Page last updated: 2024-09-03

fk 224 and histamine

fk 224 has been researched along with histamine in 4 studies

Compound Research Comparison

Studies
(fk 224)
Trials
(fk 224)
Recent Studies (post-2010)
(fk 224)
Studies
(histamine)
Trials
(histamine)
Recent Studies (post-2010) (histamine)
443037,7181,3723,457

Protein Interaction Comparison

ProteinTaxonomyfk 224 (IC50)histamine (IC50)
Histamine H1 receptorRattus norvegicus (Norway rat)0.1585
Histamine H1 receptorHomo sapiens (human)0.1585

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujii, T; Matsuda, A; Miyake, H; Morimoto, H; Yamashita, M1
Fujimura, M; Matsuda, T; Matsushima, K; Mizuguchi, M; Nomura, M; Tsujiura, M1
Amemiya, T; Fujimura, M; Matsuda, T; Mizuguchi, M; Nishi, K; Ohka, T1
Ando, M; Fujii, K; Goto, E; Hamamoto, J; Hirata, N; Honda, I; Iwagoe, H; Kohrogi, H; Yamaguchi, T1

Other Studies

4 other study(ies) available for fk 224 and histamine

ArticleYear
Effects of FR 113680 and FK 224, novel tachykinin receptor antagonists, on cigarette smoke-induced rat tracheal plasma extravasation.
    European journal of pharmacology, 1992, Nov-24, Volume: 224, Issue:1

    Topics: Amino Acid Sequence; Animals; Capillary Permeability; Histamine; Male; Molecular Sequence Data; Neurokinin A; Nicotiana; Oligopeptides; Peptides, Cyclic; Plants, Toxic; Rats; Rats, Wistar; Receptors, Neurotransmitter; Receptors, Tachykinin; Smoke; Substance P; Tachykinins; Trachea

1992
Sensory neuropeptides are not directly involved in bronchial hyperresponsiveness induced by interleukin-8 in guinea-pigs in vivo.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 1996, Volume: 26, Issue:3

    Topics: Animals; Bronchial Hyperreactivity; Bronchial Provocation Tests; Dipeptides; Guinea Pigs; Histamine; Indoles; Interleukin-8; Male; Neurokinin A; Peptides, Cyclic; Substance P

1996
Involvement of NK2 receptors rather than NK1 receptors in bronchial hyperresponsiveness induced by allergic reaction in guinea-pigs.
    British journal of pharmacology, 1996, Volume: 117, Issue:3

    Topics: Animals; Bronchial Hyperreactivity; Bronchoconstrictor Agents; Capsaicin; Dipeptides; Glycopeptides; Guinea Pigs; Histamine; Indoles; Male; Methacholine Chloride; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Protease Inhibitors; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Respiratory Hypersensitivity

1996
Tachykinin antagonist FK224 inhibits neurokinin A-, substance P- and capsaicin-induced human bronchial contraction.
    Fundamental & clinical pharmacology, 1997, Volume: 11, Issue:3

    Topics: Acetylcholine; Adult; Aged; Bronchi; Capsaicin; Glycopeptides; Histamine; Humans; In Vitro Techniques; Leukotriene D4; Middle Aged; Muscle Contraction; Muscle, Smooth; Neurokinin A; Peptides, Cyclic; Protease Inhibitors; Receptors, Tachykinin; Substance P; Tachykinins

1997