flumazenil and brotizolam

flumazenil has been researched along with brotizolam in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19904 (40.00)18.7374
1990's1 (10.00)18.2507
2000's3 (30.00)29.6817
2010's1 (10.00)24.3611
2020's1 (10.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Anzini, M; Brogi, S; Cappelli, A; Chemi, G; Di Capua, A; Di Cesare Mannelli, L; Garofalo, A; Ghelardini, C; Giorgi, G; Grande, F; Matucci, R; Paolino, M; Reale, A1
Casals-Stenzel, J1
Koot, M; Van Duin, CT; Van Miert, AS1
Bechtel, WD; Ikeda, M; Malatynska, E; Weber, KH; Yamamura, HI1
Casals-Stenzel, J; Weber, KH1
Böke-Kuhn, K; Danneberg, PB; Hommer, D; Kuhn, FJ; Lehr, E; Paul, SM; Skolnick, P; Weber, KH1
Kishore, K; Saraf, MK; Sharma, A; Singh, M; Thomas, KM1

Reviews

1 review(s) available for flumazenil and brotizolam

ArticleYear
Thieno-triazolo-1,4-diazepines as antagonists of platelet-activating factor: present status.
    Lipids, 1991, Volume: 26, Issue:12

    Topics: Animals; Azepines; Central Nervous System; Flumazenil; Humans; Platelet Activating Factor; Platelet Membrane Glycoproteins; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Structure-Activity Relationship; Triazolam; Triazoles

1991

Other Studies

9 other study(ies) available for flumazenil and brotizolam

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Design, synthesis and biological evaluation of 7-substituted 4-phenyl-6H-imidazo[1,5-a]thieno[3,2-f] [1,4]diazepines as safe anxiolytic agents.
    European journal of medicinal chemistry, 2020, Aug-15, Volume: 200

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Binding Sites; Drug Design; Locomotion; Memory Disorders; Mice; Molecular Docking Simulation; Rats; Receptors, GABA-A

2020
Appetite-modulating drugs in dwarf goats, with special emphasis on benzodiazepine-induced hyperphagia and its antagonism by flumazenil and RO 15-3505.
    Journal of veterinary pharmacology and therapeutics, 1989, Volume: 12, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Appetite Regulation; Azepines; Benzodiazepines; Benzodiazepinones; Body Weight; Diazepam; Female; Flumazenil; Goats; Hyperphagia; Ivermectin; Male; Midazolam; Time Factors

1989
Relative efficacies of 1,4-diazepines on GABA-stimulated chloride influx in rat brain vesicles.
    Life sciences, 1989, Volume: 45, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Azepines; Cell Membrane; Cerebral Cortex; Chlorides; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1989
Triazolodiazepines: dissociation of their Paf (platelet activating factor) antagonistic and CNS activity.
    British journal of pharmacology, 1987, Volume: 90, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Azepines; Benzodiazepinones; Central Nervous System; Flumazenil; Guinea Pigs; Humans; Hypnotics and Sedatives; In Vitro Techniques; Platelet Activating Factor; Platelet Aggregation; Receptors, GABA-A; Tidal Volume; Triazolam

1987
Pharmacological and neurochemical properties of 1,4-diazepines with two annelated heterocycles ('hetrazepines').
    European journal of pharmacology, 1985, Feb-12, Volume: 109, Issue:1

    Topics: Action Potentials; Aggression; Animals; Anticonvulsants; Azepines; Behavior, Animal; Benzodiazepinones; Brain Chemistry; Carbolines; Cerebral Cortex; Conflict, Psychological; Diazepam; Flumazenil; Heterocyclic Compounds; Humans; Hypnotics and Sedatives; Male; Mice; Motor Activity; Neurons; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sleep; Social Isolation; Wakefulness

1985
Role of platelet activating factor in triazolobenzodiazepines-induced retrograde amnesia.
    Behavioural brain research, 2003, Jun-16, Volume: 142, Issue:1-2

    Topics: 1-Alkyl-2-acetylglycerophosphocholine Esterase; Amnesia, Anterograde; Amnesia, Retrograde; Animals; Anti-Anxiety Agents; Azepines; Diazepam; Diterpenes; Escape Reaction; Female; Flumazenil; Ginkgolides; Lactones; Learning; Male; Mice; Phospholipases A; Platelet Activating Factor; Platelet Membrane Glycoproteins; Reaction Time; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Receptors, GABA-A; Retention, Psychology; Triazolam

2003