fg 7142 and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate

fg 7142 has been researched along with methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-199018 (69.23)18.7374
1990's5 (19.23)18.2507
2000's3 (11.54)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Andersen, KE; Frederiksen, K; Knutsen, LJ; Nielsen, EB; Suzdak, PD; Sørensen, PO1
Brain, PF; Pankaj, V1
Dragunow, M1
Cooper, SJ; Estall, LB1
Jensen, LH; Petersen, EN2
Biggio, G; Corda, MG; Giorgi, O; Longoni, B1
File, SE; Pellow, S1
Moody, EJ; Skolnick, P1
Atsoggiu, T; Concas, A; Serra, M1
Atsoggiu, T; Biggio, G; Concas, A; Serra, M1
Barber, DJ; Cooper, SJ; Gilbert, DB; Moores, WR1
Little, HJ; Nutt, DJ; Taylor, SC1
Arora, PK; Hanna, EE; Paul, SM; Skolnick, P1
Randall, JI; Rodgers, RJ1
Ableitner, A; Herz, A1
Little, HJ; Nutt, DJ; Sellars, N; Taylor, SC1
Kehr, W; Schmiechen, R; Schneider, HH; Stephens, DN1
Little, HJ; Minchin, MC; Nutt, DJ; Taylor, SC1
Braestrup, C; Honoré, T; Jensen, LH; Nielsen, M; Petersen, EN1
Biggio, G; Concas, A; Corda, MG; Crisponi, C; Gessa, GL; Nurchi, V; Salis, M; Serra, M1
Gurley, D; White, G1
Cole, BJ; Hillmann, M; Jones, GH; Klewer, M; Seidelmann, D1
Boehrer, A; Marescaux, C; Reibel, S; Simler, S; Vergnes, M1

Reviews

1 review(s) available for fg 7142 and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate

ArticleYear
Behavioural pharmacology of food, water and salt intake in relation to drug actions at benzodiazepine receptors.
    Neuroscience and biobehavioral reviews, 1985,Spring, Volume: 9, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Appetite; Appetite Depressants; Benzodiazepines; Benzodiazepinones; Carbolines; Chlordiazepoxide; Chlorides; Choice Behavior; Diazepam; Drinking Behavior; Feeding Behavior; Flumazenil; Food Deprivation; Food Preferences; gamma-Aminobutyric Acid; Ion Channels; Midazolam; Picrotoxin; Punishment; Pyrazoles; Receptors, GABA-A; Satiation; Sodium Chloride; Species Specificity

1985

Other Studies

25 other study(ies) available for fg 7142 and methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
NNC-711, a novel potent and selective gamma-aminobutyric acid uptake inhibitor: pharmacological characterization.
    European journal of pharmacology, 1992, Dec-02, Volume: 224, Issue:2-3

    Topics: Animals; Anticonvulsants; Astrocytes; Behavior, Animal; Brain; Carbolines; Cells, Cultured; Convulsants; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Motor Activity; Neurons; Nicotinic Acids; Nipecotic Acids; Oximes; Pentylenetetrazole; Rats; Seizures; Synaptosomes; Tiagabine

1992
Effects of prenatal exposure to benzodiazepine-related drugs on early development and adult social behaviour in Swiss mice--III. Inverse agonists.
    General pharmacology, 1991, Volume: 22, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Body Weight; Carbolines; Female; Growth; Male; Mice; Postural Balance; Pregnancy; Prenatal Exposure Delayed Effects; Sex Factors; Social Behavior

1991
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines

1990
Lorazepam and FG 7142 induce tolerance to the DMCM antagonistic effect of benzodiazepine receptor ligands.
    Brain research bulletin, 1987, Volume: 19, Issue:3

    Topics: Animals; Carbolines; Dose-Response Relationship, Drug; Drug Tolerance; Female; Lorazepam; Male; Mice; Receptors, GABA-A; Seizures

1987
Decreased sensitivity to diazepam induced by chronic administration of FG 7142.
    Neuroscience letters, 1988, Mar-31, Volume: 86, Issue:2

    Topics: Animals; Anticonvulsants; Azides; Benzodiazepines; Brain; Brain Chemistry; Carbolines; Convulsants; Diazepam; Drug Interactions; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures

1988
Low and high doses of benzodiazepine receptor inverse agonists respectively improve and impair performance in passive avoidance but do not affect habituation.
    Behavioural brain research, 1988, Sep-01, Volume: 30, Issue:1

    Topics: Animals; Avoidance Learning; Brain; Carbolines; Dose-Response Relationship, Drug; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; Retention, Psychology

1988
The imidazobenzodiazepine Ro 15-4513 antagonizes methoxyflurane anesthesia.
    Life sciences, 1988, Volume: 43, Issue:16

    Topics: Anesthesia, General; Animals; Azides; Benzodiazepines; Carbolines; Flumazenil; Male; Methoxyflurane; Mice; Receptors, GABA-A; Sleep

1988
[Effect of stress on the function of chloride channels associated with the GABA receptor complex].
    Annali dell'Istituto superiore di sanita, 1988, Volume: 24, Issue:4

    Topics: Animals; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbolines; Cerebral Cortex; Chloride Channels; Chlorides; Male; Membrane Proteins; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological

1988
Foot-shock stress and anxiogenic beta-carbolines increase t-[35S]butylbicyclophosphorothionate binding in the rat cerebral cortex, an effect opposite to anxiolytics and gamma-aminobutyric acid mimetics.
    Journal of neurochemistry, 1988, Volume: 51, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbolines; Cell Membrane; Cerebral Cortex; Convulsants; Diazepam; Electroshock; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Male; Muscimol; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Physiological

1988
Benzodiazepine receptor ligands and the consumption of a highly palatable diet in non-deprived male rats.
    Psychopharmacology, 1985, Volume: 86, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Drug Interactions; Feeding Behavior; Flumazenil; Ligands; Male; Midazolam; Pyrazoles; Rats; Receptors, GABA-A

1985
Chronic treatment with lorazepam and FG 7142 may change the effects of benzodiazepine receptor agonists, antagonists and inverse agonists by different mechanisms.
    European journal of pharmacology, 1987, Jan-20, Volume: 133, Issue:3

    Topics: Animals; Carbolines; Drug Interactions; Drug Tolerance; Female; Flumazenil; Lorazepam; Mice; Pentylenetetrazole; Receptors, GABA-A

1987
Selective changes in the in vivo effects of benzodiazepine receptor ligands after chemical kindling with FG 7142.
    Neuropharmacology, 1987, Volume: 26, Issue:1

    Topics: Animals; Benzodiazepines; Body Temperature; Carbolines; Flurazepam; Kindling, Neurologic; Mice; Pyrazoles; Receptors, GABA-A; Seizures

1987
Suppression of the immune response by benzodiazepine receptor inverse agonists.
    Journal of neuroimmunology, 1987, Volume: 15, Issue:1

    Topics: Animals; Appetite Depressants; Carbolines; Cells, Cultured; Convulsants; Cytotoxicity, Immunologic; Immunosuppression Therapy; Lymphocyte Activation; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A; T-Lymphocytes; T-Lymphocytes, Cytotoxic

1987
Benzodiazepine ligands, nociception and 'defeat' analgesia in male mice.
    Psychopharmacology, 1987, Volume: 91, Issue:3

    Topics: Analgesia; Animals; Appetite Depressants; Benzodiazepines; Carbolines; Chlordiazepoxide; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Nociceptors; Pyrazoles

1987
Changes in local cerebral glucose utilization induced by the beta-carbolines FG 7142 and DMCM reveal brain structures involved in the control of anxiety and seizure activity.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1987, Volume: 7, Issue:4

    Topics: Animals; Anxiety; Autoradiography; Brain; Carbolines; Convulsants; Deoxyglucose; Flumazenil; Glucose; Male; Rats; Rats, Inbred Strains; Seizures

1987
A benzodiazepine agonist and contragonist have hypothermic effects in rodents.
    Neuropharmacology, 1985, Volume: 24, Issue:1

    Topics: Animals; Benzodiazepinones; Body Temperature; Carbolines; Convulsants; Flumazenil; Flurazepam; Hypothermia; Indoles; Male; Mice; Mice, Inbred Strains; Motor Activity; Rats; Rats, Inbred Strains

1985
Beta-carbolines with agonistic and inverse agonistic properties at benzodiazepine receptors of the rat.
    Neuroscience letters, 1984, Jun-29, Volume: 47, Issue:3

    Topics: Animals; Arousal; Brain; Carbolines; Chlordiazepoxide; Conditioning, Operant; Cues; Indoles; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission

1984
Investigating benzodiazepine receptor function in vivo using an intravenous infusion of DMCM.
    European journal of pharmacology, 1984, Aug-17, Volume: 103, Issue:3-4

    Topics: Animals; Anticonvulsants; Carbolines; Convulsants; Drug Interactions; Electroshock; Indoles; Infusions, Parenteral; Male; Mice; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Sensory Thresholds

1984
Ligands for benzodiazepine receptors with positive and negative efficacy.
    Biochemical pharmacology, 1984, Mar-15, Volume: 33, Issue:6

    Topics: Animals; Benzodiazepinones; Carbolines; Flumazenil; Humans; Ligands; Radioligand Assay; Receptors, Cell Surface; Receptors, GABA-A

1984
Stress and beta-carbolines decrease the density of low affinity GABA binding sites; an effect reversed by diazepam.
    Brain research, 1984, Jul-02, Volume: 305, Issue:1

    Topics: Animals; Binding Sites; Carbolines; Cerebral Cortex; Diazepam; gamma-Aminobutyric Acid; Handling, Psychological; Indoles; Male; Rats; Rats, Inbred Strains; Stress, Physiological

1984
Benzodiazepine site inverse agonists can selectively inhibit subtypes of the GABAA receptor.
    Neuroreport, 1995, Jun-19, Volume: 6, Issue:9

    Topics: Animals; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; GABA Agonists; gamma-Aminobutyric Acid; Oocytes; Patch-Clamp Techniques; Pyrazoles; Receptors, GABA-A; Xenopus

1995
Effects of benzodiazepine receptor partial inverse agonists in the elevated plus maze test of anxiety in the rat.
    Psychopharmacology, 1995, Volume: 121, Issue:1

    Topics: Animals; Anxiety; Appetite Depressants; Behavior, Animal; Carbolines; Convulsants; Dose-Response Relationship, Drug; GABA-A Receptor Agonists; Male; Maze Learning; Rats; Rats, Wistar; Yohimbine

1995
Selective susceptibility to inhibitors of GABA synthesis and antagonists of GABA(A) receptor in rats with genetic absence epilepsy.
    Experimental neurology, 2000, Volume: 161, Issue:2

    Topics: 3-Mercaptopropionic Acid; Animals; Bicuculline; Carbolines; Convulsants; Electroencephalography; Epilepsy, Absence; Frontal Lobe; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Isoniazid; Kainic Acid; Limbic System; Male; Parietal Lobe; Picrotoxin; Proto-Oncogene Proteins c-fos; Rats; Rats, Mutant Strains; Rats, Wistar; Seizures; Strychnine

2000