fluconazole and streptomycin

fluconazole has been researched along with streptomycin in 46 studies

Research

Studies (46)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (15.22)29.6817
2010's38 (82.61)24.3611
2020's1 (2.17)2.80

Authors

AuthorsStudies
Drummond, AJ; Khalaf, AI; McGroarty, I; Pringle, B; Skellern, GG; Suckling, CJ; Waigh, RD1
Ashalatha, BV; Narayana, B; Suchetha Kumari, N; Vijaya Raj, KK1
Carle, AO; Curti, C; Gellis, A; Laget, M; Vanelle, P1
Lombardo, F; Obach, RS; Waters, NJ1
Che, Y; Jiang, L; Li, Y; Liu, S; Liu, X; Sun, B; Zhang, H1
Hosamani, KM; Keri, RS; Shingalapur, RV1
Bondock, S; Fadaly, W; Metwally, MA1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Bayrak, H; Demirbas, A; Demirbas, N; Karaoglu, SA1
Ekins, S; Williams, AJ; Xu, JJ1
Bellera, CL; Bruno-Blanch, LE; Castro, EA; Duchowicz, PR; Goodarzi, M; Ortiz, EV; Pesce, G; Talevi, A1
Isloor, AM; Isloor, N; Peethambar, SK; Rai, S; Telkar, S; Vijesh, AM1
Chen, M; Fang, H; Liu, Z; Shi, Q; Tong, W; Vijay, V1
Arulmoli, T; Isloor, AM; Isloor, NA; Peethambar, SK; Shivananda, KN; Vijesh, AM1
Chimov, A; Dimitrov, V; Dobrikov, GM; Momekov, G; Stoilova-Disheva, M; Tzvetkova, P; Valcheva, V1
Arun, Y; Balachandran, C; Bhaskar, G; Perumal, PT; Saikumar, C1
Mor, S; Narasimhan, B; Pahal, P2
Harini, ST; Kumar, HV; Naik, N; Rangaswamy, J2
Deng, Q; Ji, QG; Liu, HB; Tang, H; Yang, D; Yuan, LJ1
Lokanatha Rai, KM; Prashanth, MK; Revanasiddappa, HD; Veeresh, B1
Saundane, AR; Vaijinath, AV; Vijaykumar, K1
Almeida, RR; Alpay-Karaoğlu, S; Bektaş, H; Boyacioglu, O; Cao, W; Carlson, KR; Ceylan, S; Cunha-Neto, E; Demirbaş, N; Ferguson, S; Flandorfer, H; Fürtauer, S; Goktepe, I; Handy, E; Hua, DH; Kalil, J; Li, J; Madiyar, FR; Mairena, EC; Nguyen, TA; Prior, AM; Ribeiro, SP; Roberts, C; Rosa, DS; Sharma, M; Sökmen, BB; Sulakvelidze, A; Sun, E; Swisher, LZ; Syed, LU; Tserenjav, E; Wang, Z; Yakymovych, A; Zhang, R1
Bayrak, H; Demirbas, N; Karaoglu, SA; Mentese, MY; Mermer, A; Ulker, S; Uygun, Y1
Arulmoli, T; Kalluraya, B; Peethambar, SK; Shyma, PC; Telkar, S1
Alpay-Karaoglu, S; Basoglu, S; Demirbas, A; Demirbas, N; Ulker, S1
Chandrakantha, B; Fun, HK; Hegde, G; Isloor, AM; Shetty, P1
Chandrika, N; Harish, BG; Jasinski, JP; Jose, G; Millikan, SP; More, SS; Nagendrappa, G; Sowmya, HB; Suresha Kumara, TH1
Balaji, R; Dinesh, R; Kandhasamy, S; Karunagaran, D; Mathivanan, N; Mukesh, D; Perumal, PT; Shruthy, S; Shweta, S; Sreelatha, T1
Dufková, I; Hrabálek, A; Karabanovich, G; Klimešová, V; Němeček, J; Pávek, P; Roh, J; Smutný, T; Stolaříková, J; Vávrová, K; Vejsová, M; Vicherek, P1
Bharate, SS; Vishwakarma, RA1
Achur, R; Dalimba, U; Kumar, HS; Nayak, N; Peethambar, SK; Ramprasad, J; Sriram, D; Yogeeswari, P1
Arul Antony, S; Balachandran, C; Shahavar Sulthana, S; Syed Shafi, S1
Chen, K; Ge, Z; Huang, Y; Ji, Q; Liao, F; Liu, X; Wu, H; Yang, X; Yuan, L1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Chandrasekaran, B; Cherukupalli, S; Hampannavar, GA; Karpoormath, R; Palakollu, VN; Thapliyal, N1
Carazo, A; Hrabálek, A; Karabanovich, G; Klimešová, V; Konečná, K; Němeček, J; Pávek, P; Pavliš, O; Roh, J; Stolaříková, J; Valášková, L; Vávrová, K1
Desai, S; Desai, V; Dixit, SK; Gaonkar, SN; Joshi, SD; Palyekar, U1
Blanchet, M; Bourguet-Kondracki, ML; Brunel, JM; Cadelis, MM; Copp, BR; Li, SA; Sue, K; Vidal, N1
Bobade, VD; Chavan, A; Choudhari, P; Mhaske, PC; Modak, M; Nalawade, J; Patil, S; Shinde, A; Suryavanshi, M1
Ji, Q; Li, B; Shen, Y; Wang, K; Zhang, R1
Bai, H; Chen, L; Zhang, J; Zheng, S; Zhou, X; Zhu, R1
Gao, F; Huang, G; Xiao, J1
Liu, H; Long, S; Rakesh, KP; Zha, GF1

Reviews

4 review(s) available for fluconazole and streptomycin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
An insight on synthetic and medicinal aspects of pyrazolo[1,5-a]pyrimidine scaffold.
    European journal of medicinal chemistry, 2017, Jan-27, Volume: 126

    Topics: Animals; Chemistry Techniques, Synthetic; Humans; Pyrazoles; Pyrimidines

2017
Current scenario of tetrazole hybrids for antibacterial activity.
    European journal of medicinal chemistry, 2019, Dec-15, Volume: 184

    Topics: Anti-Bacterial Agents; Bacteria; Dose-Response Relationship, Drug; Microbial Sensitivity Tests; Molecular Structure; Structure-Activity Relationship; Tetrazoles

2019
Structure-activity relationships (SAR) of triazine derivatives: Promising antimicrobial agents.
    European journal of medicinal chemistry, 2020, Jan-01, Volume: 185

    Topics: Anti-Bacterial Agents; Antiviral Agents; Bacteria; Humans; Microbial Sensitivity Tests; Molecular Structure; Triazines; Viruses

2020

Other Studies

42 other study(ies) available for fluconazole and streptomycin

ArticleYear
Distamycin analogues with enhanced lipophilicity: synthesis and antimicrobial activity.
    Journal of medicinal chemistry, 2004, Apr-08, Volume: 47, Issue:8

    Topics: Animals; Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Cell Line; Cricetinae; Distamycins; DNA; Electrophoresis, Capillary; Humans; Hydrophobic and Hydrophilic Interactions; Microbial Sensitivity Tests; Structure-Activity Relationship

2004
Synthesis of some new bioactive 3-amino-2-mercapto-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one derivatives.
    European journal of medicinal chemistry, 2007, Volume: 42, Issue:5

    Topics: Animals; Anti-Bacterial Agents; Antifungal Agents; Female; Male; Pyrimidinones; Rats; Rats, Wistar; Spectrophotometry, Infrared

2007
Rapid synthesis of sulfone derivatives as potential anti-infectious agents.
    European journal of medicinal chemistry, 2007, Volume: 42, Issue:6

    Topics: Anti-Infective Agents; Bacteria; Fungi; Microbial Sensitivity Tests; Molecular Structure; Sulfones

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Bioactive asterric acid derivatives from the Antarctic ascomycete fungus Geomyces sp.
    Journal of natural products, 2008, Volume: 71, Issue:9

    Topics: Antifungal Agents; Ascomycota; Aspergillus fumigatus; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Phenols; Phenyl Ethers

2008
Synthesis and evaluation of in vitro anti-microbial and anti-tubercular activity of 2-styryl benzimidazoles.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:10

    Topics: Anti-Bacterial Agents; Antifungal Agents; Antitubercular Agents; Bacteria; Benzimidazoles; Fungi; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Structure-Activity Relationship

2009
Enaminonitrile in heterocyclic synthesis: synthesis and antimicrobial evaluation of some new pyrazole, isoxazole and pyrimidine derivatives incorporating a benzothiazole moiety.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:12

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Benzothiazoles; Botrytis; Drug Design; Fusarium; Heterocyclic Compounds; Heterocyclic Compounds, 2-Ring; Isoxazoles; Microbial Sensitivity Tests; Molecular Structure; Nitriles; Pyrazoles; Pyrimidines

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
Cyclization of some carbothioamide derivatives containing antipyrine and triazole moieties and investigation of their antimicrobial activities.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:11

    Topics: Anti-Infective Agents; Antipyrine; Cyclization; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Spectrophotometry, Infrared; Triazoles

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Prediction of drug intestinal absorption by new linear and non-linear QSPR.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:1

    Topics: Humans; Intestinal Absorption; Linear Models; Molecular Conformation; Nonlinear Dynamics; Permeability; Pharmaceutical Preparations; Probability; Quantitative Structure-Activity Relationship; Thermodynamics

2011
Synthesis, characterization and antimicrobial studies of some new pyrazole incorporated imidazole derivatives.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:8

    Topics: Administration, Oral; Animals; Anti-Infective Agents; Bacterial Infections; Female; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Imidazoles; Maximum Tolerated Dose; Mice; Microbial Sensitivity Tests; Molecular Structure; Mycoses; Pyrazoles

2011
FDA-approved drug labeling for the study of drug-induced liver injury.
    Drug discovery today, 2011, Volume: 16, Issue:15-16

    Topics: Animals; Benchmarking; Biomarkers, Pharmacological; Chemical and Drug Induced Liver Injury; Drug Design; Drug Labeling; Drug-Related Side Effects and Adverse Reactions; Humans; Pharmaceutical Preparations; Reproducibility of Results; United States; United States Food and Drug Administration

2011
Hantzsch reaction: synthesis and characterization of some new 1,4-dihydropyridine derivatives as potent antimicrobial and antioxidant agents.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:11

    Topics: Animals; Anti-Infective Agents; Bacteria; Behavior, Animal; Biphenyl Compounds; Chemistry Techniques, Synthetic; Dihydropyridines; Female; Free Radical Scavengers; Fungi; Mice; Picrates

2011
Synthesis and in vitro antimycobacterial activity of compounds derived from (R)- and (S)-2-amino-1-butanol - The crucial role of the configuration.
    European journal of medicinal chemistry, 2012, Volume: 48

    Topics: Amino Alcohols; Antitubercular Agents; Cell Line; Humans; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Molecular Structure; Mycobacterium tuberculosis; Optical Rotation; Spectrometry, Mass, Electrospray Ionization; Stereoisomerism

2012
Synthesis of novel spirooxindole derivatives by one pot multicomponent reaction and their antimicrobial activity.
    European journal of medicinal chemistry, 2012, Volume: 51

    Topics: Anti-Infective Agents; Bacteria; Chemistry Techniques, Synthetic; Fungi; Indoles; Microbial Sensitivity Tests; Oxindoles

2012
Synthesis, characterization, antimicrobial activities and QSAR studies of some 10a-phenylbenzo[b]indeno[1,2-e][1,4]thiazin-11(10aH)-ones.
    European journal of medicinal chemistry, 2012, Volume: 53

    Topics: Anti-Infective Agents; Bacteria; Chemistry Techniques, Synthetic; Fungi; Microbial Sensitivity Tests; Quantitative Structure-Activity Relationship; Thiazines

2012
Synthesis of benzofuran based 1,3,5-substituted pyrazole derivatives: as a new class of potent antioxidants and antimicrobials--a novel accost to amend biocompatibility.
    Bioorganic & medicinal chemistry letters, 2012, Jul-15, Volume: 22, Issue:14

    Topics: Anti-Infective Agents; Antioxidants; Benzofurans; Biocompatible Materials; Microbial Viability; Molecular Structure; Pyrazoles; Structure-Activity Relationship

2012
Synthesis and biological evaluation of novel N-acyl substituted quinolin-2(1H)-one derivatives as potential antimicrobial agents.
    Bioorganic & medicinal chemistry letters, 2012, Sep-15, Volume: 22, Issue:18

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Dose-Response Relationship, Drug; Fungi; Microbial Sensitivity Tests; Molecular Structure; Quinolones; Stereoisomerism; Structure-Activity Relationship

2012
Synthesis, characterization, biological evaluation and QSAR studies of 11-p-substituted phenyl-12-phenyl-11a,12-dihydro-11H-indeno[2,1-c][1,5]benzothiazepines as potential antimicrobial agents.
    European journal of medicinal chemistry, 2012, Volume: 57

    Topics: Anti-Bacterial Agents; Antifungal Agents; Aspergillus fumigatus; Bacillus subtilis; Candida albicans; Escherichia coli; Microbial Sensitivity Tests; Microbial Viability; Molecular Structure; Pseudomonas aeruginosa; Quantitative Structure-Activity Relationship; Staphylococcus aureus; Thiazepines

2012
Synthesis, characterization, antidepressant and antioxidant activity of novel piperamides bearing piperidine and piperazine analogues.
    Bioorganic & medicinal chemistry letters, 2012, Dec-01, Volume: 22, Issue:23

    Topics: Amides; Animals; Anti-Bacterial Agents; Antidepressive Agents; Antifungal Agents; Antioxidants; Behavior, Animal; Candida albicans; Gram-Negative Bacteria; Gram-Positive Bacteria; Mice; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Piperazine; Piperazines; Piperidines

2012
Synthesis, antioxidant and antimicrobial activity of novel vanillin derived piperidin-4-one oxime esters: preponderant role of the phenyl ester substituents on the piperidin-4-one oxime core.
    Bioorganic & medicinal chemistry letters, 2012, Dec-15, Volume: 22, Issue:24

    Topics: Anti-Bacterial Agents; Antioxidants; Aspergillus flavus; Benzaldehydes; Candida albicans; Chrysosporium; Dose-Response Relationship, Drug; Escherichia coli; Esters; Microbial Sensitivity Tests; Molecular Structure; Oximes; Piperidines; Staphylococcus aureus; Structure-Activity Relationship

2012
Synthesis of novel 2-amino-4-(5'-substituted 2'-phenyl-1H-indol-3'-yl)-6-aryl-4H-pyran-3-carbonitrile derivatives as antimicrobial and antioxidant agents.
    Bioorganic & medicinal chemistry letters, 2013, Apr-01, Volume: 23, Issue:7

    Topics: Anti-Bacterial Agents; Antifungal Agents; Antioxidants; Aspergillus flavus; Aspergillus oryzae; Dose-Response Relationship, Drug; Escherichia coli; Klebsiella pneumoniae; Microbial Sensitivity Tests; Nitriles; Pseudomonas aeruginosa; Pyrans; Staphylococcus aureus; Structure-Activity Relationship

2013
    Medicinal chemistry research : an international journal for rapid communications on design and mechanisms of action of biologically active agents, 2013, Volume: 22, Issue:8

    Topics:

2013
Microwave assisted synthesis of some hybrid molecules derived from norfloxacin and investigation of their biological activities.
    European journal of medicinal chemistry, 2013, Volume: 67

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fungi; Microbial Sensitivity Tests; Microwaves; Molecular Structure; Norfloxacin; Structure-Activity Relationship; Urease

2013
Synthesis, characterization and molecular docking studies of some new 1,3,4-oxadiazolines bearing 6-methylpyridine moiety for antimicrobial property.
    European journal of medicinal chemistry, 2013, Volume: 68

    Topics: Anti-Infective Agents; Bacteria; Crystallography, X-Ray; Molecular Docking Simulation; Molecular Structure; Oxadiazoles; Pyridines

2013
Design, synthesis and biological activities of some 7-aminocephalosporanic acid derivatives.
    European journal of medicinal chemistry, 2013, Volume: 69

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Canavalia; Cephalosporins; Dose-Response Relationship, Drug; Drug Design; Enzyme Inhibitors; Molecular Structure; Saccharomyces cerevisiae; Structure-Activity Relationship; Urease

2013
Synthesis and biological evaluation of novel substituted 1,3,4-thiadiazole and 2,6-di aryl substituted imidazo [2,1-b] [1,3,4] thiadiazole derivatives.
    European journal of medicinal chemistry, 2014, Volume: 71

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Bacterial Infections; Fungi; Humans; Microbial Sensitivity Tests; Mycoses; Thiadiazoles

2014
New polyfunctional imidazo[4,5-C]pyridine motifs: synthesis, crystal studies, docking studies and antimicrobial evaluation.
    European journal of medicinal chemistry, 2014, Apr-22, Volume: 77

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Crystallography, X-Ray; Dose-Response Relationship, Drug; Fungi; Humans; Imidazoles; Microbial Sensitivity Tests; Molecular Docking Simulation; Molecular Structure; Pyridines; Structure-Activity Relationship

2014
Synthesis and SAR study of novel anticancer and antimicrobial naphthoquinone amide derivatives.
    Bioorganic & medicinal chemistry letters, 2014, Aug-01, Volume: 24, Issue:15

    Topics: Anti-Bacterial Agents; Antifungal Agents; Antineoplastic Agents; Candida albicans; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Resistance, Fungal; Drug Screening Assays, Antitumor; Fluconazole; HeLa Cells; Humans; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Molecular Structure; Pseudomonas aeruginosa; Structure-Activity Relationship

2014
1-Substituted-5-[(3,5-dinitrobenzyl)sulfanyl]-1H-tetrazoles and their isosteric analogs: A new class of selective antitubercular agents active against drug-susceptible and multidrug-resistant mycobacteria.
    European journal of medicinal chemistry, 2014, Jul-23, Volume: 82

    Topics: Antineoplastic Agents; Antitubercular Agents; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Resistance, Multiple, Bacterial; Drug Screening Assays, Antitumor; HeLa Cells; Hep G2 Cells; Humans; Microbial Sensitivity Tests; Molecular Structure; Mycobacterium tuberculosis; Nitrobenzenes; Structure-Activity Relationship; Triazoles; Tumor Cells, Cultured

2014
Thermodynamic equilibrium solubility measurements in simulated fluids by 96-well plate method in early drug discovery.
    Bioorganic & medicinal chemistry letters, 2015, Apr-01, Volume: 25, Issue:7

    Topics: Drug Discovery; Pharmaceutical Preparations; Solubility; Thermodynamics

2015
Synthesis and biological evaluation of new imidazo[2,1-b][1,3,4]thiadiazole-benzimidazole derivatives.
    European journal of medicinal chemistry, 2015, May-05, Volume: 95

    Topics: Animals; Antifungal Agents; Antioxidants; Antitubercular Agents; Benzimidazoles; Cell Survival; Chlorocebus aethiops; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Structure-Activity Relationship; Thiadiazoles; Tuberculosis; Vero Cells

2015
Thiophene and benzodioxole appended thiazolyl-pyrazoline compounds: Microwave assisted synthesis, antimicrobial and molecular docking studies.
    Bioorganic & medicinal chemistry letters, 2015, Jul-15, Volume: 25, Issue:14

    Topics: Anti-Infective Agents; Benzodioxoles; Binding Sites; DNA Topoisomerase IV; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Microwaves; Molecular Docking Simulation; Protein Binding; Pyrazoles; Structure-Activity Relationship; Thermodynamics; Thiazoles; Thiophenes

2015
Synthesis and biological evaluation of novel phosphoramidate derivatives of coumarin as chitin synthase inhibitors and antifungal agents.
    European journal of medicinal chemistry, 2016, Jan-27, Volume: 108

    Topics: Amides; Antifungal Agents; Aspergillus flavus; Aspergillus fumigatus; Candida albicans; Candida tropicalis; Chitin Synthase; Coumarins; Cryptococcus neoformans; Dose-Response Relationship, Drug; Enzyme Inhibitors; Microbial Sensitivity Tests; Phosphoric Acids; Structure-Activity Relationship

2016
S-substituted 3,5-dinitrophenyl 1,3,4-oxadiazole-2-thiols and tetrazole-5-thiols as highly efficient antitubercular agents.
    European journal of medicinal chemistry, 2017, Jan-27, Volume: 126

    Topics: Antifungal Agents; Antitubercular Agents; Drug Design; Drug Resistance; Hep G2 Cells; Humans; Microbial Sensitivity Tests; Oxadiazoles; Structure-Activity Relationship; Sulfhydryl Compounds; Tetrazoles

2017
Novel quinoxalinyl chalcone hybrid scaffolds as enoyl ACP reductase inhibitors: Synthesis, molecular docking and biological evaluation.
    Bioorganic & medicinal chemistry letters, 2017, 05-15, Volume: 27, Issue:10

    Topics: Anti-Infective Agents; Antineoplastic Agents; Binding Sites; Candida albicans; Cell Proliferation; Chalcones; Disk Diffusion Antimicrobial Tests; Drug Design; Enoyl-CoA Hydratase; Enzyme Inhibitors; Escherichia coli; Humans; MCF-7 Cells; Molecular Docking Simulation; Mycobacterium tuberculosis; Protein Structure, Tertiary; Staphylococcus aureus

2017
6-Bromoindolglyoxylamido derivatives as antimicrobial agents and antibiotic enhancers.
    Bioorganic & medicinal chemistry, 2019, 05-15, Volume: 27, Issue:10

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Cell Line; Cell Survival; Drug Resistance, Bacterial; Erythrocytes; Fungi; Gram-Negative Bacteria; Gram-Positive Bacteria; Hemolysis; Humans; Indoles; Microbial Sensitivity Tests; Polyamines

2019
Synthesis of new thiazolyl-pyrazolyl-1,2,3-triazole derivatives as potential antimicrobial agents.
    European journal of medicinal chemistry, 2019, Oct-01, Volume: 179

    Topics: Anti-Bacterial Agents; Antifungal Agents; Aspergillus niger; Candida albicans; Dose-Response Relationship, Drug; Escherichia coli; Microbial Sensitivity Tests; Molecular Structure; Proteus mirabilis; Rhodotorula; Staphylococcus; Structure-Activity Relationship

2019
Design, synthesis and biological evaluation of novel diazaspiro[4.5]decan-1-one derivatives as potential chitin synthase inhibitors and antifungal agents.
    European journal of medicinal chemistry, 2019, Nov-15, Volume: 182

    Topics: Antifungal Agents; Aspergillus flavus; Aspergillus fumigatus; Aza Compounds; Candida albicans; Chitin Synthase; Dose-Response Relationship, Drug; Drug Design; Enzyme Inhibitors; Ketones; Microbial Sensitivity Tests; Molecular Structure; Spiro Compounds; Structure-Activity Relationship

2019
Synthesis and biological evaluation of calycanthaceous alkaloid analogs.
    Bioorganic & medicinal chemistry, 2019, 11-01, Volume: 27, Issue:21

    Topics: Acetylcholinesterase; Animals; Anti-Bacterial Agents; Antifungal Agents; Bacteria; Cholinesterase Inhibitors; Fungi; Indole Alkaloids; Microbial Sensitivity Tests; Molecular Docking Simulation; Molecular Structure; Protein Binding; Pyrroles; Structure-Activity Relationship; Torpedo

2019