flumazenil and clonazepam

flumazenil has been researched along with clonazepam in 97 studies

Research

Studies (97)

TimeframeStudies, this research(%)All Research%
pre-199040 (41.24)18.7374
1990's34 (35.05)18.2507
2000's16 (16.49)29.6817
2010's6 (6.19)24.3611
2020's1 (1.03)2.80

Authors

AuthorsStudies
Da Settimo, A; Da Settimo, F; Giannaccini, G; Greco, G; Lucacchini, A; Marini, AM; Martini, C; Novellino, E; Primofiore, G1
Da Settimo, A; Da Settimo, F; Gesi, M; Giannaccini, G; Greco, G; Lucacchini, A; Marini, AM; Martini, C; Novellino, E; Primofiore, G1
Da Settimo, F; Gesi, M; Greco, G; La Motta, C; Marini, AM; Martini, C; Novellino, E; Primofiore, G; Taliani, S; Trincavelli, L1
Topliss, JG; Yoshida, F1
Besnard, F; Costa, B; Greco, G; Lavecchia, A; Marini, AM; Martini, C; Novellino, E; Primofiore, G; Settimo, FD; Taliani, S; Trincavelli, L1
Besnard, F; Cosimelli, B; Costa, B; Da Settimo, F; Greco, G; Martini, C; Montali, M; Novellino, E; Primofiore, G; Salerno, S; Taliani, S1
Besnard, F; Calderone, V; Cosimelli, B; Da Settimo, F; Greco, G; La Motta, C; Marini, AM; Martini, C; Montali, M; Novellino, E; Patrizi, MP; Primofiore, G; Sergianni, V; Simorini, F; Taliani, S1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Järvinen, A; Männistö, PT; Rägo, L1
Almog, S; Ezra, D; Mordel, A; Tirosh, M; Winkler, E1
Fiszer de Plazas, S; Gravielle, MC1
Galpern, WR; Greenblatt, DJ; Lumpkin, M; Miller, LG; Shader, RI1
Miller, LG1
al-Tikriti, MS; Baldwin, RM; Innis, RB; Johnson, EW; Laruelle, MA; Malison, RT; Seibyl, JP; Sybirska, EH; Zimmermann, RC; Zoghbi, SS1
Blasquez, C; Braquet, P; Delbende, C; Jégou, S; Tranchand Bunel, D; Vaudry, H1
Karim, KH; Najim, RA1
De Luca, C; De Medici, D; Massotti, M1
Izquierdo, I; Medina, JH; Pereira, ME1
Elgoyhen, AB; Kazanietz, MG1
Deutsch, SI; Huntzinger, JA; Mastropaolo, J; Novitzki, MR; Rosse, RB1
Haefely, W1
Adler-Graschinsky, E; Elgoyhen, B1
al-Essa, LY; al-Jawad, FH; Najim, RA1
Bachy, A; Cordeau, LR; Croizat, BP; Gros, F; Keane, PE; Larcher, JC; Le Marquer, FJ; Vayssiere, JL1
Deutsch, SI; Kook, KA; Paul, SM; Vocci, F; Weizman, A; Weizman, R1
Fukuda, H; Hirayama, K; Inoue, O; Itoh, T; Iyo, M; Shinotoh, H; Suzuki, K; Tateno, Y; Yamada, T; Yamasaki, T1
Miller, LG; Roy, RB; Weill, CL1
Kellogg, CK; Miranda, RC; Wagner, JP1
Hanada, S; Hashimoto, S; Tanaka, C; Taniyama, K1
Greenblatt, DJ; Lopez, F; Miller, LG; Paul, SM; Shader, RI1
Ennis, C; Minchin, MC1
Concas, A; Morelli, M; Obata, T; Serra, M; Yamamura, HI1
Deutsch, SI; Greenblatt, DJ; Miller, LG; Paul, SM; Shader, RI1
Karobath, M; Supavilai, P1
Capek, R; Davies, MF; Esplin, B1
Goeders, NE; Kuhar, MJ1
Cooper, SJ; Gilbert, DB1
Chweh, AY; Swinyard, EA; Wolf, HH1
Cole, R; De Vellis, J; Noble, EP; Syapin, PJ1
Fares, F; Gavish, M1
Haefely, W; Möhler, H; Richards, JG; Schoch, P1
Bryere, P; Naquet, R; Valin, A1
Greenblatt, DJ; Miller, LG; Paul, SM; Shader, RI1
Lafaille, F; Lal, S; Nair, NP; Quirion, R; Suranyi-Cadotte, B1
Adjeroud, S; Cazin, L; Danger, JM; Gouteux, L; Lamacz, M; Leneveu, E; Tonon, MC; Vaudry, H1
Deutsch, SI; Greenblatt, DJ; Miller, LG; Paul, SM; Shader, RI; Thompson, ML1
Bryere, P; Menini, C; Rektor, I; Silva-Barrat, C1
Frey, HH; Scherkl, R1
Teo, WL; Wong, PT1
Kunert-Radek, J; Pawlikowski, M; Radek, A; Stepien, H1
Herblin, WF; Mechem, CC1
Belin, C; Carriot, T; Dubroeucq, MC; Guérémy, C; Le Fur, G; Mestre, M; Renault, C; Uzan, A1
Brown, C; Martin, IL1
Caputti, E; Cardinali, DP; Lowenstein, PR; Rosenstein, R1
Möhler, H; Richards, JG1
Carney, JM; Nakamura, M1
Möhler, H1
Camoratto, AM; Grandison, L1
Matlib, MA; Schwartz, A1
Clineschmidt, BV1
Ekström, P; Grossmann, E; Meissl, H; Yáñez, J1
Niles, LP; Tenn, CC1
Breschi, MC; Cristofani, R; Giannaccini, G; Lucacchini, A; Martini, C; Martinotti, E; Scatizzi, R1
Antonenko, YN; Kinnally, KW; McEnery, MW; Snyder, SH; Tedeschi, H; Zorov, DB1
Berigan, TR; Harazin, J; Williams, HL1
Chen, JS; Gee, KW; Johnson, D; Lan, NC1
Matthews, EK; Ratcliffe, SL1
Fuchs, K; Mossier, B; Sieghart, W; Tögel, M1
Harris, RA; Klein, RL; Whiting, PJ1
Auta, J; Costa, E; Guidotti, A; Kozikowski, A; Ma, D; Romeo, E1
Lichtensteiger, W; Ramseier, H; Schlumpf, M1
Hansen, HC; Jackson, HC; Judge, ME; Klitgaard, H; Kristiansen, M; Suzdak, PD; Swedberg, MD1
Cespuglio, R; Miachon, S1
Buldakova, S; Weiss, M1
Blanc, F; Butterworth, RF; Fabbro-Peray, P; Lavoie, J; Layrargues, GP; Mousseau, DD; Perney, P1
Kawaguchi, M; Okubo, M1
Bender, AS; Norenberg, MD1
Leeuwin, RS; van Wilgenburg, H; Zeegers, A1
Ito, K1
Contarino, A; Giusti, P; Lipartiti, M; Natolino, F; Zanotti, A1
Abekawa, T; Ito, K; Koyama, T; Ohmori, T1
Brown, SD; Skeen, GA; White, HS; Wolf, HH; Woodhead, JH1
Li, M; Rosenberg, HC; Szabo, A1
Paz, L; Peter, Y; Pick, CG; Toren, P; Weizman, R1
Bruni, F; Ciciani, G; Costa, B; Costagli, C; Costanzo, A; Guerrini, G; Martini, C; Selleri, S1
Al-Mulla Hummadi, YM; Farjou, IB; Najim, RA1
Elías, MM; Monasterolo, LA; Trumper, L1
Copolov, D; Dean, B; McLeod, M; Pralong, D1
Dean, B; McLeod, M; Scarr, E1
Arroyo Plasencia, AM; Ballentine, LM; Kao, LW; Mowry, JB1
Des Jarlais, DC; Gerra, G; Lugoboni, F; Mathewson, S; Pattaro, C; Quaglio, G; Verbanck, P1
Choi, KH; Kyong, YY; Park, JT1
Johnson, AL; Setlakwe, EL1
Cao, Y; Lian, J; Ma, Y; Muheyati, A; Su, R; Wang, N; Yu, G; Yuan, S; Zhang, S1

Reviews

4 review(s) available for flumazenil and clonazepam

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Chronic benzodiazepine administration: from the patient to the gene.
    Journal of clinical pharmacology, 1991, Volume: 31, Issue:6

    Topics: Alprazolam; Animals; Benzodiazepines; Clonazepam; Down-Regulation; Drug Tolerance; Flumazenil; Humans; Lorazepam; Mice; Receptors, GABA-A; RNA, Messenger; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors; Up-Regulation

1991
Benzodiazepine receptors resolved.
    Experientia, 1986, Feb-15, Volume: 42, Issue:2

    Topics: Animals; Antibodies, Monoclonal; Autoradiography; Benzodiazepines; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Clonazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Histocytochemistry; Humans; Immunologic Techniques; Ionophores; Muscimol; Neurons; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Spinal Cord; Synapses; Tissue Distribution

1986
Benzodiazepine receptors: mode of interaction of agonists and antagonists.
    Advances in biochemical psychopharmacology, 1983, Volume: 37

    Topics: Affinity Labels; Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Clonazepam; Drug Interactions; Flumazenil; gamma-Aminobutyric Acid; Ligands; Models, Biological; Receptors, Cell Surface; Receptors, GABA-A; Terminology as Topic; Thermodynamics

1983

Trials

1 trial(s) available for flumazenil and clonazepam

ArticleYear
High dose benzodiazepine dependence: description of 29 patients treated with flumazenil infusion and stabilised with clonazepam.
    Psychiatry research, 2012, Aug-15, Volume: 198, Issue:3

    Topics: Adult; Antidepressive Agents; Benzodiazepines; Clonazepam; Drug Therapy, Combination; Female; Flumazenil; GABA Modulators; Humans; Infusions, Intravenous; Male; Middle Aged; Substance Withdrawal Syndrome; Substance-Related Disorders

2012

Other Studies

92 other study(ies) available for flumazenil and clonazepam

ArticleYear
Synthesis, structure-activity relationships, and molecular modeling studies of N-(indol-3-ylglyoxylyl)benzylamine derivatives acting at the benzodiazepine receptor.
    Journal of medicinal chemistry, 1996, Dec-20, Volume: 39, Issue:26

    Topics: Animals; Brain; Cattle; Indoles; Mice; Models, Molecular; Radioligand Assay; Receptors, GABA-A; Structure-Activity Relationship

1996
N'-Phenylindol-3-ylglyoxylohydrazide derivatives: synthesis, structure-activity relationships, molecular modeling studies, and pharmacological action on brain benzodiazepine receptors.
    Journal of medicinal chemistry, 1998, Sep-24, Volume: 41, Issue:20

    Topics: Animals; Anticonvulsants; Binding, Competitive; Brain; Cattle; Cerebral Cortex; Convulsants; Diazepam; Flumazenil; GABA Modulators; Glyoxylates; Hydrazines; In Vitro Techniques; Indoles; Ligands; Mice; Models, Molecular; Molecular Conformation; Receptors, GABA-A; Seizures; Structure-Activity Relationship

1998
3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: tricyclic heteroaromatic derivatives as a new class of benzodiazepine receptor ligands.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Anticonvulsants; Benzimidazoles; Brain; Cattle; Convulsants; Diazepam; Flumazenil; GABA Modulators; In Vitro Techniques; Ligands; Membranes; Mice; Models, Molecular; Radioligand Assay; Receptors, GABA-A

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Novel N-(arylalkyl)indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships.
    Journal of medicinal chemistry, 2001, Jul-05, Volume: 44, Issue:14

    Topics: Amides; Animals; Brain; Cattle; Glyoxylates; In Vitro Techniques; Indoles; Ligands; Models, Molecular; Radioligand Assay; Receptors, GABA-A; Structure-Activity Relationship

2001
High affinity central benzodiazepine receptor ligands: synthesis and biological evaluation of a series of phenyltriazolobenzotriazindione derivatives.
    Journal of medicinal chemistry, 2005, Apr-21, Volume: 48, Issue:8

    Topics: Animals; Binding, Competitive; Brain; Cattle; Cell Line; Chlorides; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Humans; In Vitro Techniques; Models, Molecular; Protein Isoforms; Radioligand Assay; Rats; Recombinant Proteins; Structure-Activity Relationship; Triazines; Triazoles

2005
Novel N-substituted indol-3-ylglyoxylamides probing the LDi and L1/L2 lipophilic regions of the benzodiazepine receptor site in search for subtype-selective ligands.
    Journal of medicinal chemistry, 2007, Apr-05, Volume: 50, Issue:7

    Topics: Amides; Animals; Cattle; Cell Line; Cerebral Cortex; GABA-A Receptor Agonists; Glyoxylates; Hypnotics and Sedatives; In Vitro Techniques; Indoles; Ligands; Male; Mice; Mice, Inbred BALB C; Molecular Conformation; Motor Activity; Radioligand Assay; Rats; Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Effects of central and peripheral type benzodiazepine ligands on thyrotropin and prolactin secretion.
    Neuropeptides, 1992, Volume: 21, Issue:3

    Topics: Animals; Benzodiazepinones; Carbolines; Clonazepam; Cold Temperature; Diazepam; Flumazenil; Hypothalamo-Hypophyseal System; Isoquinolines; Male; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Secretory Rate; Thyrotropin; Thyrotropin-Releasing Hormone

1992
Seizures after flumazenil administration in a case of combined benzodiazepine and tricyclic antidepressant overdose.
    Critical care medicine, 1992, Volume: 20, Issue:12

    Topics: Adult; Clonazepam; Diazepam; Drug Overdose; Epilepsy, Tonic-Clonic; Female; Flumazenil; Humans; Imipramine; Poisoning

1992
Benzodiazepine receptor sites in the chick optic lobe: development and pharmacological characterization.
    Neurochemical research, 1991, Volume: 16, Issue:1

    Topics: Animals; Binding, Competitive; Chick Embryo; Chickens; Clonazepam; Flumazenil; Flunitrazepam; Kinetics; Receptors, GABA-A; Synaptic Membranes; Tectum Mesencephali; Time Factors

1991
Chronic benzodiazepine administration. VII. Behavioral tolerance and withdrawal and receptor alterations associated with clonazepam administration.
    Psychopharmacology, 1991, Volume: 104, Issue:2

    Topics: Animals; Behavior, Animal; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Clonazepam; Convulsants; Drug Tolerance; Flumazenil; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Substance Withdrawal Syndrome

1991
SPECT imaging of the benzodiazepine receptor: feasibility of in vivo potency measurements from stepwise displacement curves.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1991, Volume: 32, Issue:9

    Topics: Alprazolam; Animals; Benzodiazepines; Brain; Brain Chemistry; Clonazepam; Diazepam; Female; Flumazenil; Injections, Intravenous; Macaca mulatta; Male; Papio; Receptors, GABA-A; Tomography, Emission-Computed, Single-Photon

1991
Central-type benzodiazepines inhibit release of alpha-melanocyte-stimulating hormone from the rat hypothalamus.
    Neuroscience, 1991, Volume: 42, Issue:2

    Topics: Animals; Anti-Anxiety Agents; beta-Endorphin; Clonazepam; Diazepam; Flumazenil; GABA Antagonists; Hypothalamus; In Vitro Techniques; Male; Melanocyte-Stimulating Hormones; Perfusion; Pituitary Gland; Potassium Chloride; Pro-Opiomelanocortin; Pyridazines; Radioimmunoassay; Rats; Rats, Inbred Strains

1991
Protection against ethanol-induced gastric damage by drugs acting at the GABA-benzodiazepine receptor complex.
    Psychopharmacology, 1991, Volume: 103, Issue:1

    Topics: Animals; Benzodiazepinones; Clonazepam; Dose-Response Relationship, Drug; Ethanol; Flumazenil; Gastric Mucosa; Indomethacin; Male; Postural Balance; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reflex

1991
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
    Psychopharmacology, 1990, Volume: 102, Issue:4

    Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem

1990
Benzodiazepine receptor ligand influences on acquisition: suggestion of an endogenous modulatory mechanism mediated by benzodiazepine receptors.
    Behavioral and neural biology, 1990, Volume: 54, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Arousal; Avoidance Learning; Benzodiazepinones; Brain; Carbolines; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Flumazenil; Habituation, Psychophysiologic; Memory; Mental Recall; Rats; Rats, Inbred Strains; Reaction Time; Receptors, GABA-A; Retention, Psychology

1990
Relaxant effect of benzodiazepines on uterine rings isolated from estrogen-treated rats.
    European journal of pharmacology, 1990, Aug-28, Volume: 185, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Bicuculline; Clonazepam; Convulsants; Diazepam; Estradiol; Estrogens; Female; Flumazenil; In Vitro Techniques; Isoquinolines; Muscle, Smooth; Potassium Chloride; Propranolol; Rats; Rats, Inbred Strains; Uterine Contraction

1990
Profound stress-induced alterations in flurazepam's antiseizure efficacy can be attenuated.
    Brain research, 1990, Jun-18, Volume: 520, Issue:1-2

    Topics: Animals; Carbolines; Clonazepam; Cold Temperature; Diazepam; Dose-Response Relationship, Drug; Electroshock; Flumazenil; Flurazepam; Male; Mice; Mice, Inbred Strains; Midazolam; Seizures; Stress, Psychological

1990
Partial agonists of the benzodiazepine receptor: from animal data to results in patients.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Affinity Labels; Allosteric Site; Animals; Azides; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Chlorides; Clonazepam; Diazepam; Drug Interactions; Ethanol; Flumazenil; Flurazepam; Humans; Ion Channels; Ligands; Models, Neurological; Neurons; Receptors, GABA-A

1988
Diminution by benzodiazepines of the chronotropic responses to noradrenaline in rat isolated atria.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Colforsin; Cyclic AMP; Diazepam; Female; Flumazenil; Heart; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains

1989
Effect of some drugs acting at the central-type benzodiazepine receptors on blood glucose in mice.
    Clinical and experimental pharmacology & physiology, 1989, Volume: 16, Issue:1

    Topics: Animals; Benzodiazepinones; Blood Glucose; Clonazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Mice; Mice, Inbred ICR; Quinolines; Receptors, GABA-A

1989
Effects of peripheral benzodiazepines upon the O2 consumption of neuroblastoma cells.
    European journal of pharmacology, 1989, Feb-28, Volume: 161, Issue:2-3

    Topics: Animals; Benzodiazepines; Cells, Cultured; Clonazepam; Clone Cells; Diazepam; Flumazenil; Isoquinolines; Mice; Mitochondria; Neuroblastoma; Oxygen Consumption; Receptors, GABA-A

1989
Repeated swim stress alters brain benzodiazepine receptors measured in vivo.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:3

    Topics: Animals; Brain; Cerebrovascular Circulation; Clonazepam; Flumazenil; Male; Mice; Pentylenetetrazole; Receptors, GABA-A; Seizures; Stress, Physiological; Swimming; Tritium

1989
Detection of benzodiazepine receptor occupancy in the human brain by positron emission tomography.
    Psychopharmacology, 1989, Volume: 99, Issue:2

    Topics: Adult; Brain; Clonazepam; Electroencephalography; Evoked Potentials, Auditory; Female; Flumazenil; Humans; Male; Receptors, GABA-A; Tomography, Emission-Computed

1989
Chronic clonazepam administration decreases gamma-aminobutyric acidA receptor function in cultured cortical neurons.
    Molecular pharmacology, 1989, Volume: 36, Issue:5

    Topics: Animals; Benzodiazepines; Cells, Cultured; Cerebral Cortex; Chick Embryo; Chlorides; Clonazepam; Drug Administration Schedule; Flumazenil; Muscimol; Picrotoxin; Receptors, GABA-A; Sesterterpenes

1989
Early developmental exposure to benzodiazepine ligands alters brain levels of thiobarbituric acid-reactive products in young adult rats.
    Neurochemical research, 1989, Volume: 14, Issue:11

    Topics: Animals; Benzodiazepines; Brain; Clonazepam; Diazepam; Female; Flumazenil; Gestational Age; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Receptors, GABA-A; Thiobarbiturates

1989
Benzodiazepines and barbiturate potentiate the pre- and postsynaptic gamma-aminobutyric acid (GABA)A receptor-mediated response in the enteric nervous system of guinea pig small intestine.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Acetylcholine; Animals; Barbiturates; Benzodiazepines; Clonazepam; Diazepam; Female; Flumazenil; Guinea Pigs; Intestine, Small; Male; Muscimol; Pentobarbital; Potassium; Receptors, GABA-A

1988
Low-dose alprazolam augments motor activity in mice.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:2

    Topics: Alprazolam; Animals; Clonazepam; Exploratory Behavior; Flumazenil; Male; Mice; Mice, Inbred Strains; Motor Activity; Receptors, GABA-A; Triazolam

1988
Modulation of the GABA autoreceptor by benzodiazepine receptor ligands.
    Neuropharmacology, 1988, Volume: 27, Issue:10

    Topics: Animals; Bicuculline; Carbolines; Clonazepam; Flumazenil; Ligands; Male; Muscimol; Rats; Receptors, GABA-A

1988
Modulation of GABA-stimulated chloride influx into membrane vesicles from rat cerebral cortex by benzodiazepines and nonbenzodiazepines.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Anti-Anxiety Agents; Cell Membrane; Cerebral Cortex; Chlorides; Clonazepam; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Inbred Strains

1988
Acute barbiturate administration increases benzodiazepine receptor binding in vivo.
    Psychopharmacology, 1988, Volume: 96, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Barbiturates; Brain Chemistry; Clonazepam; Flumazenil; gamma-Aminobutyric Acid; Injections, Intraperitoneal; Male; Mice; Pentobarbital; Receptors, GABA-A

1988
Modulation of acetylcholine release from rat striatal slices by the GABA/benzodiazepine receptor complex.
    Life sciences, 1985, Feb-04, Volume: 36, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Baclofen; Benzodiazepinones; Clonazepam; Corpus Striatum; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Haloperidol; In Vitro Techniques; Isoxazoles; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
The effects of benzodiazepines on spinal homosynaptic depression.
    Neuropharmacology, 1985, Volume: 24, Issue:4

    Topics: Animals; Benzodiazepinones; Cats; Clonazepam; Diazepam; Female; Flumazenil; Male; Receptors, GABA-A; Reflex, Monosynaptic; Reflex, Stretch; Spinal Nerve Roots; Synapses

1985
Benzodiazepine receptor binding in vivo with [3H]-Ro 15-1788.
    Life sciences, 1985, Jul-29, Volume: 37, Issue:4

    Topics: Animals; Autoradiography; Benzodiazepinones; Brain; Clonazepam; Flumazenil; Flunitrazepam; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Receptors, GABA-A; Time Factors; Tritium

1985
Clonazepam-induced hyperphagia in nondeprived rats: tests of pharmacological specificity with Ro5-4864, Ro5-3663, Ro15-1788 and CGS 9896.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:5

    Topics: Animals; Benzodiazepinones; Clonazepam; Drug Interactions; Feeding Behavior; Flumazenil; Humans; Hyperphagia; Male; Pyrazoles; Rats; Receptors, GABA-A

1985
Benzodiazepine receptors are not involved in the neurotoxicity and anti-electroshock activity of phenytoin in mice.
    Neuroscience letters, 1985, Jun-24, Volume: 57, Issue:3

    Topics: Animals; Benzodiazepinones; Clonazepam; Drug Interactions; Electroshock; Flumazenil; Male; Mice; Phenytoin; Receptors, GABA-A; Seizures

1985
Benzodiazepine binding characteristics of embryonic rat brain neurons grown in culture.
    Journal of neurochemistry, 1985, Volume: 45, Issue:6

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cells, Cultured; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Neurons; Pyridazines; Rats; Receptors, GABA-A

1985
Solubilization of peripheral benzodiazepine-binding sites from rat kidney.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1985, Volume: 5, Issue:11

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Carbolines; Chlordiazepoxide; Clonazepam; Diazepam; Digitonin; Flumazenil; Flurazepam; Guanidine; Guanidines; Hot Temperature; Isoquinolines; Kidney; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Solubility; Time Factors; Urea

1985
Convulsant effect of Ro 5-4864, a peripheral type benzodiazepine, on the baboon (Papio papio).
    Neuroscience letters, 1986, May-15, Volume: 66, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Isoquinolines; Papio; Receptors, GABA-A; Seizures

1986
Benzodiazepine receptor occupancy in vivo: correlation with brain concentrations and pharmacodynamic actions.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:2

    Topics: Animals; Cerebral Cortex; Clonazepam; Dose-Response Relationship, Drug; Flumazenil; Lorazepam; Male; Mice; Receptors, GABA-A; Time Factors

1987
Coexistence of central and peripheral benzodiazepine binding sites in the human pineal gland.
    Life sciences, 1987, Apr-13, Volume: 40, Issue:15

    Topics: Aged; Benzodiazepinones; Binding, Competitive; Cell Membrane; Clonazepam; Female; Flumazenil; Flunitrazepam; Humans; Isoquinolines; Male; Middle Aged; Pineal Gland; Receptors, GABA-A

1987
The benzodiazepine agonist clonazepam potentiates the effects of gamma-aminobutyric acid on alpha-MSH release from neurointermediate lobes in vitro.
    Life sciences, 1987, May-11, Volume: 40, Issue:19

    Topics: Animals; Clonazepam; Drug Synergism; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Melanocyte-Stimulating Hormones; Perfusion; Pituitary Gland, Posterior; Rana ridibunda; Receptors, GABA-A

1987
Rapid increase in brain benzodiazepine receptor binding following defeat stress in mice.
    Brain research, 1987, Jun-30, Volume: 414, Issue:2

    Topics: Adrenalectomy; Animals; Brain; Cerebral Cortex; Clonazepam; Flumazenil; Lorazepam; Male; Mice; Receptors, GABA-A; Species Specificity; Stress, Psychological; Time Factors

1987
Stimulus-sensitive myoclonus of the baboon Papio papio: pharmacological studies reveal interactions between benzodiazepines and the central cholinergic system.
    Experimental neurology, 1986, Volume: 91, Issue:1

    Topics: Animals; Atropine; Benzodiazepines; Benzodiazepinones; Clonazepam; Drug Interactions; Flumazenil; Myoclonus; Neostigmine; Papio; Parasympathetic Nervous System; Physostigmine; Quinuclidinyl Benzilate

1986
Physical dependence on clonazepam in dogs.
    Pharmacology, 1986, Volume: 32, Issue:1

    Topics: Animals; Benzodiazepinones; Body Temperature; Body Weight; Clonazepam; Dogs; Female; Flumazenil; Male; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders; Tremor

1986
Diazepam-sensitive specific binding of phenytoin in rat brain.
    Journal of receptor research, 1986, Volume: 6, Issue:3-4

    Topics: Animals; Benzodiazepinones; Binding Sites; Cell Membrane; Cerebral Cortex; Clonazepam; Diazepam; Flumazenil; Male; Phenytoin; Rats; Rats, Inbred Strains

1986
Inhibition of cell proliferation of human gliomas by benzodiazepines in vitro.
    Acta neurologica Scandinavica, 1988, Volume: 77, Issue:3

    Topics: Astrocytoma; Benzodiazepines; Benzodiazepinones; Cell Division; Clonazepam; Diazepam; Female; Flumazenil; Glioma; Humans; Male; Middle Aged; Thymidine; Tumor Cells, Cultured

1988
Short-wave ultraviolet irradiation increases photo-affinity labeling of benzodiazepine sites.
    Life sciences, 1984, Jul-16, Volume: 35, Issue:3

    Topics: Affinity Labels; Animals; Benzodiazepinones; Binding Sites; Cell Membrane; Cerebellum; Cerebral Cortex; Clonazepam; Flumazenil; Flunitrazepam; In Vitro Techniques; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Ultraviolet Rays

1984
Electrophysiological and pharmacological characterization of peripheral benzodiazepine receptors in a guinea pig heart preparation.
    Life sciences, 1984, Aug-27, Volume: 35, Issue:9

    Topics: Action Potentials; Animals; Benzodiazepinones; Clonazepam; Convulsants; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; Flumazenil; Guinea Pigs; Heart; In Vitro Techniques; Isoquinolines; Myocardial Contraction; Myocardium; Receptors, Cell Surface; Receptors, GABA-A

1984
Autoradiographic localisation of benzodiazepine receptors in the rat pituitary gland.
    European journal of pharmacology, 1984, Jul-20, Volume: 102, Issue:3-4

    Topics: Animals; Autoradiography; Benzodiazepinones; Clonazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Benzodiazepine binding sites in human pineal gland.
    European journal of pharmacology, 1984, Nov-13, Volume: 106, Issue:2

    Topics: Adolescent; Adult; Aged; Animals; Benzodiazepinones; Binding, Competitive; Cerebral Cortex; Child; Child, Preschool; Clonazepam; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Infant; Kinetics; Male; Middle Aged; Pineal Gland; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Agonist and antagonist benzodiazepine receptor interaction in vitro.
    Nature, 1981, Dec-24, Volume: 294, Issue:5843

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Brain; Clonazepam; Flumazenil; Hot Temperature; Rats; Receptors, Drug; Receptors, GABA-A

1981
Separation of clonazepam-induced head twitches and muscle relaxation in mice.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:3

    Topics: Animals; Benzodiazepinones; Clonazepam; Drug Interactions; Flumazenil; Head; Male; Methysergide; Mice; Movement; Muscle Relaxants, Central; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A

1983
Inhibition of cold-induced TSH release by benzodiazepines.
    Brain research, 1983, Apr-18, Volume: 265, Issue:2

    Topics: Animals; Benzodiazepinones; Clonazepam; Cold Temperature; Depression, Chemical; Diazepam; Drug Interactions; Flumazenil; Male; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains; Thyrotropin; Thyrotropin-Releasing Hormone

1983
Selective effects of diltiazem, a benzothiazepine calcium channel blocker, and diazepam, and other benzodiazepines on the Na+/Ca2+ exchange carrier system of heart and brain mitochondria.
    Life sciences, 1983, Jun-20, Volume: 32, Issue:25

    Topics: Animals; Benzazepines; Benzodiazepines; Benzodiazepinones; Brain; Calcium; Carrier Proteins; Clonazepam; Diazepam; Diltiazem; Flumazenil; Mitochondria; Mitochondria, Heart; Rabbits; Rats; Sodium; Sodium-Calcium Exchanger

1983
Effect of the benzodiazepine receptor antagonist Ro 15-1788 on the anticonvulsant and anticonflict actions of MK-801.
    European journal of pharmacology, 1982, Oct-15, Volume: 84, Issue:1-2

    Topics: Animals; Anticonvulsants; Behavior, Animal; Benzodiazepinones; Bicuculline; Chlordiazepoxide; Clonazepam; Conflict, Psychological; Dibenzocycloheptenes; Dizocilpine Maleate; Drug Interactions; Female; Flumazenil; Mice; Phenobarbital; Rats; Rats, Inbred Strains

1982
Benzodiazepines influence melatonin secretion of the pineal organ of the trout in vitro.
    Journal of pineal research, 1994, Volume: 17, Issue:2

    Topics: 5-Methoxytryptamine; Animals; Benzodiazepines; Calcium; Clonazepam; Culture Media; Dark Adaptation; Diazepam; Flumazenil; Hydroxyindoleacetic Acid; In Vitro Techniques; Indoles; Isoquinolines; Light; Magnesium; Melatonin; Oncorhynchus mykiss; Pineal Gland

1994
Central-type benzodiazepine receptors mediate the antidopaminergic effect of clonazepam and melatonin in 6-hydroxydopamine lesioned rats: involvement of a GABAergic mechanism.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:1

    Topics: Animals; Apomorphine; Behavior, Animal; Bicuculline; Clonazepam; Corpus Striatum; Dopamine Agonists; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Isoquinolines; Male; Melatonin; Oxidopamine; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

1995
Benzodiazepine agonists reverse the effects of noise exposure on central benzodiazepine receptors and cardiac responsiveness.
    Life sciences, 1995, Volume: 57, Issue:11

    Topics: Animals; Brain; Clonazepam; Diazepam; Flumazenil; Imidazoles; Male; Myocardium; Noise; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, GABA-A; Stress, Psychological

1995
Mitochondrial benzodiazepine receptor linked to inner membrane ion channels by nanomolar actions of ligands.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Feb-15, Volume: 90, Issue:4

    Topics: Animals; Benzodiazepinones; Clonazepam; Convulsants; Flumazenil; Intracellular Membranes; Ion Channels; Isoquinolines; Male; Membrane Potentials; Mitochondria, Heart; Protoporphyrins; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Submitochondrial Particles

1993
Use of flumazenil in conjunction with electroconvulsive therapy.
    The American journal of psychiatry, 1995, Volume: 152, Issue:6

    Topics: Adult; Clonazepam; Depressive Disorder; Electroconvulsive Therapy; Female; Flumazenil; Humans; Substance Withdrawal Syndrome; Substance-Related Disorders

1995
Differential effects of 4'-chlorodiazepam on expressed human GABAA receptors.
    Journal of neurochemistry, 1995, Volume: 64, Issue:2

    Topics: Benzodiazepinones; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Clonazepam; Flumazenil; Humans; Quinolines; Receptors, GABA; Transfection

1995
Modification of the photodynamic action of delta-aminolaevulinic acid (ALA) on rat pancreatoma cells by mitochondrial benzodiazepine receptor ligands.
    British journal of cancer, 1995, Volume: 71, Issue:2

    Topics: Aminolevulinic Acid; Animals; Benzodiazepines; Benzodiazepinones; Cell Division; Cell Survival; Clonazepam; Flumazenil; Isoquinolines; Ligands; Mitochondria; Oxygen; Pancreatic Neoplasms; Photochemotherapy; Protoporphyrins; Radiation-Protective Agents; Radiation-Sensitizing Agents; Rats; Receptors, GABA-A; Singlet Oxygen; Tumor Cells, Cultured

1995
Immunoaffinity purification of gamma-aminobutyric acidA (GABAA) receptors containing gamma 1-subunits. Evidence for the presence of a single type of gamma-subunit in GABAA receptors.
    The Journal of biological chemistry, 1994, Oct-14, Volume: 269, Issue:41

    Topics: Animals; Antibody Specificity; Base Sequence; Blotting, Western; Brain Chemistry; Chromatography, Affinity; Clonazepam; Enzyme-Linked Immunosorbent Assay; Flumazenil; Flunitrazepam; Immunologic Techniques; Molecular Sequence Data; Molecular Weight; Muscimol; Peptide Fragments; Protein Conformation; Rats; Receptors, GABA-A; Recombinant Fusion Proteins

1994
Benzodiazepine treatment causes uncoupling of recombinant GABAA receptors expressed in stably transfected cells.
    Journal of neurochemistry, 1994, Volume: 63, Issue:6

    Topics: Allosteric Site; Animals; Benzodiazepines; Cattle; Cell Line; Clonazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Mice; Receptors, GABA; Recombinant Proteins; Transfection

1994
Participation of mitochondrial diazepam binding inhibitor receptors in the anticonflict, antineophobic and anticonvulsant action of 2-aryl-3-indoleacetamide and imidazopyridine derivatives.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: Aggression; Allosteric Regulation; Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Clonazepam; Desoxycorticosterone; Flumazenil; Imidazoles; Indoleacetic Acids; Isoniazid; Isoquinolines; Mitochondria; Phobic Disorders; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Seizures; Zolpidem

1993
In vitro inhibition of cellular immune responses by benzodiazepines and PK 11195. Effects on mitogen- and alloantigen-driven lymphocyte proliferation and on IL-1, IL-2 synthesis and IL-2 receptor expression.
    Immunopharmacology and immunotoxicology, 1993, Volume: 15, Issue:5

    Topics: Animals; B-Lymphocytes; Benzodiazepines; Benzodiazepinones; Clonazepam; Diazepam; Female; Flumazenil; Immunity, Cellular; In Vitro Techniques; Interleukin-1; Interleukin-2; Isoquinolines; Lymphocyte Activation; Male; Mice; Mice, Inbred A; Mice, Inbred C57BL; Neuroimmunomodulation; Receptors, GABA-A; T-Lymphocytes

1993
Anticonvulsant profile of the imidazoquinazolines NNC 14-0185 and NNC 14-0189 in rats and mice.
    European journal of pharmacology, 1996, Jul-11, Volume: 308, Issue:1

    Topics: Acoustic Stimulation; Amygdala; Animals; Anticonvulsants; Bicuculline; Carbolines; Clonazepam; Diazepam; Electroshock; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Kindling, Neurologic; Male; Mice; Mice, Inbred DBA; Mice, Inbred Strains; Pentylenetetrazole; Quinazolines; Rats; Rats, Wistar; Seizures

1996
Prevention of ACTH- and adrenalectomy-induced muricidal behavior: by benzodiazepinic ligands.
    Peptides, 1997, Volume: 18, Issue:2

    Topics: Adrenalectomy; Adrenocorticotropic Hormone; Aggression; Animals; Benzodiazepinones; Clonazepam; Flumazenil; GABA Modulators; Isoquinolines; Male; Mice; Muscimol; Rats; Rats, Wistar; Receptors, GABA-A; Time Factors

1997
Electrophysiological evidence for agonist properties of flumazenil, a benzodiazepine receptor antagonist, in rat hippocampus slices.
    Journal of the neurological sciences, 1997, Volume: 149, Issue:2

    Topics: Animals; Clonazepam; Electrophysiology; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hippocampus; Male; Organ Culture Techniques; Rats; Rats, Wistar

1997
Plasma and CSF benzodiazepine receptor ligand concentrations in cirrhotic patients with hepatic encephalopathy: relationship to severity of encephalopathy and to pharmaceutical benzodiazepine intake.
    Metabolic brain disease, 1998, Volume: 13, Issue:3

    Topics: Animals; Benzodiazepines; Binding, Competitive; Cell Fractionation; Cerebellum; Chronic Disease; Clonazepam; Diazepam; Flumazenil; GABA Modulators; Hepatic Encephalopathy; Humans; Isoquinolines; Liver Cirrhosis; Oxazepam; Radioligand Assay; Rats; Receptors, GABA-A; Tritium

1998
Inhibitory regulation of amylase release in rat parotid acinar cells by benzodiazepine receptors.
    European journal of pharmacology, 1998, Oct-23, Volume: 359, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amylases; Animals; Atropine; Benzodiazepinones; Carbachol; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoproterenol; Male; Muscarinic Agonists; Muscarinic Antagonists; Parotid Gland; Propranolol; Rats; Rats, Wistar; Receptors, GABA-A

1998
Effect of benzodiazepines and neurosteroids on ammonia-induced swelling in cultured astrocytes.
    Journal of neuroscience research, 1998, Dec-01, Volume: 54, Issue:5

    Topics: Ammonia; Astrocytes; Atrial Natriuretic Factor; Benzodiazepines; Benzodiazepinones; Brain Edema; Cell Size; Clonazepam; Dehydroepiandrosterone Sulfate; Desoxycorticosterone; Diazepam; Diazepam Binding Inhibitor; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Isoquinolines; Nerve Tissue Proteins; Neuropeptides; Peptide Fragments; Pregnanolone; Pregnenolone; Protoporphyrins; Receptors, GABA-A; Steroids; Up-Regulation

1998
Cardiac effects of benzodiazepine receptor agonists and antagonists in the isolated rat heart: a comparative study.
    Life sciences, 1998, Volume: 63, Issue:16

    Topics: Animals; Benzodiazepines; Cardiac Output; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Heart; In Vitro Techniques; Isoquinolines; Myocardial Contraction; Perfusion; Pyridines; Rats; Receptors, GABA-A; Zolpidem

1998
The role of gamma-aminobutyric acid (GABA)-benzodiazepine neurotransmission in an animal model of methamphetamine-induced psychosis.
    [Hokkaido igaku zasshi] The Hokkaido journal of medical science, 1999, Volume: 74, Issue:2

    Topics: Animals; Behavior, Animal; Central Nervous System Stimulants; Clonazepam; Depression, Chemical; Disease Models, Animal; Flumazenil; GABA Modulators; Humans; Male; Methamphetamine; Psychoses, Substance-Induced; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Transmission

1999
Abecarnil enhances recovery from diazepam tolerance.
    Neuropharmacology, 1999, Volume: 38, Issue:9

    Topics: Animals; Anticonvulsants; Benzodiazepines; Bicuculline; Carbolines; Cell Membrane; Cerebral Cortex; Clonazepam; Diazepam; Drug Interactions; Drug Tolerance; Flumazenil; Imidazoles; Ligands; Male; Mice; Receptors, GABA-A; Seizures; Tritium

1999
The role of benzodiazepine receptors in the acquisition and expression of behavioral sensitization to methamphetamine.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 65, Issue:4

    Topics: Animals; Behavior, Animal; Central Nervous System Stimulants; Clonazepam; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; Male; Methamphetamine; Motor Activity; Rats; Rats, Wistar; Receptors, GABA-A

2000
Topiramate modulates GABA-evoked currents in murine cortical neurons by a nonbenzodiazepine mechanism.
    Epilepsia, 2000, Volume: 41, Issue:S1

    Topics: Action Potentials; Animals; Anticonvulsants; Cells, Cultured; Cerebral Cortex; Clonazepam; Evoked Potentials; Flumazenil; Fructose; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Mice; Neurons; Patch-Clamp Techniques; Pentylenetetrazole; Receptors, GABA; Seizures; Topiramate

2000
Evaluation of native GABA(A) receptors containing an alpha 5 subunit.
    European journal of pharmacology, 2001, Feb-09, Volume: 413, Issue:1

    Topics: Alkynes; Animals; Anti-Anxiety Agents; Anticonvulsants; Autoradiography; Benzodiazepines; Cerebellum; Clobazam; Clonazepam; Diazepam; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Hippocampus; Imidazoles; Male; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

2001
Behavioral effects of agents active at the gamma-aminobutyric acid receptor complex in the staircase paradigm.
    Brain research, 2001, May-18, Volume: 901, Issue:1-2

    Topics: Acetates; Adjuvants, Immunologic; Amines; Animals; Anti-Anxiety Agents; Anxiety; Azabicyclo Compounds; Behavior, Animal; Brain; Clonazepam; Cyclohexanecarboxylic Acids; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; GABA Modulators; Gabapentin; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Mice; Mice, Inbred ICR; Motor Activity; Neurons; Piperazines; Receptors, GABA-A

2001
2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective peripheral benzodiazepine receptor ligands.
    Bioorganic & medicinal chemistry, 2001, Volume: 9, Issue:10

    Topics: Acetamides; Animals; Benzodiazepinones; Binding Sites; Cerebral Cortex; Clonazepam; Flumazenil; Glioma; Intracellular Membranes; Isoquinolines; Kidney; Ligands; Magnetic Resonance Spectroscopy; Molecular Structure; Pyrazoles; Pyrimidines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Thermodynamics; Tumor Cells, Cultured

2001
Benzodiazepines protect against ethanol-induced gastric mucosal damage in vitro.
    Fundamental & clinical pharmacology, 2001, Volume: 15, Issue:4

    Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Central Nervous System Depressants; Clonazepam; Ethanol; Flumazenil; GABA Modulators; Gastric Mucosa; In Vitro Techniques; Male; Rats; Rats, Wistar; Stomach Ulcer

2001
Reversal of benzodiazepine-induced renal vasculature relaxation with flumazenil.
    European journal of pharmacology, 2002, Aug-02, Volume: 449, Issue:1-2

    Topics: Animals; Clonazepam; Diazepam; Flumazenil; GABA Modulators; Male; Muscle Relaxants, Central; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Rats; Rats, Wistar; Renal Circulation; Vasoconstrictor Agents

2002
The heterogeneity of central benzodiazepine receptor subtypes in the human hippocampal formation, frontal cortex and cerebellum using [3H]flumazenil and zolpidem.
    Brain research. Molecular brain research, 2002, Aug-15, Volume: 104, Issue:2

    Topics: Cerebellum; Clonazepam; Flumazenil; Frontal Lobe; GABA Agents; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; Humans; Male; Middle Aged; Neurons; Protein Binding; Pyridines; Radioligand Assay; Receptors, GABA-A; Synaptic Transmission; Tritium; Zolpidem

2002
Changes in hippocampal GABAA receptor subunit composition in bipolar 1 disorder.
    Brain research. Molecular brain research, 2005, Aug-18, Volume: 138, Issue:2

    Topics: Adult; Aged; Binding, Competitive; Bipolar Disorder; Brain Chemistry; Clonazepam; Female; Flumazenil; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; Humans; Male; Middle Aged; Muscimol; Protein Subunits; Pyridines; Radioligand Assay; Receptors, GABA-A; Schizophrenia; Zolpidem

2005
Benzodiazepine-associated atrioventricular block.
    American journal of therapeutics, 2012, Volume: 19, Issue:1

    Topics: Acetaminophen; Alprazolam; Anti-Anxiety Agents; Anticonvulsants; Antidotes; Atrioventricular Block; Child, Preschool; Clonazepam; Drug Combinations; Electrocardiography; Flumazenil; Humans; Hydrocodone; Male; Risperidone; Young Adult

2012
Serial monitoring of sedation scores in benzodiazepine overdose.
    The American journal of emergency medicine, 2014, Volume: 32, Issue:11

    Topics: Aged; Anticonvulsants; Antidotes; Clonazepam; Drug Overdose; Female; Flumazenil; Humans; Monitoring, Physiologic; Suicide, Attempted

2014
Acute encephalopathy in a 2-year-old pot-bellied pig following accidental intoxication with clonazepam.
    Journal of veterinary emergency and critical care (San Antonio, Tex. : 2001), 2017, Volume: 27, Issue:3

    Topics: Acute Febrile Encephalopathy; Animals; Antidotes; Clonazepam; Diagnosis, Differential; Drug-Related Side Effects and Adverse Reactions; Emergencies; Female; Flumazenil; Infusions, Intravenous; Swine; Swine Diseases; Swine, Miniature

2017
High-Dose Benzodiazepines Positively Modulate GABA
    International journal of molecular sciences, 2021, Dec-21, Volume: 23, Issue:1

    Topics: Animals; Animals, Outbred Strains; Benzodiazepines; Clonazepam; Diazepam; Female; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Midazolam; Receptors, GABA-A; Xenopus laevis

2021