flumazenil has been researched along with azides in 83 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 17 (20.48) | 18.7374 |
1990's | 42 (50.60) | 18.2507 |
2000's | 19 (22.89) | 29.6817 |
2010's | 4 (4.82) | 24.3611 |
2020's | 1 (1.20) | 2.80 |
Authors | Studies |
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Colker, RE; Domangue, KR; Hicks, LH; June, HL; June, PL; Lewis, MJ; Perry, LE | 1 |
Gibert-Rahola, J; Maldonado, R; Micó, JA; Valverde, O | 1 |
Jackson, HC; Nutt, DJ | 1 |
Mehta, AK; Mhatre, M; Ticku, MK | 2 |
Inoue, O; Itoh, T; Kobayashi, K; Suhara, T; Suzuki, K; Tateno, Y | 1 |
Forster, MJ; Lal, H; Prather, PL | 1 |
Bosman, DK; Chamuleau, RA; de Haan, JG; Maas, MA; van den Buijs, CA | 1 |
Jones, EA | 1 |
Druml, W; Ferenci, P; Püspök, A; Steindl, P | 1 |
Bottlaender, M; Brouillet, E; Chavoix, C; Dodd, RH; Fournier, D; Hantraye, P; Khalili-Varasteh, M; Mazière, M | 1 |
Inoue, O; Itoh, T; Långström, B; Suhara, T; Tsukada, H; Yamasaki, T; Yonezawa, H | 1 |
Engel, JA; Söderpalm, B | 1 |
Budhram, P; Deacon, RM; Gardner, CR; Thomson, TA | 1 |
Koob, GF; Schreiber, JF; Weinger, MB | 1 |
Wettstein, JG | 1 |
Basile, AS; Gammal, SH; Geller, D; Jones, EA; Skolnick, P | 1 |
Alkana, RL; Finn, DA; Jones, BL; Kobayashi, LS; Syapin, PJ | 1 |
Borden, LA; Gibbs, TT | 1 |
Kulkarni, SK; Ticku, MK | 1 |
Becker, HC | 1 |
Mehta, AK; Ticku, MK | 1 |
Haefely, W | 1 |
Bishop, BE; Laverty, R | 1 |
Becker, HC; Hale, RL | 1 |
Biggio, G; Corda, MG; Giorgi, O; Longoni, B | 1 |
Mhatre, M; Ticku, MK | 1 |
Haraguchi, M; Sadeghi, KG; Samson, HH; Tolliver, GA | 1 |
Lister, RG | 1 |
Biggio, G; Corda, MG; Fernández, A; Giorgi, O | 1 |
Moody, EJ; Skolnick, P | 1 |
Bonetti, EP; Burkard, WP; Gabl, M; Hunkeler, W; Lorez, HP; Martin, JR; Moehler, H; Osterrieder, W; Pieri, L; Polc, P | 1 |
Crawley, JN; Glowa, JR; Paul, SM; Schwartz, RD; Skolnick, P; Suzdak, PD | 1 |
Kameyama, T; Nabeshima, T; Tohyama, K | 1 |
Slangen, JL; Woudenberg, F | 1 |
Hiltunen, AJ; Järbe, TU | 1 |
Iwasaki, T; Nakagawa, Y | 1 |
Pokk, P; Zharkovsky, A | 2 |
Miczek, KA; Tornatzky, W; Weerts, EM | 1 |
Hughes, RW; June, HL; Lewis, MJ; Spurlock, HL | 1 |
June, HL; Lewis, MJ | 1 |
Gardner, CR; Pringle, AK; Walker, RJ | 1 |
Andrews, N; File, SE | 1 |
Hu, XJ; Ticku, MK | 1 |
Langeland, BT; McKinley-McKee, JS | 1 |
Basile, AS; Jones, EA; Skolnich, P; Yurdaydin, C | 1 |
Gillard, NP; McKernan, RM; Quirk, K; Ragan, CI; Whiting, PJ | 1 |
Breese, GR; Criswell, HE | 1 |
Khan, RM; Soliman, MR | 1 |
Karim, KH; Najim, RA | 1 |
Barber, DJ; Cooper, SJ | 1 |
Mehta, AK; Shank, RP | 1 |
Inoue, O; Långström, B; Nakanishi, S; Nishiyama, S; Onoe, H; Tsukada, H; Watanabe, Y | 1 |
France, CP; Gerak, LR | 2 |
Akwa, Y; Britton, KT; Brot, MD; Koob, GF; Purdy, RH | 1 |
Benke, D; Michel, C; Mohler, H | 1 |
Cason, CR; Cheatham, G; Cook, JM; Gan, T; June, HL; Lui, R | 1 |
Boileau, AJ; Czajkowski, C; Kucken, AM; Teissére, JA; Wagner, DA; Ward, PR | 1 |
Atack, JR; Bristow, L; Brown, N; Carling, RW; Castro, JL; Cook, G; Dawson, GR; Farrar, S; Ferris, P; Garrett, L; Howell, O; Macaulay, A; Marshall, G; McKernan, RM; Moore, KW; Myers, J; Ragan, CI; Reynolds, DS; Rosahl, TW; Street, LJ; Sur, C; Wafford, KA; Whiting, PJ | 1 |
Firestone, LL; Homanics, GE; Quinlan, JJ | 1 |
France, CP; Gerak, LR; Lelas, S | 1 |
Bromidge, FA; Casula, MA; Hadingham, KL; Martin, K; Maubach, K; Pillai, GV; Seabrook, GR; Whiting, PJ; Wingrove, PB | 1 |
Paz, L; Peter, Y; Pick, CG; Weizman, R | 1 |
Cook, JM; DeLorey, TM; He, X; Lameh, J; Lin, RC; Loew, GH; McBrady, B | 1 |
Al-Mulla Hummadi, YM; Farjou, IB; Najim, RA | 1 |
Pokk, P; Väli, M | 1 |
Atack, J; Banks, G; Kelly, MD; Maubach, KA; Seabrook, GR; Smith, A; Whiting, PW; Wingrove, P | 1 |
Brooks, DJ; Cunningham, VJ; Feeney, A; Hirani, E; Hume, SP; Lingford-Hughes, A; Nutt, DJ; Osman, S; Pike, VW | 1 |
Gatch, MB; Jung, ME; Lal, H; Wallis, CJ | 1 |
Foster, AC; Grigoriadis, DE; Gross, RS; Petroski, RE; Sullivan, SK; Verge, G | 1 |
Atack, JR; Cook, SM; McKernan, RM; Pym, LJ; Rosahl, T | 1 |
Ahboucha, S; Butterworth, RF; Coyne, L; Halliwell, RF; Hirakawa, R | 1 |
Hirano, S; Kamei, J; Miyata, S | 1 |
Hanchar, HJ; Olsen, RW; Wallner, M | 1 |
France, CP; Gerak, LR; McMahon, LR | 1 |
Grant, KA; Helms, CM; Rogers, LS | 1 |
Hellsten, KS; Hyde, TM; Kleinman, JE; Korpi, ER; Maksimow, A; Särkioja, T; Sinkkonen, ST; Uusi-Oukari, M | 1 |
Abe, K; Hosoi, R; Inoue, O; Momosaki, S | 1 |
Banks, ML; Shelton, KL; Tracy, ME | 1 |
Andersson, M; Bölte, S; Borg, J; Cash, D; Farde, L; Gee, A; Halldin, C; Higgins, K; Horder, J; Howes, OD; Lingford-Hughes, A; Lundberg, J; Mendez, MA; Mick, I; Murphy, DG; Nutt, DJ; Selvaraj, S; Sementa, T; Singh, N; Spain, D; Tangen, Ä; Turkheimer, F; Veronese, M | 1 |
Benkherouf, AY; Kortesniemi, M; Laaksonen, O; Logrén, N; Salo-Ahen, OMH; Soini, SL; Somborac, T; Uusi-Oukari, M; Yang, B | 1 |
1 review(s) available for flumazenil and azides
Article | Year |
---|---|
Do benzodiazepine ligands contribute to hepatic encephalopathy?
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Disease Models, Animal; Flumazenil; GABA-A Receptor Antagonists; Hepatic Encephalopathy; Humans; Ligands; Receptors, GABA-A | 1993 |
82 other study(ies) available for flumazenil and azides
Article | Year |
---|---|
Ethanol self-administration in deprived rats: effects of Ro15-4513 alone, and in combination with flumazenil (Ro15-1788).
Topics: Alcohol Drinking; Animals; Azides; Benzodiazepines; Brain; Flumazenil; Male; Motivation; Rats; Rats, Inbred Strains; Receptors, GABA-A; Self Administration; Taste | 1992 |
Changes in benzodiazepine-receptor activity modify morphine withdrawal syndrome in mice.
Topics: Animals; Azides; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Flumazenil; Flunitrazepam; Male; Mice; Morphine; Receptors, GABA-A; Substance Withdrawal Syndrome | 1992 |
Effects of benzodiazepine receptor inverse agonists on locomotor activity and exploration in mice.
Topics: Animals; Azepines; Azides; Benzodiazepines; Benzodiazepinones; Exploratory Behavior; Flumazenil; Male; Mice; Motor Activity; Receptors, GABA-A | 1992 |
Modulation of GABAergic transmission by ethanol.
Topics: Animals; Anticonvulsants; Azides; Benzodiazepines; Brain Chemistry; Ethanol; Female; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Mice; Mice, Inbred C57BL; Pentylenetetrazole; Rats; Rats, Inbred Strains; RNA, Messenger; Seizures; Synaptic Transmission | 1992 |
In vivo binding of [11C]Ro15-4513 in human brain measured with PET.
Topics: Adult; Azides; Benzodiazepines; Brain; Flumazenil; Humans; Ligands; Male; Tomography, Emission-Computed | 1992 |
Learning and memory-enhancing effects of Ro 15-4513: a comparison with flumazenil.
Topics: Amnesia; Animals; Avoidance Learning; Azides; Benzodiazepines; Discrimination Learning; Flumazenil; Learning; Memory; Mice; Mice, Inbred ICR; Scopolamine; Stimulation, Chemical | 1992 |
The effects of benzodiazepine-receptor antagonists and partial inverse agonists on acute hepatic encephalopathy in the rat.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Electroencephalography; Evoked Potentials, Visual; Flumazenil; Hepatic Encephalopathy; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1991 |
Benzodiazepine receptor ligands and hepatic encephalopathy: further unfolding of the GABA story.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Brain; Central Nervous System; Flumazenil; gamma-Aminobutyric Acid; Hepatic Encephalopathy; Humans; Ligands; Neurons; Receptors, GABA-A; Synaptic Transmission | 1991 |
Beneficial effect of pharmacological modulation of the GABAA-benzodiazepine receptor on hepatic encephalopathy in the rat: comparison with uremic encephalopathy.
Topics: Animals; Azides; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Coma; Flumazenil; Hepatic Encephalopathy; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Uremia | 1991 |
In vivo bidirectional modulatory effect of benzodiazepine receptor ligands on GABAergic transmission evaluated by positron emission tomography in non-human primates.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Carbolines; Cerebral Cortex; Diazepam; Electroencephalography; Flumazenil; gamma-Aminobutyric Acid; Ligands; Male; Papio; Pentylenetetrazole; Receptors, GABA-A; Seizures; Synaptic Transmission; Tomography, Emission-Computed | 1991 |
Differences of distribution between RO 15-1788 and RO 15-4513 in vivo.
Topics: Animals; Azides; Benzodiazepines; Brain; Flumazenil; Male; Mice | 1991 |
Involvement of the GABAA/benzodiazepine chloride ionophore receptor complex in the 5,7-DHT Induced anticonflict effect.
Topics: 5,7-Dihydroxytryptamine; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Bicuculline; Diazepam; Drinking Behavior; Electroshock; Flumazenil; Hippocampus; Injections, Intraventricular; Limbic System; Male; Picrotoxin; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin | 1991 |
Differential interactions of Ro 15-4513 with benzodiazepines, ethanol and pentobarbital.
Topics: Anesthesia; Animals; Anti-Anxiety Agents; Azides; Behavior, Animal; Benzodiazepines; Diazepam; Drug Interactions; Ethanol; Female; Flumazenil; Male; Muscle Contraction; Muscles; Pentobarbital; Rats; Rats, Inbred Strains; Urethane; Vocalization, Animal | 1990 |
Effects of two benzodiazepine inverse agonists, RO 15-4513 and FG 7142, on recovery from pentobarbital and halothane anesthesia in the rat.
Topics: Anesthesia Recovery Period; Animals; Azides; Benzodiazepines; Carbolines; Flumazenil; Halothane; Male; Pentobarbital; Random Allocation; Rats; Rats, Inbred Strains; Reflex | 1990 |
Unusual behavioral profile of alprazolam in squirrel monkeys.
Topics: Alprazolam; Animals; Azides; Benzodiazepines; Dose-Response Relationship, Drug; Electroshock; Flumazenil; Injections, Intravenous; Lorazepam; Male; Psychomotor Performance; Saimiri | 1990 |
Reversal of the behavioral and electrophysiological abnormalities of an animal model of hepatic encephalopathy by benzodiazepine receptor ligands.
Topics: Animals; Azides; Benzodiazepines; Disease Models, Animal; Electrophysiology; Evoked Potentials, Visual; Flumazenil; Hepatic Encephalopathy; Ligands; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1990 |
Interactions between benzodiazepine antagonists, inverse agonists, and acute behavioral effects of ethanol in mice.
Topics: Animals; Azides; Benzodiazepines; Dose-Response Relationship, Drug; Ethanol; Flumazenil; GABA-A Receptor Antagonists; Hypothermia; Male; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Motor Activity; Receptors, GABA-A; Reflex | 1990 |
Flunitrazepam photoaffinity labeling of the GABA(A) receptor reduces inhibition of [3H]Ro15-4513 binding by GABA.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Brain; Chick Embryo; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Membranes; Photochemistry; Receptors, GABA-A | 1990 |
Chronic benzodiazepine antagonist treatment and its withdrawal upregulates components of GABA-benzodiazepine receptor ionophore complex in cerebral cortex of rat.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Convulsants; Flumazenil; Flunitrazepam; gamma-Aminobutyric Acid; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reference Values; Up-Regulation | 1990 |
Effects of the imidazobenzodiazepine RO15-4513 on the stimulant and depressant actions of ethanol on spontaneous locomotor activity.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Chlorides; Ethanol; Flumazenil; Ion Channels; Male; Mice; Mice, Inbred C3H; Motor Activity; Receptors, GABA-A | 1988 |
Ethanol potentiation of GABAergic transmission in cultured spinal cord neurons involves gamma-aminobutyric acidA-gated chloride channels.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Cells, Cultured; Chlorine; Ethanol; Female; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Ion Channels; Male; Mice; Mice, Inbred C57BL; Neurons; Radioisotopes; Spinal Cord | 1988 |
Partial agonists of the benzodiazepine receptor: from animal data to results in patients.
Topics: Affinity Labels; Allosteric Site; Animals; Azides; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Chlorides; Clonazepam; Diazepam; Drug Interactions; Ethanol; Flumazenil; Flurazepam; Humans; Ion Channels; Ligands; Models, Neurological; Neurons; Receptors, GABA-A | 1988 |
Dose-dependent reduction by Ro 15-4513 in mice of the effects of ethanol and some other general depressant drugs.
Topics: Anesthetics; Animals; Azides; Benzodiazepines; Central Nervous System Depressants; Dose-Response Relationship, Drug; Ethanol; Flumazenil; Mice; Sleep; Time Factors | 1989 |
Ethanol-induced locomotor stimulation in C57BL/6 mice following RO15-4513 administration.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Ethanol; Flumazenil; Male; Mice; Mice, Inbred C57BL; Motor Activity | 1989 |
Ro 15-4513, a partial inverse agonist for benzodiazepine recognition sites, has proconflict and proconvulsant effects in the rat.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Conflict, Psychological; Convulsants; Flumazenil; Isoniazid; Male; Pentobarbital; Punishment; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
Chronic ethanol treatment selectively increases the binding of inverse agonists for benzodiazepine binding sites in cultured spinal cord neurons.
Topics: Alcoholism; Animals; Azides; Benzodiazepines; Cells, Cultured; Female; Flumazenil; Flunitrazepam; Male; Mice; Mice, Inbred C57BL; Neurons; Receptors, GABA-A; Spinal Cord | 1989 |
Antagonism of ethanol-reinforced behavior by the benzodiazepine inverse agonists Ro15-4513 and FG 7142: relation to sucrose reinforcement.
Topics: Animals; Azides; Behavior, Animal; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Flumazenil; Male; Rats; Receptors, GABA-A; Reinforcement, Psychology; Self Administration; Sucrose | 1989 |
Reversal of the intrinsic effects of Ro 15-4513 on exploratory behavior by two benzodiazepine receptor antagonists.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Exploratory Behavior; Flumazenil; Male; Mice; Motor Activity; Receptors, GABA-A | 1987 |
The abstinence syndrome in diazepam-dependent cats is precipitated by Ro 15-1788 and Ro 15-4513 but not by the benzodiazepine receptor antagonist ZK 93426.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Cats; Diazepam; Flumazenil; Receptors, GABA-A; Substance Withdrawal Syndrome | 1988 |
The imidazobenzodiazepine Ro 15-4513 antagonizes methoxyflurane anesthesia.
Topics: Anesthesia, General; Animals; Azides; Benzodiazepines; Carbolines; Flumazenil; Male; Methoxyflurane; Mice; Receptors, GABA-A; Sleep | 1988 |
Chronic ethanol administration increases the binding of the benzodiazepine inverse agonist and alcohol antagonist [3H]RO15-4513 in rat brain.
Topics: Acoustic Stimulation; Animals; Azides; Benzodiazepines; Body Temperature; Brain Chemistry; Diazepam; Ethanol; Flumazenil; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures | 1988 |
Ro 15-4513: partial inverse agonism at the BZR and interaction with ethanol.
Topics: Animals; Azides; Behavior, Animal; Benzodiazepines; Brain; Brain Chemistry; Cats; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Ethanol; Flumazenil; Meta-Analysis as Topic; Mice; Phenobarbital; Rats; Receptors, GABA-A | 1988 |
A selective imidazobenzodiazepine antagonist of ethanol in the rat.
Topics: Animals; Anxiety; Azides; Benzodiazepines; Chlorides; Ethanol; Flumazenil; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes | 1986 |
Reversal of alcohol-induced amnesia by the benzodiazepine inverse agonist Ro 15-4513.
Topics: Amnesia; Animals; Avoidance Learning; Azides; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Ethanol; Flumazenil; Male; Mice; Time Factors | 1988 |
Ethanol suppression of schedule-controlled responding: interactions with Ro 15-4513, Ro 15-1788 and CGS 8216.
Topics: Alcohol Deterrents; Animals; Azides; Behavior, Animal; Benzodiazepines; Drug Interactions; Ethanol; Flumazenil; Male; Pyrazoles; Rats; Rats, Inbred Strains | 1988 |
Effects of Ro 15-4513, alone or in combination with ethanol, Ro 15-1788, diazepam, and pentobarbital on instrumental behaviors of rats.
Topics: Animals; Azides; Behavior, Animal; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Female; Flumazenil; Pentobarbital; Rats; Rats, Inbred Strains; Time Factors | 1988 |
Involvement of benzodiazepine/GABA-A receptor complex in ethanol-induced state-dependent learning in rats.
Topics: Animals; Avoidance Learning; Azides; Benzodiazepines; Bicuculline; Diazepam; Ethanol; Evaluation Studies as Topic; Flumazenil; Male; Muscimol; Picrotoxin; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A | 1995 |
The effects of drugs acting at GABA-benzodiazepine-barbiturate receptor complex on the behaviour of sleep-deprived mice.
Topics: Analysis of Variance; Animals; Azides; Behavior, Animal; Benzodiazepines; Convulsants; Diazepam; Flumazenil; Male; Mice; Receptors, GABA-A; Sleep Deprivation | 1995 |
"Anxiolytic" and "anxiogenic" benzodiazepines and beta-carbolines: effects on aggressive and social behavior in rats and squirrel monkeys.
Topics: Aggression; Animals; Anti-Anxiety Agents; Anxiety; Azides; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Motor Activity; Rats; Saimiri; Social Behavior; Species Specificity | 1993 |
Ethanol self-administration in freely feeding and drinking rats: effects of Ro15-4513 alone, and in combination with Ro15-1788 (flumazenil).
Topics: Alcohol Drinking; Animals; Azides; Benzodiazepines; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Flumazenil; GABA-A Receptor Agonists; Male; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology | 1994 |
Interactions of Ro15-4513, Ro15-1788 (flumazenil) and ethanol on measures of exploration and locomotion in rats.
Topics: Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Dose-Response Relationship, Drug; Environment; Ethanol; Exploratory Behavior; Flumazenil; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 1994 |
Different functional effect of Ro 15-4513 and Ro 19-4603 on synaptic responses of Purkinje cells in the rat cerebellar slice.
Topics: Animals; Azepines; Azides; Benzodiazepines; Cerebellum; Diazepam; Electrophysiology; Flumazenil; In Vitro Techniques; Male; Neural Inhibition; Purkinje Cells; Rats; Rats, Wistar; Receptors, GABA-A; Synapses | 1994 |
F 2692: flumazenil-reversible anxiolytic effects but inactive on [3H]-Ro 15-4513 binding.
Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding, Competitive; Carbolines; Cerebellum; Diazepam; Flumazenil; GABA-A Receptor Antagonists; In Vitro Techniques; Interpersonal Relations; Male; Membranes; Motor Activity; Pyridazines; Rats; Receptors, GABA-A | 1994 |
Development pattern of the GABAA-benzodiazepine receptor ionophore complex in primary cultures of cortical neurons.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Cells, Cultured; Cerebral Cortex; Chlorides; Flumazenil; Flunitrazepam; Mice; Mice, Inbred C57BL; Muscimol; Neurons; Receptors, GABA-A | 1994 |
Inhibition and inactivation of horse liver alcohol dehydrogenase with the imidazobenzodiazepine Ro 15-4513.
Topics: Affinity Labels; Alcohol Dehydrogenase; Animals; Azides; Benzodiazepines; Flumazenil; Horses; Hydrogen-Ion Concentration; Kinetics; Liver; Mathematics; Molecular Structure; NAD | 1994 |
Model of subunit composition of gamma-aminobutyric acid A receptor subtypes expressed in rat cerebellum with respect to their alpha and gamma/delta subunits.
Topics: Animals; Azides; Base Sequence; Benzodiazepines; Cerebellum; Escherichia coli; Flumazenil; Molecular Sequence Data; Muscimol; Precipitin Tests; Protein Conformation; Rats; Receptors, GABA-A; Recombinant Proteins | 1994 |
Similar effects of ethanol and flumazenil on acquisition of a shuttle-box avoidance response during withdrawal from chronic ethanol treatment.
Topics: Animals; Avoidance Learning; Azides; Benzodiazepines; Chlordiazepoxide; Conflict, Psychological; Dose-Response Relationship, Drug; Ethanol; Flumazenil; Male; Postural Balance; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome | 1993 |
Effects of benzodiazepine agonist, antagonist and inverse agonist on ethanol-induced changes in beta-endorphin levels in specific rat brain regions.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; beta-Endorphin; Brain Chemistry; Cerebral Cortex; Diazepam; Ethanol; Flumazenil; Hippocampus; Hypothalamus; Male; Rats; Rats, Sprague-Dawley | 1993 |
Prevention of ethanol-induced gastric damage by the imidazobenzodiazepines Ro 15-4513 and Ro 15-3505 in rats.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Ethanol; Flumazenil; Male; Rats; Rats, Wistar; Stomach Ulcer | 1993 |
The benzodiazepine receptor partial agonist bretazenil and the partial inverse agonist Ro 15-4513: effects on salt preference and aversion in the rat.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Flumazenil; Food Preferences; Male; Rats; Receptors, GABA-A; Saline Solution, Hypertonic; Sodium Chloride; Taste | 1993 |
Characterization of a benzodiazepine receptor site with exceptionally high affinity for Ro 15-4513 in the rat CNS.
Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Central Nervous System; Cerebellum; Chlorides; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; GABA Modulators; Hippocampus; Imidazoles; Male; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Spinal Cord; Tritium | 1995 |
A subclass of GABAA/benzodiazepine receptor exclusively localized in the limbic system.
Topics: Affinity Labels; Animals; Autoradiography; Azides; Benzodiazepines; Carbon Radioisotopes; Female; Flumazenil; GABA Modulators; Image Processing, Computer-Assisted; Isotope Labeling; Limbic System; Macaca mulatta; Receptors, GABA-A; Tomography, Emission-Computed | 1996 |
Discriminative stimulus effects of flumazenil in rhesus monkeys treated chronically with chlordiazepoxide.
Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Azides; Benzodiazepines; Chlordiazepoxide; Discrimination Learning; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Antagonists; Macaca mulatta; Pharmaceutical Vehicles; Time Factors | 1997 |
The anxiolytic-like effects of the neurosteroid allopregnanolone: interactions with GABA(A) receptors.
Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Anxiety; Azides; Behavior, Animal; Benzodiazepines; Binding Sites; Chloride Channels; Conflict, Psychological; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Female; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Organophosphorus Compounds; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A | 1997 |
The effects of flumazenil, Ro 15-4513 and beta-CCM on the behaviour of control and stressed mice in the plus-maze test.
Topics: Animals; Anxiety; Azides; Behavior, Animal; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; Ligands; Male; Mice; Stress, Psychological | 1997 |
GABA(A) receptors containing the alpha4-subunit: prevalence, distribution, pharmacology, and subunit architecture in situ.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Brain; Cell Membrane; Cerebellum; Diazepam; Flumazenil; Immunohistochemistry; Immunosorbent Techniques; Macromolecular Substances; Male; Muscimol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Recombinant Proteins | 1997 |
GABAA-benzodiazepine receptors in the striatum are involved in the sedation produced by a moderate, but not an intoxicating ethanol dose in outbred Wistar rats.
Topics: Alcoholic Intoxication; Analysis of Variance; Animals; Azides; Benzodiazepines; Corpus Striatum; Ethanol; Flumazenil; GABA Agents; GABA-A Receptor Agonists; Hypnotics and Sedatives; Male; Oocytes; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Xenopus | 1998 |
Discriminative stimulus effects of flumazenil in untreated and in diazepam-treated rhesus monkeys.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Diazepam; Discrimination Learning; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Modulators; Macaca mulatta; Male; Receptors, GABA-A | 1999 |
Identification of benzodiazepine binding site residues in the gamma2 subunit of the gamma-aminobutyric acid(A) receptor.
Topics: Amino Acid Sequence; Azides; Benzodiazepines; Binding Sites; Cells, Cultured; Cloning, Molecular; Flumazenil; Flunitrazepam; Humans; Molecular Sequence Data; Point Mutation; Receptors, GABA-A; Recombinant Fusion Proteins; Sequence Homology, Amino Acid | 2000 |
Sedative but not anxiolytic properties of benzodiazepines are mediated by the GABA(A) receptor alpha1 subtype.
Topics: Allosteric Site; Animals; Anti-Anxiety Agents; Anticonvulsants; Azides; Benzodiazepines; Binding, Competitive; Brain; Cell Line; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Fluorobenzenes; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Ligands; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Motor Activity; Patch-Clamp Techniques; Receptors, GABA-A; Reflex, Startle; Triazoles | 2000 |
Mice lacking the long splice variant of the gamma 2 subunit of the GABA(A) receptor are more sensitive to benzodiazepines.
Topics: Alternative Splicing; Animals; Azides; Benzodiazepines; Brain; Carbolines; Diazepam; Drug Resistance; Female; Flumazenil; GABA Modulators; Genetic Variation; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Midazolam; Pyridines; Receptors, GABA-A; Sleep; Zolpidem | 2000 |
Antagonism of the discriminative stimulus effects of positive gamma-aminobutyric acid(A) modulators in rhesus monkeys discriminating midazolam.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Diazepam; Discrimination Learning; Drug Antagonism; Female; Flumazenil; GABA Modulators; Macaca mulatta; Male; Midazolam; Receptors, GABA-A | 2000 |
Identification of amino acid residues responsible for the alpha5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABA(A) receptor.
Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Anti-Anxiety Agents; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; DNA, Complementary; Female; Flumazenil; Flunitrazepam; GABA-A Receptor Agonists; Humans; Imidazoles; Isoleucine; Ligands; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Protein Binding; Protein Structure, Tertiary; Protein Subunits; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Fusion Proteins; Sequence Alignment; Structure-Activity Relationship; Threonine; Transfection; Xenopus laevis; Zolpidem | 2001 |
Mice performance on the staircase test following acute ethanol administration.
Topics: Animals; Azides; Benzodiazepines; Central Nervous System Depressants; Diazepam; Dose-Response Relationship, Drug; Ethanol; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred ICR; Psychomotor Performance | 2001 |
Influence of benzodiazepine binding site ligands on fear-conditioned contextual memory.
Topics: Animals; Azides; Benzodiazepines; Binding Sites; Binding, Competitive; Carbolines; Conditioning, Psychological; Convulsants; Fear; Flumazenil; GABA Antagonists; GABA Modulators; Imidazoles; Ligands; Male; Memory; Mice; Mice, Inbred C57BL; Motor Activity; N-Methylscopolamine; Piperazines; Quinolines; Receptors, GABA-A; Scopolamine; Silanes; Tritium | 2001 |
Benzodiazepines protect against ethanol-induced gastric mucosal damage in vitro.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Central Nervous System Depressants; Clonazepam; Ethanol; Flumazenil; GABA Modulators; Gastric Mucosa; In Vitro Techniques; Male; Rats; Rats, Wistar; Stomach Ulcer | 2001 |
The effects of flumazenil, Ro 154513 and beta-CCM on the behaviour of control and stressed mice in the staircase test.
Topics: Animals; Arousal; Azides; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Escape Reaction; Exploratory Behavior; Fear; Flumazenil; Immobilization; Male; Mice; Mice, Inbred BALB C; Sleep Deprivation; Sleep, REM; Social Isolation; Stress, Psychological | 2001 |
Role of the histidine residue at position 105 in the human alpha 5 containing GABA(A) receptor on the affinity and efficacy of benzodiazepine site ligands.
Topics: Anticonvulsants; Arginine; Azides; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Cell Line; Cells, Cultured; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Histidine; Humans; Ligands; Mutation; Protein Subunits; Receptors, GABA-A | 2002 |
Imaging the GABA-benzodiazepine receptor subtype containing the alpha5-subunit in vivo with [11C]Ro15 4513 positron emission tomography.
Topics: Animals; Azides; Benzodiazepines; Binding, Competitive; Carbon Radioisotopes; Cerebellum; Cerebral Cortex; Flumazenil; Hippocampus; Humans; Kinetics; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Tissue Distribution; Tomography, Emission-Computed | 2002 |
Effects of GABA(A) compounds on mCPP drug discrimination in rats.
Topics: Alprazolam; Animals; Azides; Benzodiazepines; Bicuculline; Conditioning, Operant; Discrimination, Psychological; Flumazenil; GABA Agonists; GABA Antagonists; Male; Pentylenetetrazole; Piperazines; Rats; Rats, Long-Evans; Receptors, GABA-A | 2002 |
Characterization of the interaction of indiplon, a novel pyrazolopyrimidine sedative-hypnotic, with the GABAA receptor.
Topics: Acetamides; Animals; Azides; Benzodiazepines; Binding Sites; Brain; Cell Membrane; Cerebellum; Cerebral Cortex; Chloride Channels; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Kinetics; Male; Pyridines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Thiophenes; Triazolam; Tritium; Zolpidem | 2004 |
Selective labelling of diazepam-insensitive GABAA receptors in vivo using [3H]Ro 15-4513.
Topics: Animals; Azides; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Cerebellum; Flumazenil; Humans; Isotope Labeling; Ligands; Lorazepam; Male; Mice; Mice, Transgenic; Prosencephalon; Receptors, GABA-A; Receptors, GABA-B; Tritium | 2005 |
An interaction between benzodiazepines and neuroactive steroids at GABA A receptors in cultured hippocampal neurons.
Topics: Affinity Labels; Allosteric Regulation; Animals; Azides; Benzodiazepines; Cells, Cultured; Chloride Channels; Dose-Response Relationship, Drug; Drug Interactions; Female; Flumazenil; GABA Modulators; Hepatic Encephalopathy; Hippocampus; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Pregnanolone; Rats; Rats, Wistar; Receptors, GABA-A; Synaptic Transmission | 2006 |
Involvement of diazepam-insensitive benzodiazepine receptors in the suppression of DOI-induced head-twitch responses in diabetic mice.
Topics: Amphetamines; Animals; Azides; Behavior, Animal; Benzodiazepines; Bicuculline; Diabetes Mellitus, Experimental; Diazepam; Flumazenil; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Male; Mice; Mice, Inbred ICR; Receptors, GABA-A; Serotonin Receptor Agonists | 2006 |
Low-dose alcohol actions on alpha4beta3delta GABAA receptors are reversed by the behavioral alcohol antagonist Ro15-4513.
Topics: Animals; Azides; Benzodiazepines; Carbolines; Electrophysiology; Esters; Ethanol; Flumazenil; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Molecular Structure; Mutation; Oocytes; Patch-Clamp Techniques; Protein Subunits; Receptors, GABA-A; Xenopus laevis | 2006 |
Efficacy and the discriminative stimulus effects of negative GABAA modulators, or inverse agonists, in diazepam-treated rhesus monkeys.
Topics: Animals; Azides; Benzodiazepines; Conditioning, Operant; Cues; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Female; Flumazenil; GABA Agonists; GABA Modulators; Hypnotics and Sedatives; Macaca mulatta; Male; Pentobarbital; Pregnanolone; Receptors, GABA-A | 2006 |
Antagonism of the ethanol-like discriminative stimulus effects of ethanol, pentobarbital, and midazolam in cynomolgus monkeys reveals involvement of specific GABA(A) receptor subtypes.
Topics: Animals; Azides; Benzodiazepines; Discrimination Learning; Dose-Response Relationship, Drug; Ethanol; Female; Flumazenil; Macaca fascicularis; Male; Midazolam; Pentobarbital; Protein Subunits; Receptors, GABA-A | 2009 |
Human locus coeruleus neurons express the GABA(A) receptor gamma2 subunit gene and produce benzodiazepine binding.
Topics: Adult; Autoradiography; Azides; Benzodiazepines; Female; Flumazenil; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Humans; Locus Coeruleus; Male; Melanins; Neurons; Pyridines; Radioligand Assay; Receptors, GABA-A; Tyrosine 3-Monooxygenase; Zolpidem | 2010 |
Remarkable selectivity of the in vivo binding of [3H]Ro15-4513 to α5 subtype of benzodiazepine receptor in the living mouse brain.
Topics: Affinity Labels; Animals; Azides; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; Male; Mice; Protein Subunits; Receptors, GABA-A; Tritium | 2010 |
Negative allosteric modulation of GABAA receptors inhibits facilitation of brain stimulation reward by drugs of abuse in C57BL6/J mice.
Topics: Allosteric Regulation; Animals; Azides; Benzodiazepines; Brain; Diazepam; Dose-Response Relationship, Drug; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; Illicit Drugs; Male; Mice; Mice, Inbred C57BL; Microdialysis; Receptors, GABA-A; Reward; Self Stimulation | 2016 |
GABA
Topics: Adult; Animals; Autism Spectrum Disorder; Azides; Behavior; Benzodiazepines; Carbon Radioisotopes; Case-Control Studies; Disease Models, Animal; Female; Flumazenil; Gray Matter; Humans; Male; Mice; Motion Perception; Positron-Emission Tomography; Protein Subunits; Receptors, GABA-A; Task Performance and Analysis | 2018 |
Hops compounds modulatory effects and 6-prenylnaringenin dual mode of action on GABA
Topics: Animals; Azides; Benzodiazepines; Binding, Competitive; Cyclohexenes; Dose-Response Relationship, Drug; Flavonoids; Flumazenil; Flunitrazepam; GABA Modulators; Humulus; Male; Molecular Docking Simulation; Plant Extracts; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Terpenes | 2020 |