Page last updated: 2024-09-02

fk 888 and cp 99994

fk 888 has been researched along with cp 99994 in 3 studies

Compound Research Comparison

Studies
(fk 888)
Trials
(fk 888)
Recent Studies (post-2010)
(fk 888)
Studies
(cp 99994)
Trials
(cp 99994)
Recent Studies (post-2010) (cp 99994)
9723231219

Protein Interaction Comparison

ProteinTaxonomyfk 888 (IC50)cp 99994 (IC50)
Glutamate receptor 1Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 2Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 3Rattus norvegicus (Norway rat)0.0006
Glutamate receptor 4Rattus norvegicus (Norway rat)0.0006
Substance-P receptorHomo sapiens (human)0.0004

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujita, H; Kurahashi, K; Nakagiri, R; Sasaki, R; Suganuma, H; Usui, H; Yoshikawa, M1
Ngan, MP; Rudd, JA; Wai, MK1
Hamada, K; Hanioka, N; Imazumi, K; Maeda, Y; Manda, T; Matsuo, M; Mutoh, S; Yamamoto, T1

Other Studies

3 other study(ies) available for fk 888 and cp 99994

ArticleYear
Vasorelaxation by casomokinin L, a derivative of beta-casomorphin and casoxin D, is mediated by NK1 receptor.
    Peptides, 1996, Volume: 17, Issue:4

    Topics: Amino Acid Sequence; Animals; Antihypertensive Agents; Blood Pressure; Caseins; Dipeptides; Dogs; Endorphins; Endothelium, Vascular; Female; In Vitro Techniques; Indoles; Male; Mesenteric Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Oligopeptides; Piperidines; Rats; Rats, Inbred SHR; Receptors, Neurokinin-1; Sequence Homology, Amino Acid; Vasodilation

1996
Inhibition of emesis by tachykinin NK1 receptor antagonists in Suncus murinus (house musk shrew).
    European journal of pharmacology, 1999, Feb-05, Volume: 366, Issue:2-3

    Topics: Animals; Antiemetics; Copper Sulfate; Dipeptides; Dose-Response Relationship, Drug; Emetics; Female; Ganglionic Stimulants; Indoles; Infusions, Parenteral; Isoindoles; Male; Motion Sickness; Neurokinin-1 Receptor Antagonists; Nicotine; Physalaemin; Piperidines; Shrews; Stereoisomerism; Vomiting

1999
Contribution of tachykinin receptor subtypes to micturition reflex in guinea pigs.
    European journal of pharmacology, 2003, Sep-23, Volume: 477, Issue:3

    Topics: Animals; Brain; Catheterization; CHO Cells; Cricetinae; Dipeptides; Dose-Response Relationship, Drug; Guinea Pigs; Humans; Indoles; Injections, Intravenous; Iodine Radioisotopes; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Piperidines; Radioligand Assay; Receptors, Neurokinin-1; Spinal Cord; Substance P; Succinimides; Tetrazoles; Tissue Extracts; Transfection; Urinary Bladder; Urination

2003