Page last updated: 2024-09-02

fingolimod hydrochloride and mitoxantrone

fingolimod hydrochloride has been researched along with mitoxantrone in 20 studies

Compound Research Comparison

Studies
(fingolimod hydrochloride)
Trials
(fingolimod hydrochloride)
Recent Studies (post-2010)
(fingolimod hydrochloride)
Studies
(mitoxantrone)
Trials
(mitoxantrone)
Recent Studies (post-2010) (mitoxantrone)
2,7711572,0624,5551,0421,004

Protein Interaction Comparison

ProteinTaxonomyfingolimod hydrochloride (IC50)mitoxantrone (IC50)
Chain A, Probable serine/threonine-protein kinase pknBMycobacterium tuberculosis H37Rv0.8
nonstructural protein 1Influenza A virus (A/California/07/2009(H1N1))2.049
rac GTPase-activating protein 1 isoform aHomo sapiens (human)14.46
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)3.5619
Epidermal growth factor receptorHomo sapiens (human)5.3859
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)2.0352
Tyrosine-protein kinase FynHomo sapiens (human)1.2579
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)4.9898
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.219
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.6441
ATP-dependent translocase ABCB1Homo sapiens (human)1.501
Proto-oncogene tyrosine-protein kinase ROSHomo sapiens (human)2.9987
Muscarinic acetylcholine receptor M1Homo sapiens (human)0.7487
DNA topoisomerase 2-alphaHomo sapiens (human)5.3
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)1.7853
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)3.5849
Casein kinase II subunit alpha'Homo sapiens (human)0.66
Sodium-dependent noradrenaline transporter Homo sapiens (human)4.9898
5-hydroxytryptamine receptor 2CHomo sapiens (human)3.5619
Multidrug resistance-associated protein 1 Homo sapiens (human)0.0081
Casein kinase II subunit betaHomo sapiens (human)0.66
Casein kinase II subunit alphaHomo sapiens (human)0.66
Tyrosine-protein kinase BTKHomo sapiens (human)1
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.5849
TAR DNA-binding protein 43Homo sapiens (human)10
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)3.5849
Integrase Human immunodeficiency virus 15.9
Multidrug and toxin extrusion protein 2Homo sapiens (human)0.68
Casein kinase II subunit alpha 3Homo sapiens (human)0.66
Multidrug and toxin extrusion protein 1Homo sapiens (human)0.3733
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)3.39
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)0.9038

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (15.00)29.6817
2010's15 (75.00)24.3611
2020's2 (10.00)2.80

Authors

AuthorsStudies
Chun, J; Hale, J; Lariosa-Willingham, K; Lin, FF; Mandala, S; Rao, TS; Tham, CS; Webb, M; Yu, N1
Gonsette, RE1
Benedetti, MD; Invernizzi, P; Monaco, S; Poli, S1
Martin, R1
Carmona, O; Cocco, E; Drulovic, J; Duddy, M; Eggers, C; Gold, R; Haghikia, A; Zéphir, H1
Arnason, B1
Sørensen, PS1
Havla, J; Hohlfeld, R; Kümpfel, T1
Graves, D; Vernino, S1
McDonald, EA; Sedal, L; Wilson, IB1
Gündel, M; Hofmann-Apitius, M; Kotelnikova, E; Lozano-Rubi, R; Malhotra, A; Martinez-Lapiscina, EH; Martinez-Lapsicina, EH; Mevissen, HT; Mueller, B; Pastor, X; Rajput, AM; Saiz, A; Toldo, L; Villoslada, P; Zubizarreta, I1
Cocco, E; Coghe, GC; Fenu, G; Frau, F; Lorefice, L; Marrosu, MG1
Berkowitz, AL; Kaplan, TB; Samuels, MA1
Weinshenker, BG; Wingerchuk, DM1
Airody, A; Gale, RP; Heath, G1
Fernández, Ó1
Chataway, J; Doshi, A1
Axelsson, M; Dubuisson, N; Giovannoni, G; Gnanapavan, S; Lycke, J; Malmeström, C; Novakova, L1
Altincatal, A; Berdofe, A; Centonze, D; de Moor, C; Jung, E; Kim, M; Nagpal, A; Naylor, ML; Popescu, C; Radhakrishnan, M; Rajbhandari, R; Reder, AT; Sandrock, AW; Smirnakis, K1
Callegari, I; Derfuss, T; Galli, E1

Reviews

13 review(s) available for fingolimod hydrochloride and mitoxantrone

ArticleYear
Compared benefit of approved and experimental immunosuppressive therapeutic approaches in multiple sclerosis.
    Expert opinion on pharmacotherapy, 2007, Volume: 8, Issue:8

    Topics: Antibodies, Monoclonal; Cladribine; Cyclophosphamide; Drug Delivery Systems; Fingolimod Hydrochloride; Humans; Immunosuppressive Agents; Isoxazoles; Ligands; Mitoxantrone; Multiple Sclerosis; Propylene Glycols; Sphingosine

2007
Azathioprine in multiple sclerosis.
    Mini reviews in medicinal chemistry, 2008, Volume: 8, Issue:9

    Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Azathioprine; Chemistry, Pharmaceutical; Cyclophosphamide; Drug Design; Fingolimod Hydrochloride; Humans; Immunologic Factors; Immunosuppressive Agents; Methotrexate; Methyltransferases; Mitoxantrone; Models, Chemical; Multiple Sclerosis; Multiple Sclerosis, Relapsing-Remitting; Natalizumab; Propylene Glycols; Sphingosine

2008
Managing MS in a changing treatment landscape.
    Journal of neurology, 2011, Volume: 258, Issue:5

    Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Cladribine; Fingolimod Hydrochloride; Humans; Immunosuppressive Agents; Interferon-beta; Mitoxantrone; Multiple Sclerosis; Natalizumab; Propylene Glycols; Sphingosine

2011
[2012: Update on diagnosis and treatment of multiple sclerosis].
    Deutsche medizinische Wochenschrift (1946), 2012, Volume: 137, Issue:17

    Topics: Administration, Oral; Antibodies, Monoclonal, Humanized; Brain; Combined Modality Therapy; Diagnosis, Differential; Dose-Response Relationship, Drug; Drug Administration Schedule; Fingolimod Hydrochloride; Glatiramer Acetate; Glucocorticoids; Humans; Immunosuppressive Agents; Infusions, Intravenous; Interferon-beta; Methylprednisolone; Mitoxantrone; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis, Relapsing-Remitting; Natalizumab; Peptides; Plasmapheresis; Propylene Glycols; Pulse Therapy, Drug; Sphingosine; Spinal Cord

2012
Immunotherapies in neurologic disorders.
    The Medical clinics of North America, 2012, Volume: 96, Issue:3

    Topics: Adjuvants, Immunologic; Adrenal Cortex Hormones; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Azathioprine; Cyclophosphamide; Cyclosporine; Fingolimod Hydrochloride; Glatiramer Acetate; Humans; Immunoglobulins, Intravenous; Immunologic Factors; Immunosuppressive Agents; Interferon beta-1a; Interferon beta-1b; Interferon-beta; Mitoxantrone; Mycophenolic Acid; Natalizumab; Nervous System Diseases; Peptides; Plasma Exchange; Propylene Glycols; Rituximab; Sphingosine; Tacrolimus

2012
Current management of relapsing-remitting multiple sclerosis.
    Internal medicine journal, 2014, Volume: 44, Issue:10

    Topics: Administration, Intravenous; Administration, Oral; Alemtuzumab; Antibodies, Monoclonal, Humanized; Crotonates; Dimethyl Fumarate; Disease Progression; Drug Administration Schedule; Fingolimod Hydrochloride; Fumarates; Humans; Hydroxybutyrates; Immunosuppressive Agents; Mitoxantrone; Multiple Sclerosis, Relapsing-Remitting; Natalizumab; Nitriles; Propylene Glycols; Risk Assessment; Sphingosine; Toluidines

2014
Induction and escalation therapies in multiple sclerosis.
    Anti-inflammatory & anti-allergy agents in medicinal chemistry, 2015, Volume: 14, Issue:1

    Topics: Animals; Crotonates; Dimethyl Fumarate; Fingolimod Hydrochloride; Glatiramer Acetate; Humans; Hydroxybutyrates; Induction Chemotherapy; Interferon-beta; Maintenance Chemotherapy; Mitoxantrone; Multiple Sclerosis; Natalizumab; Nitriles; Randomized Controlled Trials as Topic; Toluidines; Treatment Outcome

2015
Cardiovascular Dysfunction in Multiple Sclerosis.
    The neurologist, 2015, Volume: 20, Issue:6

    Topics: Animals; Autonomic Nervous System; Blood Pressure; Cardiovascular Abnormalities; Fingolimod Hydrochloride; Heart Rate; Humans; Mitoxantrone; Multiple Sclerosis

2015
Disease modifying therapies for relapsing multiple sclerosis.
    BMJ (Clinical research ed.), 2016, Aug-22, Volume: 354

    Topics: Administration, Intravenous; Administration, Oral; Alemtuzumab; Antibodies, Monoclonal, Humanized; Crotonates; Daclizumab; Dimethyl Fumarate; Drug Substitution; Fingolimod Hydrochloride; Glatiramer Acetate; Humans; Hydroxybutyrates; Immunoglobulin G; Immunologic Factors; Injections; Interferon-beta; Magnetic Resonance Imaging; Mitoxantrone; Multiple Sclerosis; Natalizumab; Nitriles; Toluidines

2016
The Ocular Manifestations of Drugs Used to Treat Multiple Sclerosis.
    Drugs, 2017, Volume: 77, Issue:3

    Topics: Alemtuzumab; Antibodies, Monoclonal, Humanized; Eye Diseases; Fingolimod Hydrochloride; Humans; Immunosuppressive Agents; Interferons; Mitoxantrone; Multiple Sclerosis; Natalizumab

2017
Is there a change of paradigm towards more effective treatment early in the course of apparent high-risk MS?
    Multiple sclerosis and related disorders, 2017, Volume: 17

    Topics: Alemtuzumab; Antineoplastic Agents; Clinical Trials as Topic; Cyclophosphamide; Disease Progression; Fingolimod Hydrochloride; Humans; Immunologic Factors; Immunosuppressive Agents; Mitoxantrone; Multiple Sclerosis, Relapsing-Remitting; Natalizumab; Precision Medicine; Risk Assessment; Risk Factors; Treatment Outcome

2017
Multiple sclerosis, a treatable disease .
    Clinical medicine (London, England), 2017, Volume: 17, Issue:6

    Topics: Adjuvants, Immunologic; Alemtuzumab; Crotonates; Demyelinating Diseases; Dimethyl Fumarate; Fingolimod Hydrochloride; Glatiramer Acetate; Glucocorticoids; Humans; Hydroxybutyrates; Immunologic Factors; Immunosuppressive Agents; Interferon beta-1a; Interferon beta-1b; Mitoxantrone; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis, Relapsing-Remitting; Natalizumab; Nitriles; Toluidines

2017
Update on treatment in multiple sclerosis.
    Presse medicale (Paris, France : 1983), 2021, Volume: 50, Issue:2

    Topics: Abnormalities, Drug-Induced; Algorithms; Antibodies, Monoclonal, Humanized; Cladribine; Crotonates; Dimethyl Fumarate; Female; Fingolimod Hydrochloride; Hematopoietic Stem Cell Transplantation; Humans; Hydroxybutyrates; Immunologic Factors; Immunosuppressive Agents; Indans; Interferon-beta; Male; Mitoxantrone; Multiple Sclerosis; Natalizumab; Nitriles; Oxadiazoles; Pregnancy; Sphingosine 1 Phosphate Receptor Modulators; Sphingosine-1-Phosphate Receptors; Toluidines

2021

Other Studies

7 other study(ies) available for fingolimod hydrochloride and mitoxantrone

ArticleYear
Sphingosine 1-phosphate receptor agonists attenuate relapsing-remitting experimental autoimmune encephalitis in SJL mice.
    Journal of neuroimmunology, 2004, Volume: 153, Issue:1-2

    Topics: Animals; Antineoplastic Agents; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Encephalomyelitis, Autoimmune, Experimental; Female; Fingolimod Hydrochloride; Gene Expression Regulation; Granulocyte-Macrophage Colony-Stimulating Factor; Immunosuppressive Agents; Interferon-gamma; Lymphocytes; Lymphopenia; Mice; Mice, Inbred Strains; Mitoxantrone; Molecular Sequence Data; Myelin Proteins; Myelin Proteolipid Protein; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Peptide Fragments; Propylene Glycols; Receptors, G-Protein-Coupled; Receptors, Lysophospholipid; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sphingosine; Time Factors

2004
Multiple sclerosis: closing in on an oral treatment.
    Nature, 2010, Mar-18, Volume: 464, Issue:7287

    Topics: Administration, Oral; Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Clinical Trials, Phase III as Topic; Fingolimod Hydrochloride; Humans; Lysophospholipids; Mitoxantrone; Multiple Sclerosis; Natalizumab; Propylene Glycols; Randomized Controlled Trials as Topic; Sphingosine

2010
MS Forum/MS Over the Past 17 Years.
    International MS journal, 2011, Volume: 17, Issue:3

    Topics: Fingolimod Hydrochloride; Glatiramer Acetate; Humans; Interferon beta-1a; Interferon beta-1b; Interferon-beta; Mitoxantrone; Multiple Sclerosis; Recurrence

2011
Balancing the benefits and risks of disease-modifying therapy in patients with multiple sclerosis.
    Journal of the neurological sciences, 2011, Volume: 311 Suppl 1

    Topics: Administration, Oral; Antibodies, Monoclonal, Humanized; Fingolimod Hydrochloride; Glatiramer Acetate; Humans; Immunosuppressive Agents; Interferon-beta; Mitoxantrone; Multiple Sclerosis; Multiple Sclerosis, Relapsing-Remitting; Natalizumab; Peptides; Pharmacovigilance; Propylene Glycols; Risk Assessment; Sphingosine

2011
Knowledge retrieval from PubMed abstracts and electronic medical records with the Multiple Sclerosis Ontology.
    PloS one, 2015, Volume: 10, Issue:2

    Topics: Antineoplastic Agents; Antirheumatic Agents; Biological Ontologies; Computational Biology; Electronic Health Records; Fingolimod Hydrochloride; Humans; Immunosuppressive Agents; Information Storage and Retrieval; Knowledge Discovery; Mitoxantrone; Multiple Sclerosis; PubMed; Rituximab

2015
Cerebrospinal fluid NCAM levels are modulated by disease-modifying therapies.
    Acta neurologica Scandinavica, 2019, Volume: 139, Issue:5

    Topics: Adult; Biomarkers; CD56 Antigen; Enzyme-Linked Immunosorbent Assay; Female; Fingolimod Hydrochloride; Humans; Immunologic Factors; Male; Middle Aged; Mitoxantrone; Multiple Sclerosis; Multiple Sclerosis, Relapsing-Remitting; Natalizumab

2019
COVID-19 in Patients with Multiple Sclerosis: Associations with Disease-Modifying Therapies.
    CNS drugs, 2021, Volume: 35, Issue:3

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Alemtuzumab; Azathioprine; Black or African American; Cladribine; Comorbidity; COVID-19; Crotonates; Cyclophosphamide; Cyclosporine; Databases, Factual; Dimethyl Fumarate; Female; Fingolimod Hydrochloride; Hospitalization; Humans; Hydroxybutyrates; Immunologic Factors; Immunosuppressive Agents; Incidence; Interferon-beta; Logistic Models; Lupus Erythematosus, Systemic; Male; Methotrexate; Middle Aged; Mitoxantrone; Multiple Sclerosis; Mycophenolic Acid; Natalizumab; Nitriles; Obesity; Risk Factors; Rituximab; SARS-CoV-2; Toluidines; United States; White People; Young Adult

2021