Page last updated: 2024-09-02

fk 888 and phosphoramidon

fk 888 has been researched along with phosphoramidon in 8 studies

Compound Research Comparison

Studies
(fk 888)
Trials
(fk 888)
Recent Studies (post-2010)
(fk 888)
Studies
(phosphoramidon)
Trials
(phosphoramidon)
Recent Studies (post-2010) (phosphoramidon)
97237811233

Protein Interaction Comparison

ProteinTaxonomyfk 888 (IC50)phosphoramidon (IC50)
ThermolysinBacillus thermoproteolyticus0.033
NeprilysinRattus norvegicus (Norway rat)0.0578
NeprilysinOryctolagus cuniculus (rabbit)0.0028
NeprilysinHomo sapiens (human)0.0405
Angiotensin-converting enzyme Homo sapiens (human)0.615
Endothelin-converting enzyme 1Homo sapiens (human)1.0695
P2Y purinoceptor 12Homo sapiens (human)0.017

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (50.00)18.2507
2000's4 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aikawa, T; Sasaki, H; Sekizawa, K; Ujiie, Y1
Amemiya, T; Fujimura, M; Matsuda, T; Mizuguchi, M; Nishi, K; Ohka, T1
Evangelista, S; Giachetti, A; Manzini, S; Paoli, S1
Amemiya, T; Fujimura, M; Ishiura, Y; Matsuda, T; Mizuguchi, M; Myou, S; Sasaki, S1
Ando, M; Fujii, K; Hamamoto, J; Hirata, N; Iwagoe, H; Kawano, O; Kohrogi, H1
Hayashi, I; Kamijo, Y; Majima, M; Ohwada, T; Soma, K1
Bae, SJ; Hamazaki, Y; Katayama, I; Matsunaga, Y; Shimizu, K; Takenaka, M; Tanaka, Y1
De Lima, TC; Duarte, FS; Testolin, R1

Other Studies

8 other study(ies) available for fk 888 and phosphoramidon

ArticleYear
Evidence for substance P as an endogenous substance causing cough in guinea pigs.
    The American review of respiratory disease, 1993, Volume: 148, Issue:6 Pt 1

    Topics: Aerosols; Animals; Capsaicin; Cough; Dipeptides; Dose-Response Relationship, Drug; Glycopeptides; Guinea Pigs; Indoles; Male; Neprilysin; Smoking; Substance P; Tachykinins

1993
Involvement of NK2 receptors rather than NK1 receptors in bronchial hyperresponsiveness induced by allergic reaction in guinea-pigs.
    British journal of pharmacology, 1996, Volume: 117, Issue:3

    Topics: Animals; Bronchial Hyperreactivity; Bronchoconstrictor Agents; Capsaicin; Dipeptides; Glycopeptides; Guinea Pigs; Histamine; Indoles; Male; Methacholine Chloride; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Protease Inhibitors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory Hypersensitivity

1996
Involvement of tachykinin NK1 receptors in plasma protein extravasation induced by tachykinins in the guinea pig upper airways.
    Neuropeptides, 1997, Volume: 31, Issue:1

    Topics: Animals; Antigens; Blood Proteins; Capsaicin; Dextrans; Dipeptides; Extravasation of Diagnostic and Therapeutic Materials; Fluorescein-5-isothiocyanate; Glycopeptides; Guinea Pigs; Indoles; Male; Nasal Mucosa; Neurokinin A; Neurokinin-1 Receptor Antagonists; Olfactory Receptor Neurons; Peptide Fragments; Peptides, Cyclic; Protease Inhibitors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Rhinitis; Substance P

1997
Role of tachykinins in distilled water-induced bronchoconstriction in guinea-pigs.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 1998, Volume: 28, Issue:7

    Topics: Animals; Bronchoconstriction; Capsaicin; Dipeptides; Disease Models, Animal; Glycopeptides; Guinea Pigs; Indoles; Killer Cells, Natural; Male; Nebulizers and Vaporizers; Ovalbumin; Peptides, Cyclic; Respiration; Tachykinins; Water

1998
The role of substance P release in the lung with esophageal acid.
    The American journal of medicine, 2001, Dec-03, Volume: 111 Suppl 8A

    Topics: Animals; Dipeptides; Disease Models, Animal; Dose-Response Relationship, Drug; Esophagus; Extravasation of Diagnostic and Therapeutic Materials; Glycopeptides; Guinea Pigs; Hydrochloric Acid; Indoles; Lung; Reference Values; Sensitivity and Specificity; Substance P; Vagotomy

2001
Effect of neutral endopeptidase inhibitor on bradykinin-induced bronchoconstriction.
    Life sciences, 2001, Nov-21, Volume: 70, Issue:1

    Topics: Animals; Benzamides; Bradykinin; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Capsaicin; Dipeptides; Dose-Response Relationship, Drug; Drug Antagonism; Drug Interactions; Glycopeptides; Guinea Pigs; Indoles; Lung; Male; Metalloendopeptidases; Neurokinin A; Piperidines; Substance P

2001
Substance P induced preprotachykinin-a mRNA, neutral endopeptidase mRNA and substance P in cultured normal fibroblasts.
    International archives of allergy and immunology, 2002, Volume: 127, Issue:4

    Topics: Cells, Cultured; Cycloheximide; Dipeptides; Fibroblasts; Gene Expression; Glycopeptides; Humans; Immunohistochemistry; Indoles; Neprilysin; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Protease Inhibitors; Protein Precursors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Analysis, DNA; Skin; Substance P; Tachykinins

2002
Further evidence on the anxiogenic-like effect of substance P evaluated in the elevated plus-maze in rats.
    Behavioural brain research, 2004, Oct-05, Volume: 154, Issue:2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Benzamides; Dipeptides; Dose-Response Relationship, Drug; Drug Interactions; Glycopeptides; Indoles; Injections, Intraventricular; Male; Maze Learning; Microinjections; Motor Activity; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-2; Substance P; Thiorphan; Time Factors

2004