flumazenil and alfentanil

flumazenil has been researched along with alfentanil in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19905 (27.78)18.7374
1990's5 (27.78)18.2507
2000's4 (22.22)29.6817
2010's4 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Boysen, K; Crawford, ME; Krintel, JJ; Sonne, NM; Valentin, N; Wegmann, F1
Harrop-Griffiths, AW; Jewkes, DA; Watson, NA1
Andersen, P; Christiansen, C; Jarnvig, IL; Jørgensen, B; Skielboe, M; Weber, M1
Hartvig, P; Nilsson, A; Persson, MP2
Bovill, JG; Breimer, LT; Hennis, PJ; Spierdijk, J1
Hole, A; Nilsen, OG; Raeder, JC1
Hansen, PA; Jensen, AG; Lybecker, H; Møller, JT1
Blouin, RT; Conard, PF; Gross, JB; Häussler, J; Zandsberg, S1
Feng, J; Kendig, JJ1

Reviews

1 review(s) available for flumazenil and alfentanil

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

8 trial(s) available for flumazenil and alfentanil

ArticleYear
Recovery after total intravenous anaesthesia using combined midazolam/alfentanil infusion and reversal with flumazenil.
    Acta anaesthesiologica Scandinavica, 1991, Volume: 35, Issue:8

    Topics: Acoustic Stimulation; Adult; Alfentanil; Anesthesia Recovery Period; Anesthesia, Inhalation; Anesthesia, Intravenous; Blood Pressure; Female; Flumazenil; Glasgow Coma Scale; Heart Rate; Humans; Infusions, Intravenous; Male; Midazolam; Middle Aged; Nitrous Oxide; Patient Satisfaction; Reaction Time; Respiration

1991
Antagonism of diazepam sedation by flumazenil.
    British journal of anaesthesia, 1989, Volume: 63, Issue:5

    Topics: Aged; Aged, 80 and over; Alfentanil; Anesthesia, General; Carbon Dioxide; Diazepam; Double-Blind Method; Flumazenil; Humans; Middle Aged; Nitrous Oxide; Oxygen; Randomized Controlled Trials as Topic; Wakefulness

1989
Effects of flumazenil on post-operative recovery after total intravenous anesthesia with midazolam and alfentanil.
    European journal of anaesthesiology. Supplement, 1988, Volume: 2

    Topics: Alfentanil; Anesthesia Recovery Period; Anesthesia, Intravenous; Female; Fentanyl; Flumazenil; Humans; Hysterectomy; Midazolam; Postoperative Period; Receptors, GABA-A

1988
The efficacy of flumazenil versus physostigmine after midazolam-alfentanil anaesthesia in man.
    European journal of anaesthesiology. Supplement, 1988, Volume: 2

    Topics: Adult; Alfentanil; Anesthesia; Anesthesia Recovery Period; Double-Blind Method; Female; Fentanyl; Flumazenil; Humans; Male; Midazolam; Nitrous Oxide; Physostigmine; Random Allocation; Vecuronium Bromide

1988
Effects of the benzodiazepine antagonist flumazenil on postoperative performance following total intravenous anaesthesia with midazolam and alfentanil.
    Acta anaesthesiologica Scandinavica, 1988, Volume: 32, Issue:6

    Topics: Alfentanil; Anesthesia Recovery Period; Anesthesia, Intravenous; Cooperative Behavior; Female; Fentanyl; Flumazenil; Humans; Memory; Midazolam; Nitrous Oxide; Orientation; Postoperative Period; Thiopental

1988
Pharmacokinetics of midazolam and alfentanil in outpatient general anesthesia. A study with concomitant thiopentone, flumazenil or placebo administration.
    Acta anaesthesiologica Scandinavica, 1988, Volume: 32, Issue:6

    Topics: Adult; Alfentanil; Ambulatory Surgical Procedures; Anesthesia, General; Female; Fentanyl; Flumazenil; Humans; Midazolam; Middle Aged; Nitrous Oxide; Placebos; Preanesthetic Medication; Thiopental; Time Factors

1988
A random trial comparing recovery after midazolam-alfentanil anesthesia with and without reversal with flumazenil, and standardized neurolept anesthesia for major gynecologic surgery.
    Journal of clinical anesthesia, 1995, Volume: 7, Issue:1

    Topics: Adult; Aged; Alfentanil; Anesthesia Recovery Period; Anesthesia, Inhalation; Anesthesia, Intravenous; Anesthetics, Intravenous; Blood Pressure; Double-Blind Method; Female; Flumazenil; Genitalia, Female; Heart Rate; Humans; Midazolam; Middle Aged; Neuroleptanalgesia; Nitrous Oxide; Placebos; Respiration

1995
Effect of flumazenil on ventilatory drive during sedation with midazolam and alfentanil.
    Anesthesiology, 1996, Volume: 85, Issue:4

    Topics: Adult; Alfentanil; Analgesics, Opioid; Antidotes; Benzodiazepines; Carbon Dioxide; Conscious Sedation; Consciousness; Cross-Over Studies; Depression, Chemical; Double-Blind Method; Drug Interactions; Female; Flumazenil; Humans; Hypnotics and Sedatives; Hypoxia; Infusions, Intravenous; Male; Midazolam; Respiration

1996

Other Studies

9 other study(ies) available for flumazenil and alfentanil

ArticleYear
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Midazolam and flumazenil in the anaesthetic management of trigeminal nerve thermocoagulation.
    British journal of anaesthesia, 1990, Volume: 64, Issue:5

    Topics: Alfentanil; Blood Pressure; Electrocoagulation; Flicker Fusion; Flumazenil; Heart Rate; Humans; Midazolam; Middle Aged; Time Factors; Trigeminal Nerve; Trigeminal Neuralgia

1990
Synergistic interactions between midazolam and alfentanil in isolated neonatal rat spinal cord.
    British journal of anaesthesia, 1996, Volume: 77, Issue:3

    Topics: Alfentanil; Analgesics, Opioid; Animals; Bicuculline; Dose-Response Relationship, Drug; Drug Synergism; Evoked Potentials; Flumazenil; Hypnotics and Sedatives; Midazolam; Organ Culture Techniques; Rats; Rats, Sprague-Dawley; Spinal Cord

1996