flufenamic acid and niflumic acid

flufenamic acid has been researched along with niflumic acid in 56 studies

Research

Studies (56)

TimeframeStudies, this research(%)All Research%
pre-19905 (8.93)18.7374
1990's18 (32.14)18.2507
2000's14 (25.00)29.6817
2010's17 (30.36)24.3611
2020's2 (3.57)2.80

Authors

AuthorsStudies
Chang, TK; Ensom, MH; Kiang, TK1
Herz, JM; Hu, H; Tian, J; Wang, C; Wood, JD; Xiao, R; Zhu, MX; Zhu, Y1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Dai, L; Garg, V; Sanguinetti, MC1
Garg, P; Sanguinetti, MC1
Bartlett, SJ; Bauche, A; Fliegert, R; Guse, AH; Harneit, A; Kirchberger, T; Moreau, C; Potter, BV; Swarbrick, JM; Yorgan, T1
Bennis, K; Ducki, S; Lesage, F; Vivier, D1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Alexandrov, K; Capon, RJ; Cooper, MA; Fontaine, F; Francois, M; Gambin, Y; Jauch, R; Koopman, P; Lua, L; Mamidyala, S; Moustaqil, M; Narasimhan, K; Overman, J; Prokoph, N; Robertson, AAB; Salim, A; Sierecki, E; Zuegg, J1
Adihou, H; Akbarzadeh, M; Dötsch, L; Friese, A; Guéret, SM; Hahne, G; Hong, W; Kang, C; Karatas, H; Metz, M; Nowak, C; Pahl, A; Pobbati, AV; Sievers, S; Thavam, S; Waldmann, H; Yihui Ng, E; Zinken, S1
Audran, M; Boiteau, HL; Carlier, N; Hamelin, JP; Prost, A; Rossel-Renac, F1
Leynadier, F; Perrault, M1
Collas, P1
Onoda, T; Shichikawa, K1
Cook, DI; Poronnik, P; Ward, MC1
Chao, AC; Mochizuki, H1
Aylwin, M; White, MM1
Dahlem, D; Englert, HC; Gögelein, H; Lang, HJ1
Musumeci, S; Raciti, R; Romano, L; Scuteri, A1
Ottolia, M; Toro, L1
Clauss, W; Liebold, KM; Reifarth, FW; Uhr, U; Weber, WM1
Dani, JA; Dineley-Miller, K; Patrick, JW; Séguéla, P; Wadiche, J1
Martin, SC; Shuttleworth, TJ1
Oortgiesen, M; Vijverberg, HP; Zwart, R1
Busch, AE; Herzer, T; Lang, F; Raber, G; Schmidt, F; Wagner, CA; Waldegger, S1
Greenwood, IA; Large, WA1
De Smet, P; Droogmans, G; Eggermont, J; Nilius, B; Van Driessche, W; Voets, T; Wei, L1
Dixon, JE; McKinnon, D; Wang, HS1
Benos, DJ; DuVall, MD; Fuller, CM; Ji, HL; Patton, HK; Satterfield, CL1
Hamill, OP; McBride, DW; Zhang, Y1
Kinnamon, SC; Lin, W; McPheeters, M; Mierson, S; Wladkowski, SL1
Bracht, A; Ishii-Iwamoto, EL; Kelmer-Bracht, AM; Lopez, CH; Sampaio, E; Yamamoto, NS1
Baures, PW; Kelly, JW; Oza, VB; Peterson, SA1
Polásek, M; Pospísilová, M; Urbánek, M1
Katz, U; Nagel, W; Somieski, P1
Aspeslagh, S; Braet, K; Evans, WH; Leybaert, L; Martin, PE; Vandamme, W; Willecke, K1
Hotta, A; Kim, YC; Kito, Y; Nakamura, E; Suzuki, H; Yamamoto, Y1
Bauer-Brandl, A; Perlovich, GL; Surov, AO1
Gaganis, P; Knights, KM; Miners, JO1
Babini, E; Camerino, DC; Liantonio, A; Picollo, A; Pusch, M1
Arendshorst, WJ; Fellner, SK1
Guan, BC; Jiang, ZG; Ma, KT; Yang, YQ; Zhao, H1
Bates, DO; Foster, RR; Mathieson, PW; Saleem, MA; Satchell, SC; Welsh, GI; Ye, Y; Zadeh, MA1
Choi, JJ; Choi, S; Jin, M; Jun, JY; Kim, DH; Kim, SH; Koh, JW; Lee, I; Pyo, MY; Son, JP; Son, M1
Habjan, S; Vandenberg, RJ1
Perlovich, GL; Surov, AO; Szterner, P; Zielenkiewicz, W1
Domańska, U; Pelczarska, A; Pobudkowska, A2
Choi, S; Jun, JY; Kim, MY; Kim, YD; Koh, JW; Park, CG; So, I; Yeum, CH1
Han, S; Han, SE; Jung, BK; Kim, BJ; Kim, JS; Kwon, YK; Nah, SY; Nam, JH1
Bozzolan, F; Debernard, S; Demondion, E; François, A; Grauso, M; Lucas, P1
Guan, BC; Jiang, ZG; Li, L; Li, XZ; Ma, KT; Si, JQ; Zhang, ZS; Zhao, L1
Du, X; Gamper, N; Gao, H; Huang, D; Liu, Y; Qi, J; Xu, J; Zhang, H1
Hatzidimitriou, AG; Kefala, LA; Kessissoglou, DP; Papadopoulos, AN; Perdih, F; Psomas, G; Tsiliou, S; Turel, I1
Carter, JM; Diaz, MR; Gigante, ED; Landin, JD; Rieger, SP; Werner, DF1
Kumar, A; Misra, G; Pal, R1

Reviews

2 review(s) available for flufenamic acid and niflumic acid

ArticleYear
UDP-glucuronosyltransferases and clinical drug-drug interactions.
    Pharmacology & therapeutics, 2005, Volume: 106, Issue:1

    Topics: Clinical Trials as Topic; Drug Interactions; Enzyme Activation; Enzyme Induction; Glucuronides; Glucuronosyltransferase; Humans; Pharmaceutical Preparations; Pharmacogenetics; Polymorphism, Genetic

2005
Perspectives on the Two-Pore Domain Potassium Channel TREK-1 (TWIK-Related K(+) Channel 1). A Novel Therapeutic Target?
    Journal of medicinal chemistry, 2016, 06-09, Volume: 59, Issue:11

    Topics: Arrhythmias, Cardiac; Depression; Epilepsy; Humans; Inflammation; Models, Molecular; Molecular Structure; Neuroprotective Agents; Pain; Potassium Channels, Tandem Pore Domain; Structure-Activity Relationship

2016

Trials

2 trial(s) available for flufenamic acid and niflumic acid

ArticleYear
[An anti-inflammatory association in oral surgery. A report on 90 cases].
    Le Chirurgien-dentiste de France, 1977, May-26, Volume: 47, Issue:352

    Topics: Adult; Clinical Trials as Topic; Female; Flufenamic Acid; Humans; Male; Nicotinic Acids; Niflumic Acid; Postoperative Complications; Surgery, Oral

1977
[Effect of niflumic acid on chronic rheumatoid arthritis].
    Ryumachi. [Rheumatism], 1976, Volume: 16, Issue:2

    Topics: Adolescent; Adult; Arthritis, Rheumatoid; Clinical Trials as Topic; Drug Evaluation; Female; Flufenamic Acid; Humans; Male; Middle Aged; Nicotinic Acids; Niflumic Acid

1976

Other Studies

52 other study(ies) available for flufenamic acid and niflumic acid

ArticleYear
Activation of TRPA1 channels by fenamate nonsteroidal anti-inflammatory drugs.
    Pflugers Archiv : European journal of physiology, 2010, Volume: 459, Issue:4

    Topics: Animals; Ankyrins; Anti-Inflammatory Agents, Non-Steroidal; Calcium Channels; Cell Line; Fenamates; Humans; Membrane Potentials; Mice; Molecular Structure; Oocytes; Patch-Clamp Techniques; Rats; TRPA1 Cation Channel; TRPC Cation Channels; TRPM Cation Channels; TRPV Cation Channels; Xenopus laevis

2010
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Activation of Slo2.1 channels by niflumic acid.
    The Journal of general physiology, 2010, Volume: 135, Issue:3

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cells, Cultured; Dose-Response Relationship, Drug; Humans; Ion Channel Gating; Membrane Potentials; Niflumic Acid; Oocytes; Potassium Channels; Potassium Channels, Sodium-Activated; Protein Conformation; Sodium; Structure-Activity Relationship; Xenopus

2010
Structure-activity relationship of fenamates as Slo2.1 channel activators.
    Molecular pharmacology, 2012, Volume: 82, Issue:5

    Topics: Animals; Cyclooxygenase Inhibitors; Female; Fenamates; Humans; Ibuprofen; In Vitro Techniques; Large-Conductance Calcium-Activated Potassium Channel alpha Subunits; Niflumic Acid; Oocytes; ortho-Aminobenzoates; Patch-Clamp Techniques; Point Mutation; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Sodium-Activated; Structure-Activity Relationship; Xenopus laevis

2012
Structure-activity relationship of adenosine 5'-diphosphoribose at the transient receptor potential melastatin 2 (TRPM2) channel: rational design of antagonists.
    Journal of medicinal chemistry, 2013, Dec-27, Volume: 56, Issue:24

    Topics: Adenosine Diphosphate Ribose; Dose-Response Relationship, Drug; Drug Design; Humans; Models, Molecular; Molecular Structure; Structure-Activity Relationship; TRPM Cation Channels

2013
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Small-Molecule Inhibitors of the SOX18 Transcription Factor.
    Cell chemical biology, 2017, Mar-16, Volume: 24, Issue:3

    Topics: Animals; Binding Sites; Biological Products; Chlorocebus aethiops; COS Cells; DNA; Drug Design; Genes, Reporter; Immunoglobulin J Recombination Signal Sequence-Binding Protein; Inhibitory Concentration 50; Mice; Nucleic Acid Conformation; Protein Binding; Protein Interaction Maps; Protein Structure, Tertiary; Salicylic Acid; Small Molecule Libraries; SOXF Transcription Factors; Structure-Activity Relationship; Transcriptional Activation

2017
Discovery of Covalent Inhibitors Targeting the Transcriptional Enhanced Associate Domain Central Pocket.
    Journal of medicinal chemistry, 2020, 10-22, Volume: 63, Issue:20

    Topics: Dose-Response Relationship, Drug; Drug Discovery; Fluorescence; Humans; Models, Molecular; Molecular Structure; Pyrones; Small Molecule Libraries; Structure-Activity Relationship; Sulfhydryl Compounds; Transcription Factors

2020
[Ionized fluorine in the plasma and urine of subjects treated with organofluorine drugs prescribed in rheumatology].
    Revue du rhumatisme et des maladies osteo-articulaires, 1979, Volume: 46, Issue:2

    Topics: Anti-Inflammatory Agents; Flufenamic Acid; Fluorine; Humans; Nicotinic Acids; Niflumic Acid; ortho-Aminobenzoates; Rheumatic Diseases; Sulindac

1979
[Anti-inflammatory agents in current therapeutics].
    La Revue du praticien, 1975, Jan-21, Volume: 25, Issue:5

    Topics: Adrenal Cortex Hormones; Adrenocorticotropic Hormone; Anti-Inflammatory Agents; Arthritis, Rheumatoid; Aspirin; Asthma; Bursitis; Colchicine; Collagen Diseases; Dexamethasone; Drug Hypersensitivity; Drug Interactions; Flufenamic Acid; Gastrointestinal Hemorrhage; Hallucinations; Humans; Mefenamic Acid; Niflumic Acid; Phenylbutazone; Spondylitis, Ankylosing; Tendinopathy; Triamcinolone; Vertigo

1975
Intracellular Ca2+ release by flufenamic acid and other blockers of the non-selective cation channel.
    FEBS letters, 1992, Jan-27, Volume: 296, Issue:3

    Topics: Animals; Animals, Newborn; Calcium; Cell Line; Flufenamic Acid; Ion Channels; Mefenamic Acid; Mice; Molecular Structure; Niflumic Acid

1992
Niflumic and flufenamic acids are potent inhibitors of chloride secretion in mammalian airway.
    Life sciences, 1992, Volume: 51, Issue:18

    Topics: Animals; Cattle; Cells, Cultured; Chloride Channels; Chlorides; Dogs; Epithelial Cells; Epithelium; Flufenamic Acid; Ion Channels; Membrane Proteins; Niflumic Acid; Oocytes; Trachea; Xenopus laevis

1992
Niflumic and flufenamic acids are potent reversible blockers of Ca2(+)-activated Cl- channels in Xenopus oocytes.
    Molecular pharmacology, 1990, Volume: 37, Issue:5

    Topics: Animals; Calcimycin; Calcium; Chloride Channels; Chlorides; Dose-Response Relationship, Drug; Female; Flufenamic Acid; Ion Channels; Kinetics; Membrane Proteins; Nicotinic Acids; Niflumic Acid; Oocytes; Xenopus

1990
Flufenamic acid, mefenamic acid and niflumic acid inhibit single nonselective cation channels in the rat exocrine pancreas.
    FEBS letters, 1990, Jul-30, Volume: 268, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cations; Electric Conductivity; Flufenamic Acid; In Vitro Techniques; Ion Channels; Mefenamic Acid; Nicotinic Acids; Niflumic Acid; Pancreas; Rats

1990
[Interaction of anti-inflammatory substances with the transport of 35SO4 in red blood cells].
    Bollettino della Societa italiana di biologia sperimentale, 1987, Jun-30, Volume: 63, Issue:6

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adult; Biological Transport; Erythrocytes; Flufenamic Acid; Humans; Hydrogen-Ion Concentration; In Vitro Techniques; Nicotinic Acids; Niflumic Acid; Sulfates

1987
Potentiation of large conductance KCa channels by niflumic, flufenamic, and mefenamic acids.
    Biophysical journal, 1994, Volume: 67, Issue:6

    Topics: Animals; Biophysical Phenomena; Biophysics; Calcium; Charybdotoxin; Electrochemistry; Flufenamic Acid; In Vitro Techniques; Kinetics; Mefenamic Acid; Niflumic Acid; Potassium Channels; Scorpion Venoms; Tetraethylammonium; Tetraethylammonium Compounds

1994
Influence of extracellular Ca2+ on endogenous Cl- channels in Xenopus oocytes.
    Pflugers Archiv : European journal of physiology, 1995, Volume: 429, Issue:6

    Topics: Animals; Barium; Calcium; Chloride Channels; Egtazic Acid; Electric Conductivity; Female; Flufenamic Acid; Magnesium; Membrane Potentials; Niflumic Acid; Oocytes; Patch-Clamp Techniques; Potassium; Xenopus laevis

1995
Molecular cloning, functional properties, and distribution of rat brain alpha 7: a nicotinic cation channel highly permeable to calcium.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:2

    Topics: Amino Acid Sequence; Animals; Base Sequence; Brain Chemistry; Bungarotoxins; Calcium; Cations; Chloride Channels; Cloning, Molecular; Electric Conductivity; Female; Flufenamic Acid; Ion Channels; Membrane Proteins; Molecular Sequence Data; Niflumic Acid; Oocytes; Permeability; Rats; Receptors, Nicotinic; RNA, Messenger; Sodium Chloride; Tissue Distribution; Transfection; Xenopus laevis

1993
Vasoactive intestinal peptide stimulates a cAMP-mediated Cl- current in avian salt gland cells.
    Regulatory peptides, 1994, Aug-04, Volume: 52, Issue:3

    Topics: Animals; Chloride Channels; Cyclic AMP; Ducks; Electric Conductivity; Flufenamic Acid; Membrane Potentials; Niflumic Acid; Salt Gland; Stimulation, Chemical; Thionucleotides; Vasoactive Intestinal Peptide

1994
Differential modulation of alpha 3 beta 2 and alpha 3 beta 4 neuronal nicotinic receptors expressed in Xenopus oocytes by flufenamic acid and niflumic acid.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:3 Pt 2

    Topics: Animals; Chloride Channels; Dose-Response Relationship, Drug; Female; Flufenamic Acid; Gene Expression Regulation; Neurons; Niflumic Acid; Oocytes; Patch-Clamp Techniques; Receptors, Nicotinic; Recombinant Fusion Proteins; Xenopus laevis

1995
Positive regulation by chloride channel blockers of IsK channels expressed in Xenopus oocytes.
    Molecular pharmacology, 1994, Volume: 46, Issue:4

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Calcium; Chloride Channels; Flufenamic Acid; Humans; Mefenamic Acid; Membrane Potentials; Niflumic Acid; Oocytes; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Recombinant Proteins; RNA, Complementary; Xenopus

1994
Comparison of the effects of fenamates on Ca-activated chloride and potassium currents in rabbit portal vein smooth muscle cells.
    British journal of pharmacology, 1995, Volume: 116, Issue:7

    Topics: Animals; Calcium; Chloride Channels; Evoked Potentials; Female; Flufenamic Acid; In Vitro Techniques; Mefenamic Acid; Membrane Potentials; Molecular Structure; Muscle, Smooth, Vascular; Niflumic Acid; Portal Vein; Potassium Channels; Rabbits

1995
Downregulation of volume-activated Cl- currents during muscle differentiation.
    The American journal of physiology, 1997, Volume: 272, Issue:2 Pt 1

    Topics: Animals; Cell Differentiation; Cell Division; Cell Line; Chlorides; Electric Conductivity; Flufenamic Acid; Mice; Muscles; Niflumic Acid; Nitrobenzoates

1997
Unexpected and differential effects of Cl- channel blockers on the Kv4.3 and Kv4.2 K+ channels. Implications for the study of the I(to2) current.
    Circulation research, 1997, Volume: 81, Issue:5

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Calcium; Chloride Channels; Dogs; Flufenamic Acid; Humans; Ion Transport; Niflumic Acid; Oocytes; Potassium Channels; Rats; Xenopus

1997
Functional expression of a truncated Ca(2+)-activated Cl- channel and activation by phorbol ester.
    The American journal of physiology, 1998, Volume: 274, Issue:2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Calcium; Calcium Channels; Chlorides; Dithiothreitol; Electrophysiology; Flufenamic Acid; In Vitro Techniques; Ion Channel Gating; Ionophores; Molecular Weight; Mutagenesis, Site-Directed; Niflumic Acid; Oocytes; Open Reading Frames; Protein Biosynthesis; Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Xenopus laevis

1998
The ion selectivity of a membrane conductance inactivated by extracellular calcium in Xenopus oocytes.
    The Journal of physiology, 1998, May-01, Volume: 508 ( Pt 3)

    Topics: Amiloride; Animals; Anions; Anthracenes; Anti-Bacterial Agents; Anti-Inflammatory Agents, Non-Steroidal; Calcium; Cations; Diuretics; Electric Conductivity; Extracellular Space; Female; Flufenamic Acid; Gadolinium; Gentamicins; Ion Channels; Membrane Potentials; Niflumic Acid; Oocytes; Patch-Clamp Techniques; Potassium Chloride; Sodium Chloride; Tetraethylammonium; Xenopus laevis

1998
A basolateral chloride conductance in rat lingual epithelium.
    The Journal of membrane biology, 1998, Jul-01, Volume: 164, Issue:1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Calcium; Chloride Channels; Epithelial Cells; Flufenamic Acid; Membrane Potentials; Niflumic Acid; Patch-Clamp Techniques; Rats; Rats, Wistar; Taste Buds; Tongue

1998
The action of flufenamic acid and other nonsteroidal anti-inflammatories on sulfate transport in the isolated perfused rat liver.
    General pharmacology, 1999, Volume: 32, Issue:6

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Biological Transport; Dose-Response Relationship, Drug; Flufenamic Acid; In Vitro Techniques; Liver; Male; Mefenamic Acid; Naproxen; Niflumic Acid; Perfusion; Piroxicam; Rats; Rats, Wistar; Sulfates; Sulfonamides; Sulfur Radioisotopes; Time Factors

1999
Synthesis and evaluation of inhibitors of transthyretin amyloid formation based on the non-steroidal anti-inflammatory drug, flufenamic acid.
    Bioorganic & medicinal chemistry, 1999, Volume: 7, Issue:7

    Topics: Amyloid; Anti-Inflammatory Agents, Non-Steroidal; Binding Sites; Diflunisal; Drug Design; Drug Evaluation, Preclinical; Flufenamic Acid; Humans; Light; Niflumic Acid; Prealbumin; Scattering, Radiation; Structure-Activity Relationship; Sulindac; Tolmetin

1999
Capillary isotachophoretic determination of flufenamic, mefenamic, niflumic and tolfenamic acid in pharmaceuticals.
    Journal of pharmaceutical and biomedical analysis, 2000, Aug-01, Volume: 23, Issue:1

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Calibration; Dosage Forms; Electrophoresis; Flufenamic Acid; Mefenamic Acid; Niflumic Acid; ortho-Aminobenzoates; Pharmaceutical Preparations; Reproducibility of Results

2000
Selective inhibition of Cl(-) conductance in toad skin by blockers of Cl(-) channels and transporters.
    American journal of physiology. Cell physiology, 2001, Volume: 281, Issue:4

    Topics: Angiogenesis Inhibitors; Animals; Anion Transport Proteins; Anti-Inflammatory Agents, Non-Steroidal; Bufonidae; Bumetanide; Calcium Channel Blockers; Carrier Proteins; Chloride Channels; Chlorides; Cyclooxygenase Inhibitors; Diuretics; Dose-Response Relationship, Drug; Electric Conductivity; Eosine Yellowish-(YS); Flufenamic Acid; Fluorescent Dyes; Furosemide; Mefenamic Acid; Membrane Potentials; Niflumic Acid; Nitrobenzoates; ortho-Aminobenzoates; Patch-Clamp Techniques; Skin

2001
Pharmacological sensitivity of ATP release triggered by photoliberation of inositol-1,4,5-trisphosphate and zero extracellular calcium in brain endothelial cells.
    Journal of cellular physiology, 2003, Volume: 197, Issue:2

    Topics: Adenosine Triphosphate; Animals; Blood-Brain Barrier; Brain; Calcium; Cells, Cultured; Connexin 43; Connexins; Endothelium, Vascular; Extracellular Space; Flufenamic Acid; Gadolinium; Gap Junction beta-1 Protein; Gap Junctions; Glycyrrhetinic Acid; Humans; Inositol 1,4,5-Trisphosphate; Lanthanum; Niflumic Acid; Nitrobenzoates; Oligopeptides; Rats; Ultraviolet Rays

2003
Effects of inhibitors of nonselective cation channels on the acetylcholine-induced depolarization of circular smooth muscle from the guinea-pig stomach antrum.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2005, Volume: 41, Issue:6

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acetylcholine; Animals; Female; Flufenamic Acid; Guinea Pigs; Imidazoles; In Vitro Techniques; Ion Channels; Lanthanum; Male; Membrane Potentials; Muscle, Smooth; Nickel; Niflumic Acid; Pyloric Antrum; Quinidine

2005
Thermodynamic properties of flufenamic and niflumic acids--specific and non-specific interactions in solution and in crystal lattices, mechanism of solvation, partitioning and distribution.
    Journal of pharmaceutical and biomedical analysis, 2007, Nov-30, Volume: 45, Issue:4

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Calorimetry, Differential Scanning; Crystallization; Drug Design; Drug Interactions; Energy Transfer; Flufenamic Acid; Molecular Structure; Niflumic Acid; Solubility; Solutions; Solvents; Thermodynamics

2007
Glucuronidation of fenamates: kinetic studies using human kidney cortical microsomes and recombinant UDP-glucuronosyltransferase (UGT) 1A9 and 2B7.
    Biochemical pharmacology, 2007, May-15, Volume: 73, Issue:10

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Flufenamic Acid; Glucuronides; Glucuronosyltransferase; Humans; Kidney; Kidney Cortex; Kinetics; Mefenamic Acid; Microsomes; Niflumic Acid; ortho-Aminobenzoates; Recombinant Proteins; UDP-Glucuronosyltransferase 1A9

2007
Mechanism of interaction of niflumic acid with heterologously expressed kidney CLC-K chloride channels.
    The Journal of membrane biology, 2007, Volume: 216, Issue:2-3

    Topics: Animals; Chloride Channels; Drug Synergism; Flufenamic Acid; Humans; Kidney; Models, Biological; Niflumic Acid; Phenylpropionates; Rats; Xenopus laevis

2007
Angiotensin II-stimulated Ca2+ entry mechanisms in afferent arterioles: role of transient receptor potential canonical channels and reverse Na+/Ca2+ exchange.
    American journal of physiology. Renal physiology, 2008, Volume: 294, Issue:1

    Topics: Angiotensin II; Animals; Anti-Inflammatory Agents; Arterioles; Calcium; Flufenamic Acid; Kidney; Male; Microcirculation; Muscle, Smooth, Vascular; Niflumic Acid; Rats; Rats, Sprague-Dawley; Ryanodine; Sodium-Calcium Exchanger; Thiourea; TRPC Cation Channels

2008
ACh-induced depolarization in inner ear artery is generated by activation of a TRP-like non-selective cation conductance and inactivation of a potassium conductance.
    Hearing research, 2008, Volume: 239, Issue:1-2

    Topics: Acetylcholine; Amiloride; Animals; Anti-Inflammatory Agents; Ear, Inner; Electric Conductivity; Flufenamic Acid; Guinea Pigs; Indoles; Membrane Potentials; Myocytes, Smooth Muscle; Nifedipine; Niflumic Acid; Potassium; Pyridines

2008
Flufenamic acid is a tool for investigating TRPC6-mediated calcium signalling in human conditionally immortalised podocytes and HEK293 cells.
    Cell calcium, 2009, Volume: 45, Issue:4

    Topics: Boron Compounds; Calcium; Calcium Signaling; Cell Line, Transformed; Flufenamic Acid; Humans; Imidazoles; Indomethacin; Intracellular Space; Ion Channel Gating; Niflumic Acid; Podocytes; Transfection; TRPC Cation Channels; TRPC6 Cation Channel

2009
Induction of pacemaker currents by DA-9701, a prokinetic agent, in interstitial cells of Cajal from murine small intestine.
    Molecules and cells, 2009, Mar-31, Volume: 27, Issue:3

    Topics: Animals; Calcium; Female; Flufenamic Acid; Gastrointestinal Agents; Gastrointestinal Motility; Intestine, Small; Male; Membrane Potentials; Mice; Mice, Inbred BALB C; Niflumic Acid; Patch-Clamp Techniques; Plant Preparations; Type C Phospholipases

2009
Modulation of glutamate and glycine transporters by niflumic, flufenamic and mefenamic acids.
    Neurochemical research, 2009, Volume: 34, Issue:10

    Topics: Amino Acid Transport System X-AG; Animals; Dose-Response Relationship, Drug; Female; Flufenamic Acid; Glycine Plasma Membrane Transport Proteins; Mefenamic Acid; Membrane Potentials; Niflumic Acid; Xenopus laevis

2009
Thermodynamic and structural study of tolfenamic acid polymorphs.
    Journal of pharmaceutical and biomedical analysis, 2009, Dec-05, Volume: 50, Issue:5

    Topics: Buffers; Calorimetry, Differential Scanning; Flufenamic Acid; Hydrogen Bonding; Hydrogen-Ion Concentration; Ions; Models, Chemical; Niflumic Acid; ortho-Aminobenzoates; Pressure; Solubility; Solutions; Solvents; Temperature; Thermodynamics

2009
Solubility of sparingly soluble drug derivatives of anthranilic acid.
    The journal of physical chemistry. B, 2011, Mar-24, Volume: 115, Issue:11

    Topics: 1-Octanol; Anti-Inflammatory Agents, Non-Steroidal; Calorimetry, Differential Scanning; Diclofenac; Ethanol; Flufenamic Acid; Hydrogen Bonding; Hydrogen-Ion Concentration; Models, Chemical; Molecular Structure; Niflumic Acid; ortho-Aminobenzoates; Solubility; Solvents; Spectrophotometry, Ultraviolet; Thermodynamics; Transition Temperature; Water

2011
Effects of prostaglandin F2α on small intestinal interstitial cells of Cajal.
    World journal of gastroenterology, 2011, Mar-07, Volume: 17, Issue:9

    Topics: Animals; Anti-Inflammatory Agents; Biological Clocks; Calcium; Cells, Cultured; Dinoprost; Enzyme Inhibitors; Flufenamic Acid; Interstitial Cells of Cajal; Intestine, Small; Ion Channels; Membrane Potentials; Mice; Mice, Inbred BALB C; Niflumic Acid; Patch-Clamp Techniques; Type C Phospholipases

2011
Effect of 2-hydroxypropyl-β-cyclodextrin on solubility of sparingly soluble drug derivatives of anthranilic acid.
    International journal of molecular sciences, 2011, Volume: 12, Issue:4

    Topics: 2-Hydroxypropyl-beta-cyclodextrin; beta-Cyclodextrins; Flufenamic Acid; Mefenamic Acid; Niflumic Acid; ortho-Aminobenzoates; Solubility; Spectrophotometry, Ultraviolet; Temperature; Thermodynamics

2011
Effects of ginsenoside on pacemaker potentials of cultured interstitial cells of Cajal clusters from the small intestine of mice.
    Molecules and cells, 2012, Volume: 33, Issue:3

    Topics: Action Potentials; Animals; Biological Clocks; Calcium-Transporting ATPases; Cells, Cultured; Chloride Channels; Enzyme Inhibitors; Female; Flufenamic Acid; Gastrointestinal Motility; Ginsenosides; GTP-Binding Proteins; Guanosine Diphosphate; Interstitial Cells of Cajal; Intestine, Small; Male; Membrane Transport Modulators; Mice; Mice, Inbred BALB C; Niflumic Acid; Patch-Clamp Techniques; Protein Kinase C; Thionucleotides; TRPM Cation Channels; Type C Phospholipases

2012
Bestrophin-encoded Ca²⁺-activated Cl⁻ channels underlie a current with properties similar to the native current in the moth Spodoptera littoralis olfactory receptor neurons.
    PloS one, 2012, Volume: 7, Issue:12

    Topics: Amino Acid Sequence; Animals; Arthropod Antennae; Calcium; Cells, Cultured; Chloride Channels; Cloning, Molecular; Cricetinae; Flufenamic Acid; Gene Expression; Gene Expression Regulation, Developmental; Humans; Insect Proteins; Male; Membrane Potentials; Molecular Sequence Data; Niflumic Acid; Nitrobenzoates; Olfactory Receptor Neurons; Organ Specificity; Patch-Clamp Techniques; Permeability; Primary Cell Culture; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Spodoptera

2012
Fenamates block gap junction coupling and potentiate BKCa channels in guinea pig arteriolar cells.
    European journal of pharmacology, 2013, Mar-05, Volume: 703, Issue:1-3

    Topics: Animals; Arterioles; Flufenamic Acid; Gap Junctions; Guinea Pigs; In Vitro Techniques; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Niflumic Acid; Potassium Channels, Calcium-Activated

2013
Characterization of the effects of Cl⁻ channel modulators on TMEM16A and bestrophin-1 Ca²⁺ activated Cl⁻ channels.
    Pflugers Archiv : European journal of physiology, 2015, Volume: 467, Issue:7

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Anoctamin-1; Bestrophins; Chloride Channels; CHO Cells; Cricetinae; Cricetulus; Eye Proteins; Flufenamic Acid; Humans; Membrane Transport Modulators; Neoplasm Proteins; Niflumic Acid; Nitrobenzoates; Tannins

2015
Cobalt(II) complexes with non-steroidal anti-inflammatory drugs and α-diimines.
    Journal of inorganic biochemistry, 2016, Volume: 160

    Topics: 2,2'-Dipyridyl; Aminopyridines; Anti-Inflammatory Agents, Non-Steroidal; Binding Sites; Biphenyl Compounds; Cations, Divalent; Cobalt; Coordination Complexes; Crystallography, X-Ray; Diflunisal; DNA; Flufenamic Acid; Free Radical Scavengers; Intercalating Agents; Kinetics; Mefenamic Acid; Methanol; Models, Molecular; Niflumic Acid; Phenanthrolines; Picrates; Serum Albumin

2016
Inhibitors of Calcium-Activated Anion Channels Modulate Hypnotic Ethanol Responses in Adult Sprague Dawley Rats.
    Alcoholism, clinical and experimental research, 2016, Volume: 40, Issue:2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Blotting, Western; Brain Chemistry; Calcium Channel Blockers; Calcium Channels; Ethanol; Flufenamic Acid; Hypnotics and Sedatives; Male; Motor Activity; Niflumic Acid; Nitrobenzoates; Rats; Rats, Sprague-Dawley; Reflex, Righting

2016
Exploring TEAD2 as a drug target for therapeutic intervention of cancer: A multi-computational case study.
    Briefings in bioinformatics, 2021, 09-02, Volume: 22, Issue:5

    Topics: Binding Sites; Crystallization; DNA-Binding Proteins; Drug Discovery; Flufenamic Acid; Humans; Hydrophobic and Hydrophilic Interactions; Ligands; Molecular Docking Simulation; Molecular Dynamics Simulation; Molecular Targeted Therapy; Neoplasms; Niflumic Acid; Pharmaceutical Preparations; Protein Binding; TEA Domain Transcription Factors; Transcription Factors

2021