flumazenil and chlorine

flumazenil has been researched along with chlorine in 64 studies

Research

Studies (64)

TimeframeStudies, this research(%)All Research%
pre-199031 (48.44)18.7374
1990's24 (37.50)18.2507
2000's5 (7.81)29.6817
2010's2 (3.13)24.3611
2020's2 (3.13)2.80

Authors

AuthorsStudies
Facklam, M; Haefely, WE; Schoch, P1
Hood, KE; Miczek, KA; Miller, LG; Weerts, EM1
Buck, KJ; Harris, RA; Heim, H1
Galpern, WR; Greenblatt, DJ; Lumpkin, M; Miller, LG; Shader, RI1
Blakeman, DP; Im, WB1
Baker, BL; Jones, EA; Morrow, AL; Paul, SM; Vergalla, J1
Buck, KJ; Harris, RA1
Greenblatt, DJ; Heller, J; Lumpkin, M; Miller, LG; Shader, RI; Weill, CL1
Costa, E; Guidotti, A1
Hill, JL; Insel, TR; Mayor, RB1
Obata, T; Yamamura, HI1
Havoundjian, H; Skolnick, P; Trullas, R1
Greenblatt, DJ; Miller, LG; Roy, RB; Shader, RI; Summer, WR1
Becker, HC1
Haefely, W2
Costa, E; Mienville, JM; Vicini, S1
Haefely, WE2
McIntyre, TD; Skolnick, P; Trullas, R1
Aosaki, T; Kanai, Y; Manabe, S; Wada, O1
Greenblatt, DJ; Lopez, F; Miller, LG; Roy, RB; Wecker, L1
Baur, R; Peter, AB; Sigel, E; Yao, Y1
Gaver, A; Greenblatt, DJ; Lopez, F; Miller, LG; Roy, RB; Shader, RI1
Mehta, AK; Ticku, MK2
Crawley, JN; Deutsch, SI; Drugan, RC; Morrow, AL; Paul, SM; Weizman, A; Weizman, R1
Miller, LG; Roy, RB; Weill, CL1
Ikeda, M; Knapp, RJ; Malatynska, E; Yamamura, HI1
Lucki, I; Rowan, GA1
Bechtel, WD; Ikeda, M; Malatynska, E; Weber, KH; Yamamura, HI1
Cooper, SJ; Estall, LB1
Dan'ura, T; Ishibashi, S; Kurokawa, T; Yamashita, A; Yanagiuchi, H1
Concas, A; Morelli, M; Obata, T; Serra, M; Yamamura, HI1
Kempner, ES; Paul, SM; Schwartz, RD; Skolnick, P; Thomas, JW1
Haefely, W; Möhler, H; Richards, JG; Schoch, P1
Crawley, JN; Glowa, JR; Paul, SM; Schwartz, RD; Skolnick, P; Suzdak, PD1
Chiu, TH; Rosenberg, HC; Yu, O1
Corda, MG; Costa, E; Guidotti, A1
Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Jacobsen, EJ; Pregenzer, JF1
Biggio, G; Concas, A; Cuccheddu, T; Maciocco, E; Santoro, G; Serra, M1
Hu, XJ; Ticku, MK2
Harris, RA; Klein, RL; McQuilkin, SJ; Sanna, E; Whiting, PJ1
Carter, DB; Gammill, RB; Hamilton, BJ; Im, HK; Im, WB; Judge, TM; Pregenzer, JF1
Harris, RA; McQuilkin, SJ; Mihic, SJ; Whatley, VJ1
Hara, M; Ikemoto, Y; Kai, Y1
Davies, MF; Loew, GH; Maguire, PA1
Alastra, AJ; Cohen, C; Goldberg, SR; Marley, RJ; Sannerud, CA; Serdikoff, SL1
Dalton, CR; Dudley, MW; Kane, JM; Kehne, JH; Ketteler, HJ; McCloskey, TC; Miller, FP; Ogden, AM; Senyah, Y; Staeger, MA1
Deutsch, SI; Hitri, A; Lukacs, LG; Park, CH1
Mehta, AK; Shank, RP1
Hatta, S; Saito, T; Takahata, N; Toki, S1
Matsumoto, K; Ojima, K; Watanabe, H2
Betti, L; Bistocchi, M; Giannaccini, G; Gori, M; Lucacchini, A1
Biggio, F; Biggio, G; Busonero, F; Cagetti, E; Carta, M; Desole, MS; Follesa, P; Maciocco, E; Manca, A; Mancuso, L; Massa, F; Sanna, E1
Firestone, LL; Gyulai, FE; Mintun, MA1
Kawaguchi, M; Kujirai, M; Sawaki, K1
Furtmueller, B; Furtmueller, R; Huck, S; Marder, M; Paladini, AC; Ramerstorfer, J; Sieghart, W; Wasowski, C1
Alcaro, S; Anzini, M; Betti, L; Biggio, G; Braile, C; Cappelli, A; Daniele, S; Di Cesare Mannelli, L; Ghelardini, C; Giannaccini, G; Giorgi, G; Limongelli, V; Lucacchini, A; Marinelli, L; Martini, C; Mascia, MP; Novellino, E; Ortuso, F; Valenti, S; Vomero, S1
Absalom, NL; Chebib, M; Chua, HC; Hanrahan, JR; Viswas, R1
Amari, M; Bonato, F; Brioschi, FA; Di Cesare, F; Giordano, A; Magnone, W; Moretti, P; Pecile, A; Rabbogliatti, V; Ravasio, G1
Chai, X; Chen, S; Gao, X; Huang, L; Jiao, S; Li, J; Ma, X; Tu, P; Wuken, S1

Reviews

5 review(s) available for flumazenil and chlorine

ArticleYear
Endogenous ligands for benzodiazepine recognition sites.
    Biochemical pharmacology, 1985, Oct-01, Volume: 34, Issue:19

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Brain; Caffeine; Carrier Proteins; Chlorides; Conflict, Psychological; Diazepam Binding Inhibitor; Flumazenil; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Humans; Hypoxanthine; Hypoxanthines; Inosine; Ion Channels; Membrane Proteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neuroglia; Neurons; Niacinamide; Organic Anion Transporters; Peptides; Phosphorylation; Protein Conformation; Protein Precursors; Receptors, GABA-A; Synaptic Membranes; Tissue Distribution; Trypsin

1985
Benzodiazepines.
    International anesthesiology clinics, 1988,Winter, Volume: 26, Issue:4

    Topics: Animals; Benzodiazepines; Chlorides; Flumazenil; Humans; Ion Channels; Receptors, GABA-A

1988
Behavioural pharmacology of food, water and salt intake in relation to drug actions at benzodiazepine receptors.
    Neuroscience and biobehavioral reviews, 1985,Spring, Volume: 9, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Appetite; Appetite Depressants; Benzodiazepines; Benzodiazepinones; Carbolines; Chlordiazepoxide; Chlorides; Choice Behavior; Diazepam; Drinking Behavior; Feeding Behavior; Flumazenil; Food Deprivation; Food Preferences; gamma-Aminobutyric Acid; Ion Channels; Midazolam; Picrotoxin; Punishment; Pyrazoles; Receptors, GABA-A; Satiation; Sodium Chloride; Species Specificity

1985
Benzodiazepine receptors resolved.
    Experientia, 1986, Feb-15, Volume: 42, Issue:2

    Topics: Animals; Antibodies, Monoclonal; Autoradiography; Benzodiazepines; Benzodiazepinones; Bicuculline; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Chlorides; Clonazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Histocytochemistry; Humans; Immunologic Techniques; Ionophores; Muscimol; Neurons; Radioisotopes; Radioligand Assay; Receptors, GABA-A; Spinal Cord; Synapses; Tissue Distribution

1986
On a brain polypeptide functioning as a putative effector for the recognition sites of benzodiazepine and beta-carboline derivatives.
    Neuropharmacology, 1983, Volume: 22, Issue:12B

    Topics: Animals; Benzodiazepinones; Brain Chemistry; Carbolines; Carrier Proteins; Chlorides; Flumazenil; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Humans; Ionophores; Ligands; Membrane Proteins; Membrane Transport Proteins; Nerve Tissue Proteins; Organic Anion Transporters; Peptides; Receptors, Cell Surface; Receptors, GABA-A

1983

Other Studies

59 other study(ies) available for flumazenil and chlorine

ArticleYear
Relationship between benzodiazepine receptor occupancy and potentiation of gamma-aminobutyric acid-stimulated chloride flux in vitro of four ligands of differing intrinsic efficacies.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Animals; Benzodiazepinones; Cell Membrane; Cerebral Cortex; Chlorides; Diazepam; Drug Synergism; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Rats; Receptors, GABA-A; Triazolam

1992
Increased GABAA-dependent chloride uptake in mice selectively bred for low aggressive behavior.
    Psychopharmacology, 1992, Volume: 108, Issue:1-2

    Topics: Aggression; Animals; Chlorides; Flumazenil; gamma-Aminobutyric Acid; Genetics, Behavioral; Male; Mice; Mice, Inbred ICR; Phenotype; Receptors, GABA-A

1992
Reversal of alcohol dependence and tolerance by a single administration of flumazenil.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:3

    Topics: Alcoholism; Animals; Ataxia; Behavior, Animal; Brain; Carbolines; Chlorides; Drug Administration Schedule; Drug Tolerance; Ethanol; Flumazenil; Hypothermia; Male; Mice; Mice, Inbred ICR; Neurons; Receptors, GABA-A

1991
Chronic benzodiazepine administration. VII. Behavioral tolerance and withdrawal and receptor alterations associated with clonazepam administration.
    Psychopharmacology, 1991, Volume: 104, Issue:2

    Topics: Animals; Behavior, Animal; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Clonazepam; Convulsants; Drug Tolerance; Flumazenil; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Substance Withdrawal Syndrome

1991
Correlation between gamma-aminobutyric acidA receptor ligand-induced changes in t-butylbicyclophosphoro[35S]thionate binding and 36Cl- uptake in rat cerebrocortical membranes.
    Molecular pharmacology, 1991, Volume: 39, Issue:3

    Topics: Animals; Bicuculline; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Desoxycorticosterone; Diazepam; Ethanol; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ligands; Membrane Proteins; Pentobarbital; Pregnanolone; Rats; Receptors, GABA-A; Synaptosomes

1991
Gamma-aminobutyric acid (GABAA) receptor-function in a rat model of hepatic encephalopathy.
    Metabolic brain disease, 1990, Volume: 5, Issue:4

    Topics: Animals; Cerebral Cortex; Chlorides; Disease Models, Animal; Flumazenil; Hepatic Encephalopathy; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Statistics as Topic; Synaptosomes

1990
Benzodiazepine agonist and inverse agonist actions on GABAA receptor-operated chloride channels. I. Acute effects of ethanol.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:2

    Topics: Animals; Benzodiazepines; Brain; Carbolines; Chloride Channels; Chlorides; Convulsants; Ethanol; Flumazenil; Flunitrazepam; Injections, Intraperitoneal; Male; Membrane Proteins; Mice; Mice, Inbred ICR; Tritium

1990
Augmentation of GABAA receptor function by chronic exposure to GABA-neutral and GABA-negative benzodiazepine ligands in cultured cortical neurons.
    Biochemical pharmacology, 1990, Sep-15, Volume: 40, Issue:6

    Topics: Animals; Appetite Depressants; Binding Sites; Carbolines; Chick Embryo; Chlorides; Culture Techniques; Flumazenil; Muscimol; Neurons; Ouabain; Receptors, GABA-A

1990
Rat pup ultrasonic isolation calls: possible mediation by the benzodiazepine receptor complex.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:5

    Topics: Animals; Benzodiazepinones; Chlorides; Diazepam; Flumazenil; Ion Channels; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sex Factors; Temperature; Vocalization, Animal

1986
The effect of benzodiazepines and beta-carbolines on GABA-stimulated chloride influx by membrane vesicles from the rat cerebral cortex.
    Biochemical and biophysical research communications, 1986, Nov-26, Volume: 141, Issue:1

    Topics: Animals; Benzodiazepines; Biological Transport; Carbolines; Cerebral Cortex; Chlorides; Drug Synergism; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channels; Rats; Receptors, GABA-A; Synaptic Vesicles

1986
Stress-induced changes in t-[35S]butylbicyclophosphorothionate binding to gamma-aminobutyric acid-gated chloride channels are mimicked by in vitro occupation of benzodiazepine receptors.
    Journal of neurochemistry, 1987, Volume: 49, Issue:3

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cerebral Cortex; Chlorides; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Ion Channels; Kinetics; Male; Membranes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Swimming

1987
Chronic benzodiazepine administration. II. Discontinuation syndrome is associated with upregulation of gamma-aminobutyric acidA receptor complex binding and function.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1

    Topics: Animals; Binding Sites; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Drug Tolerance; Flumazenil; Flunitrazepam; Ion Channels; Lorazepam; Male; Mice; Motor Activity; Muscimol; Receptors, GABA-A; Time Factors

1988
Effects of the imidazobenzodiazepine RO15-4513 on the stimulant and depressant actions of ethanol on spontaneous locomotor activity.
    Life sciences, 1988, Volume: 43, Issue:7

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Chlorides; Ethanol; Flumazenil; Ion Channels; Male; Mice; Mice, Inbred C3H; Motor Activity; Receptors, GABA-A

1988
Partial agonists of the benzodiazepine receptor: from animal data to results in patients.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Affinity Labels; Allosteric Site; Animals; Azides; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Chlorides; Clonazepam; Diazepam; Drug Interactions; Ethanol; Flumazenil; Flurazepam; Humans; Ion Channels; Ligands; Models, Neurological; Neurons; Receptors, GABA-A

1988
Chloride channel modulation through the benzodiazepine recognition site.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Bicuculline; Carbolines; Cells, Cultured; Chlorides; Convulsants; Flumazenil; Flunitrazepam; Ion Channels; Neurons; Receptors, GABA-A

1988
Asymmetrical activation of GABA-gated chloride channels in cerebral cortex.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Flumazenil; Functional Laterality; Ion Channels; Kinetics; Male; Organ Specificity; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
The story and activity of flumazenil (Anexate).
    Acta anaesthesiologica Belgica, 1989, Volume: 40, Issue:1

    Topics: Animals; Chemical Phenomena; Chemistry; Chlorides; Flumazenil; Humans; Ion Channels; Models, Chemical; Receptors, GABA-A

1989
Suppression of GABA-induced chloride current by 3-amino-1-methyl-5H-pyrido[4,3-b]indole (Trp-P-2).
    European journal of pharmacology, 1989, Aug-03, Volume: 166, Issue:3

    Topics: Alanine; Animals; Carbolines; Chlorides; Flumazenil; GABA Antagonists; Ganglia, Spinal; Male; Membrane Potentials; Mice; Mice, Inbred Strains; Muscimol; Neurons, Afferent; Taurine

1989
Dietary choline intake modulates benzodiazepine receptor binding and gamma-aminobutyric acidA receptor function in mouse brain.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:1

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Chlorides; Choline; Diet; Flumazenil; Male; Membrane Proteins; Mice; Motor Activity; Receptors, GABA-A

1989
The tremorigen aflatrem is a positive allosteric modulator of the gamma-aminobutyric acidA receptor channel expressed in Xenopus oocytes.
    Molecular pharmacology, 1989, Volume: 35, Issue:3

    Topics: Allosteric Regulation; Animals; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Indoles; Membrane Proteins; Mycotoxins; Oocytes; Pentobarbital; Picrotoxin; Receptors, GABA-A; Xenopus

1989
Chronic benzodiazepine administration. III. Upregulation of gamma-aminobutyric acidA receptor binding and function associated with chronic benzodiazepine antagonist administration.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3

    Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Flumazenil; Male; Membrane Proteins; Mice; Motor Activity; Receptors, GABA-A

1989
Benzodiazepine and beta-carboline interactions with GABAA receptor-gated chloride channels in mammalian cultured spinal cord neurons.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:2

    Topics: Animals; Benzodiazepines; Carbolines; Cells, Cultured; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Female; Flumazenil; Male; Membrane Proteins; Mice; Mice, Inbred C57BL; Neurons; Receptors, GABA-A; Spinal Cord

1989
Stress-induced behavioral depression in the rat is associated with a decrease in GABA receptor-mediated chloride ion flux and brain benzodiazepine receptor occupancy.
    Brain research, 1989, May-15, Volume: 487, Issue:1

    Topics: Animals; Brain; Chlorides; Depression; Flumazenil; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological; Synaptosomes

1989
Chronic clonazepam administration decreases gamma-aminobutyric acidA receptor function in cultured cortical neurons.
    Molecular pharmacology, 1989, Volume: 36, Issue:5

    Topics: Animals; Benzodiazepines; Cells, Cultured; Cerebral Cortex; Chick Embryo; Chlorides; Clonazepam; Drug Administration Schedule; Flumazenil; Muscimol; Picrotoxin; Receptors, GABA-A; Sesterterpenes

1989
Amoxapine inhibition of GABA-stimulated chloride conductance: investigations of potential sites of activity.
    Life sciences, 1989, Volume: 45, Issue:20

    Topics: Amoxapine; Animals; Cerebral Cortex; Chlorides; Dibenzoxazepines; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; GABA Antagonists; Ligands; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Discrimination of the benzodiazepine receptor antagonist Ro 15-1788 using the conditioned taste aversion procedure.
    NIDA research monograph, 1989, Volume: 95

    Topics: Animals; Brain; Chlorides; Conditioning, Classical; Discrimination Learning; Dose-Response Relationship, Drug; Drinking; Flumazenil; Generalization, Stimulus; Lithium; Lithium Chloride; Rats; Receptors, GABA-A; Taste

1989
Relative efficacies of 1,4-diazepines on GABA-stimulated chloride influx in rat brain vesicles.
    Life sciences, 1989, Volume: 45, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Azepines; Cell Membrane; Cerebral Cortex; Chlorides; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1989
Inhibition of rat brain adenylate cyclase activity by benzodiazepine through the effects on Gi and catalytic proteins.
    Life sciences, 1988, Volume: 42, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Aluminum; Aluminum Chloride; Aluminum Compounds; Animals; Benzodiazepines; Brain; Chlorides; Diazepam; Flumazenil; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptic Membranes

1988
Modulation of GABA-stimulated chloride influx into membrane vesicles from rat cerebral cortex by benzodiazepines and nonbenzodiazepines.
    Advances in biochemical psychopharmacology, 1988, Volume: 45

    Topics: Animals; Anti-Anxiety Agents; Cell Membrane; Cerebral Cortex; Chlorides; Clonazepam; Diazepam; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Inbred Strains

1988
Radiation inactivation studies of the benzodiazepine/gamma-aminobutyric acid/chloride ionophore receptor complex.
    Journal of neurochemistry, 1985, Volume: 45, Issue:1

    Topics: Animals; Barbiturates; Benzodiazepines; Benzodiazepinones; Binding Sites; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Flumazenil; Flunitrazepam; Ionophores; Male; Molecular Weight; Muscimol; Picrotoxin; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
A selective imidazobenzodiazepine antagonist of ethanol in the rat.
    Science (New York, N.Y.), 1986, Dec-05, Volume: 234, Issue:4781

    Topics: Animals; Anxiety; Azides; Benzodiazepines; Chlorides; Ethanol; Flumazenil; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes

1986
Modulation of GABA-gated chloride ion flux in rat brain by acute and chronic benzodiazepine administration.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1

    Topics: Animals; Benzodiazepines; Brain; Chlorides; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred Strains

1988
Antagonists of benzodiazepines: functional aspects.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Carbolines; Chlorides; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Ion Channels; Narcotic Antagonists; Parasympathomimetics; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A; Substance-Related Disorders; Xanthines

1983
Characterization of U-97775 as a GABAA receptor ligand of dual functionality in cloned rat GABAA receptor subtypes.
    British journal of pharmacology, 1995, Volume: 115, Issue:1

    Topics: Animals; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Line; Chlorides; Electrophysiology; Flumazenil; Humans; Imidazoles; Ligands; Quinoxalines; Rats; Receptors, GABA-A; Recombinant Proteins

1995
The effect of cyclopyrrolones on GABAA receptor function is different from that of benzodiazepines.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 350, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlorides; Chlorine; Flumazenil; Hypnotics and Sedatives; Kinetics; Male; Mice; Mice, Inbred Strains; Muscimol; Naphthyridines; Piperazines; Radioisotopes; Receptors, GABA-A; Sulfur Compounds; Sulfur Radioisotopes; Tritium

1994
Development pattern of the GABAA-benzodiazepine receptor ionophore complex in primary cultures of cortical neurons.
    Brain research. Developmental brain research, 1994, Jul-15, Volume: 80, Issue:1-2

    Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Cells, Cultured; Cerebral Cortex; Chlorides; Flumazenil; Flunitrazepam; Mice; Mice, Inbred C57BL; Muscimol; Neurons; Receptors, GABA-A

1994
Effects of 5-HT3 receptor antagonists on binding and function of mouse and human GABAA receptors.
    European journal of pharmacology, 1994, Jul-15, Volume: 268, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flunitrazepam; Humans; Indazoles; Indoles; Male; Mice; Mice, Inbred ICR; Receptors, GABA-A; Serotonin Antagonists; Tropanes; Tropisetron; Xenopus laevis

1994
Substituted pyrazinones, a new class of allosteric modulators for gamma-aminobutyric acidA receptors.
    Molecular pharmacology, 1993, Volume: 44, Issue:2

    Topics: Allosteric Regulation; Benzyl Compounds; Cell Line; Chlorides; Dose-Response Relationship, Drug; Flumazenil; Furans; gamma-Aminobutyric Acid; Humans; Pyrazines; Receptors, GABA-A

1993
Chronic flurazepam treatment produces decreased efficacy of the benzodiazepine ligands and pentobarbital with gamma-aminobutyric acidA receptors in cortical neurons.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:2

    Topics: Animals; Benzodiazepines; Biological Transport; Cells, Cultured; Cerebral Cortex; Chlorides; Female; Flumazenil; Flurazepam; Ligands; Male; Mice; Mice, Inbred C57BL; Neurons; Pentobarbital; Receptors, GABA

1994
beta-Lumicolchicine interacts with the benzodiazepine binding site to potentiate GABAA receptor-mediated currents.
    Journal of neurochemistry, 1994, Volume: 62, Issue:5

    Topics: Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Cerebral Cortex; Chlorides; DNA, Complementary; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Kinetics; Lumicolchicines; Mice; Mice, Inbred ICR; Oocytes; Receptors, GABA-A; Xenopus laevis

1994
Propofol activates GABAA receptor-chloride ionophore complex in dissociated hippocampal pyramidal neurons of the rat.
    Anesthesiology, 1993, Volume: 79, Issue:4

    Topics: Animals; Central Nervous System; Chloride Channels; Chlorides; Diazepam; Flumazenil; Hippocampus; Kinetics; Membrane Potentials; Neurons; Propofol; Pyramidal Tracts; Rats; Rats, Wistar; Receptors, GABA

1993
Zinc selectively inhibits flux through benzodiazepine-insensitive gamma-aminobutyric acid chloride channels in cortical and cerebellar microsacs.
    Molecular pharmacology, 1993, Volume: 44, Issue:4

    Topics: Animals; Benzodiazepines; Cerebellum; Cerebral Cortex; Chloride Channels; Chlorides; Chlorine; Drug Synergism; Flumazenil; Flunitrazepam; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Kinetics; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stimulation, Chemical; Tritium; Zinc

1993
Tolerance to the behavioral effects of chlordiazepoxide: pharmacological and biochemical selectivity.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:3

    Topics: Amphetamine; Animals; Behavior, Animal; Caffeine; Carbolines; Chlordiazepoxide; Chlorides; Chlorine; Dose-Response Relationship, Drug; Drug Tolerance; Flumazenil; gamma-Aminobutyric Acid; Male; Midazolam; Morphine; Pentobarbital; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sensitivity and Specificity; Stimulation, Chemical

1993
5-Aryl-3-(alkylthio)-4H-1,2,4-triazoles as selective antagonists of strychnine-induced convulsions and potential antispastic agents.
    Journal of medicinal chemistry, 1994, Jan-07, Volume: 37, Issue:1

    Topics: Animals; Anticonvulsants; Cerebellum; Cerebral Cortex; Chlorides; Electroshock; Flumazenil; Male; Mice; Molecular Structure; Muscle Spasticity; Paralysis; Rats; Rats, Sprague-Dawley; Seizures; Structure-Activity Relationship; Strychnine; Triazoles

1994
Swim stress selectively alters the specific binding of a benzodiazepine antagonist in mice.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:2

    Topics: Animals; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flumazenil; Flurazepam; In Vitro Techniques; Kinetics; Male; Mice; Receptors, GABA-A; Stress, Physiological; Swimming; Tissue Distribution

1993
Characterization of a benzodiazepine receptor site with exceptionally high affinity for Ro 15-4513 in the rat CNS.
    Brain research, 1995, Dec-18, Volume: 704, Issue:2

    Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Central Nervous System; Cerebellum; Chlorides; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; GABA Modulators; Hippocampus; Imidazoles; Male; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Spinal Cord; Tritium

1995
Diazepam physical dependence and withdrawal in rats is associated with alteration in GABAA receptor function.
    Life sciences, 1996, Volume: 59, Issue:19

    Topics: Animals; Benzodiazepines; Cerebral Cortex; Chloride Channels; Chlorides; Diazepam; Flumazenil; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred F344; Receptors, GABA-A; Substance Withdrawal Syndrome; Substance-Related Disorders

1996
Flumazenil reverses the decrease in the hypnotic activity of pentobarbital by social isolation stress: are endogenous benzodiazepine receptor ligands involved?
    Brain research, 1997, Jan-16, Volume: 745, Issue:1-2

    Topics: Animals; Carbolines; Chlorides; Diazepam; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Hypnotics and Sedatives; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred Strains; Pentobarbital; Receptors, GABA-A; Sleep; Social Isolation; Stress, Psychological; Synaptosomes

1997
Central corticotropin-releasing factor and benzodiazepine receptor systems are involved in the social isolation stress-induced decrease in ethanol sleep in mice.
    Brain research, 1997, Apr-11, Volume: 753, Issue:2

    Topics: Animals; Brain; Central Nervous System Depressants; Chlorides; Corticotropin-Releasing Hormone; Ethanol; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Hormone Antagonists; Housing, Animal; Male; Mice; Receptors, GABA-A; Sleep; Social Isolation; Stress, Psychological; Synaptosomes

1997
[3H]Ro 15-1788 binding sites to brain membrane of the saltwater Mugil cephalus.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2001, Volume: 128, Issue:3

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Female; Fishes; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Imidazoles; Ionophores; Male; Pyridines; Receptors, GABA-A; Synaptosomes; Tritium; Zolpidem

2001
Increase in expression of the GABA(A) receptor alpha(4) subunit gene induced by withdrawal of, but not by long-term treatment with, benzodiazepine full or partial agonists.
    Brain research. Molecular brain research, 2001, Aug-15, Volume: 92, Issue:1-2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Cell Membrane; Cells, Cultured; Cerebellum; Chloride Channels; Chlorides; Diazepam; Drug Tolerance; Female; Flumazenil; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Imidazoles; Ion Transport; Membrane Potentials; Microinjections; Nerve Tissue Proteins; Neurons; Oocytes; Protein Subunits; Rats; Receptors, GABA-A; RNA, Messenger; Substance Withdrawal Syndrome; Substance-Related Disorders; Up-Regulation; Xenopus laevis

2001
Dose-dependent enhancement of in vivo GABA(A)-benzodiazepine receptor binding by isoflurane.
    Anesthesiology, 2001, Volume: 95, Issue:3

    Topics: Adult; Anesthetics, Inhalation; Blood-Brain Barrier; Cerebrovascular Circulation; Chlorides; Dose-Response Relationship, Drug; Female; Flumazenil; Humans; Isoflurane; Male; Protein Binding; Receptors, GABA-A

2001
Inhibitory effect of diazepam on muscarinic receptor-stimulated inositol 1,4,5-trisphosphate production in rat parotid acinar cells.
    British journal of pharmacology, 2002, Volume: 137, Issue:7

    Topics: Animals; Anticonvulsants; Calcium; Carbachol; Chlorides; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; GABA-A Receptor Antagonists; GTP-Binding Proteins; Inositol 1,4,5-Trisphosphate; Isoquinolines; Male; Parotid Gland; Phenylephrine; Phosphoinositide Phospholipase C; Phosphoric Diester Hydrolases; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Muscarinic; Time Factors

2002
6,3'-Dinitroflavone is a low efficacy modulator of GABA(A) receptors.
    European journal of pharmacology, 2008, Sep-04, Volume: 591, Issue:1-3

    Topics: Animals; Anti-Anxiety Agents; Cell Line; Chlorides; Female; Flavonoids; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Oocytes; Patch-Clamp Techniques; Protein Binding; Protein Subunits; Receptors, GABA-A; Transfection; Xenopus

2008
New insight into the central benzodiazepine receptor-ligand interactions: design, synthesis, biological evaluation, and molecular modeling of 3-substituted 6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and related compounds.
    Journal of medicinal chemistry, 2011, Aug-25, Volume: 54, Issue:16

    Topics: Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Cattle; Cerebral Cortex; Chlorides; Flumazenil; HEK293 Cells; Humans; Ligands; Male; Mice; Models, Molecular; Molecular Structure; Motor Activity; Protein Structure, Tertiary; Protein Subunits; Radioligand Assay; Receptors, GABA-A; Synaptosomes; Tritium; Xenopus laevis

2011
The Direct Actions of GABA, 2'-Methoxy-6-Methylflavone and General Anaesthetics at β3γ2L GABAA Receptors: Evidence for Receptors with Different Subunit Stoichiometries.
    PloS one, 2015, Volume: 10, Issue:10

    Topics: Anesthetics, Intravenous; Animals; Cells, Cultured; Chlorides; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Etomidate; Female; Flavones; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Humans; Propofol; Protein Subunits; Receptors, GABA-A; Xenopus laevis; Zinc Compounds

2015
Comparison of two injectable anaesthetic protocols in Egyptian fruit bats (Rousettus aegyptiacus) undergoing gonadectomy.
    Scientific reports, 2022, 09-24, Volume: 12, Issue:1

    Topics: Anesthetics; Animals; Butorphanol; Castration; Chiroptera; Chlorides; Dexmedetomidine; Flumazenil; Hypnotics and Sedatives; Isoflurane; Ketamine; Midazolam; Sodium

2022
Zerumbone, a major sesquiterpene from Syringa pinnatifolia Hemsl., exerts the sedative effect by regulating GABAergic nervous system.
    Journal of ethnopharmacology, 2023, Jan-30, Volume: 301

    Topics: Animals; Bicuculline; Chlorides; Flumazenil; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Mice; Molecular Docking Simulation; Nervous System; Pentobarbital; Plant Extracts; Rats; Receptors, GABA-A; Sesquiterpenes; Syringa

2023
Ethanol potentiation of GABAergic transmission in cultured spinal cord neurons involves gamma-aminobutyric acidA-gated chloride channels.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:2

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Cells, Cultured; Chlorine; Ethanol; Female; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Mice; Mice, Inbred C57BL; Neurons; Radioisotopes; Spinal Cord

1988