Injections, Intraperitoneal; Male; Mice; Mice, Inbred BALB C; Naloxone; Narcotic Antagonists; Passiflora; Pentylenetetrazole; Phytotherapy; Plant Components, Aerial; Plant Extracts; Receptors, GABA-A; Receptors, Opioid; Sodium Chloride; Treatment Outcome

2007
Effect of withdrawal of diazepam or morphine treatment on gastric motility (charcoal meal test) in mice: possible role of different central and peripheral receptors.
    Indian journal of experimental biology, 2007, Volume: 45, Issue:7

    Topics: Analgesics; Analgesics, Opioid; Animals; Central Nervous System; Chemistry, Pharmaceutical; Diazepam; Drug Evaluation, Preclinical; Flumazenil; Gastric Mucosa; Male; Mice; Morphine; Naloxone; Peripheral Nervous System; Stomach; Substance Withdrawal Syndrome

2007
Treatment with haloperidol and diazepam alters GABA(A) receptor density in the rat brain.
    Progress in neuro-psychopharmacology & biological psychiatry, 2008, Feb-15, Volume: 32, Issue:2

    Topics: Animals; Antipsychotic Agents; Autoradiography; Benzodiazepines; Binding Sites; Brain; Diazepam; Disease Models, Animal; Drug Combinations; Flumazenil; Haloperidol; Hippocampus; Humans; Injections, Intraperitoneal; Muscimol; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Schizophrenia; Thalamus; Tissue Distribution

2008
The anxiolytic-like effect of the selective 5-HT6 receptor antagonist SB-399885: the impact of benzodiazepine receptors.
    European journal of pharmacology, 2008, Feb-12, Volume: 580, Issue:3

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Behavior, Animal; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drinking; Electroshock; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Injections, Intraperitoneal; Male; p-Chloroamphetamine; Piperazines; Rats; Rats, Wistar; Receptors, GABA; Receptors, GABA-A; Receptors, Serotonin; Serotonin Antagonists; Sulfonamides

2008
Reduced GABA neurotransmission underlies hyperalgesia induced by repeated forced swimming stress.
    Behavioural brain research, 2008, May-16, Volume: 189, Issue:1

    Topics: Analysis of Variance; Animals; Diazepam; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Hyperalgesia; Male; Microdialysis; Pain; Pain Threshold; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Spinal Cord; Stress, Psychological; Swimming

2008
Reversal of paradoxical excitement to diazepam sedation.
    Paediatric anaesthesia, 2008, Volume: 18, Issue:6

    Topics: Anti-Anxiety Agents; Antidotes; Child; Conscious Sedation; Diazepam; Flumazenil; Humans; Male; Psychomotor Agitation; Treatment Outcome

2008
Long-lasting modulation of glutamatergic transmission in VTA dopamine neurons after a single dose of benzodiazepine agonists.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2009, Volume: 34, Issue:2

    Topics: Animals; Benzodiazepines; Diazepam; Dizocilpine Maleate; Ethanol; Excitatory Postsynaptic Potentials; Female; Flumazenil; GABA-A Receptor Agonists; Glutamic Acid; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Morphine; Neurons; Patch-Clamp Techniques; Pyridines; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Ventral Tegmental Area; Zolpidem

2009
Anxiolytic activity of a phytochemically characterized Passiflora incarnata extract is mediated via the GABAergic system.
    Planta medica, 2008, Volume: 74, Issue:15

    Topics: Animals; Anti-Anxiety Agents; Buspirone; Chromatography, High Pressure Liquid; Diazepam; Flavonoids; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Maze Learning; Mice; Mice, Inbred C57BL; Passiflora; Phytotherapy; Piperazines; Plant Extracts; Pyridines; Serotonin Antagonists

2008
GABAA receptor alpha5 subunits contribute to GABAA,slow synaptic inhibition in mouse hippocampus.
    Journal of neurophysiology, 2009, Volume: 101, Issue:3

    Topics: Animals; Biophysical Phenomena; Biophysics; Diazepam; Electric Stimulation; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Transgenic; Neural Inhibition; Patch-Clamp Techniques; Point Mutation; Pyramidal Cells; Receptors, GABA-A; Synapses

2009
A high-throughput functional assay for characterization of gamma-aminobutyric acid(A) channel modulators using cryopreserved transiently transfected cells.
    Assay and drug development technologies, 2008, Volume: 6, Issue:6

    Topics: Carbolines; Cell Culture Techniques; Cell Line; Cell Membrane; Cryopreservation; Diazepam; DNA; Dose-Response Relationship, Drug; Drug Discovery; Flumazenil; Flunitrazepam; Fluorescent Dyes; Fluorobenzenes; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Receptors, GABA-A; Reproducibility of Results; Spectrometry, Fluorescence; Transfection; Triazoles; Tritium

2008
[Pharmacodynamic and pharmacokinetic effects of flumazenil and theophylline application in rats acutely intoxicated by diazepam].
    Vojnosanitetski pregled, 2009, Volume: 66, Issue:2

    Topics: Animals; Antidotes; Diazepam; Flumazenil; GABA Modulators; Hypnotics and Sedatives; Male; Motor Activity; Phosphodiesterase Inhibitors; Rats; Rats, Wistar; Theophylline

2009
The effects of benzodiazepines on urotensin II-stimulated norepinephrine release from rat cerebrocortical slices.
    Anesthesia and analgesia, 2009, Volume: 108, Issue:4

    Topics: Animals; Benzodiazepines; Benzoxazoles; Calcium Signaling; Cell Line; Cerebral Cortex; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Humans; Hypnotics and Sedatives; In Vitro Techniques; Male; Midazolam; Naphthyridines; Norepinephrine; Orexin Receptors; Rats; Rats, Wistar; Receptors, G-Protein-Coupled; Receptors, GABA-A; Receptors, Neuropeptide; Transfection; Urea; Urotensins

2009
Kaempferol from the leaves of Apocynum venetum possesses anxiolytic activities in the elevated plus maze test in mice.
    Phytomedicine : international journal of phytotherapy and phytopharmacology, 2009, Volume: 16, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Apocynum; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Kaempferols; Male; Maze Learning; Mice; Mice, Inbred BALB C; Phytotherapy; Piperazines; Plant Extracts; Plant Leaves; Pyridines

2009
Central action of Araucaria angustifolia seed lectin in mice.
    Epilepsy & behavior : E&B, 2009, Volume: 15, Issue:3

    Topics: Analysis of Variance; Animals; Anticonvulsants; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Lectins; Locomotion; Male; Mice; Pentylenetetrazole; Phytotherapy; Plant Extracts; Reaction Time; Seeds; Seizures; Strychnine

2009
A novel operant conflict procedure using incrementing shock intensities to assess the anxiolytic and anxiogenic effects of drugs.
    Behavioural pharmacology, 2009, Volume: 20, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Aripiprazole; Benzodiazepines; Chlordiazepoxide; Conditioning, Operant; Conflict, Psychological; Dextroamphetamine; Diazepam; Electroshock; Flumazenil; Male; Piperazines; Punishment; Pyridazines; Quinolones; Rats; Rats, Sprague-Dawley; Triazoles; Yohimbine

2009
Impairment of the cortical GABAergic inhibitory system in catatonic stupor: a case report with neuroimaging.
    Epileptic disorders : international epilepsy journal with videotape, 2009, Volume: 11, Issue:2

    Topics: Acute Disease; Adult; Catatonia; Cerebral Cortex; Diazepam; Electroencephalography; Encephalitis; Flumazenil; Fluorodeoxyglucose F18; Frontal Lobe; Functional Laterality; GABA Modulators; Glucose; Humans; Male; Positron-Emission Tomography; Radiopharmaceuticals; Stupor; Temporal Lobe; Tomography, Emission-Computed, Single-Photon

2009
Relative positioning of diazepam in the benzodiazepine-binding-pocket of GABA receptors.
    Journal of neurochemistry, 2009, Volume: 111, Issue:5

    Topics: Allosteric Regulation; Animals; Anti-Anxiety Agents; Benzodiazepines; Binding Sites; Biophysics; Cell Line, Transformed; Cysteine; Diazepam; Dizocilpine Maleate; Dose-Response Relationship, Drug; Electric Stimulation; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Oocytes; Point Mutation; Protein Binding; Receptors, GABA-A; Structure-Activity Relationship; Transfection; Xenopus

2009
Discriminative stimulus effects of L-838,417 (7-tert-butyl-3-(2,5-difluoro-phenyl)-6-(2-methyl-2H-[1,2,4]triazol-3-ylmethoxy)-[1,2,4]triazolo[4,3-b]pyridazine): role of GABA(A) receptor subtypes.
    Neuropharmacology, 2010, Volume: 58, Issue:2

    Topics: Animals; Barbiturates; Carbolines; Catheterization; Central Nervous System Depressants; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Ethanol; Flumazenil; Fluorobenzenes; GABA Agonists; GABA Antagonists; GABA Modulators; Neuropsychological Tests; Pyridines; Receptors, GABA-A; Saimiri; Triazoles; Zolpidem

2010
Neurosteroid withdrawal regulates GABA-A receptor α4-subunit expression and seizure susceptibility by activation of progesterone receptor-independent early growth response factor-3 pathway.
    Neuroscience, 2010, Oct-27, Volume: 170, Issue:3

    Topics: Animals; Diazepam; Drug Administration Schedule; Early Growth Response Protein 3; Female; Flumazenil; Gene Expression Regulation; Hippocampus; Kindling, Neurologic; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurotransmitter Agents; Oligodeoxyribonucleotides, Antisense; Pregnanolone; Progesterone; Receptors, GABA-A; Receptors, Progesterone; Signal Transduction; Up-Regulation

2010
Metabotropic glutamate receptor 4 novel agonist LSP1-2111 with anxiolytic, but not antidepressant-like activity, mediated by serotonergic and GABAergic systems.
    Neuropharmacology, 2010, Volume: 59, Issue:7-8

    Topics: Aminobutyrates; Animals; Anti-Anxiety Agents; Antidepressive Agents; Diazepam; Fever; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Maze Learning; Mice; Phosphinic Acids; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Stress, Psychological

2010
Diazepam decreases action potential firing of neocortical neurons via two distinct mechanisms.
    Anesthesia and analgesia, 2010, Volume: 111, Issue:6

    Topics: Action Potentials; Anesthetics; Animals; Binding Sites; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Hypnotics and Sedatives; Male; Mice; Mice, Inbred C57BL; Neocortex; Neural Inhibition; Neurons; Receptors, GABA-A; Time Factors; Tissue Culture Techniques

2010
Chronic benzodiazepine treatment does not alter interactions between positive GABA(A) modulators and flumazenil or pentylenetetrazole in monkeys.
    Behavioural pharmacology, 2011, Volume: 22, Issue:1

    Topics: Animals; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Drug Interactions; Female; Flumazenil; GABA Modulators; Macaca mulatta; Male; Midazolam; Pentylenetetrazole; Receptors, GABA-A

2011
Sedative effects of Iranian Artemisia annua in mice: possible benzodiazepine receptors involvement.
    Pharmaceutical biology, 2011, Volume: 49, Issue:8

    Topics: Acetates; Alkanes; Animals; Antidotes; Antimalarials; Artemisia annua; Artemisinins; Chloroform; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Hypnotics and Sedatives; Immobilization; Iran; Male; Mice; Phytotherapy; Plant Components, Aerial; Plant Extracts; Receptors, GABA-A; Solvents

2011
Stress-induced hyperalgesia is associated with a reduced and delayed GABA inhibitory control that enhances post-synaptic NMDA receptor activation in the spinal cord.
    Pain, 2011, Volume: 152, Issue:8

    Topics: Analgesics; Animals; Diazepam; Disease Models, Animal; Excitatory Postsynaptic Potentials; Flumazenil; Formaldehyde; GABA Modulators; gamma-Aminobutyric Acid; Glutamic Acid; Hyperalgesia; Ketamine; Male; Pain Measurement; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Stress, Psychological; Swimming; Time Factors

2011
3-Hydroxy-2'-methoxy-6-methylflavone: a potent anxiolytic with a unique selectivity profile at GABA(A) receptor subtypes.
    Biochemical pharmacology, 2011, Dec-15, Volume: 82, Issue:12

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Dose-Response Relationship, Drug; Fatty Acids, Volatile; Flavones; Flumazenil; gamma-Aminobutyric Acid; Humans; Male; Mice; Mice, Inbred BALB C; Molecular Structure; Motor Activity; Oocytes; Pentylenetetrazole; Receptors, GABA-A; Recombinant Proteins; Thiopental; Xenopus

2011
The role of α1 and α5 subunit-containing GABAA receptors in motor impairment induced by benzodiazepines in rats.
    Behavioural pharmacology, 2012, Volume: 23, Issue:2

    Topics: Animals; Ataxia; Benzodiazepines; Benzodiazepinones; Carbolines; Diazepam; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hand Strength; Imidazoles; Male; Muscle Relaxation; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Rotarod Performance Test; Zolpidem

2012
Evaluation of acute toxicity of a natural compound (+)-limonene epoxide and its anxiolytic-like action.
    Brain research, 2012, Apr-11, Volume: 1448

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Cyclohexane Monoterpenes; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Hypnotics and Sedatives; Injections, Intraperitoneal; Male; Mice; Monoterpenes; Motor Activity; Postural Balance; Stereoisomerism

2012
Participation of the GABAergic system in the anesthetic effect of Lippia alba (Mill.) N.E. Brown essential oil.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 2012, Volume: 45, Issue:5

    Topics: Anesthetics; Animals; Catfishes; Diazepam; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Lippia; Models, Animal; Oils, Volatile; Plant Leaves; Receptors, GABA-A

2012
Magnolol, a major bioactive constituent of the bark of Magnolia officinalis, induces sleep via the benzodiazepine site of GABA(A) receptor in mice.
    Neuropharmacology, 2012, Volume: 63, Issue:6

    Topics: Animals; Arousal; Biphenyl Compounds; Diazepam; Drug Interactions; Electroencephalography; Electromyography; Flumazenil; GABA Modulators; Gene Expression; Genes, fos; Hypothalamic Area, Lateral; Immunohistochemistry; Lignans; Magnolia; Male; Mice; Mice, Inbred C57BL; Plant Bark; Polysomnography; Preoptic Area; Receptors, GABA-A; Sleep; Sleep, REM

2012
GABA(A) receptor α subunits differentially contribute to diazepam tolerance after chronic treatment.
    PloS one, 2012, Volume: 7, Issue:8

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Benzodiazepinones; Body Temperature; Brain; Diazepam; DNA Primers; Drug Tolerance; Flumazenil; Hypnotics and Sedatives; In Situ Hybridization; Male; Mice; Mice, Mutant Strains; Pyridazines; Pyridines; Receptors, GABA-A; Triazoles; Zolpidem

2012
Effects of diazepam and flumazenil on forebrain ischaemia in a rat model of benzodiazepine tolerance.
    British journal of anaesthesia, 2012, Volume: 109, Issue:6

    Topics: Analysis of Variance; Animals; Benzodiazepines; Brain Ischemia; Diazepam; Disease Models, Animal; Drug Tolerance; Flumazenil; GABA Modulators; Male; Neuroprotective Agents; Prosencephalon; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Severity of Illness Index

2012
βCCT, an antagonist selective for α(1)GABA(A) receptors, reverses diazepam withdrawal-induced anxiety in rats.
    Brain research bulletin, 2013, Volume: 91

    Topics: Animals; Anxiety; Carbolines; Diazepam; Flumazenil; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Male; Maze Learning; Rats; Rats, Wistar; Receptors, GABA-A; Substance Withdrawal Syndrome

2013
Piperine decreases pilocarpine-induced convulsions by GABAergic mechanisms.
    Pharmacology, biochemistry, and behavior, 2013, Volume: 104

    Topics: Alkaloids; Amino Acids; Animals; Anticonvulsants; Antioxidants; Atropine; Benzodioxoles; Biogenic Monoamines; Brain; Diazepam; Disease Models, Animal; Epilepsy; Flumazenil; gamma-Aminobutyric Acid; Humans; Male; Memantine; Mice; Nimodipine; Nitrites; Pilocarpine; Piperidines; Polyunsaturated Alkamides; Seizures; Tumor Necrosis Factor-alpha

2013
Potentiating effect of glabridin on GABAA receptor-mediated responses in dorsal raphe neurons.
    Planta medica, 2013, Volume: 79, Issue:15

    Topics: Animals; Anti-Anxiety Agents; Brain; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Agents; gamma-Aminobutyric Acid; Glycyrrhiza; Hypnotics and Sedatives; Isoflavones; Neurons; Pentobarbital; Phenols; Plant Extracts; Plant Roots; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Zolpidem

2013
A possible mechanism for the anxiolytic-like effect of gallic acid in the rat elevated plus maze.
    Pharmacology, biochemistry, and behavior, 2014, Volume: 117

    Topics: Animals; Anti-Anxiety Agents; Buspirone; Diazepam; Flumazenil; Gallic Acid; Male; Maze Learning; Rats; Rats, Wistar

2014
Potential antioxidant and anxiolytic effects of (+)-limonene epoxide in mice after marble-burying test.
    Pharmacology, biochemistry, and behavior, 2014, Volume: 118

    Topics: Animals; Anti-Anxiety Agents; Antioxidants; Anxiety; Catalase; Cyclohexane Monoterpenes; Diazepam; Flumazenil; Free Radical Scavengers; Hippocampus; Male; Mice; Monoterpenes; Reactive Nitrogen Species; Reactive Oxygen Species; Superoxide Dismutase

2014
Marine polyphenol phlorotannins promote non-rapid eye movement sleep in mice via the benzodiazepine site of the GABAA receptor.
    Psychopharmacology, 2014, Volume: 231, Issue:14

    Topics: Animals; Diazepam; Dioxanes; Dose-Response Relationship, Drug; Electroencephalography; Flumazenil; Heterocyclic Compounds, 4 or More Rings; Hypnotics and Sedatives; Male; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Polyphenols; Receptors, GABA-A; Sleep; Tannins

2014
S-(+)-Linalool from Lippia alba: sedative and anesthetic for silver catfish (Rhamdia quelen).
    Veterinary anaesthesia and analgesia, 2014, Volume: 41, Issue:6

    Topics: Acyclic Monoterpenes; Anesthesia; Anesthetics; Animals; Catfishes; Central Nervous System; Diazepam; Flumazenil; Hypnotics and Sedatives; Lippia; Monoterpenes; Plant Oils

2014
Effects of chronic mild stress on the development of drug dependence in rats.
    Behavioural pharmacology, 2014, Volume: 25, Issue:5-6

    Topics: Animals; Chronic Disease; Citalopram; Depressive Disorder; Diazepam; Disease Models, Animal; Flumazenil; GABA Modulators; Male; Mecamylamine; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Stress, Psychological; Substance Withdrawal Syndrome; Substance-Related Disorders

2014
Potential mechanisms involved in the anticonvulsant effect of walnut extract on pentylenetetrazole-induced seizure.
    Medical principles and practice : international journal of the Kuwait University, Health Science Centre, 2014, Volume: 23, Issue:6

    Topics: Animals; Anticonvulsants; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Ethosuximide; Flumazenil; Juglans; Male; Pentylenetetrazole; Plant Extracts; Rats; Rats, Wistar; Seizures

2014
Women with PTSD have a changed sensitivity to GABA-A receptor active substances.
    Psychopharmacology, 2016, Volume: 233, Issue:11

    Topics: Adolescent; Adult; Anxiety; Diagnostic and Statistical Manual of Mental Disorders; Diazepam; Female; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; Humans; Hypnotics and Sedatives; Pregnanolone; Psychiatric Status Rating Scales; Receptors, GABA-A; Saccades; Stress Disorders, Post-Traumatic; Young Adult

2016
Positive modulation of synaptic and extrasynaptic GABAA receptors by an antagonist of the high affinity benzodiazepine binding site.
    Neuropharmacology, 2015, Volume: 95

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding Sites; Diazepam; Flumazenil; GABA Agents; gamma-Aminobutyric Acid; HEK293 Cells; Humans; Membrane Potentials; Mutation; Neurons; Oocytes; Patch-Clamp Techniques; Protein Isoforms; Quinolines; Radioligand Assay; Receptors, GABA-A; Recombinant Proteins; Thiazoles; Transfection; Xenopus laevis

2015
Negative allosteric modulation of GABAA receptors inhibits facilitation of brain stimulation reward by drugs of abuse in C57BL6/J mice.
    Psychopharmacology, 2016, Volume: 233, Issue:4

    Topics: Allosteric Regulation; Animals; Azides; Benzodiazepines; Brain; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Illicit Drugs; Male; Mice; Mice, Inbred C57BL; Microdialysis; Receptors, GABA-A; Reward; Self Stimulation

2016
Effect of (+)-dehydrofukinone on GABAA receptors and stress response in fish model.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 2016, Volume: 49, Issue:1

    Topics: Anesthetics; Animals; Catfishes; Diazepam; Flame Ionization; Flumazenil; GABA Modulators; Gas Chromatography-Mass Spectrometry; Hydrocortisone; Hypnotics and Sedatives; Lauraceae; Oils, Volatile; Plant Extracts; Plant Leaves; Receptors, GABA-A; Sesquiterpenes; Stress, Physiological

2016
A microPET comparison of the effects of etifoxine and diazepam on [(11)C]flumazenil uptake in rat brains.
    Neuroscience letters, 2016, Jan-26, Volume: 612

    Topics: Animals; Anti-Anxiety Agents; Brain; Carbon Isotopes; Diazepam; Flumazenil; Magnetic Resonance Imaging; Male; Oxazines; Positron-Emission Tomography; Protein Binding; Radiopharmaceuticals; Rats, Wistar; Receptors, GABA-A

2016
Inhibition of Neuropathic Pain by a Single Intraperitoneal Injection of Diazepam in the Rat: Possible Role of Neurosteroids.
    The Chinese journal of physiology, 2016, 02-29, Volume: 59, Issue:1

    Topics: Animals; Benzodiazepinones; Carrier Proteins; Diazepam; Flumazenil; Injections, Intraperitoneal; Interleukin-1beta; Male; Neuralgia; Neurotransmitter Agents; Pregnenolone; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

2016
Determination of flumazenil in serum by liquid chromatography-mass spectrometry: Application to kinetics study in acute diazepam overdose.
    Vojnosanitetski pregled, 2016, Volume: 73, Issue:2

    Topics: Aminophylline; Antidotes; Chromatography, Liquid; Diazepam; Dimensional Measurement Accuracy; Dose-Response Relationship, Drug; Drug Interactions; Drug Overdose; Flumazenil; Half-Life; Humans; Hypnotics and Sedatives; Mass Spectrometry; Phosphodiesterase Inhibitors; Reproducibility of Results

2016
Benzodiazepine poisoning in elderly.
    Vojnosanitetski pregled, 2016, Volume: 73, Issue:3

    Topics: Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Antidotes; Benzodiazepines; Bromazepam; Cohort Studies; Coma; Diazepam; Drug Overdose; Female; Flumazenil; Humans; Incidence; Length of Stay; Lorazepam; Male; Middle Aged; Pneumonia, Aspiration; Respiratory Insufficiency; Retrospective Studies; Serbia; Suicide, Attempted; Young Adult

2016
Kavain, the Major Constituent of the Anxiolytic Kava Extract, Potentiates GABAA Receptors: Functional Characteristics and Molecular Mechanism.
    PloS one, 2016, Volume: 11, Issue:6

    Topics: Anesthetics; Animals; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Drug Interactions; Drug Synergism; Etomidate; Flumazenil; Humans; Kava; Mutation; Propofol; Protein Subunits; Pyrones; Receptors, GABA-A; Xenopus laevis

2016
Diazepam Inhibits Electrically Evoked and Tonic Dopamine Release in the Nucleus Accumbens and Reverses the Effect of Amphetamine.
    ACS chemical neuroscience, 2017, 02-15, Volume: 8, Issue:2

    Topics: Amphetamine; Analysis of Variance; Animals; Central Nervous System Stimulants; Diazepam; Dopamine; Dose-Response Relationship, Drug; Electric Stimulation; Electrochemical Techniques; Flumazenil; GABA Modulators; Mice; Microdialysis; Nucleus Accumbens

2017
The anxiolytic-like effect of rutin in rats involves GABAA receptors in the basolateral amygdala.
    Behavioural pharmacology, 2017, Volume: 28, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Basolateral Nuclear Complex; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Male; Maze Learning; Rats; Rats, Wistar; Receptors, GABA-A; Rutin

2017
Curcumol allosterically modulates GABA(A) receptors in a manner distinct from benzodiazepines.
    Scientific reports, 2017, 04-24, Volume: 7

    Topics: Allosteric Regulation; Animals; Benzodiazepines; CA1 Region, Hippocampal; Cells, Cultured; Diazepam; Drugs, Chinese Herbal; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; HEK293 Cells; Humans; Membrane Potentials; Pyramidal Cells; Receptors, GABA-A; Sesquiterpenes

2017
Intra-hippocampal microinjection of oxytocin produced antiepileptic effect on the pentylenetetrazol-induced epilepsy in rats.
    Pharmacological reports : PR, 2017, Volume: 69, Issue:4

    Topics: Animals; Anticonvulsants; Diazepam; Epilepsy; Flumazenil; Hippocampus; Male; Microinjections; Oxytocics; Oxytocin; Pentylenetetrazole; Rats; Tocolytic Agents; Vasotocin

2017
Diazepam Concurrently Increases the Frequency and Decreases the Amplitude of Transient Dopamine Release Events in the Nucleus Accumbens.
    The Journal of pharmacology and experimental therapeutics, 2018, Volume: 364, Issue:1

    Topics: Animals; Diazepam; Dopamine; Flumazenil; Male; Nucleus Accumbens; Rats; Time Factors

2018
The anxiolytic-like effect of 6-styryl-2-pyrone in mice involves GABAergic mechanism of action.
    Metabolic brain disease, 2018, Volume: 33, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Hippocampus; Imipramine; Male; Mice; Pyrones; Styrenes

2018
Subregion-Specific Impacts of Genetic Loss of Diazepam Binding Inhibitor on Synaptic Inhibition in the Murine Hippocampus.
    Neuroscience, 2018, 09-15, Volume: 388

    Topics: Animals; Central Nervous System Agents; Diazepam; Diazepam Binding Inhibitor; Female; Flumazenil; Hippocampus; Inhibitory Postsynaptic Potentials; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Miniature Postsynaptic Potentials; Neurons; Receptors, GABA-A; Tissue Culture Techniques

2018
Gephyrin Palmitoylation in Basolateral Amygdala Mediates the Anxiolytic Action of Benzodiazepine.
    Biological psychiatry, 2019, 02-01, Volume: 85, Issue:3

    Topics: Acyltransferases; Animals; Anti-Anxiety Agents; Anxiety; Basolateral Nuclear Complex; Benzodiazepines; Diazepam; Flumazenil; Gene Knockdown Techniques; Lipoylation; Male; Membrane Proteins; Rats; Receptors, GABA-A

2019
Biological profiling of piperazinediones for the management of anxiety.
    Pharmacology, biochemistry, and behavior, 2019, Volume: 176

    Topics: Amygdala; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Benzodiazepines; Catalytic Domain; Diazepam; Diketopiperazines; Flumazenil; GABA Modulators; Hypnotics and Sedatives; Male; Maze Learning; Models, Animal; Norepinephrine; Rats; Rats, Wistar; Receptors, GABA-A; Serotonin

2019
Benzodiazepines Suppress Neuromodulatory Effects of Pudendal Nerve Stimulation on Rat Bladder Nociception.
    Anesthesia and analgesia, 2020, Volume: 130, Issue:4

    Topics: Animals; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Female; Flumazenil; GABA Modulators; Midazolam; Motor Neurons; Muscle Contraction; Muscle, Smooth; Nociception; Pudendal Nerve; Rats; Rats, Sprague-Dawley; Sensory Receptor Cells; Urinary Bladder

2020
Shared structural mechanisms of general anaesthetics and benzodiazepines.
    Nature, 2020, Volume: 585, Issue:7824

    Topics: Allosteric Regulation; Anesthetics, General; Barbiturates; Benzodiazepines; Bicuculline; Binding Sites; Binding, Competitive; Cryoelectron Microscopy; Diazepam; Electrophysiology; Etomidate; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Ligands; Models, Molecular; Molecular Conformation; Molecular Dynamics Simulation; Phenobarbital; Picrotoxin; Propofol; Receptors, GABA-A

2020
Potential modulating effect of the Ascaris suum nicotinic acetylcholine receptor (nAChR) by compounds GSK575594A, diazepam and flumazenil discovered by structure-based virtual screening approach.
    Molecular and biochemical parasitology, 2021, Volume: 242

    Topics: Acetylcholine; Animals; Anthelmintics; Ascaris suum; Binding Sites; Caenorhabditis elegans Proteins; Databases, Chemical; Diazepam; Flumazenil; Gene Expression; Helminth Proteins; High-Throughput Screening Assays; Humans; Ligands; Molecular Docking Simulation; Muscles; Piperazines; Protein Binding; Protein Conformation, alpha-Helical; Protein Conformation, beta-Strand; Protein Interaction Domains and Motifs; Receptors, Nicotinic; Structural Homology, Protein; Tissue Culture Techniques; User-Computer Interface

2021
How does α
    Physical chemistry chemical physics : PCCP, 2021, Feb-19, Volume: 23, Issue:6

    Topics: Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Histidine; Humans; Molecular Dynamics Simulation; Protein Conformation; Protein Subunits; Protons; Receptors, GABA-A

2021
The biologically active compound of
    Journal of psychopharmacology (Oxford, England), 2021, Volume: 35, Issue:10

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Ethanol; Flumazenil; Male; Maze Learning; Mice; Plant Extracts; Reflex, Righting; Withania

2021
Bumetanide prevents diazepam-modified anxiety-like behavior in lipopolysaccharide-treated mice.
    European journal of pharmacology, 2021, Aug-05, Volume: 904

    Topics: Animals; Anti-Anxiety Agents; Anti-Bacterial Agents; Anxiety; Behavior, Animal; Bicuculline; Bumetanide; Diazepam; Emotions; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Inflammation; Lipopolysaccharides; Male; Mice, Inbred ICR; Minocycline; Motor Activity; Sodium Potassium Chloride Symporter Inhibitors

2021
Sedative-hypnotic, anxiolytic and possible side effects of Salvia limbata C. A. Mey. Extracts and the effects of phenological stage and altitude on the rosmarinic acid content.
    Journal of ethnopharmacology, 2022, Jan-10, Volume: 282

    Topics: Altitude; Animals; Antidotes; Cinnamates; Depsides; Diazepam; Flumazenil; Hypnotics and Sedatives; Male; Memory; Mice; Plant Components, Aerial; Plant Extracts; Rosmarinic Acid; Salvia; Toxicity Tests

2022
High-Dose Benzodiazepines Positively Modulate GABA
    International journal of molecular sciences, 2021, Dec-21, Volume: 23, Issue:1

    Topics: Animals; Animals, Outbred Strains; Benzodiazepines; Clonazepam; Diazepam; Female; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Midazolam; Receptors, GABA-A; Xenopus laevis

2021
Anxiolytic-like Effect of Quercetin Possibly through GABA Receptor Interaction Pathway: In Vivo and In Silico Studies.
    Molecules (Basel, Switzerland), 2022, Oct-22, Volume: 27, Issue:21

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Diazepam; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Maze Learning; Mice; Quercetin; Receptors, GABA; Receptors, GABA-A

2022