Page last updated: 2024-09-02

fk 888 and fk 224

fk 888 has been researched along with fk 224 in 14 studies

Compound Research Comparison

Studies
(fk 888)
Trials
(fk 888)
Recent Studies (post-2010)
(fk 888)
Studies
(fk 224)
Trials
(fk 224)
Recent Studies (post-2010) (fk 224)
97234430

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's13 (92.86)18.2507
2000's1 (7.14)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Church, MK; Featherstone, R; Polak, JM; Salmon, M; Walsh, DA; Wharton, J1
Buckley, TL; Koster, AS; Kraneveld, AD; Nijkamp, FP; van Heuven-Nolsen, D; van Schaik, Y1
Barnes, PJ; Hirayama, Y; Lei, YH; Rogers, DF1
Fujii, T1
Fujimura, M; Matsuda, T; Matsushima, K; Mizuguchi, M; Nomura, M; Tsujiura, M1
Amemiya, T; Fujimura, M; Matsuda, T; Mizuguchi, M; Nishi, K; Ohka, T1
Fujimura, M; Ishiura, Y; Matsuda, T; Myou, S; Tsujiura, M1
Asakura, K; Kataura, A; Narita, S; Shirasaki, H; Watanabe, M1
Ferrell, WR; Karimian, SM; Lockhart, JC1
Kraneveld, AD; Nijkamp, FP; Van Oosterhout, AJ1
Katahashi, T; Konno, A1
Amemiya, T; Fujimura, M; Ishiura, Y; Matsuda, T; Mizuguchi, M; Myou, S; Sasaki, S1
Dong, F; Hasegawa, S; Iijima, H; Nomura, A; Uchida, Y; Xiang, A; Zhang, MJ1
Bae, SJ; Hamazaki, Y; Katayama, I; Matsunaga, Y; Shimizu, K; Takenaka, M; Tanaka, Y1

Reviews

1 review(s) available for fk 888 and fk 224

ArticleYear
[Discovery and pharmacological properties of selective neurokinin-receptor antagonists, FK224 and FK888].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1995, Volume: 106, Issue:3

    Topics: Animals; Bronchoconstriction; Cricetinae; Dipeptides; Humans; Indoles; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Rats; Receptors, Neurokinin-2; Receptors, Neurokinin-3

1995

Other Studies

13 other study(ies) available for fk 888 and fk 224

ArticleYear
Differences in the distribution and characteristics of tachykinin NK1 binding sites between human and guinea pig lung.
    British journal of pharmacology, 1994, Volume: 113, Issue:4

    Topics: Animals; Autoradiography; Dipeptides; Guinea Pigs; Humans; Immunohistochemistry; In Vitro Techniques; Indoles; Iodine Radioisotopes; Lung; Male; Neurokinin-1 Receptor Antagonists; Ovalbumin; Peptides, Cyclic; Pulmonary Artery; Receptors, Neurokinin-1; Respiratory Hypersensitivity; Species Specificity; Substance P; Succinimides

1994
Delayed-type hypersensitivity-induced increase in vascular permeability in the mouse small intestine: inhibition by depletion of sensory neuropeptides and NK1 receptor blockade.
    British journal of pharmacology, 1995, Volume: 114, Issue:7

    Topics: Animals; Capillary Permeability; Capsaicin; Dipeptides; Hypersensitivity, Delayed; Indoles; Intestine, Small; Isoindoles; Male; Mice; Mice, Inbred BALB C; Neurokinin-1 Receptor Antagonists; Neuropeptides; Peptides, Cyclic

1995
Effects of two novel tachykinin antagonists, FK224 and FK888, on neurogenic airway plasma exudation, bronchoconstriction and systemic hypotension in guinea-pigs in vivo.
    British journal of pharmacology, 1993, Volume: 108, Issue:3

    Topics: Animals; Blood Pressure; Bronchoconstriction; Capsaicin; Dipeptides; Electric Stimulation; Evans Blue; Exudates and Transudates; Guinea Pigs; Hypotension; Indoles; Male; Neurokinin A; Peptide Fragments; Peptides, Cyclic; Platelet Activating Factor; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Respiratory Mechanics; Smoking; Substance P; Vagus Nerve

1993
Sensory neuropeptides are not directly involved in bronchial hyperresponsiveness induced by interleukin-8 in guinea-pigs in vivo.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 1996, Volume: 26, Issue:3

    Topics: Animals; Bronchial Hyperreactivity; Bronchial Provocation Tests; Dipeptides; Guinea Pigs; Histamine; Indoles; Interleukin-8; Male; Neurokinin A; Peptides, Cyclic; Substance P

1996
Involvement of NK2 receptors rather than NK1 receptors in bronchial hyperresponsiveness induced by allergic reaction in guinea-pigs.
    British journal of pharmacology, 1996, Volume: 117, Issue:3

    Topics: Animals; Bronchial Hyperreactivity; Bronchoconstrictor Agents; Capsaicin; Dipeptides; Glycopeptides; Guinea Pigs; Histamine; Indoles; Male; Methacholine Chloride; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Protease Inhibitors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory Hypersensitivity

1996
Role of sensory neuropeptides in post-allergic propranolol-induced bronchoconstriction in guinea pigs in vivo.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 1996, Volume: 26, Issue:12

    Topics: Adrenergic beta-Antagonists; Animals; Asthma; Bronchial Hyperreactivity; Bronchoconstriction; Dipeptides; Guinea Pigs; Indoles; Male; Neurokinin A; Peptides, Cyclic; Propranolol; Substance P

1996
The effects of NK1 receptor antagonists (FK224 and FK888) on agonist- and antigen-induced nasal microvascular leakage in guinea pigs.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1997, Volume: 46, Issue:1

    Topics: Animals; Antigens; Capillary Permeability; Dipeptides; Guinea Pigs; Indoles; Male; Neurokinin-1 Receptor Antagonists; Nose; Ovalbumin; Peptides, Cyclic; Receptors, Neurokinin-1; Respiratory Hypersensitivity; Substance P

1997
Tachykinin regulation of basal synovial blood flow.
    British journal of pharmacology, 1997, Volume: 121, Issue:1

    Topics: Administration, Topical; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Benzamides; Dipeptides; Dose-Response Relationship, Drug; Drug Interactions; Hindlimb; Indoles; Joints; Laser-Doppler Flowmetry; Male; Microscopy, Electron; Nerve Fibers; Peptides, Cyclic; Phenoxybenzamine; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Tachykinin; Regional Blood Flow; Synovial Membrane; Tachykinins; Vasoconstriction

1997
Role for neurokinin-2 receptor in interleukin-5-induced airway hyperresponsiveness but not eosinophilia in guinea pigs.
    American journal of respiratory and critical care medicine, 1997, Volume: 156, Issue:2 Pt 1

    Topics: Airway Resistance; Animals; Bronchial Hyperreactivity; Bronchoalveolar Lavage Fluid; Dipeptides; Eosinophilia; Eosinophils; Guinea Pigs; Indoles; Interleukin-5; Leukocyte Count; Male; Peptides, Cyclic; Receptors, Neurokinin-2; Specific Pathogen-Free Organisms; Substance P

1997
Effects of tachykinin receptor antagonists, FK224 and FK888, in a guinea-pig model of nasal allergy.
    Rhinology, 1997, Volume: 35, Issue:2

    Topics: Airway Resistance; Animals; Antigens; Capillary Permeability; Dipeptides; Female; Guinea Pigs; Indoles; Neurokinin-1 Receptor Antagonists; Ovalbumin; Peptides, Cyclic; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory Hypersensitivity; Sneezing; Statistics, Nonparametric

1997
Role of tachykinins in distilled water-induced bronchoconstriction in guinea-pigs.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 1998, Volume: 28, Issue:7

    Topics: Animals; Bronchoconstriction; Capsaicin; Dipeptides; Disease Models, Animal; Glycopeptides; Guinea Pigs; Indoles; Killer Cells, Natural; Male; Nebulizers and Vaporizers; Ovalbumin; Peptides, Cyclic; Respiration; Tachykinins; Water

1998
Effects of airway inflammation on cough response in the guinea pig.
    Journal of applied physiology (Bethesda, Md. : 1985), 1998, Volume: 85, Issue:5

    Topics: Animals; Antitussive Agents; Benzamides; Bronchoalveolar Lavage Fluid; Capsaicin; Codeine; Cough; Dipeptides; Female; Guinea Pigs; Indoles; Inflammation; Peptides, Cyclic; Piperidines; Quinuclidines; Receptors, Neurokinin-2; Receptors, Tachykinin; Respiratory Hypersensitivity; Respiratory Tract Diseases

1998
Substance P induced preprotachykinin-a mRNA, neutral endopeptidase mRNA and substance P in cultured normal fibroblasts.
    International archives of allergy and immunology, 2002, Volume: 127, Issue:4

    Topics: Cells, Cultured; Cycloheximide; Dipeptides; Fibroblasts; Gene Expression; Glycopeptides; Humans; Immunohistochemistry; Indoles; Neprilysin; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Protease Inhibitors; Protein Precursors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Analysis, DNA; Skin; Substance P; Tachykinins

2002