flumazenil and cl 218872

flumazenil has been researched along with cl 218872 in 46 studies

Research

Studies (46)

TimeframeStudies, this research(%)All Research%
pre-199024 (52.17)18.7374
1990's17 (36.96)18.2507
2000's4 (8.70)29.6817
2010's1 (2.17)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barone, D; Gallico, L; Luzzani, F; Tarzia, G; Toja, E1
Lüddens, H; Wieland, HA1
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Clayton, T; Cook, JM; Cromer, BA; Ma, C; Majumder, S; Namjoshi, OA; Petrou, S; Platt, DM; Roth, BL; VanLinn, ML; Yin, W1
Arbilla, S; Benavides, J; Durand, A; Peny, B; Scatton, B1
McNamara, RK; Skelton, RW1
Borsini, F; Gragnani, L; Lecci, A; Meli, A; Volterra, G1
Franklin, SR; Tang, AH1
De Luca, C; De Medici, D; Massotti, M1
Lüddens, H; Pritchett, DB; Seeburg, PH1
Evans, SM; Johanson, CE1
Benavides, J; Dubois, A; Morel, E; Peny, B; Perrault, G; Scatton, B; Zivkovic, B1
Arbilla, S; Langer, SZ; Lista, A1
De Medici, D; Gatta, F; Longo, VG; Massotti, M1
File, SE; Pellow, S; Wilks, L1
Chan, CY; Farb, DH1
Ator, NA; Griffiths, RR1
File, SE; Pellow, S1
Spealman, RD; Wettstein, JG1
de la Garza, R; Evans, S; Johanson, CE1
Dewey, WL; Glennon, RA; Young, R1
Kuriyama, K; Taguchi, J1
Spealman, RD1
Cole, R; De Vellis, J; Noble, EP; Syapin, PJ1
Meiners, BA; Salama, AI1
De Vry, J; Slangen, JL1
Macdonald, RL; Skerritt, JH1
Villiger, JW1
Morin, AM1
Goldberg, ME; Malick, JB; Patel, JB; Salama, AI1
Vellucci, SV; Webster, RA1
Garrett, KM; Melchior, CL; Tabakoff, B1
Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Vonvoigtlander, PF1
Corcoran, ME; McNamara, RK1
Pritchett, DB; Williamson, RE1
Bannwarth, W; Benke, D; Fritschy, JM; Mohler, H; Trzeciak, A1
Berman, JA; Pritchett, DB; Roberts, JL1
Benavides, J; Peny, B; Ruano, D; Scatton, B; Vitorica, J1
Hadingham, KL; Palmer, KJ; Thompson, SA; Wafford, KA; Whiting, PJ1
Aguayo, LG; Cisternas, C; Pancetti, FC; Tapia, JC1
Araujo, F; Benavides, J; Ruano, D; Schoemaker, H; Tan, S; Vitorica, J1
Atack, JR; Emms, F; McKernan, RM; Smith, AJ1
Araujo, F; Ruano, D; Vitorica, J1
Bromidge, FA; Casula, MA; Hadingham, KL; Martin, K; Maubach, K; Pillai, GV; Seabrook, GR; Whiting, PJ; Wingrove, PB1
Safo, P; Thompson, SA; Wafford, KA; Wheat, L; Whiting, PJ; Wingrove, PB1

Reviews

1 review(s) available for flumazenil and cl 218872

ArticleYear
Novel non-benzodiazepine anxiolytics.
    Neuropharmacology, 1983, Volume: 22, Issue:12B

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Benzodiazepinones; Conflict, Psychological; Flumazenil; Flunitrazepam; Hypnotics and Sedatives; Mice; Piperazines; Pyrazoles; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983

Other Studies

45 other study(ies) available for flumazenil and cl 218872

ArticleYear
Benzodiazepine receptor binding and anticonflict activity in a series of 3,6-disubstituted pyridazino[4,3-c]isoquinolines devoid of anticonvulsant properties.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:9

    Topics: Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Conflict, Psychological; Diazepam; Isoquinolines; Male; Mice; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Structure-Activity Relationship

1985
Four amino acid exchanges convert a diazepam-insensitive, inverse agonist-preferring GABAA receptor into a diazepam-preferring GABAA receptor.
    Journal of medicinal chemistry, 1994, Dec-23, Volume: 37, Issue:26

    Topics: Amino Acid Sequence; Azides; Base Sequence; Benzodiazepines; Binding Sites; Diazepam; GABA Agonists; Humans; Molecular Sequence Data; Mutation; Receptors, GABA-A; Structure-Activity Relationship

1994
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Design, synthesis, and subtype selectivity of 3,6-disubstituted β-carbolines at Bz/GABA(A)ergic receptors. SAR and studies directed toward agents for treatment of alcohol abuse.
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Alcoholism; Animals; Benzodiazepines; Binding Sites; Carbolines; Cell Line; Computer Simulation; GABA-A Receptor Antagonists; Humans; Protein Subunits; Rats; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship

2010
Comparative in vivo and in vitro regional selectivity of central omega (benzodiazepine) site ligands in inhibiting [3H]flumazenil binding in the rat central nervous system.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Brain Chemistry; Cell Membrane; Central Nervous System; Flumazenil; Hypnotics and Sedatives; Pyridazines; Pyridines; Rats; Receptors, GABA-A; Triazolam; Zolpidem

1992
Like diazepam, CL 218,872, a selective ligand for the benzodiazepine omega 1 receptor subtype, impairs place learning in the Morris water maze.
    Psychopharmacology, 1992, Volume: 107, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Flumazenil; Learning; Male; Memory; Motor Activity; Pyridazines; Rats; Receptors, GABA-A

1992
Effect of psychotomimetics and some putative anxiolytics on stress-induced hyperthermia.
    Journal of neural transmission. General section, 1991, Volume: 83, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Body Temperature; Dextroamphetamine; Dizocilpine Maleate; Fever; Flumazenil; Male; Mice; Phencyclidine; Pyrazoles; Pyridazines; Quinolines; Receptors, GABA-A; Receptors, Serotonin; Single-Blind Method; Stress, Physiological

1991
The discriminative stimulus effects of diazepam in rats at two training doses.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: Alprazolam; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Male; Morphine; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Triazolam

1991
Relative efficacies of benzodiazepine receptor agonists in affecting red nucleus electrical activity in rabbits.
    Psychopharmacology, 1990, Volume: 102, Issue:4

    Topics: Animals; Bicuculline; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Imidazoles; Isoquinolines; Male; Pentylenetetrazole; Pyridazines; Pyridines; Rabbits; Receptors, GABA-A; Red Nucleus; Zolpidem

1990
Type I and type II GABAA-benzodiazepine receptors produced in transfected cells.
    Science (New York, N.Y.), 1989, Sep-22, Volume: 245, Issue:4924

    Topics: Cell Line; Diazepam; Flumazenil; Flunitrazepam; Humans; Molecular Weight; Pyridazines; Receptors, GABA-A; Recombinant Proteins; Transfection

1989
Discriminative stimulus properties of midazolam in the pigeon.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Buspirone; Columbidae; Discrimination Learning; Dose-Response Relationship, Drug; Flumazenil; Midazolam; Pentobarbital; Pyridazines

1989
In vivo interaction of zolpidem with central benzodiazepine (BZD) binding sites (as labeled by [3H]Ro 15-1788) in the mouse brain. Preferential affinity of zolpidem for the omega 1 (BZD1) subtype.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:3

    Topics: Animals; Autoradiography; Binding Sites; Brain; Flumazenil; Flunitrazepam; Hypnotics and Sedatives; In Vitro Techniques; Male; Mice; Pyridazines; Pyridines; Receptors, GABA-A; Zolpidem

1988
Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.
    Journal of neurochemistry, 1988, Volume: 51, Issue:5

    Topics: Animals; Benzodiazepines; Carbolines; Cerebral Cortex; Diazepam; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Monoamine Oxidase Inhibitors; Pargyline; Pyrazoles; Pyridazines; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin

1988
Effects of drugs on the electrical activity of the red nucleus in the rabbit. Activation of benzodiazepine and barbiturate receptors.
    Annali dell'Istituto superiore di sanita, 1988, Volume: 24, Issue:3

    Topics: Animals; Bicuculline; Carbolines; Diazepam; Drug Interactions; Electroencephalography; Flumazenil; Muscle Relaxation; Pentobarbital; Pyridazines; Rabbits; Receptors, GABA-A; Receptors, Neurotransmitter; Red Nucleus

1988
The sedative effects of CL 218,872, like those of chlordiazepoxide, are reversed by benzodiazepine antagonists.
    Psychopharmacology, 1985, Volume: 85, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepinones; Chlordiazepoxide; Convulsants; Flumazenil; Hypnotics and Sedatives; Male; Mice; Motor Activity; Pyrazoles; Pyridazines

1985
Modulation of neurotransmitter action: control of the gamma-aminobutyric acid response through the benzodiazepine receptor.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1985, Volume: 5, Issue:9

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Chick Embryo; Electric Conductivity; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Neurotransmitter Agents; Picrotoxin; Pyridazines; Receptors, GABA-A

1985
Discriminative stimulus effects of atypical anxiolytics in baboons and rats.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepinones; Buspirone; Discrimination Learning; Flumazenil; Isoxazoles; Lorazepam; Male; Papio; Piperazines; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
Anxiolytic and anxiogenic drug effects on exploratory activity in an elevated plus-maze: a novel test of anxiety in the rat.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Convulsants; Exploratory Behavior; Flumazenil; Male; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats

1986
Behavioral effects of zopiclone, CL 218,872 and diazepam in squirrel monkeys: antagonism by Ro 15-1788 and CGS 8216.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepinones; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Piperazines; Pyrazoles; Pyridazines; Saimiri

1986
Discriminative stimulus properties of oxazepam in the pigeon.
    Life sciences, 1987, Jan-05, Volume: 40, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Columbidae; Discrimination Learning; Flumazenil; Oxazepam; Pentobarbital; Pyridazines

1987
Effects of pyrazolopyridines and a triazolopyridazine on the pentobarbital discriminative stimulus.
    Psychopharmacology, 1987, Volume: 93, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Discrimination Learning; Discrimination, Psychological; Flumazenil; Generalization, Stimulus; Male; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains

1987
Functional coupling of gamma-aminobutyric acid (GABA)A and benzodiazepine type II receptors: analysis using purified GABA/benzodiazepine receptor complex from bovine cerebral cortex.
    Neuropharmacology, 1987, Volume: 26, Issue:12

    Topics: Animals; Antipsychotic Agents; Bicuculline; Cattle; Cerebral Cortex; Flumazenil; Flunitrazepam; In Vitro Techniques; Kinetics; Muscimol; Pyridazines; Receptors, GABA-A

1987
Discriminative-stimulus effects of midazolam in squirrel monkeys: comparison with other drugs and antagonism by Ro 15-1788.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Azabicyclo Compounds; Barbital; Benzodiazepines; Benzodiazepinones; Buspirone; Caffeine; Chlordiazepoxide; Cinanserin; Clozapine; Conditioning, Operant; Cyproheptadine; Diazepam; Diphenhydramine; Discrimination Learning; Electroshock; Flumazenil; Male; Midazolam; Muscimol; Nordazepam; Pentobarbital; Piperazines; Pyridazines; Pyrimidines; Saimiri; Tripelennamine

1985
Benzodiazepine binding characteristics of embryonic rat brain neurons grown in culture.
    Journal of neurochemistry, 1985, Volume: 45, Issue:6

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Cells, Cultured; Clonazepam; Diazepam; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Neurons; Pyridazines; Rats; Receptors, GABA-A

1985
Enhancement of GABA binding by the benzodiazepine partial agonist CGS9896.
    European journal of pharmacology, 1985, Dec-10, Volume: 119, Issue:1-2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Calcium Chloride; Diazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Magnesium; Pyrazoles; Pyridazines; Rats; Receptors, GABA-A

1985
The Ro 15-1788 cue: evidence for benzodiazepine agonist and inverse agonist properties.
    European journal of pharmacology, 1985, Dec-17, Volume: 119, Issue:3

    Topics: Animals; Anticonvulsants; Barbiturates; Benzodiazepines; Benzodiazepinones; Convulsants; Discrimination, Psychological; Flumazenil; Male; Pyridazines; Rats; Rats, Inbred Strains

1985
Benzodiazepine receptor ligand actions on GABA responses. Benzodiazepines, CL 218872, zopiclone.
    European journal of pharmacology, 1984, May-18, Volume: 101, Issue:1-2

    Topics: Animals; Azabicyclo Compounds; Benzodiazepines; Benzodiazepinones; Cells, Cultured; Drug Interactions; Flumazenil; gamma-Aminobutyric Acid; Ligands; Mice; Neurons; Piperazines; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord

1984
CL 218,872 binding to benzodiazepine receptors in rat spinal cord: modulation by gamma-aminobutyric acid and evidence for receptor heterogeneity.
    Journal of neurochemistry, 1984, Volume: 43, Issue:4

    Topics: Animals; Benzodiazepinones; Cerebral Cortex; Flumazenil; gamma-Aminobutyric Acid; Male; Muscimol; Pyridazines; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord

1984
Beta-carboline kindling of the benzodiazepine receptor.
    Brain research, 1984, Oct-29, Volume: 321, Issue:1

    Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Flumazenil; Indoles; Kindling, Neurologic; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
Is Ro15-1788 a partial agonist at benzodiazepine receptors?
    European journal of pharmacology, 1983, Jun-03, Volume: 90, Issue:2-3

    Topics: Animals; Benzodiazepinones; Bicuculline; Convulsants; Diazepam; Flumazenil; Male; Mice; Mice, Inbred C3H; Phenobarbital; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A

1983
A benzodiazepine antagonist action of CL 218,872.
    Life sciences, 1984, May-28, Volume: 34, Issue:22

    Topics: Animals; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Convulsants; Diazepam; Flumazenil; Male; Mice; Mice, Inbred C57BL; Pyridazines; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1984
Potentiation of gamma-aminobutyric acid-induced chloride currents by various benzodiazepine site agonists with the alpha 1 gamma 2, beta 2 gamma 2 and alpha 1 beta 2 gamma 2 subtypes of cloned gamma-aminobutyric acid type A receptors.
    Molecular pharmacology, 1993, Volume: 44, Issue:4

    Topics: Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Binding Sites; Cells, Cultured; Chloride Channels; Cloning, Molecular; Drug Synergism; Flumazenil; gamma-Aminobutyric Acid; Humans; Hypnotics and Sedatives; Imidazoles; Kidney; Kinetics; Membrane Potentials; Piperazines; Pyridazines; Pyridines; Receptors, GABA-A; Triazolam

1993
CL 218,872 a triazolopyridazine with a selective affinity for the benzodiazepine BZ1 receptor subtype, retards the development and expression of amygdaloid-kindled seizures: effects of flumazenil.
    Epilepsy research, 1993, Volume: 16, Issue:1

    Topics: Amygdala; Animals; Anti-Anxiety Agents; Drug Interactions; Flumazenil; Kindling, Neurologic; Male; Pyridazines; Rats; Receptors, GABA-A; Seizures

1993
Levels of benzodiazepine receptor subtypes and GABAA receptor alpha-subunit mRNA do not correlate during development.
    Journal of neurochemistry, 1994, Volume: 63, Issue:2

    Topics: Aging; Animals; Animals, Newborn; Anti-Anxiety Agents; Binding, Competitive; Cerebellum; Flumazenil; Hippocampus; Kinetics; Macromolecular Substances; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger

1994
Distribution, prevalence, and drug binding profile of gamma-aminobutyric acid type A receptor subtypes differing in the beta-subunit variant.
    The Journal of biological chemistry, 1994, Oct-28, Volume: 269, Issue:43

    Topics: Animals; Brain Chemistry; Carbolines; Flumazenil; Flunitrazepam; Genetic Variation; Immunohistochemistry; Male; Microscopy, Confocal; Molecular Weight; Precipitin Tests; Protein Conformation; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tissue Distribution; Zolpidem

1994
Molecular and pharmacological characterization of GABAA receptors in the rat pituitary.
    Journal of neurochemistry, 1994, Volume: 63, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; DNA; Flumazenil; Male; Muscimol; Pituitary Gland; Polymerase Chain Reaction; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; RNA, Messenger; Tritium

1994
Comparative autoradiographic distribution of central omega (benzodiazepine) modulatory site subtypes with high, intermediate and low affinity for zolpidem and alpidem.
    Brain research, 1993, Feb-26, Volume: 604, Issue:1-2

    Topics: Animals; Animals, Newborn; Anti-Anxiety Agents; Autoradiography; Binding, Competitive; Brain; Flumazenil; Hypnotics and Sedatives; Imidazoles; Kinetics; Male; Organ Specificity; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Spinal Cord; Tritium; Zolpidem

1993
Expression and pharmacology of human GABAA receptors containing gamma 3 subunits.
    European journal of pharmacology, 1995, Nov-30, Volume: 291, Issue:3

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Base Sequence; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Molecular Sequence Data; Pyrazoles; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Proteins; Sequence Homology, Amino Acid; Triazolam; Xenopus; Zolpidem

1995
Effects of benzodiazepine receptor ligands on isolated rat superior cervical ganglia neurons.
    Pharmacology, 1996, Volume: 52, Issue:6

    Topics: Age Factors; Animals; Animals, Newborn; Anti-Anxiety Agents; Diazepam; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Ligands; Neurons; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Superior Cervical Ganglion

1996
Molecular and pharmacological characterization of native cortical gamma-aminobutyric acidA receptors containing both alpha1 and alpha3 subunits.
    The Journal of biological chemistry, 1996, Nov-01, Volume: 271, Issue:44

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Antibodies; Binding Sites; Cattle; Cell Membrane; Cerebral Cortex; Chromatography, Affinity; Flumazenil; Hypnotics and Sedatives; Immunoblotting; Kinetics; Macromolecular Substances; Models, Structural; Peptide Fragments; Pyridazines; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Zolpidem

1996
Regional differences in the inhibition of mouse in vivo [3H]Ro 15-1788 binding reflect selectivity for alpha 1 versus alpha 2 and alpha 3 subunit-containing GABAA receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1999, Volume: 20, Issue:3

    Topics: Animals; Benzodiazepines; Binding Sites; Cerebellum; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; In Vitro Techniques; Ligands; Male; Mice; Pyridazines; Pyridines; Receptors, GABA-A; Spinal Cord; Time Factors; Tritium; Zolpidem

1999
Native gamma-aminobutyric acid type A receptors from rat hippocampus, containing both alpha 1 and alpha 5 subunits, exhibit a single benzodiazepine binding site with alpha 5 pharmacological properties.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding Sites; Chromatography, Affinity; Flumazenil; GABA Modulators; Hippocampus; Hypnotics and Sedatives; Macromolecular Substances; Precipitin Tests; Pyridazines; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Tritium; Zolpidem

1999
Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; DNA, Complementary; Female; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Humans; Imidazoles; Isoleucine; Ligands; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Protein Binding; Protein Structure, Tertiary; Protein Subunits; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Fusion Proteins; Sequence Alignment; Structure-Activity Relationship; Threonine; Transfection; Xenopus laevis; Zolpidem

2001
Mechanism of alpha-subunit selectivity of benzodiazepine pharmacology at gamma-aminobutyric acid type A receptors.
    European journal of pharmacology, 2002, Feb-15, Volume: 437, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Cell Line; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Mutation; Oocytes; Protein Subunits; Pyridazines; Pyridines; Radioligand Assay; Receptors, GABA-A; Tritium; Xenopus laevis; Zolpidem

2002