Page last updated: 2024-09-02

fk 888 and sr 48968

fk 888 has been researched along with sr 48968 in 14 studies

Compound Research Comparison

Studies
(fk 888)
Trials
(fk 888)
Recent Studies (post-2010)
(fk 888)
Studies
(sr 48968)
Trials
(sr 48968)
Recent Studies (post-2010) (sr 48968)
9723338213

Protein Interaction Comparison

ProteinTaxonomyfk 888 (IC50)sr 48968 (IC50)
Substance-K receptorHomo sapiens (human)0.0001
Substance-P receptorHomo sapiens (human)0.8

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (50.00)18.2507
2000's7 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gerard, NP; Gether, U; Jensen, CJ; Schwartz, TW1
Calixto, JB; Campos, AH; Cechinel Filho, V; Dias, MA; Yunes, RA1
Hirayama, Y; Hiroi, J; Imai, T; Miyayasu, K; Yasumitsu, R1
Calixto, JB; De Lima, TC; Rae, GA; Ribeiro, SJ; Santos, AR; Teixeira, RM1
Ferrell, WR; Karimian, SM; Lockhart, JC1
Calixto, JB; Medeiros, YS; Saleh, TS1
Dong, F; Hasegawa, S; Iijima, H; Nomura, A; Uchida, Y; Xiang, A; Zhang, MJ1
Abe, S; Kaneko, S; Tanaka, H; Teramoto, S2
Lam, FF; Yip, AL1
Hayashi, I; Kamijo, Y; Majima, M; Ohwada, T; Soma, K1
Beirith, A; Calixto, JB; Santos, AR1
Calixto, JB; El Sayah, M1
De Lima, TC; Duarte, FS; Testolin, R1

Other Studies

14 other study(ies) available for fk 888 and sr 48968

ArticleYear
The species selectivity of chemically distinct tachykinin nonpeptide antagonists is dependent on common divergent residues of the rat and human neurokinin-1 receptors.
    Molecular pharmacology, 1994, Volume: 45, Issue:2

    Topics: Amino Acid Sequence; Animals; Benzamides; Biphenyl Compounds; Cell Line; Dipeptides; Humans; Indoles; Molecular Sequence Data; Mutation; Neurokinin-1 Receptor Antagonists; Piperidines; Rats; Receptors, Neurokinin-1; Recombinant Proteins; Substance P

1994
Analysis of the mechanisms underlying the contractile response induced by the hydroalcoholic extract of Phyllanthus urinaria in the guinea-pig urinary bladder in-vitro.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:10

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Benzamides; Dipeptides; Ethanol; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ion Channels; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurokinin A; Piperidines; Plant Extracts; Plants, Medicinal; Receptors, Tachykinin; Substance P; Urinary Bladder

1995
Effects of specific tachykinin receptor antagonists on citric acid-induced cough and bronchoconstriction in unanesthetized guinea pigs.
    European journal of pharmacology, 1996, Apr-11, Volume: 300, Issue:3

    Topics: Animals; Antacids; Benzamides; Bronchoconstriction; Citric Acid; Cough; Dipeptides; Guinea Pigs; Indoles; Male; Piperidines

1996
Effects of central administration of tachykinin receptor agonists and antagonists on plus-maze behavior in mice.
    European journal of pharmacology, 1996, Sep-05, Volume: 311, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzamides; Dipeptides; Dose-Response Relationship, Drug; Indoles; Injections, Intraventricular; Male; Mice; Motor Activity; Neurokinin A; Neurokinin-1 Receptor Antagonists; Piperidines; Postural Balance; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Substance P

1996
Tachykinin regulation of basal synovial blood flow.
    British journal of pharmacology, 1997, Volume: 121, Issue:1

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Benzamides; Dipeptides; Dose-Response Relationship, Drug; Drug Interactions; Hindlimb; Indoles; Joints; Laser-Doppler Flowmetry; Male; Microscopy, Electron; Nerve Fibers; Peptides, Cyclic; Phenoxybenzamine; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Tachykinin; Regional Blood Flow; Synovial Membrane; Tachykinins; Vasoconstriction

1997
Pro-inflammatory effects induced by bradykinin in a murine model of pleurisy.
    European journal of pharmacology, 1997, Jul-16, Volume: 331, Issue:1

    Topics: Animals; Benzamides; Bradykinin; Bradykinin Receptor Antagonists; Cell Movement; Dipeptides; Dose-Response Relationship, Drug; Female; Indoles; Inflammation; Leukocyte Count; Male; Mice; Neutrophils; Oligopeptides; Piperidines; Pleura; Pleurisy; Receptor, Bradykinin B2; Time Factors

1997
Effects of airway inflammation on cough response in the guinea pig.
    Journal of applied physiology (Bethesda, Md. : 1985), 1998, Volume: 85, Issue:5

    Topics: Animals; Antitussive Agents; Benzamides; Bronchoalveolar Lavage Fluid; Capsaicin; Codeine; Cough; Dipeptides; Female; Guinea Pigs; Indoles; Inflammation; Peptides, Cyclic; Piperidines; Quinuclidines; Receptors, Neurokinin-2; Receptors, Tachykinin; Respiratory Hypersensitivity; Respiratory Tract Diseases

1998
Neurokinin-1 receptor antagonist inhibits short-term sulfuric-acid-induced airway hyperresponsiveness in sensitized guinea pigs.
    International archives of allergy and immunology, 2000, Volume: 121, Issue:1

    Topics: Aerosols; Airway Resistance; Animals; Benzamides; Bronchial Hyperreactivity; Bronchial Provocation Tests; Bronchoconstriction; Dipeptides; Guinea Pigs; Indoles; Male; Methacholine Chloride; Nebulizers and Vaporizers; Neurokinin-1 Receptor Antagonists; Ovalbumin; Piperidines; Receptors, Neurokinin-2; Sulfuric Acids

2000
Unique gradual and sustained vasodilator response to substance P in the rabbit knee joint.
    European journal of pharmacology, 2000, Jul-21, Volume: 400, Issue:2-3

    Topics: Administration, Topical; Animals; Benzamides; Cyclooxygenase Inhibitors; Dipeptides; Evans Blue; Extravasation of Diagnostic and Therapeutic Materials; Flurbiprofen; Hindlimb; Indoles; Injections, Intra-Articular; Joints; Neurokinin-1 Receptor Antagonists; Piperidines; Rabbits; Receptors, Neurokinin-2; Regional Blood Flow; Substance P; Vasodilation

2000
Effect of neutral endopeptidase inhibitor on bradykinin-induced bronchoconstriction.
    Life sciences, 2001, Nov-21, Volume: 70, Issue:1

    Topics: Animals; Benzamides; Bradykinin; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Capsaicin; Dipeptides; Dose-Response Relationship, Drug; Drug Antagonism; Drug Interactions; Glycopeptides; Guinea Pigs; Indoles; Lung; Male; Metalloendopeptidases; Neurokinin A; Piperidines; Substance P

2001
Neurokinin-1 and neurokinin-2 antagonism inhibits long-term acid fog-induced airway hyperresponsiveness.
    Chest, 2003, Volume: 123, Issue:2

    Topics: Airway Resistance; Animals; Benzamides; Bronchial Hyperreactivity; Bronchial Provocation Tests; Bronchoalveolar Lavage Fluid; Dipeptides; Eosinophilia; Guinea Pigs; Indoles; Leukocyte Count; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Sulfuric Acids; Weather

2003
The role of neuropeptides and capsaicin-sensitive fibres in glutamate-induced nociception and paw oedema in mice.
    Brain research, 2003, Apr-18, Volume: 969, Issue:1-2

    Topics: Animals; Benzamides; Bradykinin Receptor Antagonists; Calcitonin Gene-Related Peptide; Capsaicin; Dipeptides; Edema; Foot; Glutamic Acid; Indoles; Male; Mice; Nerve Fibers; Neurokinin-1 Receptor Antagonists; Nociceptors; Pain; Piperidines; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Calcitonin Gene-Related Peptide; Receptors, Neurokinin-1; Receptors, Neurokinin-2

2003
New evidence on the mechanisms underlying bradykinin-mediated contraction of the pig iris sphincter in vitro.
    Peptides, 2003, Volume: 24, Issue:7

    Topics: Animals; Benzamides; Bradykinin; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Calcium; Calcium Channels; Capsaicin; Carbazoles; Conotoxins; Dipeptides; Dose-Response Relationship, Drug; Egtazic Acid; In Vitro Techniques; Indoles; Iris; Maleimides; Muscle Contraction; Nicardipine; omega-Agatoxin IVA; Peptide Fragments; Piperidines; Protein Kinase Inhibitors; Protein Kinases; Pyrroles; Receptors, Calcitonin Gene-Related Peptide; Receptors, Drug; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Swine; Tachykinins

2003
Further evidence on the anxiogenic-like effect of substance P evaluated in the elevated plus-maze in rats.
    Behavioural brain research, 2004, Oct-05, Volume: 154, Issue:2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Benzamides; Dipeptides; Dose-Response Relationship, Drug; Drug Interactions; Glycopeptides; Indoles; Injections, Intraventricular; Male; Maze Learning; Microinjections; Motor Activity; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-2; Substance P; Thiorphan; Time Factors

2004