flumazenil and beta-carboline-3-carboxylic acid methyl ester

flumazenil has been researched along with beta-carboline-3-carboxylic acid methyl ester in 51 studies

Research

Studies (51)

TimeframeStudies, this research(%)All Research%
pre-199020 (39.22)18.7374
1990's16 (31.37)18.2507
2000's15 (29.41)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cecchi, L; Colotta, V; Filacchioni, G; Giannaccini, G; Lucacchini, A; Martini, C; Melani, F1
Da Settimo, A; Da Settimo, F; Gesi, M; Giannaccini, G; Greco, G; Lucacchini, A; Marini, AM; Martini, C; Novellino, E; Primofiore, G1
Da Settimo, F; Gesi, M; Greco, G; La Motta, C; Marini, AM; Martini, C; Novellino, E; Primofiore, G; Taliani, S; Trincavelli, L1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Clayton, T; Cook, J; DeLorey, TM; Furtmüller, R; Halliwell, RF; Harris, D; Huck, S; Sahbaie, P; Sieghart, W1
Chapouthier, G; Cherkaoui, J; Dellu, F; Dodd, RH; Le Moal, M; Mayo, W; Simon, H1
Bottlaender, M; Brouillet, E; Chavoix, C; Dodd, RH; Fournier, D; Hantraye, P; Khalili-Varasteh, M; Mazière, M1
Belzung, C; Cabib, S; Fabiani, L; Puglisi-Allegra, S; Tolentino, P1
Nagatani, T; Sugihara, T; Takao, K; Ueki, S; Yamamoto, T1
Kovács, I; Maksay, G; Simonyi, M1
Biggio, G; Corda, MG; Giorgi, O; Longoni, B1
Ozaki, T; Shibata, S; Ueki, S; Yamamoto, E; Yamashita, K1
Nagatani, T; Sugihara, T; Ueki, S; Yamamoto, T1
Gerhardt, S; Liebman, JM1
Moura, D; Soares-da-Silva, P1
Ikonomidou, C; Klockgether, T; Schwarz, M; Sontag, KH; Turski, L1
Brouillet, E; Chavoix, C; Crouzel, M; Dodd, RH; Fukuda, H; Guibert, B; Hantraye, P; Mazière, M; Naquet, R; Prenant, C1
Costello, MJ; Nutt, DJ1
Conti-Tronconi, B; Costa, E; Ferrero, P; Guidotti, A; Santi, MR1
Bortolotto, ZA; Cavalheiro, EA; Ikonomidou, C; Mello, LE; Turski, L; Turski, WA1
Little, HJ1
Bonetti, EP; Haefely, W; Polc, P; Schaffner, R1
Cavalheiro, E; Chapouthier, G; Dodd, RH; Kaijima, M; Potier, P; Prado de Carvalho, L; Rossier, J; Valin, A; Venault, P1
Crawley, JN; Paul, SM; Skolnick, P1
Paul, SM; Skolnick, P1
Biggio, G; Concas, A; Fanni, B; Mereu, G; Serra, M1
Biggio, G; Mereu, G1
Cavalheiro, EA; Chapouthier, G; Dodd, RH; Grecksch, G; Prado de Carvalho, L; Rossier, J1
Cain, M; Cook, J; Paul, S; Schweri, M; Skolnick, P1
Morel, E; Perrault, G; Sanger, DJ; Zivkovic, B1
Bannwarth, W; Benke, D; Fritschy, JM; Mohler, H; Trzeciak, A1
Emerich, DF; Stackman, RW; Taylor, LA; Walsh, TJ1
Hadingham, KL; Palmer, KJ; Thompson, SA; Wafford, KA; Whiting, PJ1
Chimirri, A; De Sarro, A; De Sarro, G; Guisti, P; Lipartiti, M; Zappala, M1
Bondoux, D; Chapouthier, G; Clément, Y; Launay, JM1
Pokk, P; Zharkovsky, A1
Chimirri, A; De Sarro, A; De Sarro, G; Giusti, P; McKernan, R; Quirk, K1
Breton, C; Chapouthier, G; Crusio, WE; Launay, JM; Roubertoux, PL; Venault, P1
D'Amato, FR; Mandillo, S1
Chapouthier, G; Dodd, RH; Launay, JM; Rössler, AS; Venault, P1
Kamei, J; Ohsawa, M1
Firestone, LL; Homanics, GE; Quinlan, JJ1
Bondoux, D; Chapouthier, G; Clément, Y; Launay, JM; Martin, B; Venault, P1
Beaujean, D; Do-Rego, JL; Leprince, J; Luu-The, V; Mensah-Nyagan, AG; Pelletier, G; Tonon, MC; Vaudry, H1
Betti, L; Bistocchi, M; Giannaccini, G; Gori, M; Lucacchini, A1
Béracochéa, D; Borde, N; Krazem, A1
Bromidge, FA; Casula, MA; Hadingham, KL; Martin, K; Maubach, K; Pillai, GV; Seabrook, GR; Whiting, PJ; Wingrove, PB1
Kamei, J; Matsumiya, T; Ohsawa, M; Takeda, H; Tsuji, M1
Pokk, P; Väli, M1
France, CP; McMahon, LR1
Hirano, S; Kamei, J; Miyata, S1

Reviews

1 review(s) available for flumazenil and beta-carboline-3-carboxylic acid methyl ester

ArticleYear
[Drug activation of GABAergic transmission in the central nervous system: benzodiazepines and GABAergic agonists].
    Acta medica portuguesa, 1985, Volume: 6, Issue:2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Chemical Phenomena; Chemistry; Cyclic GMP; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Humans; Receptors, GABA-A; Synaptic Transmission; Valproic Acid

1985

Other Studies

50 other study(ies) available for flumazenil and beta-carboline-3-carboxylic acid methyl ester

ArticleYear
Tricyclic heteroaromatic systems. [1]benzopyranopyrrol-4-ones and [1]benzopyrano-1,2,3-triazol-4-ones as benzodiazepine receptor ligands. Synthesis and structure-activity relationships.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:9

    Topics: Animals; Azoles; Benzopyrans; Cattle; Chemical Phenomena; Chemistry; Dibenzazepines; Ligands; Pyrroles; Receptors, GABA-A; Structure-Activity Relationship

1990
N'-Phenylindol-3-ylglyoxylohydrazide derivatives: synthesis, structure-activity relationships, molecular modeling studies, and pharmacological action on brain benzodiazepine receptors.
    Journal of medicinal chemistry, 1998, Sep-24, Volume: 41, Issue:20

    Topics: Animals; Anticonvulsants; Binding, Competitive; Brain; Cattle; Cerebral Cortex; Convulsants; Diazepam; Flumazenil; GABA Modulators; Glyoxylates; Hydrazines; In Vitro Techniques; Indoles; Ligands; Mice; Models, Molecular; Molecular Conformation; Receptors, GABA-A; Seizures; Structure-Activity Relationship

1998
3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: tricyclic heteroaromatic derivatives as a new class of benzodiazepine receptor ligands.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Anticonvulsants; Benzimidazoles; Brain; Cattle; Convulsants; Diazepam; Flumazenil; GABA Modulators; In Vitro Techniques; Ligands; Membranes; Mice; Models, Molecular; Radioligand Assay; Receptors, GABA-A

2000
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.
    Journal of medicinal chemistry, 2008, Jul-10, Volume: 51, Issue:13

    Topics: Animals; Behavior, Animal; Benzodiazepines; Chemical Phenomena; Chemistry, Physical; Computer Simulation; Databases, Factual; Electrophysiology; Female; Ligands; Male; Memory; Mice; Models, Molecular; Molecular Structure; Oocytes; Protein Isoforms; Protein Subunits; Quantitative Structure-Activity Relationship; Receptors, GABA-A; Structure-Activity Relationship; Xenopus laevis

2008
Cognitive enhancing properties of beta-CCM infused into the nucleus basalis magnocellularis of the rat.
    Brain research, 1992, Aug-28, Volume: 589, Issue:1

    Topics: Animals; Carbolines; Cognition; Flumazenil; Memory; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Reproducibility of Results; Substantia Innominata; Synaptic Transmission

1992
In vivo bidirectional modulatory effect of benzodiazepine receptor ligands on GABAergic transmission evaluated by positron emission tomography in non-human primates.
    Brain research, 1991, Aug-23, Volume: 557, Issue:1-2

    Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Carbolines; Cerebral Cortex; Diazepam; Electroencephalography; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Papio; Pentylenetetrazole; Receptors, GABA-A; Seizures; Synaptic Transmission; Tomography, Emission-Computed

1991
LY 171555-induced hyperdefensiveness in the mouse does not implicate benzodiazepine receptors.
    Psychopharmacology, 1991, Volume: 103, Issue:4

    Topics: Aggression; Animals; Behavior, Animal; Carbolines; Chlordiazepoxide; Convulsants; Dopamine Agents; Dose-Response Relationship, Drug; Ergolines; Flumazenil; Mice; Mice, Inbred C57BL; Quinpirole; Receptors, GABA-A; Social Behavior

1991
beta-CCM inhibits muricide induced by olfactory bulbectomy in rats.
    Japanese journal of pharmacology, 1990, Volume: 52, Issue:3

    Topics: Aggression; Animals; Brain; Carbolines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Injections, Intravenous; Male; Mice; Motor Activity; Muscle Relaxants, Central; Olfactory Bulb; Phenoxybenzamine; Postural Balance; Rats; Rats, Inbred Strains; Receptors, GABA-A

1990
Inhibition of high-affinity synaptosomal uptake of gamma-aminobutyric acid by a bicyclo-heptane derivative.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:3

    Topics: Animals; Anticonvulsants; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Camphanes; Carbolines; Cerebral Cortex; Diazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Synaptic Membranes; Synaptosomes

1989
Ro 15-4513, a partial inverse agonist for benzodiazepine recognition sites, has proconflict and proconvulsant effects in the rat.
    European journal of pharmacology, 1989, Jan-17, Volume: 159, Issue:3

    Topics: Animals; Azides; Benzodiazepines; Carbolines; Conflict, Psychological; Convulsants; Flumazenil; Isoniazid; Male; Pentobarbital; Punishment; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
Effects of benzodiazepine and GABA antagonists on anticonflict effects of antianxiety drugs injected into the rat amygdala in a water-lick suppression test.
    Psychopharmacology, 1989, Volume: 98, Issue:1

    Topics: Amygdala; Animals; Anti-Anxiety Agents; Behavior, Animal; Body Weight; Carbolines; Conflict, Psychological; Dose-Response Relationship, Drug; Drinking; Flumazenil; GABA Antagonists; Injections; Male; Rats; Rats, Inbred Strains

1989
The effect of agonists at the GABA-benzodiazepine-receptor-complex on the proconflict effect induced by beta-CCM and pentetrazol in rats.
    Japanese journal of pharmacology, 1988, Volume: 46, Issue:3

    Topics: Aminooxyacetic Acid; Animals; Azabicyclo Compounds; Carbolines; Conflict, Psychological; Convulsants; Diazepam; Flumazenil; Hypnotics and Sedatives; Male; Pentylenetetrazole; Phenobarbital; Piperazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Self-regulation of ICSS duration: effects of anxiogenic substances, benzodiazepine antagonists and antidepressants.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Anti-Anxiety Agents; Antidepressive Agents; Anxiety; Benzodiazepinones; Caffeine; Carbolines; Conditioning, Operant; Convulsants; Flumazenil; Humans; Male; Pentylenetetrazole; Pyrazoles; Rats; Rats, Inbred F344; Self Stimulation; Time Factors

1985
Effects of methyl beta-carboline-3-carboxylate, Ro 15-1788 and CGS 8216 on muscle tone in genetically spastic rats.
    European journal of pharmacology, 1985, Jul-17, Volume: 113, Issue:2

    Topics: Animals; Benzodiazepinones; Carbolines; Dose-Response Relationship, Drug; Electromyography; Female; Flumazenil; Male; Muscle Spasticity; Muscle Tonus; Pyrazoles; Rats; Rats, Mutant Strains; Receptors, GABA-A

1985
Benzodiazepine receptors studied in living primates by positron emission tomography: inverse agonist interactions.
    European journal of pharmacology, 1987, Jun-19, Volume: 138, Issue:2

    Topics: Animals; Binding, Competitive; Carbolines; Cerebral Cortex; Convulsants; Dose-Response Relationship, Drug; Electroencephalography; Flumazenil; Male; Papio; Receptors, GABA-A; Tomography, Emission-Computed

1987
Rapid induction of lorazepam dependence and reversal with flumazenil.
    Life sciences, 1988, Volume: 43, Issue:13

    Topics: Animals; Carbolines; Flumazenil; Lorazepam; Male; Mice; Mice, Inbred Strains; Seizures; Substance-Related Disorders

1988
Study of an octadecaneuropeptide derived from diazepam binding inhibitor (DBI): biological activity and presence in rat brain.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:3

    Topics: Amino Acid Sequence; Animals; Behavior, Animal; Benzodiazepinones; Brain Chemistry; Carbolines; Chromatography, High Pressure Liquid; Diazepam Binding Inhibitor; Enzyme-Linked Immunosorbent Assay; Flumazenil; Flunitrazepam; Male; Nerve Tissue Proteins; Neuropeptides; Peptide Fragments; Rats; Rats, Inbred Strains; Seizures; Synaptic Membranes

1986
Effects of aminophylline and 2-chloroadenosine on seizures produced by pilocarpine in rats: morphological and electroencephalographic correlates.
    Brain research, 1985, Dec-30, Volume: 361, Issue:1-2

    Topics: 2-Chloroadenosine; Adenosine; Aminophylline; Animals; Benzodiazepinones; Bicuculline; Brain; Carbolines; Convulsants; Electroencephalography; Flumazenil; Male; Motor Activity; Pilocarpine; Rats; Rats, Inbred Strains; Seizures

1985
The effects of benzodiazepine agonists, inverse agonists and Ro 15-1788 on the responses of the superior cervical ganglion to GABA in vitro.
    British journal of pharmacology, 1984, Volume: 83, Issue:1

    Topics: Animals; Barbiturates; Benzodiazepinones; Bicuculline; Carbolines; Chlordiazepoxide; Flumazenil; Flurazepam; gamma-Aminobutyric Acid; Ganglia, Sympathetic; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1984
A three-state model of the benzodiazepine receptor explains the interactions between the benzodiazepine antagonist Ro 15-1788, benzodiazepine tranquilizers, beta-carbolines, and phenobarbitone.
    Naunyn-Schmiedeberg's archives of pharmacology, 1982, Volume: 321, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Carbolines; Cats; Female; Flumazenil; Hippocampus; In Vitro Techniques; Indoles; Male; Mice; Models, Biological; Phenobarbital; Rats; Receptors, Cell Surface; Receptors, GABA-A; Spinal Cord

1982
Distinct behavioral and pharmacological effects of two benzodiazepine antagonists: Ro 15-1788 and methyl beta-carboline.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepinones; Carbolines; Cats; Drug Synergism; Electroencephalography; Electrophysiology; Flumazenil; Indoles; Mice; Papio; Pentylenetetrazole; Seizures; Species Specificity

1983
Absence of intrinsic antagonist actions of benzodiazepine antagonists on an exploratory model of anxiety in the mouse.
    Neuropharmacology, 1984, Volume: 23, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Carbolines; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Humans; Male; Mice; Pyrazoles

1984
New concepts in the neurobiology of anxiety.
    The Journal of clinical psychiatry, 1983, Volume: 44, Issue:11 Pt 2

    Topics: Animals; Anxiety; Barbiturates; Behavior; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Carbolines; Central Nervous System; Flumazenil; Humans; Macaca mulatta; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A

1983
beta-Carbolines activate neurons in the substantia nigra pars reticulata: an effect reversed by diazepam and Ro15-1788.
    European journal of pharmacology, 1983, Dec-09, Volume: 96, Issue:1-2

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Drug Interactions; Flumazenil; Indoles; Injections, Intravenous; Male; Rats; Rats, Inbred Strains; Substantia Nigra; Synaptic Transmission

1983
Effect of agonists, inverse agonists, and antagonists of benzodiazepine receptors on the firing rate of substantia nigra pars reticulata neurons.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electrophysiology; Flumazenil; Male; Neurons; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substantia Nigra

1983
Characterization of convulsions induced by methyl beta-carboline-3-carboxylate in mice.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electroencephalography; Flumazenil; Hypnotics and Sedatives; Indoles; Male; Mice; Pentylenetetrazole; Postural Balance; Time Factors

1984
Blockade of 3-carbomethoxy-beta-carboline induced seizures by diazepam and the benzodiazepine antagonists, Ro 15-1788 and CGS 8216.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:3

    Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Harmaline; Indoles; Male; Mice; Pyrazoles; Seizures; Tremor

1982
Repeated treatment with alpidem, a new anxiolytic, does not induce tolerance or physical dependence.
    Neuropharmacology, 1993, Volume: 32, Issue:9

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Bicuculline; Carbolines; Convulsants; Diazepam; Drug Tolerance; Flumazenil; Imidazoles; Isoniazid; Male; Mice; Pentylenetetrazole; Pyridines; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
Distribution, prevalence, and drug binding profile of gamma-aminobutyric acid type A receptor subtypes differing in the beta-subunit variant.
    The Journal of biological chemistry, 1994, Oct-28, Volume: 269, Issue:43

    Topics: Animals; Brain Chemistry; Carbolines; Flumazenil; Flunitrazepam; Genetic Variation; Immunohistochemistry; Male; Microscopy, Confocal; Molecular Weight; Precipitin Tests; Protein Conformation; Pyridazines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tissue Distribution; Zolpidem

1994
Intraseptal injection of GABA and benzodiazepine receptor ligands alters high-affinity choline transport in the hippocampus.
    Brain research bulletin, 1993, Volume: 31, Issue:3-4

    Topics: Acetylcholinesterase; Animals; Baclofen; Brain; Carbolines; Chlordiazepoxide; Choline; Convulsants; Flumazenil; gamma-Aminobutyric Acid; Hippocampus; Injections; Male; Muscimol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptosomes

1993
Expression and pharmacology of human GABAA receptors containing gamma 3 subunits.
    European journal of pharmacology, 1995, Nov-30, Volume: 291, Issue:3

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Base Sequence; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Molecular Sequence Data; Pyrazoles; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Proteins; Sequence Homology, Amino Acid; Triazolam; Xenopus; Zolpidem

1995
Azirino[1, 2-d][1, 4]benzodiazepine derivatives and related 1,4-benzodiazepines as anticonvulsant agents in DBA/2 mice.
    General pharmacology, 1996, Volume: 27, Issue:7

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Benzodiazepines; Binding, Competitive; Carbolines; Cell Membrane; Cerebellum; Cerebral Cortex; Chemical Phenomena; Chemistry, Physical; Convulsants; Flumazenil; GABA Modulators; Male; Mice; Mice, Inbred DBA; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1996
Convulsive effects of a benzodiazepine receptor inverse agonist: are they related to anxiogenic processes?
    Journal of physiology, Paris, 1997, Volume: 91, Issue:1

    Topics: Animals; Anxiety; Behavior, Animal; Carbolines; Convulsants; Female; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Ligands; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Receptors, GABA-A; Seizures

1997
The effects of flumazenil, Ro 15-4513 and beta-CCM on the behaviour of control and stressed mice in the plus-maze test.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 1997, Volume: 48, Issue:2

    Topics: Animals; Anxiety; Azides; Behavior, Animal; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Ligands; Male; Mice; Stress, Psychological

1997
Anticonvulsant activity of azirino[1,2-d][1,4]benzodiazepines and related 1,4-benzodiazepines in mice.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:1

    Topics: Animals; Anticonvulsants; Benzodiazepines; Carbolines; Cell Line; Convulsants; Flumazenil; GABA Modulators; Male; Membranes; Mice; Mice, Inbred DBA; Movement; Pentylenetetrazole; Radioligand Assay; Receptors, GABA-A; Seizures

1997
Genetic selection of mouse lines differing in sensitivity to a benzodiazepine receptor inverse agonist.
    Brain research, 1998, Mar-16, Volume: 787, Issue:1

    Topics: Animals; Carbolines; Convulsants; Female; Flumazenil; GABA Agents; Male; Mice; Mice, Inbred Strains; Radioligand Assay; Selection, Genetic; Species Specificity

1998
Male olfactory cues affect mothers' behavior in mice: effects of benzodiazepines.
    Psychopharmacology, 1999, Volume: 146, Issue:3

    Topics: Animals; Benzodiazepines; Carbolines; Chlordiazepoxide; Cues; Female; Flumazenil; Lactation; Male; Maternal Behavior; Mice; Odorants; Reaction Time

1999
Changes in benzodiazepine binding in a subkindling situation.
    Epilepsia, 2000, Volume: 41, Issue:6

    Topics: Animals; Carbolines; Convulsants; Disease Models, Animal; Epilepsy; Flumazenil; GABA Antagonists; Kindling, Neurologic; Male; Mice; Receptors, GABA-A; Seizures; Tritium

2000
Socio-psychological stress-induced antinociception in diabetic mice.
    Psychopharmacology, 2000, Volume: 149, Issue:4

    Topics: Animals; Anti-Bacterial Agents; Anticonvulsants; Carbolines; Convulsants; Diabetes Mellitus, Experimental; Diazepam; Flumazenil; GABA Modulators; Male; Mice; Mice, Inbred ICR; Pain Measurement; Streptozocin; Stress, Psychological

2000
Mice lacking the long splice variant of the gamma 2 subunit of the GABA(A) receptor are more sensitive to benzodiazepines.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 66, Issue:2

    Topics: Alternative Splicing; Animals; Azides; Benzodiazepines; Brain; Carbolines; Diazepam; Drug Resistance; Female; Flumazenil; GABA Modulators; Genetic Variation; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Midazolam; Pyridines; Receptors, GABA-A; Sleep; Zolpidem

2000
Chromosomes 4 and 13 in beta-carboline-induced seizures in mice: benzodiazepine binding.
    Neuroreport, 2000, Jul-14, Volume: 11, Issue:10

    Topics: Animals; Brain; Carbolines; Chromosome Mapping; Convulsants; Flumazenil; Mice; Mice, Inbred Strains; Mice, Mutant Strains; Radioligand Assay; Receptors, GABA-A; Seizures; Species Specificity; Tritium

2000
The octadecaneuropeptide ODN stimulates neurosteroid biosynthesis through activation of central-type benzodiazepine receptors.
    Journal of neurochemistry, 2001, Volume: 76, Issue:1

    Topics: 17-alpha-Hydroxypregnenolone; 17-alpha-Hydroxyprogesterone; 3-Hydroxysteroid Dehydrogenases; Animals; Carbolines; Chromatography, High Pressure Liquid; Dehydroepiandrosterone; Diazepam Binding Inhibitor; Dihydrotestosterone; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hydroxysteroids; Hypothalamus; Immunohistochemistry; In Vitro Techniques; Ligands; Male; Neuroglia; Neurons; Neuropeptides; Peptide Fragments; Pregnenolone; Progesterone; Rana ridibunda; Receptors, GABA-A

2001
[3H]Ro 15-1788 binding sites to brain membrane of the saltwater Mugil cephalus.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2001, Volume: 128, Issue:3

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Female; Fishes; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Imidazoles; Ionophores; Male; Pyridines; Receptors, GABA-A; Synaptosomes; Tritium; Zolpidem

2001
Effects of diazepam and beta-CCM on working memory in mice: relationships with emotional reactivity.
    Pharmacology, biochemistry, and behavior, 2001, Volume: 68, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Carbolines; Convulsants; Diazepam; Emotions; Flumazenil; GABA Modulators; Male; Memory; Mice; Mice, Inbred BALB C; Time Factors

2001
Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; DNA, Complementary; Female; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Humans; Imidazoles; Isoleucine; Ligands; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Protein Binding; Protein Structure, Tertiary; Protein Subunits; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Fusion Proteins; Sequence Alignment; Structure-Activity Relationship; Threonine; Transfection; Xenopus laevis; Zolpidem

2001
Modification of the effects of benzodiazepines on the exploratory behaviors of mice on a hole-board by diabetes.
    Japanese journal of pharmacology, 2001, Volume: 86, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Carbolines; Convulsants; Diabetes Mellitus, Experimental; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Injections, Intraperitoneal; Male; Mice; Mice, Inbred ICR

2001
The effects of flumazenil, Ro 154513 and beta-CCM on the behaviour of control and stressed mice in the staircase test.
    Journal of psychopharmacology (Oxford, England), 2001, Volume: 15, Issue:3

    Topics: Animals; Arousal; Azides; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Escape Reaction; Exploratory Behavior; Fear; Flumazenil; Immobilization; Male; Mice; Mice, Inbred BALB C; Sleep Deprivation; Sleep, REM; Social Isolation; Stress, Psychological

2001
Negative GABA(A) modulators attenuate the discriminative stimulus effects of benzodiazepines and the neuroactive steroid pregnanolone in rhesus monkeys.
    Psychopharmacology, 2005, Volume: 181, Issue:4

    Topics: Animals; Benzodiazepines; Carbolines; Discrimination Learning; Dose-Response Relationship, Drug; Drug Interactions; Female; Flumazenil; Macaca mulatta; Male; Midazolam; Pregnanolone; Receptors, GABA-A; Serotonin Antagonists; Serotonin Receptor Agonists

2005
Abnormal benzodiazepine receptor function in the depressive-like behavior of diabetic mice.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 82, Issue:4

    Topics: Animals; Behavior, Animal; Carbolines; Depression; Diabetes Mellitus, Experimental; Flumazenil; gamma-Aminobutyric Acid; Hindlimb Suspension; Male; Mice; Mice, Inbred ICR; Motor Activity; Receptors, GABA-A

2005