flumazenil and 2-(4-chlorophenyl)-2,5-dihydropyrazolo(4,3-c)quinoline-3(3h)-one

flumazenil has been researched along with 2-(4-chlorophenyl)-2,5-dihydropyrazolo(4,3-c)quinoline-3(3h)-one in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-199012 (70.59)18.7374
1990's5 (29.41)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bernasconi, R; Leonhardt, T; Martin, P; Portet, C; Schmutz, M; Steulet, AF1
Borsini, F; Gragnani, L; Lecci, A; Meli, A; Volterra, G1
Karim, KH; Najim, RA1
Bianchi, M; Fumagalli, P; Mantegazza, P; Panerai, AE; Rovati, LC; Sacerdote, P1
Randall, JI; Rodgers, RJ1
Leidenheimer, NJ; Schechter, MD1
Ator, NA; Griffiths, RR1
Crawley, JN; Smith, CB1
De Deyn, PP; Macdonald, RL2
Cooper, SJ; Gilbert, DB1
Meiners, BA; Salama, AI1
Spealman, RD; Wettstein, JG1
Goldberg, ME; Malick, JB; Patel, JB; Salama, AI1
Bernard, P; Cassidy, JP; Czernik, AJ; Petrack, B; Yokoyama, N1
Griffiths, RR; Lamb, RJ1
Rowlett, JK; Woolverton, WL1

Reviews

2 review(s) available for flumazenil and 2-(4-chlorophenyl)-2,5-dihydropyrazolo(4,3-c)quinoline-3(3h)-one

ArticleYear
Novel non-benzodiazepine anxiolytics.
    Neuropharmacology, 1983, Volume: 22, Issue:12B

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepines; Benzodiazepinones; Conflict, Psychological; Flumazenil; Flunitrazepam; Hypnotics and Sedatives; Mice; Piperazines; Pyrazoles; Pyridazines; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
Assessment of benzodiazepine receptor heterogeneity in vivo: apparent pA2 and pKB analyses from behavioral studies.
    Psychopharmacology, 1996, Volume: 128, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Discrimination Learning; Flumazenil; GABA Modulators; GABA-A Receptor Agonists; Pyrazoles

1996

Other Studies

15 other study(ies) available for flumazenil and 2-(4-chlorophenyl)-2,5-dihydropyrazolo(4,3-c)quinoline-3(3h)-one

ArticleYear
Effects of benzodiazepine receptor ligands with different intrinsic activities on seizures induced by inhibition of GAD.
    Epilepsy research. Supplement, 1992, Volume: 8

    Topics: Animals; Anti-Anxiety Agents; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hippocampus; Isoniazid; Male; Mice; Mice, Inbred Strains; Pyrazoles; Reaction Time; Receptors, GABA-A; Seizures

1992
Effect of psychotomimetics and some putative anxiolytics on stress-induced hyperthermia.
    Journal of neural transmission. General section, 1991, Volume: 83, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Body Temperature; Dextroamphetamine; Dizocilpine Maleate; Fever; Flumazenil; Male; Mice; Phencyclidine; Pyrazoles; Pyridazines; Quinolines; Receptors, GABA-A; Receptors, Serotonin; Single-Blind Method; Stress, Physiological

1991
Effect of CGS 9896 on stress-induced gastric ulcer in rat.
    Clinical and experimental pharmacology & physiology, 1990, Volume: 17, Issue:2

    Topics: Animals; Benzodiazepines; Chlordiazepoxide; Cold Temperature; Drug Therapy, Combination; Flumazenil; Hyperglycemia; Male; Pyrazoles; Rats; Rats, Inbred Strains; Stomach Ulcer; Stress, Physiological

1990
Benzodiazepines and their antagonists interfere with opioid-dependent stress-induced analgesia.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:1

    Topics: Analgesia; Animals; Benzodiazepines; Drug Interactions; Electroshock; Flumazenil; In Vitro Techniques; Male; Mesencephalon; Naloxone; Pain; Pyrazoles; Rats; Rats, Inbred Strains; Sensory Thresholds; Stress, Physiological

1990
Are the analgesic effects of social defeat mediated by benzodiazepine receptors?
    Physiology & behavior, 1987, Volume: 41, Issue:3

    Topics: Analgesia; Animals; Behavior, Animal; Carbolines; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Pyrazoles; Receptors, GABA-A; Social Behavior

1987
Discriminative stimulus properties of CGS 9896: interactions within the GABA/benzodiazepine receptor complex.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 31, Issue:2

    Topics: Animals; Carbolines; Chlordiazepoxide; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; gamma-Aminobutyric Acid; Male; Pentobarbital; Pentylenetetrazole; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Discriminative stimulus effects of atypical anxiolytics in baboons and rats.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Azabicyclo Compounds; Benzodiazepinones; Buspirone; Discrimination Learning; Flumazenil; Isoxazoles; Lorazepam; Male; Papio; Piperazines; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1986
Anxiolytic action of CGS 9896 on mouse exploratory behavior.
    European journal of pharmacology, 1986, Dec-16, Volume: 132, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Exploratory Behavior; Flumazenil; Male; Mice; Motor Activity; Pyrazoles

1986
Effects of non-sedative anxiolytic drugs on responses to GABA and on diazepam-induced enhancement of these responses on mouse neurones in cell culture.
    British journal of pharmacology, 1988, Volume: 95, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Buspirone; Carbolines; Cells, Cultured; Convulsants; Diazepam; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Mice; Neurons; Pyrazoles; Quinolines; Spinal Cord

1988
Clonazepam-induced hyperphagia in nondeprived rats: tests of pharmacological specificity with Ro5-4864, Ro5-3663, Ro15-1788 and CGS 9896.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:5

    Topics: Animals; Benzodiazepinones; Clonazepam; Drug Interactions; Feeding Behavior; Flumazenil; Humans; Hyperphagia; Male; Pyrazoles; Rats; Receptors, GABA-A

1985
Enhancement of GABA binding by the benzodiazepine partial agonist CGS9896.
    European journal of pharmacology, 1985, Dec-10, Volume: 119, Issue:1-2

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain; Calcium Chloride; Diazepam; Flumazenil; gamma-Aminobutyric Acid; In Vitro Techniques; Magnesium; Pyrazoles; Pyridazines; Rats; Receptors, GABA-A

1985
CGS 9896 and ZK 91296, but not CGS 8216 and RO 15-1788, are pure benzodiazepine receptor antagonists on mouse neurons in culture.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:1

    Topics: Animals; Brain; Carbolines; Cells, Cultured; Diazepam; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Mice; Neurons; Pyrazoles; Receptors, GABA-A; Spinal Cord

1987
Behavioral effects of the pyrazoloquinoline CGS 9896: agonist and antagonist actions in squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:1

    Topics: Animals; Azabicyclo Compounds; Behavior, Animal; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Lorazepam; Male; Piperazines; Pyrazoles; Saimiri

1987
Benzodiazepine receptor ligands with opposing pharmacologic actions.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Diazepam; Flumazenil; Flunitrazepam; Kinetics; Ligands; Membranes; Models, Psychological; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, GABA-A; Temperature

1983
Precipitated and spontaneous withdrawal in baboons after chronic dosing with lorazepam and CGS 9896.
    Drug and alcohol dependence, 1984, Volume: 14, Issue:1

    Topics: Animals; Benzodiazepinones; Flumazenil; Humans; Lorazepam; Male; Papio; Pyrazoles; Substance Withdrawal Syndrome; Substance-Related Disorders

1984