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flesinoxan and eltoprazine

flesinoxan has been researched along with eltoprazine in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
IJzerman, AP; Kruse, CG; Kuipers, W; Spek, AL; Standaar, PJ; Tulp, MT; van Wijngaarden, I; Veldman, N1
Herremans, AH; Mos, J; Olivier, B; Van Drimmelen, M; Van Hest, A1
Ronken, E; Soudijn, W; van Steen, BJ; van Wijngaarden, I1
Cryan, JF; Kelliher, P; Kelly, JP; Leonard, BE1
Bloemarts, E; Groenink, L; Olivier, B; Oosting, RS; van den Bergh, FS1

Other Studies

5 other study(ies) available for flesinoxan and eltoprazine

ArticleYear
5-HT1A-versus D2-receptor selectivity of flesinoxan and analogous N4-substituted N1-arylpiperazines.
    Journal of medicinal chemistry, 1997, Jan-31, Volume: 40, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amino Acid Sequence; Animals; Binding Sites; Binding, Competitive; Brain; CHO Cells; Cricetinae; Crystallography, X-Ray; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Conformation; Molecular Sequence Data; Molecular Structure; Piperazines; Protein Binding; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Spiperone; Structure-Activity Relationship

1997
The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons.
    European journal of pharmacology, 1997, May-01, Volume: 325, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Columbidae; Discrimination Learning; Fluvoxamine; Indoles; Pindolol; Piperazines; Pyridines; Pyrimidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles

1997
Functional characteristics of a series of N4-substituted 1-(2,3-dihydro-1,4-benzodioxin-5-yl)piperazines as 5-HT1A receptor ligands. Structure-activity relationships.
    Bioorganic & medicinal chemistry letters, 1998, Sep-22, Volume: 8, Issue:18

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; CHO Cells; Cricetinae; Frontal Lobe; Humans; Ligands; Models, Chemical; Piperazines; Pyridines; Pyrimidines; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship

1998
Comparative effects of serotonergic agonists with varying efficacy at the 5-HT(1A) receptor on core body temperature: modification by the selective 5-HT(1A) receptor antagonist WAY 100635.
    Journal of psychopharmacology (Oxford, England), 1999, Volume: 13, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Dose-Response Relationship, Drug; Hypothermia; Male; Piperazines; Pyridines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists

1999
Delay aversion: effects of 7-OH-DPAT, 5-HT1A/1B-receptor stimulation and D-cycloserine.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 85, Issue:4

    Topics: Animals; Central Nervous System Stimulants; Cycloserine; Dextroamphetamine; Impulsive Behavior; Male; Oxadiazoles; Piperazines; Rats; Rats, Wistar; Receptors, Dopamine D3; Receptors, N-Methyl-D-Aspartate; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Tetrahydronaphthalenes

2006
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