Page last updated: 2024-09-02

fingolimod and sotrastaurin

fingolimod has been researched along with sotrastaurin in 1 studies

Compound Research Comparison

Studies
(fingolimod)
Trials
(fingolimod)
Recent Studies (post-2010)
(fingolimod)
Studies
(sotrastaurin)
Trials
(sotrastaurin)
Recent Studies (post-2010) (sotrastaurin)
65051881269

Protein Interaction Comparison

ProteinTaxonomyfingolimod (IC50)sotrastaurin (IC50)
Serine/threonine-protein kinase D3Homo sapiens (human)0.0021
Tyrosine-protein kinase ABL1Homo sapiens (human)3.3
Protein kinase C beta typeHomo sapiens (human)0.0025
Tyrosine-protein kinase FynHomo sapiens (human)5.5
Cytochrome P450 3A4Homo sapiens (human)0.001
Serine/threonine-protein kinase pim-1Homo sapiens (human)0.0501
Protein kinase C alpha typeHomo sapiens (human)0.0026
Cyclin-A2Homo sapiens (human)2.3
Tyrosine-protein kinase JAK1Homo sapiens (human)7.3
Protein kinase C eta typeHomo sapiens (human)0.0041
Cyclin-dependent kinase 2Homo sapiens (human)2.3
Tyrosine-protein kinase receptor UFOHomo sapiens (human)9.1
Vascular endothelial growth factor receptor 3Homo sapiens (human)4.6
Vascular endothelial growth factor receptor 2Homo sapiens (human)3.9
Glycogen synthase kinase-3 betaHomo sapiens (human)0.87
Tyrosine-protein kinase JAK3Homo sapiens (human)1.5
Protein kinase C beta type Mus musculus (house mouse)0.234
Cyclin-A1Homo sapiens (human)2.3
Protein kinase C epsilon typeHomo sapiens (human)0.0041
Protein kinase C theta typeHomo sapiens (human)0.0094
Focal adhesion kinase 1Homo sapiens (human)8.3
Protein kinase C zeta typeHomo sapiens (human)5.4
Protein kinase C delta typeHomo sapiens (human)0.0025
Peroxisome proliferator-activated receptor alphaHomo sapiens (human)0.0031
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrialHomo sapiens (human)6.7

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Angst, D; Bassilana, F; Beerli, C; Berst, F; Bollbuck, B; Bruns, C; Buehlmayer, P; Hersperger, R; Janser, P; Oberer, L; Pally, C; Quancard, J; Streiff, M1

Other Studies

1 other study(ies) available for fingolimod and sotrastaurin

ArticleYear
An oral sphingosine 1-phosphate receptor 1 (S1P(1)) antagonist prodrug with efficacy in vivo: discovery, synthesis, and evaluation.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Administration, Oral; Aminobutyrates; Animals; Heart Transplantation; Lymphocytes; Magnetic Resonance Spectroscopy; Male; Molecular Structure; Prodrugs; Rats; Rats, Inbred Lew; Receptors, Lysosphingolipid; Sulfonamides

2012