flumazenil has been researched along with 2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one in 98 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 83 (84.69) | 18.7374 |
1990's | 13 (13.27) | 18.2507 |
2000's | 2 (2.04) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S | 1 |
Lucki, I; Rowan, GA | 1 |
Kucharik, RF; Lucki, I | 1 |
Morse, WH; Teeple, ES; Wettstein, JG | 1 |
Brain, PF; Pankaj, V | 1 |
Bianchi, M; Fumagalli, P; Mantegazza, P; Panerai, AE; Rovati, LC; Sacerdote, P | 1 |
Falk, JL; Lau, CE; Tang, M | 1 |
Dragunow, M | 1 |
Wettstein, JG | 1 |
Albertson, TE; Joy, RM | 1 |
Bizière, K; Fournier, M; Keane, P; Santucci, V; Worms, P | 1 |
Cooper, SJ; Estall, LB | 2 |
Green, S; Hodges, H | 1 |
Randall, JI; Rodgers, RJ | 2 |
Arbilla, S; Langer, SZ; Lista, A | 1 |
Rodgers, RJ; Waters, AJ | 1 |
File, SE | 3 |
Gerhardt, S; Liebman, JM | 1 |
File, SE; Pellow, S; Wilks, L | 1 |
Harris, C; Lal, H | 1 |
File, SE; Pellow, S | 8 |
Spealman, RD; Wettstein, JG | 2 |
Danchev, N | 1 |
Albertson, TE; Foulke, GE | 1 |
Treit, D | 1 |
Bassett, ML; Jones, EA; Martin, JV; Mendelson, WB; Mullen, KD | 1 |
De Deyn, PP; Macdonald, RL | 2 |
Braestrup, C; Petersen, EN; Scheel-Krüger, J | 1 |
Kempner, ES; Paul, SM; Schwartz, RD; Skolnick, P; Thomas, JW | 1 |
Caporali, MG; Gatta, F; Lucantoni, D; Massotti, M; Mele, L | 1 |
Barber, DJ; Cooper, SJ; Gilbert, DB; Moores, WR | 1 |
Ikonomidou, C; Klockgether, T; Schwarz, M; Sontag, KH; Turski, L | 1 |
Barber, DJ; Cooper, SJ; Jackson, A; Moores, WR | 1 |
Meiners, BA; Salama, AI | 1 |
De Vry, J; Slangen, JL | 1 |
Kulkarni, SK; Kunchandy, J | 1 |
Crawley, JN; Glowa, JR; Paul, SM; Schwartz, RD; Skolnick, P; Suzdak, PD | 1 |
Bender, AS; Hertz, L | 1 |
Berridge, KC; Schultz, CE; Treit, D | 1 |
Goldstein, JM; Malick, JB; Sutton, EB | 1 |
Martin, WR; McNicholas, LF | 1 |
Katzman, NJ; Shannon, HE | 1 |
Biziere, K; Calassi, R; Chambon, JP; Heaulme, M; Perio, A | 1 |
Sanger, DJ | 1 |
Boisse, NR; Guarino, JJ; Kruger, HS; Periana, RM; Samoriski, GM | 1 |
Albertson, TE; Walby, WF | 1 |
Cooper, SJ; Kirkham, TC | 1 |
Ascioti, C; De Sarro, GB; Libri, V; Nistico, G; Testa, R | 1 |
Iwasawa, H; Naito, H; Tonoue, T | 1 |
Griffiths, RR; Lamb, RJ | 1 |
Martin, WR; McNicholas, LF; Sloan, JW; Wala, E | 1 |
Slangen, JL; Woudenberg, F | 1 |
Cooper, SJ; Moores, WR | 1 |
Braestrup, C; Honoré, T; Jensen, LH; Kehr, W; Petersen, EN; Schmiechen, R; Schneider, H; Seidelmann, D; Stephens, DN | 1 |
Carney, JM; Nakamura, M | 2 |
Mendelson, WB | 1 |
Bernard, P; Cassidy, JP; Czernik, AJ; Petrack, B; Yokoyama, N | 1 |
Haefely, W | 2 |
Amato, M; Bizzi, A; Garattini, S; Ricci, MR; Veneroni, E | 1 |
Crawley, JN; Paul, SM; Skolnick, P | 1 |
Clemmitt, M; Rodgers, RJ | 1 |
Risley, EA; Williams, M | 1 |
Braestrup, C; Jensen, LH; Petersen, EN | 1 |
Gee, KW; Yamamura, HI | 1 |
File, SE; Lister, RG | 1 |
Paul, SM; Skolnick, P | 1 |
Robertson, HA | 1 |
Black, DA; Peterson, MR; Riives, M; Robertson, HA | 1 |
Barbaz, BS; Bergen, KM; Bernard, PS; Boast, CA | 1 |
File, SE; Tucker, JC | 1 |
Lloyd, HG; Morgan, PF; Stone, TW | 1 |
File, SE; Herberg, LJ; Pellow, S | 1 |
Schwarz, M; Sontag, KH; Turski, L | 1 |
Katz, RJ; Wagner, JA | 1 |
Falk, JL; Tang, M | 1 |
Cain, M; Cook, J; Paul, S; Schweri, M; Skolnick, P | 1 |
Bayley, P; Curnow, R; Dawson, GR; Rambridge, A; Tricklebank, MD | 1 |
Kawasaki, K; Matsushita, A; Satoh, M; Yasui, M | 1 |
Grahn, RE; Maier, SF; Maswood, S; Watkins, LR | 1 |
Hadingham, KL; Palmer, KJ; Thompson, SA; Wafford, KA; Whiting, PJ | 1 |
Cason, CR; Cox, R; Duemler, SE; Greene, TL; Hite, ML; June, HL; Li, TK; Lumeng, L; Mellon-Burke, J; Murphy, JM; Torres, L; Williams, JA | 1 |
Allen, A; Braun, MR; Cason, CR; Craig, KS; DeLong, J; June, HL; Murphy, JM; Torres, L; Zuccarelli, D | 1 |
Campagna, F; Carotti, A; De Sarro, A; De Sarro, G; Falconi, U; Giusti, P; Mckernan, R; Palluotto, F; Rettore, C; Rizzo, M | 1 |
7 review(s) available for flumazenil and 2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one
Article | Year |
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Behavioural pharmacology of food, water and salt intake in relation to drug actions at benzodiazepine receptors.
Topics: Animals; Anti-Anxiety Agents; Appetite; Appetite Depressants; Benzodiazepines; Benzodiazepinones; Carbolines; Chlordiazepoxide; Chlorides; Choice Behavior; Diazepam; Drinking Behavior; Feeding Behavior; Flumazenil; Food Deprivation; Food Preferences; gamma-Aminobutyric Acid; Ion Channels; Midazolam; Picrotoxin; Punishment; Pyrazoles; Receptors, GABA-A; Satiation; Sodium Chloride; Species Specificity | 1985 |
Benzodiazepines and their antagonists: a pharmacoethological analysis with particular reference to effects on "aggression".
Topics: Aggression; Agonistic Behavior; Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Chlordiazepoxide; Conflict, Psychological; Environment; Flumazenil; Humans; Midazolam; Predatory Behavior; Pyrazoles; Social Behavior; Species Specificity; Time Factors | 1985 |
What can be learned from the effects of benzodiazepines on exploratory behavior?
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Carbolines; Environment; Exploratory Behavior; Flumazenil; Lorazepam; Mice; Motor Activity; Pyrazoles; Rats; Receptors, GABA-A | 1985 |
Could an endogenous benzodiazepine ligand contribute to hepatic encephalopathy?
Topics: Benzodiazepines; Flumazenil; Hepatic Encephalopathy; Humans; Ligands; Pyrazoles; Receptors, GABA-A; Synaptic Transmission | 1988 |
Behavioural actions of Ro 5-4864: a peripheral-type benzodiazepine?
Topics: Animals; Behavior, Animal; Benzodiazepinones; Binding Sites; Brain; Convulsants; Drug Interactions; Flumazenil; Humans; Isoquinolines; Kidney; Phenytoin; Picrotoxin; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Antagonists of benzodiazepines.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Binding, Competitive; Carbolines; Flumazenil; gamma-Aminobutyric Acid; Humans; Models, Chemical; Molecular Conformation; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Synaptic Transmission | 1983 |
The neuropharmacology of various diazepam antagonists.
Topics: Animals; Benzodiazepinones; Caffeine; Carbolines; Diazepam; Flumazenil; Humans; Physostigmine; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A; Theophylline | 1983 |
91 other study(ies) available for flumazenil and 2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one
Article | Year |
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Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship | 2000 |
Discriminative stimulus properties of the benzodiazepine receptor antagonist flumazenil.
Topics: Analysis of Variance; Animals; Anticonvulsants; Behavior, Animal; Benzodiazepines; Carbolines; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; GABA-A Receptor Antagonists; Male; Pyrazoles; Rats; Rats, Inbred Strains | 1992 |
Increased sensitivity to benzodiazepine antagonists in rats following chronic treatment with a low dose of diazepam.
Topics: Animals; Anti-Anxiety Agents; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Food; Male; Pyrazoles; Rats; Rats, Inbred Strains; Reinforcement Schedule; Reinforcement, Psychology | 1990 |
Respiratory effects of benzodiazepine-related drugs in awake rhesus monkeys.
Topics: Administration, Inhalation; Alprazolam; Animals; Anti-Anxiety Agents; Appetite Depressants; Benzodiazepines; Buspirone; Carbolines; Carbon Dioxide; Drug Therapy, Combination; Female; Flumazenil; Lorazepam; Macaca mulatta; Male; Pentobarbital; Plethysmography; Pyrazoles; Respiration | 1990 |
Effects of prenatal exposure to benzodiazepine-related drugs on early development and adult social behaviour in Swiss mice--II. Antagonists.
Topics: Animals; Behavior, Animal; Benzodiazepines; Body Weight; Female; Flumazenil; Growth; Male; Mice; Postural Balance; Pregnancy; Prenatal Exposure Delayed Effects; Pyrazoles; Sex Factors; Social Behavior | 1991 |
Benzodiazepines and their antagonists interfere with opioid-dependent stress-induced analgesia.
Topics: Analgesia; Animals; Benzodiazepines; Drug Interactions; Electroshock; Flumazenil; In Vitro Techniques; Male; Mesencephalon; Naloxone; Pain; Pyrazoles; Rats; Rats, Inbred Strains; Sensory Thresholds; Stress, Physiological | 1990 |
Motor performance decrement by midazolam: antagonism by Ro 15-1788 and CGS 8216.
Topics: Animals; Benzodiazepines; Drug Interactions; Flumazenil; Male; Midazolam; Motor Activity; Pyrazoles; Rats | 1990 |
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines | 1990 |
Behavioral studies with the beta-carboline FG 7142 combined with related drugs in monkeys.
Topics: Animals; Appetite Depressants; Behavior, Animal; Benzodiazepines; Carbolines; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Lorazepam; Male; Pyrazoles; Reinforcement Schedule; Saimiri | 1989 |
Modification of evoked hippocampal dentate inhibition by diazepam and three antagonists in urethane-anesthetized rats.
Topics: Anesthesia; Animals; Diazepam; Evoked Potentials; Flumazenil; gamma-Aminobutyric Acid; Hippocampus; Isoquinolines; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synapses; Urethane | 1989 |
Cerebral-activating (EEG) properties of two inverse agonists and of an antagonist at the benzodiazepine receptor in the rat.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Central Nervous System Stimulants; Chlorpromazine; Diazepam; Electroencephalography; Flumazenil; Imipramine; Male; Pentobarbital; Pyrazoles; Pyridazines; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1989 |
Are the effects of benzodiazepines on discrimination and punishment dissociable?
Topics: Amygdala; Animals; Behavior, Animal; Benzodiazepines; Carbolines; Chlordiazepoxide; Discrimination, Psychological; Ethanolamines; Flumazenil; gamma-Aminobutyric Acid; Midazolam; Punishment; Pyrazoles; Rats; Receptors, GABA-A | 1987 |
Are the analgesic effects of social defeat mediated by benzodiazepine receptors?
Topics: Analgesia; Animals; Behavior, Animal; Carbolines; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Pyrazoles; Receptors, GABA-A; Social Behavior | 1987 |
Modulation of the electrically evoked release of 5-[3H]hydroxytryptamine from rat cerebral cortex: effects of alpidem, CL 218872, and diazepam.
Topics: Animals; Benzodiazepines; Carbolines; Cerebral Cortex; Diazepam; Electric Stimulation; Flumazenil; gamma-Aminobutyric Acid; Imidazoles; Male; Monoamine Oxidase Inhibitors; Pargyline; Pyrazoles; Pyridazines; Pyridines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Serotonin | 1988 |
Self-regulation of ICSS duration: effects of anxiogenic substances, benzodiazepine antagonists and antidepressants.
Topics: Adrenergic alpha-Antagonists; Animals; Anti-Anxiety Agents; Antidepressive Agents; Anxiety; Benzodiazepinones; Caffeine; Carbolines; Conditioning, Operant; Convulsants; Flumazenil; Humans; Male; Pentylenetetrazole; Pyrazoles; Rats; Rats, Inbred F344; Self Stimulation; Time Factors | 1985 |
The sedative effects of CL 218,872, like those of chlordiazepoxide, are reversed by benzodiazepine antagonists.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepinones; Chlordiazepoxide; Convulsants; Flumazenil; Hypnotics and Sedatives; Male; Mice; Motor Activity; Pyrazoles; Pyridazines | 1985 |
Interoceptive stimuli produced by an anxiogenic drug are mimicked by benzodiazepine antagonists in rats pretreated with isoniazid.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Brain Chemistry; Convulsants; Discrimination, Psychological; Flumazenil; gamma-Aminobutyric Acid; Humans; Isoniazid; Male; Pentobarbital; Pentylenetetrazole; Pyrazoles; Rats | 1985 |
Anxiolytic and anxiogenic drug effects on exploratory activity in an elevated plus-maze: a novel test of anxiety in the rat.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Convulsants; Exploratory Behavior; Flumazenil; Male; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats | 1986 |
Behavioral effects of zopiclone, CL 218,872 and diazepam in squirrel monkeys: antagonism by Ro 15-1788 and CGS 8216.
Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepinones; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Piperazines; Pyrazoles; Pyridazines; Saimiri | 1986 |
[Benzodiazepines and benzodiazepine receptors].
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Bicuculline; Brain; Flumazenil; gamma-Aminobutyric Acid; Mice; Muscle Relaxants, Central; Pyrazoles; Rats; Receptors, GABA-A; Receptors, Neurotransmitter; Synaptic Transmission | 1986 |
Interactions of aminophylline and three benzodiazepine compounds with amygdala-kindled seizures in rats.
Topics: Aminophylline; Amygdala; Animals; Anti-Anxiety Agents; Diazepam; Drug Interactions; Flumazenil; Kindling, Neurologic; Male; Pyrazoles; Rats; Rats, Inbred Strains; Seizures | 1987 |
Ro 15-1788, CGS 8216, picrotoxin, and pentylenetetrazol: do they antagonize anxiolytic drug effects through an anxiogenic action?
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Drug Interactions; Flumazenil; Humans; Injections, Intraperitoneal; Male; Pentylenetetrazole; Picrotoxin; Pyrazoles; Rats; Receptors, GABA-A | 1987 |
Effects of non-sedative anxiolytic drugs on responses to GABA and on diazepam-induced enhancement of these responses on mouse neurones in cell culture.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Buspirone; Carbolines; Cells, Cultured; Convulsants; Diazepam; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Mice; Neurons; Pyrazoles; Quinolines; Spinal Cord | 1988 |
The anxiogenic action of RO 5-4864 in the social interaction test: effect of chlordiazepoxide, RO 15-1788 and CGS 8216.
Topics: Animals; Anxiety; Benzodiazepinones; Chlordiazepoxide; Convulsants; Drug Interactions; Flumazenil; Humans; Male; Motor Activity; Pyrazoles; Rats; Receptors, GABA-A; Social Behavior | 1985 |
Evidence that the anticonflict effect of midazolam in amygdala is mediated by the specific benzodiazepine receptors.
Topics: Amygdala; Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Conflict, Psychological; Flumazenil; Male; Midazolam; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Radiation inactivation studies of the benzodiazepine/gamma-aminobutyric acid/chloride ionophore receptor complex.
Topics: Animals; Barbiturates; Benzodiazepines; Benzodiazepinones; Binding Sites; Brain; Carbolines; Cell Membrane; Chlorides; Diazepam; Flumazenil; Flunitrazepam; Ionophores; Male; Molecular Weight; Muscimol; Picrotoxin; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Supraspinal convulsions induced by inverse benzodiazepine agonists in rabbits.
Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electroencephalography; Flumazenil; Male; Pyrazoles; Rabbits; Receptors, GABA-A; Seizures | 1985 |
Benzodiazepine receptor ligands and the consumption of a highly palatable diet in non-deprived male rats.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Drug Interactions; Feeding Behavior; Flumazenil; Ligands; Male; Midazolam; Pyrazoles; Rats; Receptors, GABA-A | 1985 |
Effects of methyl beta-carboline-3-carboxylate, Ro 15-1788 and CGS 8216 on muscle tone in genetically spastic rats.
Topics: Animals; Benzodiazepinones; Carbolines; Dose-Response Relationship, Drug; Electromyography; Female; Flumazenil; Male; Muscle Spasticity; Muscle Tonus; Pyrazoles; Rats; Rats, Mutant Strains; Receptors, GABA-A | 1985 |
Effects of tifluadom on food consumption compared with chlordiazepoxide and kappa agonists in the rat.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzodiazepinones; Benzomorphans; Chlordiazepoxide; Convulsants; Cyclazocine; Drug Interactions; Eating; Ethylketocyclazocine; Flumazenil; Male; Naloxone; Pyrazoles; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa | 1985 |
The effects of putative anxiogenic compounds (FG 7142, CGS 8216 and Ro 15-1788) on the rat corticosterone response.
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Corticosterone; Flumazenil; Male; Pyrazoles; Rats; Receptors, GABA-A; Stress, Psychological | 1985 |
Enhancement of GABA binding by the benzodiazepine partial agonist CGS9896.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Calcium Chloride; Diazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Magnesium; Pyrazoles; Pyridazines; Rats; Receptors, GABA-A | 1985 |
Differential interactions between chlordiazepoxide, pentobarbital and benzodiazepine antagonists Ro 15-1788 and CGS 8216 in a drug discrimination procedure.
Topics: Animals; Benzodiazepinones; Chlordiazepoxide; Conditioning, Operant; Cues; Discrimination Learning; Drug Interactions; Flumazenil; Generalization, Stimulus; Male; Pentobarbital; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1986 |
Benzodiazepine receptor-mediated effect of CGS 8216 on milk consumption in the non-deprived rat.
Topics: Animals; Benzodiazepinones; Brain; Cattle; Depression, Chemical; Drinking; Flumazenil; Milk; Pyrazoles; Rats; Receptors, GABA-A | 1986 |
Apparent pA2 estimation of benzodiazepine receptor antagonists.
Topics: Animals; Diazepam; Drug Interactions; Female; Flumazenil; Male; Pentylenetetrazole; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures | 1986 |
A selective imidazobenzodiazepine antagonist of ethanol in the rat.
Topics: Animals; Anxiety; Azides; Benzodiazepines; Chlorides; Ethanol; Flumazenil; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes | 1986 |
Dissimilarities between benzodiazepine-binding sites and adenosine uptake sites in astrocytes and neurons in primary cultures.
Topics: Adenosine; Animals; Astrocytes; Benzodiazepines; Binding Sites; Cells, Cultured; Diazepam; Flumazenil; Isoquinolines; Neurons; Pyrazoles; Receptors, GABA-A | 1987 |
The direct enhancement of positive palatability by chlordiazepoxide is antagonized by Ro 15-1788 and CGS 8216.
Topics: Animals; Chlordiazepoxide; Consummatory Behavior; Flumazenil; Food Preferences; Male; Pyrazoles; Rats; Receptors, GABA-A; Solutions; Taste | 1987 |
CGS 9896 and ZK 91296, but not CGS 8216 and RO 15-1788, are pure benzodiazepine receptor antagonists on mouse neurons in culture.
Topics: Animals; Brain; Carbolines; Cells, Cultured; Diazepam; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Mice; Neurons; Pyrazoles; Receptors, GABA-A; Spinal Cord | 1987 |
Interactions of Ro 15-1788, CGS 8216 and diazepam on head-turning in rats.
Topics: Animals; Benzodiazepinones; Diazepam; Drug Interactions; Electric Stimulation; Flumazenil; Head; Male; Movement; Muscimol; Pyrazoles; Rats; Rats, Inbred Strains | 1986 |
Benzodiazepine antagonist, CGS-8216, in diazepam- or pentobarbital-dependent and non-dependent rats.
Topics: Animals; Arousal; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Pentobarbital; Pyrazoles; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Substance-Related Disorders | 1986 |
CGS 8216: agonist and diazepam-antagonist effects in rodents.
Topics: Animals; Ataxia; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Male; Mice; Pentylenetetrazole; Pyrazoles; Rats; Rats, Inbred F344; Reinforcement, Psychology | 1986 |
Evaluation of two anticonvulsant amino-pyridazine derivatives in the conflict test in rats.
Topics: Animals; Anticonvulsants; Conflict, Psychological; Diazepam; Flumazenil; Meprobamate; Mice; Papio; Pentobarbital; Pyrazoles; Pyridazines; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Valproic Acid | 1986 |
Investigation of the actions of the benzodiazepine antagonists Ro 15-1788 and CGS 8216 using the schedule-controlled behavior of rats.
Topics: Animals; Anxiety; Behavior, Animal; Benzodiazepines; Diazepam; Drug Interactions; Flumazenil; Male; Pyrazoles; Pyridines; Rats; Rats, Inbred Strains; Zolpidem | 1986 |
Pharmacologic characterization of acute chlordiazepoxide dependence in the rat.
Topics: Animals; Behavior, Animal; Chlordiazepoxide; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Flumazenil; Male; Pyrazoles; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors | 1986 |
Effects of the benzodiazepine antagonists RO 15-1788, CGS-8216 and PK-11195 on amygdaloid kindled seizures and the anticonvulsant efficacy of diazepam.
Topics: Amygdala; Animals; Diazepam; Flumazenil; Isoquinolines; Kindling, Neurologic; Male; Pyrazoles; Rats; Rats, Inbred Strains | 1986 |
Benzodiazepine ligands, nociception and 'defeat' analgesia in male mice.
Topics: Analgesia; Animals; Appetite Depressants; Benzodiazepines; Carbolines; Chlordiazepoxide; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Nociceptors; Pyrazoles | 1987 |
The pyrazoloquinoline, CGS 8216, reduces sham feeding in the rat.
Topics: Animals; Dose-Response Relationship, Drug; Drinking; Eating; Flumazenil; Gastric Fistula; Male; Pyrazoles; Rats; Rats, Inbred Strains; Time Factors | 1987 |
Anticonvulsant effect of denzimol in DBA/2 mice.
Topics: Acoustic Stimulation; Aminophylline; Animals; Anticonvulsants; Flumazenil; Imidazoles; Mice; Mice, Inbred DBA; Pyrazoles; Seizures | 1987 |
Diazepam and endorphin independently inhibit ultrasonic distress calls in rats.
Topics: Animals; Convulsants; Depression, Chemical; Diazepam; Endorphins; Flumazenil; Injections, Subcutaneous; Male; Pyrazoles; Rats; Rats, Inbred Strains; Ultrasonics; Vocalization, Animal | 1987 |
Effects of Ro 15-1788 and CGS 8216 in diazepam-dependent baboons.
Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Papio; Pyrazoles; Substance Withdrawal Syndrome; Substance-Related Disorders | 1987 |
Precipitation of abstinence in nordiazepam- and diazepam-dependent dogs.
Topics: Analysis of Variance; Animals; Diazepam; Dogs; Flumazenil; Nordazepam; Oxazepam; Pyrazoles; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders | 1988 |
Distinctive behavioral effects of the pyrazoloquinoline CGS 8216 in squirrel monkeys.
Topics: Animals; Behavior, Animal; Benzodiazepines; Clonidine; Diazepam; Flumazenil; Male; Pyrazoles; Saimiri | 1988 |
Ethanol suppression of schedule-controlled responding: interactions with Ro 15-4513, Ro 15-1788 and CGS 8216.
Topics: Alcohol Deterrents; Animals; Azides; Behavior, Animal; Benzodiazepines; Drug Interactions; Ethanol; Flumazenil; Male; Pyrazoles; Rats; Rats, Inbred Strains | 1988 |
Chlordiazepoxide-induced hyperphagia in non-food-deprived rats: effects of Ro15-1788, CGS 8216 and ZK 93 426.
Topics: Animals; Benzodiazepinones; Carbolines; Chlordiazepoxide; Convulsants; Dose-Response Relationship, Drug; Drug Interactions; Eating; Flumazenil; Indoles; Male; Pyrazoles; Rats | 1985 |
Chlordiazepoxide enhances the anxiogenic action of CGS 8216 in the social interaction test: evidence for benzodiazepine withdrawal?
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Chlordiazepoxide; Flumazenil; Humans; Male; Pyrazoles; Rats; Social Behavior; Species Specificity; Substance Withdrawal Syndrome | 1985 |
Evaluation of the beta-carboline ZK 93 426 as a benzodiazepine receptor antagonist.
Topics: Animals; Anticonvulsants; Ataxia; Benzodiazepinones; Binding, Competitive; Carbolines; Diazepam; Discrimination, Psychological; Drinking; Exploratory Behavior; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Mice; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Sleep | 1984 |
Behavioural effects of PK 8165 that are not mediated by benzodiazepine binding sites.
Topics: Animals; Behavior, Animal; Benzodiazepinones; Exploratory Behavior; Flumazenil; Male; Motor Activity; Pyrazoles; Quinolines; Rats; Receptors, GABA-A | 1984 |
Antagonism by CGS 8216 and Ro 15-1788, benzodiazepines antagonists, of the action of chlordiazepoxide on a timing behavior in rats.
Topics: Animals; Benzodiazepinones; Chlordiazepoxide; Conditioning, Psychological; Flumazenil; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Reinforcement Schedule | 1984 |
The benzodiazepine receptor and sleep.
Topics: Animals; Barbiturates; Benzodiazepines; Benzodiazepinones; Calcium; Carbolines; Diazepam; Flumazenil; Flurazepam; Humans; Motor Activity; Nifedipine; Phenobarbital; Pyrazoles; Rats; Receptors, GABA-A; Sleep; Synaptosomes | 1984 |
Benzodiazepine receptor ligands with opposing pharmacologic actions.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Flumazenil; Flunitrazepam; Kinetics; Ligands; Membranes; Models, Psychological; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Temperature | 1983 |
Antagonists of benzodiazepines: functional aspects.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Carbolines; Chlorides; Flumazenil; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Ion Channels; Narcotic Antagonists; Parasympathomimetics; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A; Substance-Related Disorders; Xanthines | 1983 |
Benzodiazepine receptor antagonists reverse the effect of diazepam on plasma corticosterone in stressed rats.
Topics: Animals; Benzodiazepinones; Corticosterone; Diazepam; Flumazenil; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Stress, Physiological | 1984 |
Absence of intrinsic antagonist actions of benzodiazepine antagonists on an exploratory model of anxiety in the mouse.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Carbolines; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Humans; Male; Mice; Pyrazoles | 1984 |
CGS 8216 fails to modify novelty-related behaviour in mice: further evidence for differential actions of benzodiazepine antagonists.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepinones; Flumazenil; Male; Mice; Pyrazoles | 1984 |
Modification of seizures elicited by the benzodiazepine Ro 5-3663--a comparison with picrotoxin.
Topics: Animals; Benzodiazepinones; Chemical Phenomena; Chemistry; Convulsants; Diazepam; Drug Synergism; Flumazenil; Male; Mice; Picrotoxin; Pyrazoles; Quinolines; Seizures | 1984 |
Interaction of the benzodiazepine antagonists, CGS 8216 and Ro 15-1788, with central adenosine A-1 receptors.
Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Brain; Flumazenil; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, Purinergic | 1982 |
Audiogenic seizures in DBA/2 mice discriminate sensitively between low efficacy benzodiazepine receptor agonists and inverse agonists.
Topics: Acoustic Stimulation; Animals; Anticonvulsants; Benzodiazepines; Benzodiazepinones; Carbolines; Convulsants; Flumazenil; Male; Mice; Mice, Inbred DBA; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A; Seizures | 1983 |
RO5-4864, a ligand for benzodiazepine micromolar and peripheral binding sites: antagonism and enhancement of behavioural effects.
Topics: Animals; Behavior, Animal; Benzodiazepinones; Drug Interactions; Flumazenil; Male; Motor Activity; Phenytoin; Picrotoxin; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Photoaffinity labeling of benzodiazepine receptors in rat brain with flunitrazepam alters the affinity of benzodiazepine receptor agonist but not antagonist binding.
Topics: Affinity Labels; Animals; Benzodiazepines; Benzodiazepinones; Brain; Carbolines; Flumazenil; Flunitrazepam; Male; Photochemistry; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Substrate Specificity | 1983 |
Interactions of ethyl-beta-carboline-3-carboxylate and Ro 15-1788 with CGS 8216 in an animal model of anxiety.
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Disease Models, Animal; Drug Interactions; Flumazenil; Humans; Indoles; Male; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Social Behavior | 1983 |
Separation of clonazepam-induced head twitches and muscle relaxation in mice.
Topics: Animals; Benzodiazepinones; Clonazepam; Drug Interactions; Flumazenil; Head; Male; Methysergide; Mice; Movement; Muscle Relaxants, Central; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
New concepts in the neurobiology of anxiety.
Topics: Animals; Anxiety; Barbiturates; Behavior; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Carbolines; Central Nervous System; Flumazenil; Humans; Macaca mulatta; Pyrazoles; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Evidence for distinct benzodiazepine receptors for anticonvulsant and sedative actions: implications for the treatment of temporal lobe epilepsy.
Topics: Amygdala; Animals; Anticonvulsants; Benzodiazepinones; Diazepam; Epilepsy, Temporal Lobe; Flumazenil; Kindling, Neurologic; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
A partial agonist at the anticonvulsant benzodiazepine receptor: reversal of the anticonvulsant effects of Ro 15-1788 with CGS-8216.
Topics: Amygdala; Animals; Benzodiazepinones; Convulsants; Flumazenil; Kindling, Neurologic; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1984 |
Chronic neonatal treatment with CGS 8216: effects on the behaviour of adolescent rats.
Topics: Animals; Animals, Newborn; Behavior, Animal; Benzodiazepinones; Brain; Chlordiazepoxide; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Flumazenil; Motor Activity; Pregnancy; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Social Behavior | 1984 |
Benzodiazepine inhibition of adenosine uptake is not prevented by benzodiazepine antagonists.
Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Flumazenil; Flurazepam; Hexobendine; In Vitro Techniques; Pyrazoles; Rats; Rats, Inbred Strains; Synaptosomes; Temperature | 1983 |
Proconvulsant action of CGS 8216.
Topics: Animals; Benzodiazepinones; Convulsants; Drug Synergism; Flumazenil; Male; Mice; Pentylenetetrazole; Picrotoxin; Pyrazoles; Seizures | 1983 |
Intracranial self-stimulation distinguishes between two benzodiazepine antagonists.
Topics: Animals; Benzodiazepinones; Chlordiazepoxide; Drug Combinations; Flumazenil; Hypothalamic Area, Lateral; Male; Pyrazoles; Rats; Self Stimulation | 1984 |
CGS 8216, Ro 15-1788 and methyl-beta-carboline-3-carboxylate, but not EMD 41717 antagonize the muscle relaxant effect of diazepam in genetically spastic rats.
Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Electromyography; Female; Flumazenil; Imidazoles; Kinetics; Male; Muscle Contraction; Muscle Relaxation; Muscle Spasticity; Pyrazoles; Rats; Rats, Mutant Strains | 1984 |
Anxiogenic action of benzodiazepine antagonists Ro 15-1788 and CGS 8216 in the rat.
Topics: Animals; Anxiety; Benzodiazepines; Benzodiazepinones; Convulsants; Dose-Response Relationship, Drug; Flumazenil; Humans; Male; Pyrazoles; Rats; Rats, Inbred Strains | 1984 |
The anxiogenic action of FG 7142 in the social interaction test is reversed by chlordiazepoxide and Ro 15-1788 but not by CGS 8216.
Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Chlordiazepoxide; Convulsants; Flumazenil; Humans; Indoles; Male; Motor Activity; Pyrazoles; Rats; Social Behavior | 1984 |
Midazolam-induced increase in NaCl solution ingestion: differential effect of the benzodiazepine antagonists Ro 15-1788 and CGS 8216.
Topics: Animals; Appetite; Benzodiazepines; Benzodiazepinones; Drug Interactions; Flumazenil; Male; Midazolam; Pyrazoles; Rats; Sodium Chloride | 1984 |
Blockade of 3-carbomethoxy-beta-carboline induced seizures by diazepam and the benzodiazepine antagonists, Ro 15-1788 and CGS 8216.
Topics: Animals; Benzodiazepinones; Carbolines; Convulsants; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Harmaline; Indoles; Male; Mice; Pyrazoles; Seizures; Tremor | 1982 |
Lack of effect of flumazenil and CGS 8216 on the anxiolytic-like properties of loreclezole.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Convulsants; Drug Interactions; Flumazenil; Injections, Intraperitoneal; Male; Pyrazoles; Rats; Triazoles | 1994 |
Benzodiazepine inverse agonists augment long-term potentiation in CA1 and CA3 of guinea pig hippocampal slices.
Topics: Animals; Benzodiazepines; Carbolines; Electric Stimulation; Evoked Potentials; Flumazenil; Guinea Pigs; Hippocampus; In Vitro Techniques; Male; Neuronal Plasticity; Psychotropic Drugs; Pyrazoles; Quinolones | 1993 |
The benzodiazepine receptor antagonists flumazenil and CGS8216 block the enhancement of fear conditioning and interference with escape behavior produced by inescapable shock.
Topics: Animals; Behavior, Animal; Electroshock; Escape Reaction; Flumazenil; GABA Antagonists; Male; Pyrazoles; Rats; Reaction Time; Stress, Physiological; Time Factors | 1995 |
Expression and pharmacology of human GABAA receptors containing gamma 3 subunits.
Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Base Sequence; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Molecular Sequence Data; Pyrazoles; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Proteins; Sequence Homology, Amino Acid; Triazolam; Xenopus; Zolpidem | 1995 |
Effects of the benzodiazepine inverse agonist RO19-4603 alone and in combination with the benzodiazepine receptor antagonists flumazenil, ZK 93426 and CGS 8216, on ethanol intake in alcohol-preferring (P) rats.
Topics: Alcohol Drinking; Animals; Azepines; Benzodiazepines; Dose-Response Relationship, Drug; Drinking; Drug Combinations; Eating; Ethanol; Female; Flumazenil; GABA-A Receptor Antagonists; Pyrazoles; Rats; Saccharin; Solutions; Time Factors | 1996 |
High-affinity benzodiazepine antagonists reduce responding maintained by ethanol presentation in ethanol-preferring rats.
Topics: Animals; Carbolines; Dose-Response Relationship, Drug; Ethanol; Flumazenil; GABA-A Receptor Antagonists; Male; Pyrazoles; Rats; Reinforcement, Psychology; Saccharin | 1998 |
Benzodiazepine receptor affinities, behavioral, and anticonvulsant activity of 2-aryl-2,5-dihydropyridazino[4,3-b]indol- 3(3H)-ones in mice.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Benzodiazepines; Body Temperature; Flumazenil; Hypnotics and Sedatives; Indoles; Ketones; Male; Mice; Mice, Inbred DBA; Motor Activity; Pyrazoles; Receptors, GABA-A; Seizures; Synaptosomes | 2000 |