Page last updated: 2024-09-03

fk 224 and phosphoramidon

fk 224 has been researched along with phosphoramidon in 6 studies

Compound Research Comparison

Studies
(fk 224)
Trials
(fk 224)
Recent Studies (post-2010)
(fk 224)
Studies
(phosphoramidon)
Trials
(phosphoramidon)
Recent Studies (post-2010) (phosphoramidon)
44307811233

Protein Interaction Comparison

ProteinTaxonomyfk 224 (IC50)phosphoramidon (IC50)
ThermolysinBacillus thermoproteolyticus0.033
NeprilysinRattus norvegicus (Norway rat)0.0578
NeprilysinOryctolagus cuniculus (rabbit)0.0028
NeprilysinHomo sapiens (human)0.0405
Angiotensin-converting enzyme Homo sapiens (human)0.615
Endothelin-converting enzyme 1Homo sapiens (human)1.0695
P2Y purinoceptor 12Homo sapiens (human)0.017

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (83.33)18.2507
2000's1 (16.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ando, M; Fujii, K; Hamamoto, J; Hirata, N; Iwagoe, H; Kawano, O; Kohrogi, H; Yamaguchi, T1
Amemiya, T; Fujimura, M; Matsuda, T; Mizuguchi, M; Nishi, K; Ohka, T1
Ando, M; Fujii, K; Hamamoto, J; Iwagoe, H; Kawano, O; Kohrogi, H; Yamaguchi, T1
Ando, M; Fujii, K; Goto, E; Hamamoto, J; Hirata, N; Honda, I; Iwagoe, H; Kohrogi, H; Yamaguchi, T1
Amemiya, T; Fujimura, M; Ishiura, Y; Matsuda, T; Mizuguchi, M; Myou, S; Sasaki, S1
Bae, SJ; Hamazaki, Y; Katayama, I; Matsunaga, Y; Shimizu, K; Takenaka, M; Tanaka, Y1

Other Studies

6 other study(ies) available for fk 224 and phosphoramidon

ArticleYear
Evidence that PGF2 alpha-induced contraction of isolated guinea pig bronchi is mediated in part by release of tachykinins.
    Journal of applied physiology (Bethesda, Md. : 1985), 1995, Volume: 79, Issue:5

    Topics: Animals; Bronchi; Bronchoconstriction; Capsaicin; Dinoprost; Glycopeptides; Guinea Pigs; In Vitro Techniques; Male; Peptides, Cyclic; Protease Inhibitors; Tachykinins; Tetrodotoxin

1995
Involvement of NK2 receptors rather than NK1 receptors in bronchial hyperresponsiveness induced by allergic reaction in guinea-pigs.
    British journal of pharmacology, 1996, Volume: 117, Issue:3

    Topics: Animals; Bronchial Hyperreactivity; Bronchoconstrictor Agents; Capsaicin; Dipeptides; Glycopeptides; Guinea Pigs; Histamine; Indoles; Male; Methacholine Chloride; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Protease Inhibitors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory Hypersensitivity

1996
Evidence that allergen-induced contraction of guinea pig bronchi is mediated in part by the release of tachykinins.
    International archives of allergy and immunology, 1997, Volume: 112, Issue:3

    Topics: Allergens; Animals; Bronchoconstriction; Drug Hypersensitivity; Glycopeptides; Guinea Pigs; Male; Metalloendopeptidases; Ovalbumin; Peptides, Cyclic; Protease Inhibitors; Tachykinins; Tetrodotoxin

1997
Tachykinin antagonist FK224 inhibits neurokinin A-, substance P- and capsaicin-induced human bronchial contraction.
    Fundamental & clinical pharmacology, 1997, Volume: 11, Issue:3

    Topics: Acetylcholine; Adult; Aged; Bronchi; Capsaicin; Glycopeptides; Histamine; Humans; In Vitro Techniques; Leukotriene D4; Middle Aged; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptides, Cyclic; Protease Inhibitors; Receptors, Tachykinin; Substance P; Tachykinins

1997
Role of tachykinins in distilled water-induced bronchoconstriction in guinea-pigs.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 1998, Volume: 28, Issue:7

    Topics: Animals; Bronchoconstriction; Capsaicin; Dipeptides; Disease Models, Animal; Glycopeptides; Guinea Pigs; Indoles; Killer Cells, Natural; Male; Nebulizers and Vaporizers; Ovalbumin; Peptides, Cyclic; Respiration; Tachykinins; Water

1998
Substance P induced preprotachykinin-a mRNA, neutral endopeptidase mRNA and substance P in cultured normal fibroblasts.
    International archives of allergy and immunology, 2002, Volume: 127, Issue:4

    Topics: Cells, Cultured; Cycloheximide; Dipeptides; Fibroblasts; Gene Expression; Glycopeptides; Humans; Immunohistochemistry; Indoles; Neprilysin; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Protease Inhibitors; Protein Precursors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Analysis, DNA; Skin; Substance P; Tachykinins

2002