fg 7142 and 2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one

fg 7142 has been researched along with 2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-199018 (81.82)18.7374
1990's4 (18.18)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davies, MF; Loew, GH; Pryor, GT; Uyeno, ET1
Morse, WH; Teeple, ES; Wettstein, JG1
Dragunow, M1
Crawley, JN; Paul, SM; Suzdak, PD1
Wettstein, JG1
Cooper, SJ; Estall, LB1
Cooper, SJ; Kirkham, TC1
Green, S; Hodges, H1
File, SE; Pellow, S5
Braestrup, C; Petersen, EN; Scheel-Krüger, J1
Caporali, MG; Gatta, F; Lucantoni, D; Massotti, M; Mele, L1
Barber, DJ; Cooper, SJ; Gilbert, DB; Moores, WR1
Cooper, SJ2
Little, HJ; Nutt, DJ; Taylor, SC1
Randall, JI; Rodgers, RJ1
Crawley, JN; Paul, SM; Skolnick, P1
Gurley, D; White, G1

Reviews

1 review(s) available for fg 7142 and 2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one

ArticleYear
Behavioural pharmacology of food, water and salt intake in relation to drug actions at benzodiazepine receptors.
    Neuroscience and biobehavioral reviews, 1985,Spring, Volume: 9, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Appetite; Appetite Depressants; Benzodiazepines; Benzodiazepinones; Carbolines; Chlordiazepoxide; Chlorides; Choice Behavior; Diazepam; Drinking Behavior; Feeding Behavior; Flumazenil; Food Deprivation; Food Preferences; gamma-Aminobutyric Acid; Ion Channels; Midazolam; Picrotoxin; Punishment; Pyrazoles; Receptors, GABA-A; Satiation; Sodium Chloride; Species Specificity

1985

Other Studies

21 other study(ies) available for fg 7142 and 2-phenylpyrazolo(4,3-c)quinolin-3(5h)-one

ArticleYear
Selective effect on punished versus unpunished responding in a conflict test as the criterion for anxiogenic activity.
    Life sciences, 1990, Volume: 47, Issue:15

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Carbolines; Conflict, Psychological; Electroshock; Male; Pentylenetetrazole; Punishment; Pyrazoles; Rats; Rats, Inbred Strains; Water Deprivation

1990
Respiratory effects of benzodiazepine-related drugs in awake rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:3

    Topics: Administration, Inhalation; Alprazolam; Animals; Anti-Anxiety Agents; Appetite Depressants; Benzodiazepines; Buspirone; Carbolines; Carbon Dioxide; Drug Therapy, Combination; Female; Flumazenil; Lorazepam; Macaca mulatta; Male; Pentobarbital; Plethysmography; Pyrazoles; Respiration

1990
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines

1990
Effects of Ro15-4513 and other benzodiazepine receptor inverse agonists on alcohol-induced intoxication in the rat.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:3

    Topics: Alcoholic Intoxication; Animals; Azides; Benzodiazepines; Carbolines; Chlorides; Ethanol; Ion Channels; Male; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Behavioral studies with the beta-carboline FG 7142 combined with related drugs in monkeys.
    European journal of pharmacology, 1989, Apr-25, Volume: 163, Issue:2-3

    Topics: Animals; Appetite Depressants; Behavior, Animal; Benzodiazepines; Carbolines; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Flumazenil; Lorazepam; Male; Pyrazoles; Reinforcement Schedule; Saimiri

1989
Adrenalectomy and the anorectic effects of benzodiazepine inverse agonists and opiate antagonists in rats fed a palatable diet.
    Physiology & behavior, 1987, Volume: 40, Issue:4

    Topics: Adrenal Glands; Adrenalectomy; Animals; Appetite; Appetite Depressants; Carbolines; Clonazepam; Diprenorphine; Eating; Hunger; Male; Morphinans; Naltrexone; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Taste

1987
Are the effects of benzodiazepines on discrimination and punishment dissociable?
    Physiology & behavior, 1987, Volume: 41, Issue:3

    Topics: Amygdala; Animals; Behavior, Animal; Benzodiazepines; Carbolines; Chlordiazepoxide; Discrimination, Psychological; Ethanolamines; Flumazenil; gamma-Aminobutyric Acid; Midazolam; Punishment; Pyrazoles; Rats; Receptors, GABA-A

1987
Pro- and anti-convulsant drug effects in combination with the convulsant benzodiazepine Ro 5-4864.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Carbolines; Convulsants; Drug Interactions; Male; Mice; Mice, Inbred Strains; Pyrazoles; Pyridazines; Quinolines

1985
Anxiolytic and anxiogenic drug effects on exploratory activity in an elevated plus-maze: a novel test of anxiety in the rat.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Benzodiazepinones; Buspirone; Carbolines; Convulsants; Exploratory Behavior; Flumazenil; Male; Pyrazoles; Pyridazines; Pyrimidines; Quinolines; Rats

1986
Evidence that the anticonflict effect of midazolam in amygdala is mediated by the specific benzodiazepine receptors.
    Neuroscience letters, 1985, Feb-04, Volume: 53, Issue:3

    Topics: Amygdala; Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Conflict, Psychological; Flumazenil; Male; Midazolam; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Supraspinal convulsions induced by inverse benzodiazepine agonists in rabbits.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 234, Issue:1

    Topics: Animals; Benzodiazepinones; Carbolines; Diazepam; Electroencephalography; Flumazenil; Male; Pyrazoles; Rabbits; Receptors, GABA-A; Seizures

1985
Benzodiazepine receptor ligands and the consumption of a highly palatable diet in non-deprived male rats.
    Psychopharmacology, 1985, Volume: 86, Issue:3

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Carbolines; Drug Interactions; Feeding Behavior; Flumazenil; Ligands; Male; Midazolam; Pyrazoles; Rats; Receptors, GABA-A

1985
The anorectic effect of FG 7142, a partial inverse agonist at benzodiazepine recognition sites, is reversed by CGS 8216 and clonazepam but not food deprivation.
    Brain research, 1985, Oct-28, Volume: 346, Issue:1

    Topics: Animals; Appetite Depressants; Carbolines; Clonazepam; Food Deprivation; Male; Pyrazoles; Rats; Receptors, GABA-A

1985
The effects of putative anxiogenic compounds (FG 7142, CGS 8216 and Ro 15-1788) on the rat corticosterone response.
    Physiology & behavior, 1985, Volume: 35, Issue:4

    Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Corticosterone; Flumazenil; Male; Pyrazoles; Rats; Receptors, GABA-A; Stress, Psychological

1985
Selective changes in the in vivo effects of benzodiazepine receptor ligands after chemical kindling with FG 7142.
    Neuropharmacology, 1987, Volume: 26, Issue:1

    Topics: Animals; Benzodiazepines; Body Temperature; Carbolines; Flurazepam; Kindling, Neurologic; Mice; Pyrazoles; Receptors, GABA-A; Seizures

1987
Benzodiazepine ligands, nociception and 'defeat' analgesia in male mice.
    Psychopharmacology, 1987, Volume: 91, Issue:3

    Topics: Analgesia; Animals; Appetite Depressants; Benzodiazepines; Carbolines; Chlordiazepoxide; Diazepam; Flumazenil; Male; Mice; Mice, Inbred DBA; Nociceptors; Pyrazoles

1987
Hyperphagic and anorectic effects of beta-carbolines in a palatable food consumption test: comparisons with triazolam and quazepam.
    European journal of pharmacology, 1986, Jan-29, Volume: 120, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Appetite Depressants; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; Eating; Male; Pyrazoles; Rats; Triazolam

1986
Chlordiazepoxide enhances the anxiogenic action of CGS 8216 in the social interaction test: evidence for benzodiazepine withdrawal?
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:1

    Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Chlordiazepoxide; Flumazenil; Humans; Male; Pyrazoles; Rats; Social Behavior; Species Specificity; Substance Withdrawal Syndrome

1985
Absence of intrinsic antagonist actions of benzodiazepine antagonists on an exploratory model of anxiety in the mouse.
    Neuropharmacology, 1984, Volume: 23, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Carbolines; Disease Models, Animal; Dose-Response Relationship, Drug; Exploratory Behavior; Flumazenil; Humans; Male; Mice; Pyrazoles

1984
The anxiogenic action of FG 7142 in the social interaction test is reversed by chlordiazepoxide and Ro 15-1788 but not by CGS 8216.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 271, Issue:2

    Topics: Animals; Anxiety; Benzodiazepinones; Carbolines; Chlordiazepoxide; Convulsants; Flumazenil; Humans; Indoles; Male; Motor Activity; Pyrazoles; Rats; Social Behavior

1984
Benzodiazepine site inverse agonists can selectively inhibit subtypes of the GABAA receptor.
    Neuroreport, 1995, Jun-19, Volume: 6, Issue:9

    Topics: Animals; Benzodiazepines; Carbolines; Dose-Response Relationship, Drug; GABA Agonists; gamma-Aminobutyric Acid; Oocytes; Patch-Clamp Techniques; Pyrazoles; Receptors, GABA-A; Xenopus

1995