fluconazole has been researched along with ergosterol in 120 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 18 (15.00) | 18.2507 |
2000's | 25 (20.83) | 29.6817 |
2010's | 54 (45.00) | 24.3611 |
2020's | 23 (19.17) | 2.80 |
Authors | Studies |
---|---|
Cannon, RD; Holmes, AR; Lamping, E; Nakamura, K; Niimi, K; Niimi, M; Ranchod, A; Tyndall, JD | 1 |
Pfaller, M; Riley, J | 1 |
Ballard, SA; Ellis, SW; Kelly, SL; Troke, PF | 1 |
Denning, DW; Kelly, SL; Manning, NJ; Venkateswarlu, K | 2 |
Baldwin, BC; Corran, A; Kelly, SL; Kwon-Chung, J; Lamb, DC | 1 |
Casadevall, A; Currie, B; Edwards, JE; Ghannoum, MA; Ibrahim, AS; Ritchie, JA; Spellberg, BJ; Spitzer, ED | 1 |
Bartlett, MS; Queener, SF; Richardson, JD; Shaw, MM; Smith, JW | 1 |
Hof, H; Kretschmar, M | 1 |
Capobianco, JO; Goldman, RC; Griffin, JH; Sharpe, BA; Zakula, D | 1 |
Abecia, LC; Arévalo, JM; López, MJ | 1 |
Connolly, P; Le Monte, A; Marichal, P; Vanden Bossche, H; Wheat, J | 1 |
Baldwin, BC; Corran, AJ; Kelly, DE; Kelly, SL; Lamb, DC | 1 |
Denning, DW; Kelly, SL; Venkateswarlu, K | 1 |
Bowden, RA; Lyons, CN; Marr, KA; Rustad, T; Rustad, TR; White, TC | 1 |
Falconer, D; Filler, SG; Ghannoum, MA; Higginbotham, LM; Hitchcock, CA; Ibrahim, AS; Orozco, AS; Parkinson, T | 1 |
Krishnamurthy, SS; Prasad, R | 1 |
Einsele, H; Kelly, DE; Kelly, SL; Lamb, DC; Loeffler, J | 1 |
Arthington-Skaggs, BA; Desai, T; Jradi, H; Morrison, CJ | 1 |
Daum, G; Einsele, H; Hebart, H; Hrastnik, C; Löffler, J; Schumacher, U | 1 |
Arthington-Skaggs, BA; Morrison, CJ; Warnock, DW | 1 |
Kontoyiannis, DP | 2 |
Arthington-Skaggs, BA; Brandt, ME; Ciblak, MA; Frade, JP; Hajjeh, RA; Harrison, LH; Lee-Yang, W; Sofair, AN; Warnock, DW | 1 |
Kudoh, M; Maebashi, K; Makimura, K; Mori, T; Nishiyama, Y; Uchida, K; Yamaguchi, H | 1 |
Barker, KS; Rogers, PD | 1 |
Kamai, Y; Kudoh, M; Maebashi, K; Makimura, K; Nishiyama, Y; Uchida, K; Yamaguchi, H | 1 |
Daneshtalab, M; Kurosawa, T; Mori, Y; Sardari, S | 1 |
Holleman, S; Lyons, CN; Oliver, BG; Song, JL; White, TC | 1 |
Barbuch, R; Bard, M; Bareither, B; Barker, KS; Crisp, S; Eckstein, J; Lewis, RE; Rogers, PD; Wiederhold, N | 1 |
Gao, Y; Ling, X; Lou, H; Sun, S | 1 |
Kamai, Y; Kudoh, M; Maebashi, K; Makimura, K; Naka, W; Uchida, K; Yamaguchi, H | 1 |
Jung, WH; Nunn, CD; Popolo, L; Ragni, E; Stateva, L; Turner, MP; Warn, P | 1 |
Cowen, LE; Lindquist, S | 1 |
Park, S; Perlin, DS | 1 |
Paula, CR; Ribeiro, MA | 1 |
Berman, J; Forche, A; Selmecki, A | 1 |
Chandra, A; Mukhopadhyay, CK; Prasad, R; Prasad, T | 1 |
Berdicevsky, I; Eads, E; Heitman, J; Horwitz, BA; Kaufman, G; Onyewu, C; Perfect, JR; Schell, WA; Ullmann, Y | 1 |
Barker, KS; Dunkel, N; Homayouni, R; Liu, TT; Morschhäuser, J; Rogers, PD | 1 |
Borecká-Melkusová, S; Bujdáková, H; Chorvát, D; Kucharíková, S; Moran, GP; Sullivan, DJ | 1 |
Cheng, AX; Lou, HX; Lv, BB; Sun, LM; Wu, XZ | 1 |
Costa-de-Oliveira, S; Pina-Vaz, C; Pinto e Silva, AT; Rodrigues, AG; Silva-Dias, A | 1 |
Ando, A; Hata, M; Ishii, C; Otani, T; Yoshida, K | 1 |
Gamarra, S; Park, S; Perlin, DS; Rao, R; Rocha, EM; Zhang, YQ | 1 |
Gamarra, S; Garcia-Effron, G; Park, S; Perlin, DS; Rao, R; Zhang, YQ | 1 |
Bader, O; Gross, U; Kelly, DE; Kelly, SL; Martel, CM; Parker, JE; Rolley, N; Warrilow, AG; Weig, M | 1 |
Kelly, DE; Kelly, SL; Martel, CM; Parker, JE; Rolley, NJ; Warrilow, AG | 1 |
Brown, RP; Hoot, SJ; Smith, AR; White, TC | 1 |
Aoyama, T; Bard, M; Chibana, H; Higashi, S; Kajiwara, S; Miyazaki, Y; Nagi, M; Nakayama, H; Niimi, M; Ohno, H; Okano, M; Tanabe, K; Ueno, K; Umeyama, T; Yamagoe, S | 1 |
Khan, LA; Muralidhar, S; Neelofar, K; Nikhat, M; Rimple, B; Shreaz, S | 1 |
Blaško, J; Borecká, S; Bujdáková, H; Kuchler, K; Kulková, N; Pinjon, E; Sullivan, DJ | 1 |
Khan, LA; Manzoor, N; Rizvi, MM; Shreaz, S | 1 |
Blakely, KM; Brown, E; Curak, J; De Pascale, G; Ejim, L; Griffiths, E; Rossi, L; Spitzer, M; Tyers, M; Wildenhain, J; Wright, GD | 1 |
Alvarez-Rueda, N; Fleury, A; Gastinel, L; Le Pape, P; Morio, F; Pagniez, F | 1 |
Blosser, SJ; Cramer, RA | 1 |
César, IC; Gouveia, LF; Pianetti, GA; Resende-Stoianoff, MA; Santos, DA; Santos, JR; Taylor, EL | 1 |
Bader, O; Gross, U; Hull, CM; Kelly, DE; Kelly, SL; Parker, JE; Warrilow, AG; Weig, M | 1 |
Barker, KS; Berkow, EL; Chadwick, SG; Flowers, SA; Gygax, SE; Morschhäuser, J; Rogers, PD; Toner, G | 1 |
Cadieux, B; Cho, YJ; Choi, J; Chun, J; Do, E; Hu, G; Jung, WH; Kim, J; Kronstad, JW; Lee, Y | 1 |
Calderone, R; Chen, H; Fonzi, W; She, X; Sun, N; Zhang, L | 1 |
Hakariya, M; Kaneko, Y; Matsumoto, S; Miyagawa, S; Miyazaki, Y; Ohno, H; Takeda, O | 1 |
Bandeira, Tde J; Brilhante, RS; Caetano, EP; Castelo-Branco, Dde S; Cordeiro, Rde A; de Lima, RA; Leite, JJ; Monteiro, AJ; Ribeiro, JF; Rocha, MF; Sidrim, JJ | 1 |
Hoot, SJ; White, TC; Zavrel, M | 1 |
Coste, A; Eddouzi, J; Ischer, F; Kelly, S; Manai, M; Parker, JE; Sanglard, D; Vale-Silva, LA | 1 |
Ban, X; Chen, Y; Ma, B; Tian, J; Wang, Y; Zeng, H | 1 |
Coleman, K; Dahl, T; Ghannoum, M; Keating, J; Lafleur, MD; Lee, RE; Lewis, K; Lister, I; Long, L; Nantel, A; North, J; Sun, L | 1 |
Calucci, L; Castellano, S; Cicogna, F; Forte, C; Pinzino, C; Porta, A | 1 |
Barker, KS; Caudle, KE; Chadwick, SG; Gygax, SE; Rogers, PD; Toner, G; Vermitsky, JP; Whaley, SG | 1 |
Fiori, A; Van Dijck, P; Van Hauwenhuyse, F | 1 |
Liang, S; Liao, K; Sun, LM; Wang, DY; Yu, PH | 1 |
Eom, SH; Ha, S; Im, YJ; Lee, CW; Tong, J; Yang, H | 1 |
Li, WJ; Liu, JY; Shi, C; Wang, Y; Xiang, MJ; Zhao, Y | 1 |
Lu, KQ; Shao, J; Shi, GX; Wang, CZ; Wang, TM; Yan, YY; Zhang, MX | 1 |
Bracher, F; Burger-Kentischer, A; Eickhoff, H; Engelhardt, I; Hiller, E; Keller, P; Lemuth, K; Müller, C; Rupp, S; Wiesmüller, KH | 1 |
Bandeira, Tde J; Brilhante, RS; Cordeiro, Rde A; de Melo, CV; Evangelista, AJ; Marques, FJ; Mota, VF; Rocha, MF; Serpa, R; Sidrim, JJ | 1 |
Kodedová, M; Sychrová, H | 1 |
Alencar, LP; Bandeira, TJPG; Brilhante, RSN; Cordeiro, RA; Evangelista, AJJ; Franco, JDS; Marques, FJF; Melo, CVS; Oliveira, JS; Rocha, MFG; Serpa, R; Sidrim, JJC | 1 |
Alencar, LP; Bandeira, SP; Bandeira, TJ; Brandine, GS; Brilhante, RS; Castelo-Branco, DS; Cordeiro, RA; Guedes, GM; Melo, LM; Moreira, JL; Paiva, MA; Pereira-Neto, WA; Ponte, YB; Rocha, MF; Sales, JA; Sidrim, JJ | 1 |
Cao, YB; Chen, J; Han, B; Jiang, YY; Yu, YQ | 1 |
Alvarez-Rueda, N; Fleury, A; Le Pape, P; Logé, C; Morio, F; Pagniez, F; Robert, E | 1 |
Garvey, EP; Hoekstra, WJ; Kelly, DE; Kelly, SL; Nes, WD; Parker, JE; Price, CL; Schotzinger, RJ; Warrilow, AG | 1 |
Koli, SH; Patil, CD; Patil, SV; Suryawanshi, RK | 1 |
Hampe, IAI; Hertlein, T; Morschhäuser, J; Ohlsen, K; Popp, C; Rogers, PD | 1 |
Adelantado, N; Daum, G; Ferrer, P; Feussner, I; García-Ortega, X; Grillitsch, K; Monforte, S; Tarazona, P; Valero, F | 1 |
Shao, J; Shi, G; Wang, C; Wang, T; Wu, D | 1 |
Demuyser, L; Fiori, A; Herrera-Malaver, B; Swinnen, E; Van Dijck, P; Vestrepen, K | 1 |
Elkahoui, S; Essid, R; Gharbi, D; Hammami, M; Hamouda, TB; Karkouch, I; Limam, F; Tabbene, O | 1 |
Bujdáková, H; Černáková, L; Dižová, S | 1 |
Huang, Z; Liu, W; Ma, K; Shi, P; Wang, Q; Yang, Z | 1 |
Bhattacharya, S; Fries, BC | 1 |
Altamirano, S; Kozubowski, L; Simmons, C | 1 |
Bhattacharya, S; Esquivel, BD; White, TC | 1 |
Deng, L; Liu, JF; Wang, F; Wang, SQ; Wang, T | 1 |
Keniya, MV; Monk, BC; Ruma, YN; Tyndall, JDA | 1 |
Ahmad, K; Fatima, Z; Hameed, S; Singh, S | 1 |
Chen, J; Ding, X; Hu, S; Tan, X; Wang, C; Xia, Z; Yang, R; Yu, H; Zhang, D | 1 |
Franz, KJ; Hunsaker, EW | 1 |
Bosch, C; Botha, A; Toplis, B; Volschenk, H; Vreulink, JM | 1 |
Bandara, HMHN; Cheung, BPK; Hugenholtz, P; Samaranayake, LP; Vanwonterghem, I; Wood, DLA | 1 |
Butler, G; Califórnia, R; Cavalheiro, M; Chibana, H; Galocha, M; Ola, M; Pais, P; Takahashi-Nakaguchi, A; Teixeira, MC; Viana, R | 1 |
Capilla, J; Guarro, J; López-Fernández, L; Martin-Vicente, A; Navarro-Rodríguez, P | 1 |
Carmello, JC; Dias, LM; Jordão, CC; Klein, MI; Pavarina, AC | 1 |
Fattouh, N; Geukgeuzian, G; Hdayed, D; Khalaf, RA; Tokajian, S | 1 |
Bernat, P; Krasowska, A; Muraszko, J; Suchodolski, J | 1 |
Doorley, L; Kelly, SL; Krysan, DJ; Moye-Rowley, WS; Murante, D; Ollinger, TL; Parker, JE; Rogers, PD; Simonicova, L; Stamnes, MA; Vu, B | 1 |
Afonso, G; Amaral, C; da Silva, SM; Gaspar-Cordeiro, A; Pimentel, C | 1 |
Basu, P; Elias, R; Fridman, M | 1 |
Bautista-Crescencio, C; Chamorro-Cevallos, G; Escalante, CH; Gonzalez-Silva, A; Hernández-Rodríguez, C; Madrigal-Aguilar, DA; Ortiz-Álvarez, J; Rosales-Acosta, B; Sánchez-Navarrete, J; Tamariz, J; Villa-Tanaca, L | 1 |
Bácskay, I; Balla, N; Csillag, K; Jakab, Á; Kovács, ÁT; Kovács, F; Kovács, R; Majoros, L; Nagy-Köteles, C; Nemes, D; Pócsi, I; Ragyák, Á; Sajtos, Z; Tóth, Z | 1 |
Esfahani, A; Eybpoosh, S; Ghane, M; Omran, AN; Razzaghi-Abyaneh, M; Salehi, Z; Shams-Ghahfarokhi, M | 1 |
Moye-Rowley, WS; Vu, BG | 1 |
Lao, AR; Moron-Espiritu, LS; Yu, PK | 1 |
Behbehani, JM; Irshad, M; Karched, M; Shreaz, S | 1 |
Derkacz, D; Krasowska, A | 1 |
Beilharz, TH; Koch, B; Lo, TL; Olivier, FAB; Powell, DR; Traven, A; Weerasinghe, H; Yau, KPS | 1 |
Benedetti, MD; Braga, SFP; Caldas, IS; Campos Péret, VA; Carvalho, DT; Johann, S; Reis, RCFM; Santana, LFA; Souza, TB | 1 |
Chang, L; Cheng, X; Duan, C; Li, Y; Li, Z; Sui, X; Wang, Y; Xu, P; Yan, R; Zhang, Z | 1 |
Chen, Z; Cheng, JX; Dong, PT; Eldesouky, HE; Jusuf, S; Lin, H; Salama, EA; Seleem, MN; Wang, Z; Zhan, Y; Zhang, M; Zong, C | 1 |
Choy, HL; Doering, TL; Gaylord, EA | 1 |
3 review(s) available for fluconazole and ergosterol
Article | Year |
---|---|
[Rational use of antimycotics against yeast infections].
Topics: Amphotericin B; Antifungal Agents; Candida; Candida albicans; Candidiasis; Chemistry, Pharmaceutical; Drug Resistance, Microbial; Ergosterol; Fluconazole; Humans; Mycoses; Yeasts | 1995 |
Molecular epidemiology, antifungal susceptibility, and ERG11 gene mutation of Candida species isolated from vulvovaginal candidiasis: Comparison between recurrent and non-recurrent infections.
Topics: Antifungal Agents; Candida; Candida albicans; Candida glabrata; Candida parapsilosis; Candida tropicalis; Candidiasis, Vulvovaginal; Drug Resistance, Fungal; Ergosterol; Female; Fluconazole; Fungal Proteins; Humans; Microbial Sensitivity Tests; Molecular Epidemiology; Mutation; Peptide Hydrolases; Phospholipases | 2022 |
Quantitative proteomics revealed the transition of ergosterol biosynthesis and drug transporters processes during the development of fungal fluconazole resistance.
Topics: Antifungal Agents; Candida albicans; Ergosterol; Fluconazole; Membrane Transport Proteins; Proteome; Proteomics; Sterols | 2023 |
117 other study(ies) available for fluconazole and ergosterol
Article | Year |
---|---|
Abc1p is a multidrug efflux transporter that tips the balance in favor of innate azole resistance in Candida krusei.
Topics: Amino Acid Sequence; Animals; Antifungal Agents; ATP-Binding Cassette Transporters; Azoles; Blotting, Northern; Blotting, Southern; Candida; Candidiasis; Cell Membrane; Chromosomes, Fungal; Drug Resistance, Fungal; Endoplasmic Reticulum; Humans; Phenotype; Plasmids; Reverse Transcriptase Polymerase Chain Reaction; Saccharomyces cerevisiae | 2009 |
Effects of fluconazole on the sterol and carbohydrate composition of four species of Candida.
Topics: Candida; Candida albicans; Carbohydrates; Cell Wall; Chitin; Ergosterol; Fluconazole; Glucans; Lanosterol; Mannans; Sterols | 1992 |
A novel method for studying ergosterol biosynthesis by a cell-free preparation of Aspergillus fumigatus and its inhibition by azole antifungal agents.
Topics: Antifungal Agents; Aspergillus fumigatus; Autoradiography; Azoles; Chromatography, Thin Layer; Ergosterol; Fluconazole; Gas Chromatography-Mass Spectrometry; Hydrogen-Ion Concentration; Itraconazole; Ketoconazole; Molecular Structure | 1990 |
Resistance to fluconazole in Candida albicans from AIDS patients correlated with reduced intracellular accumulation of drug.
Topics: AIDS-Related Opportunistic Infections; Antifungal Agents; Candida albicans; Candidiasis, Chronic Mucocutaneous; Cholestadienols; Cytochrome P-450 Enzyme System; Drug Resistance, Microbial; Ergosterol; Fluconazole; Humans; Lanosterol; Microbial Sensitivity Tests; Oxidoreductases; Sterol 14-Demethylase | 1995 |
Resistant P45051A1 activity in azole antifungal tolerant Cryptococcus neoformans from AIDS patients.
Topics: AIDS-Related Opportunistic Infections; Cryptococcosis; Cryptococcus neoformans; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Resistance, Microbial; Drug Tolerance; Ergosterol; Fluconazole; Humans; Itraconazole; Ketoconazole; Microbial Sensitivity Tests; Microsomes; Oxidoreductases; Sterol 14-Demethylase; Sterols; Treatment Failure | 1995 |
Sterol composition of Cryptococcus neoformans in the presence and absence of fluconazole.
Topics: Cholestadienols; Cryptococcus neoformans; Ergosterol; Fluconazole; Humans; Microbial Sensitivity Tests; Phytosterols; Sterols | 1994 |
Pneumocystis carinii is resistant to imidazole antifungal agents.
Topics: Animals; Antifungal Agents; Ergosterol; Female; Fluconazole; Gas Chromatography-Mass Spectrometry; Itraconazole; Ketoconazole; Miconazole; Pneumocystis; Rats; Rats, Sprague-Dawley; Triazoles | 1994 |
Comparison of D0870, a new triazole antifungal agent, to fluconazole for inhibition of Candida albicans cytochrome P-450 by using in vitro assays.
Topics: Antifungal Agents; Candida albicans; Cytochrome P-450 Enzyme System; Ergosterol; Fluconazole; Gas Chromatography-Mass Spectrometry; Humans; Microbial Sensitivity Tests; Microsomes; Structure-Activity Relationship; Triazoles | 1996 |
Inhibition of 2,3-oxidosqualene-lanosterol cyclase in Candida albicans by pyridinium ion-based inhibitors.
Topics: Amphotericin B; Antifungal Agents; Candida albicans; Drug Resistance, Microbial; Enzyme Inhibitors; Ergosterol; Fluconazole; Intramolecular Transferases; Isomerases; Pyridinium Compounds | 1996 |
In vitro activity of fluconazole on Candida albicans.
Topics: Antifungal Agents; Candida albicans; Ergosterol; Fluconazole; Microbial Sensitivity Tests | 1996 |
Hypothesis on the mechanism of resistance to fluconazole in Histoplasma capsulatum.
Topics: Adult; AIDS-Related Opportunistic Infections; Antifungal Agents; Drug Resistance, Microbial; Ergosterol; Fluconazole; Histoplasma; Histoplasmosis; Humans; Itraconazole; Male; Microbial Sensitivity Tests; Polymerase Chain Reaction | 1997 |
Characterization of Saccharomyces cerevisiae CYP61, sterol delta22-desaturase, and inhibition by azole antifungal agents.
Topics: Antifungal Agents; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Ergosterol; Fluconazole; Ketoconazole; Oxidoreductases; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Spectrophotometry, Atomic; Sterol 14-Demethylase | 1997 |
In-vitro activity of D0870, a new triazole antifungal drug, in comparison with fluconazole and itraconazole against Aspergillus fumigatus and Candida krusei.
Topics: Antifungal Agents; Aspergillus fumigatus; Candida; Carbon Monoxide; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Ergosterol; Fluconazole; Itraconazole; Time Factors; Triazoles | 1997 |
Rapid, transient fluconazole resistance in Candida albicans is associated with increased mRNA levels of CDR.
Topics: Antifungal Agents; ATP-Binding Cassette Transporters; Candida albicans; Drug Resistance, Microbial; Ergosterol; Fluconazole; RNA, Messenger | 1998 |
Mechanism of fluconazole resistance in Candida krusei.
Topics: Antifungal Agents; Candida; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Resistance, Microbial; Ergosterol; Fluconazole; Oxidoreductases; Sterol 14-Demethylase | 1998 |
Membrane fluidity affects functions of Cdr1p, a multidrug ABC transporter of Candida albicans.
Topics: ATP-Binding Cassette Transporters; Candida albicans; Drug Resistance, Microbial; Drug Resistance, Multiple; Ergosterol; Estradiol; Fluconazole; Fungal Proteins; Membrane Fluidity; Membrane Transport Proteins; Rhodamines; Saccharomyces cerevisiae; Transformation, Genetic | 1999 |
The G464S amino acid substitution in Candida albicans sterol 14alpha-demethylase causes fluconazole resistance in the clinic through reduced affinity.
Topics: Amino Acid Sequence; Amino Acid Substitution; Antifungal Agents; Candida albicans; Carbon Monoxide; Catalysis; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Resistance, Microbial; Ergosterol; Fluconazole; Heme; Inhibitory Concentration 50; Kinetics; Mutagenesis, Site-Directed; Oxidation-Reduction; Oxidoreductases; Protein Binding; Saccharomyces cerevisiae; Spectrum Analysis; Sterol 14-Demethylase | 1999 |
Quantitation of ergosterol content: novel method for determination of fluconazole susceptibility of Candida albicans.
Topics: Antifungal Agents; Candida albicans; Drug Resistance, Microbial; Ergosterol; Fluconazole; Microbial Sensitivity Tests; Reproducibility of Results | 1999 |
Phospholipid and sterol analysis of plasma membranes of azole-resistant Candida albicans strains.
Topics: AIDS-Related Opportunistic Infections; Antifungal Agents; Candida albicans; Candidiasis; Cell Membrane; Drug Resistance, Microbial; Ergosterol; Fluconazole; Hematologic Neoplasms; Humans; Microbial Sensitivity Tests; Phospholipids | 2000 |
Quantitation of Candida albicans ergosterol content improves the correlation between in vitro antifungal susceptibility test results and in vivo outcome after fluconazole treatment in a murine model of invasive candidiasis.
Topics: Animals; Antifungal Agents; Candida albicans; Candidiasis; Disease Models, Animal; Ergosterol; Female; Fluconazole; Kidney; Mice; Microbial Sensitivity Tests; Statistics as Topic; Treatment Outcome | 2000 |
Modulation of fluconazole sensitivity by the interaction of mitochondria and erg3p in Saccharomyces cerevisiae.
Topics: Antifungal Agents; Culture Media; Drug Resistance, Microbial; Ergosterol; Fluconazole; Microbial Sensitivity Tests; Mitochondria; Mutation; Oxidative Phosphorylation; Oxidoreductases; Saccharomyces cerevisiae; Sterols | 2000 |
Efflux-mediated resistance to fluconazole could be modulated by sterol homeostasis in Saccharomyces cerevisiae.
Topics: Antifungal Agents; ATP-Binding Cassette Transporters; Cloning, Molecular; Culture Media; DNA-Binding Proteins; Drug Resistance, Microbial; Ergosterol; Fluconazole; Homeostasis; Membrane Proteins; Microbial Sensitivity Tests; Mutation; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Sterols; Trans-Activators; Transcription Factors | 2000 |
Comparison of visual and spectrophotometric methods of broth microdilution MIC end point determination and evaluation of a sterol quantitation method for in vitro susceptibility testing of fluconazole and itraconazole against trailing and nontrailing Cand
Topics: Antifungal Agents; Candida; Candidiasis; Endpoint Determination; Ergosterol; Fluconazole; Indicator Dilution Techniques; Itraconazole; Microbial Sensitivity Tests; Spectrophotometry; Sterols | 2002 |
A novel mechanism of fluconazole resistance associated with fluconazole sequestration in Candida albicans isolates from a myelofibrosis patient.
Topics: Antifungal Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Candida albicans; Candidiasis; Cytochrome P-450 Enzyme System; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Humans; Membrane Transport Proteins; Microscopy, Electron; Oxidoreductases; Primary Myelofibrosis; Reverse Transcriptase Polymerase Chain Reaction; RNA, Fungal; Spheroplasts; Sterol 14-Demethylase | 2002 |
Evaluation of differential gene expression in fluconazole-susceptible and -resistant isolates of Candida albicans by cDNA microarray analysis.
Topics: Antifungal Agents; Candida albicans; Carbohydrate Metabolism; Cell Wall; DNA Probes; DNA, Complementary; DNA, Fungal; Drug Resistance, Fungal; Ergosterol; Fluconazole; Gene Expression Regulation, Fungal; Iron; Microbial Sensitivity Tests; Oligonucleotide Array Sequence Analysis; Reverse Transcriptase Polymerase Chain Reaction; RNA, Bacterial | 2002 |
Proliferation of intracellular structure corresponding to reduced affinity of fluconazole for cytochrome P-450 in two low-susceptibility strains of Candida albicans isolated from a Japanese AIDS patient.
Topics: AIDS-Related Opportunistic Infections; Amino Acid Substitution; Antifungal Agents; Candida albicans; Candidiasis, Oral; Cytochrome P-450 Enzyme System; Drug Resistance, Fungal; Ergosterol; Fluconazole; Humans; Japan; Microbial Sensitivity Tests; Microscopy, Electron; Multienzyme Complexes; Oxidoreductases | 2003 |
Modulatory effect of cAMP on fungal ergosterol level and inhibitory activity of azole drugs.
Topics: Amphotericin B; Antifungal Agents; Atropine; Bucladesine; Candida albicans; Chromatography, Gas; Cryptococcus neoformans; Cyclic AMP; Drug Synergism; Ergosterol; Fluconazole; Ketoconazole; Microbial Sensitivity Tests; Phosphodiesterase Inhibitors | 2003 |
Antifungal activity of fluconazole in combination with lovastatin and their effects on gene expression in the ergosterol and prenylation pathways in Candida albicans.
Topics: Base Sequence; Candida albicans; DNA Primers; Drug Synergism; Ergosterol; Fluconazole; Gene Expression Regulation, Fungal; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Lovastatin; Microbial Sensitivity Tests; Protein Prenylation; Reverse Transcriptase Polymerase Chain Reaction | 2003 |
Genome-wide expression profiling reveals genes associated with amphotericin B and fluconazole resistance in experimentally induced antifungal resistant isolates of Candida albicans.
Topics: Amphotericin B; Antifungal Agents; Candida albicans; Candidiasis; Cytochrome P-450 Enzyme System; DNA Primers; DNA, Complementary; Drug Resistance, Fungal; Ergosterol; Fluconazole; Gene Expression Profiling; Genes, Fungal; Genome, Fungal; Humans; Microbial Sensitivity Tests; Oligonucleotide Array Sequence Analysis; Oxidoreductases; Phenotype; Protein Folding; Reverse Transcriptase Polymerase Chain Reaction; RNA, Fungal; Saccharomyces cerevisiae; Sterol 14-Demethylase; Sterols | 2004 |
The combination effects of phenolic compounds and fluconazole on the formation of ergosterol in Candida albicans determined by high-performance liquid chromatography/tandem mass spectrometry.
Topics: Caffeic Acids; Candida albicans; Chromatography, High Pressure Liquid; Ergosterol; Fluconazole; Lanosterol; Naphthalenes; Phenols; Resveratrol; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization; Squalene; Stilbenes | 2005 |
Characterization of mechanisms of fluconazole resistance in a Candida albicans isolate from a Japanese patient with chronic mucocutaneous candidiasis.
Topics: Antifungal Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Candida albicans; Candidiasis, Chronic Mucocutaneous; Cytochrome P-450 Enzyme System; DNA, Fungal; Drug Resistance, Multiple, Fungal; Ergosterol; Female; Fluconazole; Fungal Proteins; Humans; Membrane Transport Proteins; Microbial Sensitivity Tests; Oxidoreductases; Point Mutation; Polymerase Chain Reaction; RNA, Messenger; Sequence Analysis, DNA; Sterol 14-Demethylase | 2004 |
Deletion of PDE2, the gene encoding the high-affinity cAMP phosphodiesterase, results in changes of the cell wall and membrane in Candida albicans.
Topics: Antifungal Agents; Candida albicans; Cell Wall; Cyclic Nucleotide Phosphodiesterases, Type 2; Ergosterol; Fluconazole; Glucans; Membranes; Microbial Sensitivity Tests; Microscopy, Electron, Transmission; Mutation; Phosphoric Diester Hydrolases; Sodium Dodecyl Sulfate | 2005 |
Hsp90 potentiates the rapid evolution of new traits: drug resistance in diverse fungi.
Topics: AIDS-Related Opportunistic Infections; Antifungal Agents; Aspergillosis; Aspergillus; Biological Evolution; Calcineurin; Calcineurin Inhibitors; Candida albicans; Candidiasis; Caspofungin; Cyclophilin A; Drug Resistance, Fungal; Echinocandins; Ergosterol; Fluconazole; HSP90 Heat-Shock Proteins; Humans; Lipopeptides; Mutation; Peptides, Cyclic; Phenotype; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Selection, Genetic | 2005 |
Establishing surrogate markers for fluconazole resistance in Candida albicans.
Topics: Antifungal Agents; Biomarkers; Candida albicans; Candidiasis; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Membrane Transport Proteins; Microbial Sensitivity Tests; Mutation | 2005 |
Up-regulation of ERG11 gene among fluconazole-resistant Candida albicans generated in vitro: is there any clinical implication?
Topics: Antifungal Agents; Candida albicans; Candidiasis; Drug Resistance, Fungal; Ergosterol; Female; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Humans; Microbial Sensitivity Tests; Up-Regulation | 2007 |
Aneuploidy and isochromosome formation in drug-resistant Candida albicans.
Topics: Aneuploidy; Antifungal Agents; Azoles; Candida albicans; Centromere; Chromosomes, Fungal; Cytochrome P-450 Enzyme System; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Dosage; Gene Expression Profiling; Genes, Fungal; Isochromosomes; Karyotyping; Molecular Sequence Data; Repetitive Sequences, Nucleic Acid; Sequence Analysis, DNA; Transcription Factors; Trisomy | 2006 |
Unexpected link between iron and drug resistance of Candida spp.: iron depletion enhances membrane fluidity and drug diffusion, leading to drug-susceptible cells.
Topics: Antifungal Agents; Candida; Copper; Culture Media; Diffusion; Down-Regulation; Drug Resistance, Fungal; Drug Synergism; Ergosterol; Fluconazole; Fluorescence Polarization Immunoassay; Genotype; Hybridization, Genetic; Iron; Iron Chelating Agents; Membrane Fluidity; Microbial Sensitivity Tests; RNA, Fungal | 2006 |
Targeting the calcineurin pathway enhances ergosterol biosynthesis inhibitors against Trichophyton mentagrophytes in vitro and in a human skin infection model.
Topics: Antifungal Agents; Calcineurin; Colony Count, Microbial; Culture Media; Cyclosporine; Drug Synergism; Drug Therapy, Combination; Ergosterol; Fluconazole; Humans; Immunosuppressive Agents; Naphthalenes; Signal Transduction; Skin; Tacrolimus; Terbinafine; Tinea; Trichophyton | 2007 |
A gain-of-function mutation in the transcription factor Upc2p causes upregulation of ergosterol biosynthesis genes and increased fluconazole resistance in a clinical Candida albicans isolate.
Topics: Antifungal Agents; Candida albicans; Candidiasis; Codon, Nonsense; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Humans; Mutation; Transcription Factors; Up-Regulation | 2008 |
The expression of genes involved in the ergosterol biosynthesis pathway in Candida albicans and Candida dubliniensis biofilms exposed to fluconazole.
Topics: Antifungal Agents; Biofilms; Candida; Candida albicans; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Humans; Microbial Sensitivity Tests | 2009 |
The effect of plagiochin E alone and in combination with fluconazole on the ergosterol biosynthesis of Candida albicans.
Topics: Antifungal Agents; Bridged-Ring Compounds; Candida albicans; Ergosterol; Fluconazole; Gene Expression Regulation, Fungal; Sterols; Stilbenes | 2009 |
Dynamics of in vitro acquisition of resistance by Candida parapsilosis to different azoles.
Topics: Antifungal Agents; Biosynthetic Pathways; Candida; Drug Resistance, Fungal; Ergosterol; Fluconazole; Humans; Microbial Sensitivity Tests; Mutation; Pyrimidines; Triazoles; Voriconazole | 2009 |
In vitro and in vivo antifungal activities of aminopiperidine derivatives, novel ergosterol synthesis inhibitors.
Topics: Animals; Antifungal Agents; Candida albicans; Candidiasis; Ergosterol; Female; Fluconazole; Fungi; Inhibitory Concentration 50; Kaplan-Meier Estimate; Mice; Microbial Sensitivity Tests; Molecular Structure; Piperidines | 2010 |
Mechanism of the synergistic effect of amiodarone and fluconazole in Candida albicans.
Topics: Amiodarone; Animals; Antifungal Agents; Calcium; Candida albicans; Candidiasis; Down-Regulation; Drug Resistance, Fungal; Drug Synergism; Enzyme Inhibitors; Ergosterol; Female; Fluconazole; Gene Expression Profiling; Genes, Fungal; Hyphae; Lysosomes; Mice; Mice, Inbred BALB C; Up-Regulation; Vacuoles | 2010 |
Requirement for ergosterol in V-ATPase function underlies antifungal activity of azole drugs.
Topics: Amiodarone; Animals; Antifungal Agents; Candida albicans; Drug Synergism; Enzyme Inhibitors; Ergosterol; Female; Fluconazole; Mice; Mice, Inbred BALB C; Protons; Saccharomyces cerevisiae; Vacuolar Proton-Translocating ATPases; Vacuoles | 2010 |
Identification and characterization of four azole-resistant erg3 mutants of Candida albicans.
Topics: Amphotericin B; Antifungal Agents; Azoles; Candida albicans; Clotrimazole; Drug Resistance, Fungal; Ergosterol; Fluconazole; Itraconazole; Ketoconazole; Microbial Sensitivity Tests; Mutation; Oxidoreductases; Pyrimidines; Triazoles; Voriconazole | 2010 |
Complementation of a Saccharomyces cerevisiae ERG11/CYP51 (sterol 14α-demethylase) doxycycline-regulated mutant and screening of the azole sensitivity of Aspergillus fumigatus isoenzymes CYP51A and CYP51B.
Topics: Anti-Bacterial Agents; Aspergillus fumigatus; Azoles; Clotrimazole; Cytochrome P-450 Enzyme System; Doxycycline; Ergosterol; Fluconazole; Fungal Proteins; Genetic Complementation Test; Itraconazole; Pyrimidines; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Triazoles; Voriconazole | 2010 |
An A643V amino acid substitution in Upc2p contributes to azole resistance in well-characterized clinical isolates of Candida albicans.
Topics: Amino Acid Substitution; Antifungal Agents; Azoles; Candida albicans; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Humans; Microbial Sensitivity Tests; Sequence Analysis, DNA; Trans-Activators | 2011 |
Transcription factors CgUPC2A and CgUPC2B regulate ergosterol biosynthetic genes in Candida glabrata.
Topics: Antifungal Agents; Candida glabrata; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Genes, Fungal; Lovastatin; Saccharomyces cerevisiae Proteins; Sterols; Trans-Activators; Transcription Factors | 2011 |
Curcumin as a promising anticandidal of clinical interest.
Topics: Antifungal Agents; Candida albicans; Candida glabrata; Curcumin; Ergosterol; Fluconazole; Glucose; Microbial Sensitivity Tests; Peptide Hydrolases; Proton-Translocating ATPases | 2011 |
Cdr2p contributes to fluconazole resistance in Candida dubliniensis clinical isolates.
Topics: Antifungal Agents; Candida; Cell Membrane; DNA, Ribosomal Spacer; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Genes, Fungal; Genotyping Techniques; Humans; Membrane Transport Proteins; Microbial Sensitivity Tests | 2011 |
Anticandidal activity of Cassia fistula and its effect on ergosterol biosynthesis.
Topics: Anthraquinones; Antifungal Agents; Candida albicans; Candida glabrata; Candida tropicalis; Cassia; Cell Membrane; Ergosterol; Fluconazole; Fruit; Medicine, Traditional; Microbial Sensitivity Tests; Plant Extracts; Seeds | 2011 |
Cross-species discovery of syncretic drug combinations that potentiate the antifungal fluconazole.
Topics: Animals; Antifungal Agents; Candida; Computational Biology; Cryptococcus; Drug Resistance, Fungal; Drug Synergism; Ergosterol; Fluconazole; Gene Expression Profiling; Insecta; Microbial Sensitivity Tests; Saccharomyces; Species Specificity | 2011 |
Amino acid substitutions at the major insertion loop of Candida albicans sterol 14alpha-demethylase are involved in fluconazole resistance.
Topics: Amino Acid Sequence; Amino Acid Substitution; Antifungal Agents; Candida albicans; Drug Resistance, Microbial; Ergosterol; Fluconazole; Molecular Sequence Data; Mutagenesis, Site-Directed; Sterol 14-Demethylase | 2011 |
SREBP-dependent triazole susceptibility in Aspergillus fumigatus is mediated through direct transcriptional regulation of erg11A (cyp51A).
Topics: Animals; Antifungal Agents; Aspergillosis; Aspergillus fumigatus; Cytochrome P-450 Enzyme System; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Genetic Complementation Test; Genotype; Humans; Microbial Sensitivity Tests; Organisms, Genetically Modified; Pyrimidines; Real-Time Polymerase Chain Reaction; Sterol Regulatory Element Binding Proteins; Transcription, Genetic; Triazoles; Voriconazole | 2012 |
Dynamic interaction between fluconazole and amphotericin B against Cryptococcus gattii.
Topics: Amphotericin B; Antifungal Agents; Cell Membrane; Cryptococcus gattii; Culture Media; Dose-Response Relationship, Drug; Drug Antagonism; Drug Synergism; Ergosterol; Fluconazole; Humans; Microbial Sensitivity Tests; Species Specificity; Spectrophotometry | 2012 |
Facultative sterol uptake in an ergosterol-deficient clinical isolate of Candida glabrata harboring a missense mutation in ERG11 and exhibiting cross-resistance to azoles and amphotericin B.
Topics: Amphotericin B; Antifungal Agents; Azoles; Base Sequence; Biological Transport; Candida glabrata; Drug Resistance, Multiple, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Humans; Microbial Sensitivity Tests; Mutation, Missense; Pyrimidines; Saccharomyces cerevisiae; Sequence Analysis, DNA; Sterol 14-Demethylase; Sterols; Triazoles; Voriconazole | 2012 |
Gain-of-function mutations in UPC2 are a frequent cause of ERG11 upregulation in azole-resistant clinical isolates of Candida albicans.
Topics: Antifungal Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Candida albicans; Cytochrome P-450 Enzyme System; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Genome, Fungal; Mutation, Missense; Transcription Factors; Transcription, Genetic; Up-Regulation | 2012 |
A defect in iron uptake enhances the susceptibility of Cryptococcus neoformans to azole antifungal drugs.
Topics: Antifungal Agents; Azoles; Biological Transport; Ceruloplasmin; Cryptococcosis; Cryptococcus neoformans; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Deletion; Gene Expression Regulation, Fungal; Humans; Iron; Microbial Sensitivity Tests | 2012 |
Azole susceptibility and transcriptome profiling in Candida albicans mitochondrial electron transport chain complex I mutants.
Topics: Antifungal Agents; ATP-Binding Cassette Transporters; Candida albicans; Drug Resistance, Fungal; Electron Transport; Electron Transport Complex I; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Profiling; Gene Expression Regulation, Fungal; Microbial Sensitivity Tests; Mitochondria; Mutation; Peroxisomes; Transcriptome | 2013 |
Real-time microscopic observation of Candida biofilm development and effects due to micafungin and fluconazole.
Topics: Antifungal Agents; Biofilms; Candida albicans; Echinocandins; Ergosterol; Fluconazole; Glucans; Hyphae; Kinetics; Lipopeptides; Micafungin; Microscopy; Time-Lapse Imaging | 2013 |
Effect of farnesol on growth, ergosterol biosynthesis, and cell permeability in Coccidioides posadasii.
Topics: Antifungal Agents; Cell Membrane Permeability; Coccidioides; Drug Synergism; Drug Therapy, Combination; Ergosterol; Farnesol; Fluconazole; Microbial Sensitivity Tests; Osmolar Concentration; Osmotic Pressure; Sodium Chloride | 2013 |
Comparison of sterol import under aerobic and anaerobic conditions in three fungal species, Candida albicans, Candida glabrata, and Saccharomyces cerevisiae.
Topics: Aerobiosis; Anaerobiosis; Antifungal Agents; Candida albicans; Candida glabrata; Cholesterol; Culture Media; Ergosterol; Esterification; Fluconazole; Gene Knockout Techniques; Microbial Sensitivity Tests; Saccharomyces cerevisiae | 2013 |
Molecular mechanisms of drug resistance in clinical Candida species isolated from Tunisian hospitals.
Topics: Amino Acid Sequence; Amino Acid Substitution; Amphotericin B; Antifungal Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azoles; Base Sequence; Candida albicans; Candida glabrata; Candida tropicalis; Candidiasis; Cytochrome P-450 Enzyme System; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Humans; Microbial Sensitivity Tests; Molecular Sequence Data; Mutation; Polyenes; Pyrimidines; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Sequence Analysis, DNA; Triazoles; Tunisia; Voriconazole | 2013 |
Antifungal mechanism of essential oil from Anethum graveolens seeds against Candida albicans.
Topics: Anethum graveolens; Antifungal Agents; Candida albicans; Cell Membrane; Cysteine; Ergosterol; Flow Cytometry; Fluconazole; Membrane Potential, Mitochondrial; Microbial Sensitivity Tests; Mitochondria; Nystatin; Oils, Volatile; Oxidoreductases; Plant Oils; Reactive Oxygen Species; Seeds | 2013 |
Potentiation of azole antifungals by 2-adamantanamine.
Topics: Amantadine; Animals; Antifungal Agents; Biofilms; Candida albicans; Candidiasis, Cutaneous; Culture Media; Drug Evaluation, Preclinical; Drug Synergism; Ergosterol; Fluconazole; Gene Expression Profiling; Guinea Pigs; Hep G2 Cells; Hepatocytes; Humans; Miconazole | 2013 |
Interaction of azole compounds with DOPC and DOPC/ergosterol bilayers by spin probe EPR spectroscopy: implications for antifungal activity.
Topics: Antifungal Agents; Azoles; Candida albicans; Cyclic N-Oxides; Electron Spin Resonance Spectroscopy; Ergosterol; Fluconazole; Lipid Bilayers; Phosphatidylcholines; Spin Labels; Temperature | 2013 |
UPC2A is required for high-level azole antifungal resistance in Candida glabrata.
Topics: Antifungal Agents; Azoles; Candida albicans; Candida glabrata; Cytochrome P-450 Enzyme System; Drug Resistance, Fungal; Ergosterol; Fluconazole; Gene Expression Regulation, Fungal; Microbial Sensitivity Tests; Protein Isoforms; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Sequence Homology, Amino Acid; Trans-Activators; Transcription Factors; Transcription, Genetic | 2014 |
Ascorbic acid inhibition of Candida albicans Hsp90-mediated morphogenesis occurs via the transcriptional regulator Upc2.
Topics: Ascorbic Acid; Benzoquinones; Candida albicans; Cytochrome P-450 Enzyme System; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; HSP90 Heat-Shock Proteins; Hyphae; Lactams, Macrocyclic; Morphogenesis; Temperature; Trans-Activators | 2014 |
Synergistic activity of magnolol with azoles and its possible antifungal mechanism against Candida albicans.
Topics: Antifungal Agents; Azoles; Biphenyl Compounds; Candida albicans; Drug Synergism; Ergosterol; Fluconazole; Fungal Proteins; Lignans; Membrane Transport Proteins; Up-Regulation | 2015 |
Structural mechanism of ergosterol regulation by fungal sterol transcription factor Upc2.
Topics: Antifungal Agents; Binding Sites; Cell Nucleus; Chromatography, Gel; Chromatography, High Pressure Liquid; Chromatography, Reverse-Phase; Crystallography, X-Ray; Cytosol; Drug Resistance, Microbial; Ergosterol; Fluconazole; Green Fluorescent Proteins; Ligands; Mass Spectrometry; Models, Biological; Mutant Proteins; Protein Multimerization; Protein Structure, Secondary; Protein Structure, Tertiary; Reference Standards; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Spectrometry, Fluorescence; Trans-Activators; Zinc Fingers | 2015 |
Mechanisms of azole resistance in Candida albicans clinical isolates from Shanghai, China.
Topics: Amino Acid Substitution; Antifungal Agents; Azoles; Candida albicans; China; Drug Resistance, Fungal; Ergosterol; Flow Cytometry; Fluconazole; Genes, Fungal; Genes, MDR; Humans; Lanosterol; Mutation, Missense; Real-Time Polymerase Chain Reaction; Sequence Analysis, DNA | 2015 |
[Effect of Huanglian Jiedu decoction in combination with fluconazole on ergosterol of fluconazole-resistant Candida albicans].
Topics: Antifungal Agents; Candida albicans; Drug Resistance, Fungal; Drug Synergism; Drugs, Chinese Herbal; Ergosterol; Fluconazole; Microbial Sensitivity Tests | 2015 |
An Antifungal Benzimidazole Derivative Inhibits Ergosterol Biosynthesis and Reveals Novel Sterols.
Topics: Antifungal Agents; Benzimidazoles; Candida; Candida albicans; Candida glabrata; Ergosterol; Fluconazole; Fungal Proteins; High-Throughput Screening Assays; Nocodazole; Small Molecule Libraries; Sterol 14-Demethylase | 2015 |
Inhibitory activity of isoniazid and ethionamide against Cryptococcus biofilms.
Topics: Antifungal Agents; Biofilms; Cell Membrane Permeability; Cryptococcus gattii; Cryptococcus neoformans; Ergosterol; Ethionamide; Fluconazole; Isoniazid; Microbial Sensitivity Tests | 2015 |
Changes in the Sterol Composition of the Plasma Membrane Affect Membrane Potential, Salt Tolerance and the Activity of Multidrug Resistance Pumps in Saccharomyces cerevisiae.
Topics: Antifungal Agents; ATP-Binding Cassette Transporters; Biosynthetic Pathways; Cell Membrane; Drug Resistance, Multiple, Fungal; Ergosterol; Fluconazole; Hydrogen-Ion Concentration; Membrane Potentials; Methyltransferases; Microscopy, Fluorescence; Molecular Structure; Mutation; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Salt Tolerance | 2015 |
Inhibition of heat-shock protein 90 enhances the susceptibility to antifungals and reduces the virulence of Cryptococcus neoformans/Cryptococcus gattii species complex.
Topics: Amphotericin B; Animals; Antifungal Agents; Biofilms; Caenorhabditis elegans; Cell Membrane; Cryptococcosis; Cryptococcus gattii; Cryptococcus neoformans; Ergosterol; Fluconazole; HSP90 Heat-Shock Proteins; Humans; Itraconazole; Melanins; Microbial Sensitivity Tests; Plankton; Voriconazole | 2016 |
Cross-resistance to fluconazole induced by exposure to the agricultural azole tetraconazole: an environmental resistance school?
Topics: Animals; Anti-Allergic Agents; Antifungal Agents; ATP-Binding Cassette Transporters; Candida; Chlorobenzenes; Drug Resistance, Microbial; Ergosterol; Fluconazole; Fungicides, Industrial; Gene Expression Regulation, Fungal; Humans; Itraconazole; Malathion; Microbial Sensitivity Tests; Promethazine; Rhodamines; Sterol 14-Demethylase; Triazoles; Voriconazole | 2016 |
Antifungal activity of Rubus chingii extract combined with fluconazole against fluconazole-resistant Candida albicans.
Topics: Antifungal Agents; Apoptosis; Candida albicans; Cell Cycle; Cell Membrane; Drug Resistance, Fungal; Drug Synergism; Ergosterol; Fluconazole; Microbial Sensitivity Tests; Microscopy, Electron, Transmission; Plant Extracts; Rhodamines; Rubus | 2016 |
The amino acid substitution N136Y in Candida albicans sterol 14alpha-demethylase is involved in fluconazole resistance.
Topics: 14-alpha Demethylase Inhibitors; Amino Acid Substitution; Antifungal Agents; Binding Sites; Candida albicans; Drug Resistance, Fungal; Ergosterol; Fluconazole; Gas Chromatography-Mass Spectrometry; Models, Molecular; Mutagenesis, Site-Directed; Mutant Proteins; Mutation, Missense; Pichia; Protein Conformation; Sterol 14-Demethylase; Transformation, Genetic | 2016 |
The Investigational Drug VT-1129 Is a Highly Potent Inhibitor of Cryptococcus Species CYP51 but Only Weakly Inhibits the Human Enzyme.
Topics: Antifungal Agents; Clotrimazole; Cryptococcus; Enzyme Activation; Ergosterol; Fluconazole; Humans; Itraconazole; Ketoconazole; Lanosterol; Pyridines; Sterol 14-Demethylase; Tetrazoles; Voriconazole | 2016 |
Fluconazole treatment enhances extracellular release of red pigments in the fungus Monascus purpureus.
Topics: Antifungal Agents; Chromatography, Thin Layer; Ergosterol; Fluconazole; Hydrogen-Ion Concentration; Mass Spectrometry; Microbial Sensitivity Tests; Monascus; Pigments, Biological | 2017 |
Competitive Fitness of Fluconazole-Resistant Clinical Candida albicans Strains.
Topics: Antifungal Agents; Candida albicans; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Mutation | 2017 |
The effect of hypoxia on the lipidome of recombinant Pichia pastoris.
Topics: Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Profiling; Glycolysis; Lipid Metabolism; Membrane Lipids; Oxygen; Pichia; Promoter Regions, Genetic; Protein Transport; Proteomics; Recombinant Proteins; Sphingolipids; Sterols; Unfolded Protein Response | 2017 |
Mechanism of berberine-mediated fluconazole-susceptibility enhancement in clinical fluconazole-resistant Candida tropicalis isolates.
Topics: Antifungal Agents; Berberine; Biofilms; Candida tropicalis; Candidiasis; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Humans; Membrane Transport Proteins; Microbial Sensitivity Tests; RNA, Messenger | 2017 |
Mitochondrial Cochaperone Mge1 Is Involved in Regulating Susceptibility to Fluconazole in
Topics: Antifungal Agents; Candida albicans; Candida glabrata; Drug Resistance, Fungal; Ergosterol; Fluconazole; HSP70 Heat-Shock Proteins; Iron; Mitochondrial Membrane Transport Proteins; Mitochondrial Proteins; Molecular Chaperones; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins | 2017 |
Antifungal mechanism of the combination of Cinnamomum verum and Pelargonium graveolens essential oils with fluconazole against pathogenic Candida strains.
Topics: Antifungal Agents; Candida; Cinnamomum zeylanicum; Drug Synergism; Ergosterol; Fluconazole; Oils, Volatile; Pelargonium; Plant Oils | 2017 |
The impact of farnesol in combination with fluconazole on Candida albicans biofilm: regulation of ERG20, ERG9, and ERG11 genes.
Topics: Antifungal Agents; Biofilms; Candida albicans; Dose-Response Relationship, Drug; Drug Synergism; Ergosterol; Farnesol; Fluconazole; Gene Expression Regulation, Fungal; Genes, Fungal; Hyphae; Metabolic Networks and Pathways; Microbial Sensitivity Tests | 2018 |
Fluconazole inhibits cellular ergosterol synthesis to confer synergism with berberine against yeast cells.
Topics: Antifungal Agents; Berberine; Cell Membrane Permeability; Drug Synergism; Ergosterol; Fluconazole; Microbial Sensitivity Tests; Saccharomyces cerevisiae | 2018 |
Enhanced Efflux Pump Activity in Old Candida glabrata Cells.
Topics: Amphotericin B; Antifungal Agents; ATP-Binding Cassette Transporters; Biological Transport; Candida glabrata; Cell Division; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Genes, MDR; Glucosyltransferases; Micafungin; Microbial Sensitivity Tests | 2018 |
Colony and Single Cell Level Analysis of the Heterogeneous Response of
Topics: Antifungal Agents; Biological Variation, Population; Cell Membrane; Cryptococcosis; Cryptococcus neoformans; Drug Resistance, Fungal; Ergosterol; Fluconazole; Humans; Microbial Sensitivity Tests; Optical Imaging; Single-Cell Analysis | 2018 |
Overexpression or Deletion of Ergosterol Biosynthesis Genes Alters Doubling Time, Response to Stress Agents, and Drug Susceptibility in
Topics: Amphotericin B; Antifungal Agents; Biosynthetic Pathways; Drug Resistance, Fungal; Ergosterol; Fluconazole; Gene Deletion; Gene Expression Regulation, Fungal; Genes, Fungal; Saccharomyces cerevisiae | 2018 |
Overexpression of Ecm22 improves ergosterol biosynthesis in Saccharomyces cerevisiae.
Topics: Antifungal Agents; Bioreactors; DNA, Fungal; Ergosterol; Fluconazole; Gene Expression Regulation, Fungal; Microbial Sensitivity Tests; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Transcription Factors | 2018 |
Heterologous Expression of Full-Length Lanosterol 14α-Demethylases of Prominent Fungal Pathogens Candida albicans and Candida glabrata Provides Tools for Antifungal Discovery.
Topics: Amphotericin B; Antifungal Agents; Azoles; Candida albicans; Candida glabrata; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Humans; Itraconazole; Lanosterol; Microbial Sensitivity Tests; Saccharomyces cerevisiae; Sterol 14-Demethylase; Triazoles; Voriconazole | 2018 |
Fungicidal action of geraniol against Candida albicans is potentiated by abrogated CaCdr1p drug efflux and fluconazole synergism.
Topics: Acyclic Monoterpenes; Animals; Antifungal Agents; Biofilms; Caenorhabditis elegans; Candida albicans; Cell Adhesion; Drug Resistance, Fungal; Drug Synergism; Epithelial Cells; Ergosterol; Fluconazole; Fungal Proteins; Humans; Membrane Potential, Mitochondrial; Membrane Transport Proteins; Molecular Docking Simulation; Phospholipases; Protein Binding; Terpenes | 2018 |
Genomic and transcriptome identification of fluconazole-resistant genes for Trichosporon asahii.
Topics: Antifungal Agents; Biosynthetic Pathways; Drug Resistance, Fungal; Ergosterol; Female; Fluconazole; Fungal Proteins; Genomics; Humans; Invasive Fungal Infections; Mutation, Missense; Point Mutation; Saccharomyces cerevisiae; Skin; Transcriptome; Trichosporon; Young Adult | 2020 |
Candida albicans reprioritizes metal handling during fluconazole stress.
Topics: Adaptation, Physiological; Antifungal Agents; Biosynthetic Pathways; Candida albicans; Drug Resistance, Fungal; Ergosterol; Fluconazole; Homeostasis; Metals; Microbial Sensitivity Tests | 2019 |
Nitrogen concentration affects amphotericin B and fluconazole tolerance of pathogenic cryptococci.
Topics: Ammonium Chloride; Amphotericin B; Antifungal Agents; Biosynthetic Pathways; Cryptococcus; Cryptococcus gattii; Cryptococcus neoformans; Culture Media; Ergosterol; Fluconazole; Melanins; Microbial Sensitivity Tests; Nitrogen | 2020 |
Fluconazole resistance in Candida albicans is induced by Pseudomonas aeruginosa quorum sensing.
Topics: Antifungal Agents; Biosynthetic Pathways; Candida albicans; Drug Resistance, Fungal; Ergosterol; Fluconazole; Gene Expression Regulation, Fungal; Microbial Interactions; Pseudomonas aeruginosa; Quorum Sensing | 2020 |
Candida glabrata Transcription Factor Rpn4 Mediates Fluconazole Resistance through Regulation of Ergosterol Biosynthesis and Plasma Membrane Permeability.
Topics: Antifungal Agents; Candida glabrata; Cell Membrane; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Permeability; Transcription Factors | 2020 |
Topics: Antifungal Agents; Azoles; Candida albicans; Candida tropicalis; Candidiasis; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Humans; Microbial Sensitivity Tests; Permeability; Voriconazole | 2020 |
Consecutive treatments with photodynamic therapy and nystatin altered the expression of virulence and ergosterol biosynthesis genes of a fluconazole-resistant Candida albicans in vivo.
Topics: Animals; Antifungal Agents; Candida albicans; Ergosterol; Fluconazole; Mice; Nystatin; Photochemotherapy; Photosensitizing Agents; Virulence | 2021 |
Molecular mechanism of fluconazole resistance and pathogenicity attributes of Lebanese Candida albicans hospital isolates.
Topics: Amino Acid Substitution; Animals; Antifungal Agents; Biofilms; Candida albicans; Candidiasis; Cell Wall; Chitin; Cross Infection; Drug Resistance, Fungal; Ergosterol; Female; Fluconazole; Frameshift Mutation; Fungal Proteins; Genes, Fungal; Humans; Lebanon; Mice; Virulence | 2021 |
Lactate Like Fluconazole Reduces Ergosterol Content in the Plasma Membrane and Synergistically Kills
Topics: Antifungal Agents; Candida albicans; Cell Membrane; Drug Resistance, Fungal; Drug Synergism; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Glucose; Lactic Acid; Membrane Transport Proteins; Microbial Sensitivity Tests; Protein Transport | 2021 |
Loss-of-Function
Topics: Antifungal Agents; Candida glabrata; Ergosterol; Fluconazole; Gene Expression Regulation, Fungal; Methyltransferases; Mutation; Oxidoreductases; Repressor Proteins; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Trans-Activators | 2021 |
Zap1 is required for Candida glabrata response to fluconazole.
Topics: Antifungal Agents; Candida; Candida glabrata; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Microbial Sensitivity Tests | 2022 |
Fluconazole-COX Inhibitor Hybrids: A Dual-Acting Class of Antifungal Azoles.
Topics: Antifungal Agents; Candida; Cyclooxygenase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P450 Family 51; Ergosterol; Fluconazole; Microbial Sensitivity Tests; Stereoisomerism | 2022 |
Antifungal Activity of Fibrate-Based Compounds and Substituted Pyrroles That Inhibit the Enzyme 3-Hydroxy-methyl-glutaryl-CoA Reductase of
Topics: Acyl Coenzyme A; Animals; Antifungal Agents; Candida glabrata; COVID-19; Drug Resistance, Fungal; Ergosterol; Fibric Acids; Fluconazole; Humans; Hydroxymethylglutaryl CoA Reductases; Microbial Sensitivity Tests; Pandemics; Pyrroles | 2022 |
Physiological and transcriptional profiling of surfactin exerted antifungal effect against Candida albicans.
Topics: Antifungal Agents; Candida albicans; Drug Resistance, Fungal; Ergosterol; Ethanol; Fluconazole; Fungal Proteins; Iron; Microbial Sensitivity Tests | 2022 |
Nonidentical function of Upc2A binding sites in the Candida glabrata CDR1 promoter.
Topics: Adenosine Triphosphate; Antifungal Agents; ATP-Binding Cassette Transporters; Binding Sites; Candida albicans; Candida glabrata; DNA; Drug Resistance, Fungal; Ergosterol; Fluconazole; Fungal Proteins; Gene Expression Regulation, Fungal; Sterols; Transcription Factors; Zinc | 2022 |
Mathematical Modeling of Fluconazole Resistance in the Ergosterol Pathway of
Topics: Antifungal Agents; Azoles; Candida; Candida albicans; Candidiasis; Ergosterol; Fluconazole; Methyltransferases; Microbial Sensitivity Tests; Models, Theoretical; Mycoses; Sterols | 2022 |
Anticandidal Activity of Capsaicin and Its Effect on Ergosterol Biosynthesis and Membrane Integrity of
Topics: Antifungal Agents; Candida; Candida albicans; Candidiasis; Capsaicin; Ergosterol; Fluconazole; Microbial Sensitivity Tests | 2023 |
Alterations in the Level of Ergosterol in
Topics: Antifungal Agents; Azoles; Candida albicans; Candidiasis; Cell Membrane; Drug Resistance, Fungal; Ergosterol; Female; Fluconazole; Humans; Microbial Sensitivity Tests; Virulence; Virulence Factors | 2023 |
The proteasome regulator Rpn4 controls antifungal drug tolerance by coupling protein homeostasis with metabolic responses to drug stress.
Topics: Antifungal Agents; Candida albicans; Drug Resistance, Fungal; Drug Tolerance; Ergosterol; Fluconazole; Humans; Microbial Sensitivity Tests; Proteasome Endopeptidase Complex; Proteostasis | 2023 |
New miconazole-based azoles derived from eugenol show activity against Candida spp. and Cryptococcus gattii by inhibiting the fungal ergosterol biosynthesis.
Topics: Antifungal Agents; Azoles; Candida; Candida albicans; Cryptococcus gattii; Ergosterol; Eugenol; Fluconazole; Imidazoles; Miconazole; Microbial Sensitivity Tests | 2023 |
Fingerprint Stimulated Raman Scattering Imaging Unveils Ergosteryl Ester as a Metabolic Signature of Azole-Resistant
Topics: Animals; Antifungal Agents; Azoles; Candida albicans; Ergosterol; Esters; Fluconazole; Mice; Microbial Sensitivity Tests; Oleic Acid; Spectrum Analysis, Raman | 2023 |
Ergosterol distribution controls surface structure formation and fungal pathogenicity.
Topics: Antifungal Agents; Cryptococcosis; Cryptococcus neoformans; Ergosterol; Fluconazole; Fungal Proteins; Humans; Membrane Transport Proteins; Saccharomyces cerevisiae; Sterols; Virulence | 2023 |