fexofenadine and naringin

fexofenadine has been researched along with naringin in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (20.00)29.6817
2010's4 (80.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Bailey, DG; Dresser, GK; Kim, RB; Leake, BF1
Alexander, N; Dahlke, M; Hanna, I; Hariry, S; Jarugula, V; Rebello, S; Vapurcuyan, A; Zhao, S1
Chen, Y; Jiang, S; Li, F; Li, Y; Liu, L; Liu, X; Xu, P; Zhang, M; Zhao, K; Zhao, W; Zhong, Z1

Reviews

1 review(s) available for fexofenadine and naringin

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010

Trials

2 trial(s) available for fexofenadine and naringin

ArticleYear
Naringin is a major and selective clinical inhibitor of organic anion-transporting polypeptide 1A2 (OATP1A2) in grapefruit juice.
    Clinical pharmacology and therapeutics, 2007, Volume: 81, Issue:4

    Topics: Adult; Anticoagulants; Beverages; Citrus paradisi; Cross-Over Studies; Data Interpretation, Statistical; Double-Blind Method; Drug Interactions; Female; Flavanones; Furocoumarins; HeLa Cells; Hesperidin; Histamine H1 Antagonists; Humans; Male; Middle Aged; Organic Anion Transporters; Reproducibility of Results; Terfenadine

2007
Intestinal OATP1A2 inhibition as a potential mechanism for the effect of grapefruit juice on aliskiren pharmacokinetics in healthy subjects.
    European journal of clinical pharmacology, 2012, Volume: 68, Issue:5

    Topics: Adult; Amides; Antihypertensive Agents; Beverages; Biological Transport; Citrus paradisi; Cross-Over Studies; Flavanones; Food-Drug Interactions; Fruit; Fumarates; Half-Life; HEK293 Cells; Humans; Intestinal Mucosa; Male; Organic Anion Transporters; Recombinant Proteins; Renin; Terfenadine; Young Adult

2012

Other Studies

2 other study(ies) available for fexofenadine and naringin

ArticleYear
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Paroxetine decreased plasma exposure of glyburide partly via inhibiting intestinal absorption in rats.
    Drug metabolism and pharmacokinetics, 2015, Volume: 30, Issue:3

    Topics: Animals; Antidepressive Agents, Second-Generation; Biological Transport; Caco-2 Cells; Drug Interactions; Drug Therapy, Combination; Feces; Flavanones; Glyburide; Humans; Hypoglycemic Agents; Intestinal Absorption; Male; Microsomes, Liver; Organic Anion Transporters, Sodium-Independent; Paroxetine; Rats, Sprague-Dawley; Terfenadine

2015