fg 7142 and beta-carboline-3-carboxylic acid ethyl ester

fg 7142 has been researched along with beta-carboline-3-carboxylic acid ethyl ester in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-199010 (58.82)18.7374
1990's6 (35.29)18.2507
2000's0 (0.00)29.6817
2010's1 (5.88)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chapouthier, G; Dodd, RH; Dorey, G; Poissonnet, G; Potier, MC; Potier, P; Prado de Carvalho, L; Rossier, J; Venault, P1
Donát, P; Krsiak, M; Sulcová, A1
McCullough, LD; Salamone, JD1
Allen, M; Cook, JM; Griffiths, RR; Sannerud, CA1
Holtzman, SG; Mumford, GK1
Morse, WH; Teeple, ES; Wettstein, JG1
Crawley, JN; Paul, SM; Suzdak, PD1
Dubroeucq, MC; Gauthier, A; Guérémy, C; Le Fur, G; Mizoule, J; Renault, C; Uzan, A1
Caporali, MG; Gatta, F; Lucantoni, D; Massotti, M; Mele, L1
Sanger, D; Soubrié, P; Thiébot, MH1
File, SE; Pellow, S1
Nutt, D1
Braestrup, C; Kehr, W; Nielsen, M; Paschelke, G; Petersen, EN1
Braestrup, C; Honoré, T; Jensen, LH; Nielsen, M; Petersen, EN1
Biggio, G; Concas, A; Corda, MG; Crisponi, C; Gessa, GL; Nurchi, V; Salis, M; Serra, M1
Auta, J; Faust, WB; Lambert, P; Moerschbaecher, JM; Winsauer, PJ1
Dickson, CT; Hughes, AM; Lu, L; Treit, D; Yeung, M1

Reviews

1 review(s) available for fg 7142 and beta-carboline-3-carboxylic acid ethyl ester

ArticleYear
Anxiogenic properties of beta-CCE and FG 7142: a review of promises and pitfalls.
    Psychopharmacology, 1988, Volume: 94, Issue:4

    Topics: Animals; Anxiety; Appetite Depressants; Carbolines; Humans; Ligands

1988

Other Studies

16 other study(ies) available for fg 7142 and beta-carboline-3-carboxylic acid ethyl ester

ArticleYear
Synthesis and benzodiazepine receptor affinities of rigid analogues of 3-carboxy-beta-carbolines: demonstration that the benzodiazepine receptor recognizes preferentially the s-cis conformation of the 3-carboxy group.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:8

    Topics: Animals; Carbolines; Chemical Phenomena; Chemistry; In Vitro Techniques; Mice; Receptors, GABA-A; Stereoisomerism; Structure-Activity Relationship

1989
Beta--CCE and FG 7142 increase defensiveness during intraspecies encounters in mice.
    Psychopharmacology, 1992, Volume: 108, Issue:1-2

    Topics: Aggression; Animals; Anxiety; Carbolines; Escape Reaction; GABA-A Receptor Antagonists; Interpersonal Relations; Male; Mice; Mice, Inbred ICR; Motor Activity

1992
Anxiogenic drugs beta-CCE and FG 7142 increase extracellular dopamine levels in nucleus accumbens.
    Psychopharmacology, 1992, Volume: 109, Issue:3

    Topics: Analysis of Variance; Animals; Anxiety; Carbolines; Dopamine; Male; Microdialysis; Motor Activity; Nucleus Accumbens; Rats; Rats, Sprague-Dawley

1992
Behavioral effects of benzodiazepine ligands in non-dependent, diazepam-dependent and diazepam-withdrawn baboons.
    European journal of pharmacology, 1991, Sep-17, Volume: 202, Issue:2

    Topics: Animals; Behavior, Animal; Benzodiazepines; Carbolines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Ligands; Male; Midazolam; Papio; Receptors, GABA-A; Social Behavior; Substance Withdrawal Syndrome; Substance-Related Disorders

1991
Do adenosinergic substrates mediate methylxanthine effects upon reinforcement thresholds for electrical brain stimulation in the rat?
    Brain research, 1991, May-31, Volume: 550, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Brain; Carbolines; Chlordiazepoxide; Electric Stimulation; Hypothalamic Area, Lateral; Male; Midazolam; Phenylisopropyladenosine; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Purinergic; Reinforcement, Psychology; Self Stimulation; Sensory Thresholds; Theophylline; Triazoles

1991
Respiratory effects of benzodiazepine-related drugs in awake rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:3

    Topics: Administration, Inhalation; Alprazolam; Animals; Anti-Anxiety Agents; Appetite Depressants; Benzodiazepines; Buspirone; Carbolines; Carbon Dioxide; Drug Therapy, Combination; Female; Flumazenil; Lorazepam; Macaca mulatta; Male; Pentobarbital; Plethysmography; Pyrazoles; Respiration

1990
Effects of Ro15-4513 and other benzodiazepine receptor inverse agonists on alcohol-induced intoxication in the rat.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:3

    Topics: Alcoholic Intoxication; Animals; Azides; Benzodiazepines; Carbolines; Chlorides; Ethanol; Ion Channels; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Opposite effects of two ligands for peripheral type benzodiazepine binding sites, PK 11195 and RO5-4864, in a conflict situation in the rat.
    Life sciences, 1985, Mar-18, Volume: 36, Issue:11

    Topics: Animals; Benzodiazepinones; Carbolines; Conditioning, Operant; Conflict, Psychological; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Flumazenil; Isoquinolines; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Supraspinal convulsions induced by inverse benzodiazepine agonists in rabbits.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 234, Issue:1

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electroencephalography; Flumazenil; Male; Pyrazoles; Rabbits; Receptors, GABA-A; Seizures

1985
Chlordiazepoxide enhances the anxiogenic action of CGS 8216 in the social interaction test: evidence for benzodiazepine withdrawal?
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:1

    Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Chlordiazepoxide; Flumazenil; Humans; Male; Pyrazoles; Rats; Social Behavior; Species Specificity; Substance Withdrawal Syndrome

1985
Pharmacological and behavioural studies of benzodiazepine antagonists and contragonists.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepinones; Carbolines; Conditioning, Operant; Conflict, Psychological; Flumazenil; Ganglia, Spinal; Hippocampus; Male; Rats; Seizures; Social Behavior

1983
Does the reversal of the anticonflict effect of phenobarbital by beta-CCE and FG 7142 indicate benzodiazepine receptor-mediated anxiogenic properties?
    European journal of pharmacology, 1982, Aug-27, Volume: 82, Issue:3-4

    Topics: Animals; Anxiety; Carbolines; Conflict, Psychological; Diazepam; Flunitrazepam; Humans; Indoles; Male; Phenobarbital; Punishment; Rats; Rats, Inbred Strains; Receptors, Drug; Receptors, GABA-A

1982
Ligands for benzodiazepine receptors with positive and negative efficacy.
    Biochemical pharmacology, 1984, Mar-15, Volume: 33, Issue:6

    Topics: Animals; Benzodiazepinones; Carbolines; Flumazenil; Humans; Ligands; Radioligand Assay; Receptors, Cell Surface; Receptors, GABA-A

1984
Stress and beta-carbolines decrease the density of low affinity GABA binding sites; an effect reversed by diazepam.
    Brain research, 1984, Jul-02, Volume: 305, Issue:1

    Topics: Animals; Binding Sites; Carbolines; Cerebral Cortex; Diazepam; gamma-Aminobutyric Acid; Handling, Psychological; Indoles; Male; Rats; Rats, Inbred Strains; Stress, Physiological

1984
Effects of negative allosteric modulators of gamma-aminobutyric acidA receptors on complex behavioral processes in monkeys.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:1

    Topics: Allosteric Regulation; Alprazolam; Animals; Carbolines; Conditioning, Psychological; Discrimination Learning; Dose-Response Relationship, Drug; Erythrocebus patas; Female; Flumazenil; Receptors, GABA-A

1997
FG7142, yohimbine, and βCCE produce anxiogenic-like effects in the elevated plus-maze but do not affect brainstem activated hippocampal theta.
    Neuropharmacology, 2013, Volume: 75

    Topics: Adrenergic alpha-2 Receptor Antagonists; Analysis of Variance; Animals; Anxiety; Biophysics; Brain Stem; Carbolines; Disease Models, Animal; Electric Stimulation; GABA Antagonists; Hippocampus; Male; Maze Learning; Rats; Rats, Sprague-Dawley; Theta Rhythm; Yohimbine

2013