fentanyl and etorphine

fentanyl has been researched along with etorphine in 62 studies

Research

Studies (62)

TimeframeStudies, this research(%)All Research%
pre-199024 (38.71)18.7374
1990's17 (27.42)18.2507
2000's10 (16.13)29.6817
2010's8 (12.90)24.3611
2020's3 (4.84)2.80

Authors

AuthorsStudies
Govoni, S; Kumakura, K; Spano, PF; Tonon, GC; Trabucchi, M1
Green, CJ1
Patenaude, RP1
Kocher, FH; Williams, TD1
Mortelmans, J1
Ebedes, H1
Smuts, GL1
Coghill, RC; Frenk, H; Leshem, M; Mayer, DJ1
Kreeger, TJ; Seal, US1
Dickenson, AH; McQuay, HJ; Sullivan, AF1
Blake, JW; DeQuick, D; Kamerling, S; Tai, C; Tobin, T; Weckman, TJ; Wood, T1
Ashraf, M; Gordon, B; Granley, K; Mishra, U; Rao, MM; Singh, AK1
He, BL; Jin, B; Li, H1
Andrews, P; Martin, J1
Garzón, J; Herz, A; Schulz, R1
Hynes, MD; Leander, JD; Reel, JK; Zimmerman, DM1
Cheney, CS; Hattingh, J1
von Hegel, G; Wiesner, H1
Day, AR; Freer, RJ; Liao, CS1
Grevel, J; Richards, ML; Rosenbaum, JS; Sadée, W1
Cochin, J; Miller, JM; Pelikan, EW; Rosow, CE1
Field, M; Kachur, JF; Miller, RJ1
Holford, NH; Rosenbaum, JS; Sadée, W1
Aman, RA; Holford, NH; Richards, ML; Rosenbaum, JS; Sadée, W1
Flecknell, PA; John, M; Mitchell, M; Shurey, C; Simpkin, S1
Doyle, R; Glenn, BL; Kocan, AA; Kubat, G; Shaw, MG; Thedford, TR; Waldrup, K1
Duttaroy, A; Yoburn, BC1
Davis, T; Duttaroy, A; Shah, S; Yoburn, BC2
House, JD; Makhay, MM; Walker, EA; Young, AM1
Chi, ZQ; Li, GF; Lu, YF1
Brine, GA; Carroll, FI; Ni, Q; Partilla, JS; Rothman, RB; Stark, PA; Xu, H1
Billings, B; Duttaroy, A; Yoburn, BC1
Butour, JL; Meunier, JC; Moisand, C; Mollereau, C; Parmentier, M1
Freye, E; Neruda, B; Smith, OW1
Harris, LS; Kim, SA; Martin, TJ; Smith, JE1
Brine, GA; Carroll, FI; Chen, C; Lai, J; Liu-Chen, LY; Lu, YF; Partilla, JS; Porreca, F; Rice, KC; Rothman, RB; Sadee, W; Xu, H1
Hairston, CT; Harris, LS; Lutz, PO; Martin, TJ; Porreca, F1
Chen, J; Chi, ZQ; Li, CL; Pei, G; Shen, QX; Wang, CH; Wei, Q; Zhou, DH1
Akil, H; Lee, KO; Traynor, JR; Woods, JH1
Cao, Y; Chen, KX; Huang, XQ; Ji, RY; Jiang, HL; Luo, XM; Zhu, YC1
Enserink, M; Stone, R1
David Clark, J; Demirci, H; Gharagozlou, P; Lameh, J1
Aibak, H; Beaudet, A; Cahill, CM; Collier, B; Esdaile, MJ; Kieffer, BL; Morinville, A1
Chen, XJ; Chi, ZQ; He, Y; Jin, WQ; Liu, ZH; Shen, QX; Zhang, HP1
Portas, TJ1
Clippinger, TL; Howard, LL; Kearns, KS; Larsen, RS; Morris, PJ1
Drevemo, SA; Grootenhuis, JG; Karstad, L1
Virk, MS; Williams, JT1
Fick, LG; Fuller, A; Hetem, RS; Matthee, A; Meyer, LC; Mitchell, D1
Chi, ZQ; Liu, JG; Sun, JF; Tao, YM; Wang, YH; Xu, XJ1
Chu, J; Law, PY; Loh, HH; Zhang, Y; Zheng, H1
Akbarali, HI; Dewey, WL; Maguma, HT1
Edner, A; Fahlman, Å; Foggin, C; Nyman, G; Wenger, S1
Meyer, LCR; Zeiler, GE2
Bdolah-Abram, T; King, R; Lapid, R; Shilo-Benjamini, Y1
Bryant, B; Jordan, NR; McMahon, CR; Pittard, S1
Laubscher, L; Laurence, M; Meyer, LRC; Pfitzer, S; Raath, JP; Vaughan-Higgins, R; Warren, K1
Laubscher, L; Laurence, M; Meyer, L; Pfitzer, S; Raath, JP; Vaughan-Higgins, R; Warren, K2
Baert, B; Beetens, J; Bodé, S; De Spiegeleer, B; Deconinck, E; Lambert, J; Slegers, G; Slodicka, M; Stoppie, P; Van Gele, M; Vander Heyden, Y1

Reviews

2 review(s) available for fentanyl and etorphine

ArticleYear
Narcotic analgesics, their detection and pain measurement in the horse: a review.
    Equine veterinary journal, 1989, Volume: 21, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Butorphanol; Chromatography, Thin Layer; Cyclazocine; Ethylketocyclazocine; Etorphine; Fentanyl; Horses; Morphine; Pain Measurement; Pentazocine; Pyrrolidines; Radioimmunoassay; Receptors, Opioid

1989
A review of drugs and techniques used for sedation and anaesthesia in captive rhinoceros species.
    Australian veterinary journal, 2004, Volume: 82, Issue:9

    Topics: Adrenergic alpha-Agonists; Analgesics, Opioid; Anesthetics, Combined; Animals; Animals, Zoo; Azaperone; Butyrophenones; Etorphine; Fentanyl; Hypnotics and Sedatives; Perissodactyla

2004

Other Studies

60 other study(ies) available for fentanyl and etorphine

ArticleYear
Interaction of narcotic analgesics with dopamine receptors in rat brain.
    Pharmacological research communications, 1975, Volume: 07, Issue:1

    Topics: Adenylyl Cyclases; Analgesics, Opioid; Animals; Corpus Striatum; Cyclic AMP; Depression, Chemical; Dextromoramide; Dextropropoxyphene; Dopamine; Enzyme Activation; Etorphine; Fentanyl; In Vitro Techniques; Male; Methadone; Rats; Receptors, Drug

1975
Neuroleptanalgesic drug combinations in the anaesthetic management of small laboratory animals.
    Laboratory animals, 1975, Volume: 9, Issue:3

    Topics: Alfaxalone Alfadolone Mixture; Anesthesia, Inhalation; Anesthetics; Animals; Animals, Laboratory; Butyrophenones; Cricetinae; Diazepam; Drug Combinations; Ethanol; Etorphine; Fentanyl; Guinea Pigs; Halothane; Imidazoles; Ketamine; Methohexital; Methotrimeprazine; Mice; Neuroleptanalgesia; Pentobarbital; Piperazines; Rabbits; Rats; Xylazine

1975
Evaluation of fentanyl citrate, etorphine hydrochloride, and naloxone hydrochloride in captive polar bears.
    Journal of the American Veterinary Medical Association, 1979, Nov-01, Volume: 175, Issue:9

    Topics: Anesthesia; Animals; Carnivora; Etorphine; Female; Fentanyl; Immobilization; Male; Morphinans; Naloxone; Ursidae

1979
Comparison of anesthetic agents in the sea otter.
    Journal of the American Veterinary Medical Association, 1978, Nov-01, Volume: 173, Issue:9

    Topics: Anesthetics; Animals; Carnivora; Diazepam; Drug Combinations; Etorphine; Female; Fentanyl; Halothane; Immobilization; Ketamine; Male; Tiletamine; Zolazepam

1978
Anaesthesia in okapis.
    Acta zoologica et pathologica Antverpiensia, 1978, Issue:71

    Topics: Anesthesia; Animals; Artiodactyla; Azaperone; Etorphine; Fentanyl; Immobilization; Male; Nalorphine; Xylazine

1978
The capture and translocation of gemsbok Oryx gazella gazella in the Nambi Desert with the aid of fentanyl, etorphine and tranquillizers.
    Journal of the South African Veterinary Association, 1975, Volume: 46, Issue:4

    Topics: Acepromazine; Animals; Artiodactyla; Azaperone; Chlorpromazine; Etorphine; Female; Fentanyl; Immobilization; Male; Morphinans; South Africa; Tranquilizing Agents; Transportation; Triflupromazine

1975
An appraisal of naloxone hydrochloride as a narcotic antagonist in the capture and release of wild herbivores.
    Journal of the American Veterinary Medical Association, 1975, Oct-01, Volume: 167, Issue:7

    Topics: Animals; Antelopes; Artiodactyla; Buffaloes; Elephants; Etorphine; Fentanyl; Male; Mammals; Naloxone; Perissodactyla; Swine

1975
Paradoxical opiate specific paralytic effects of high doses of intracerebroventricular etorphine and fentanyl in rats.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 38, Issue:2

    Topics: Animals; Etorphine; Fentanyl; Injections, Intraventricular; Injections, Spinal; Male; Naloxone; Paralysis; Rats; Rats, Inbred Strains; Receptors, Opioid

1991
Immobilization of gray wolves (Canis lupus) with sufentanil citrate.
    Journal of wildlife diseases, 1990, Volume: 26, Issue:4

    Topics: Anesthetics; Animals; Arousal; Carnivora; Etorphine; Female; Fentanyl; Immobilization; Male; Naloxone; Sufentanil; Xylazine; Yohimbine

1990
Intrathecal etorphine, fentanyl and buprenorphine on spinal nociceptive neurones in the rat.
    Pain, 1990, Volume: 42, Issue:2

    Topics: Animals; Buprenorphine; Dose-Response Relationship, Drug; Etorphine; Fentanyl; Injections, Intravenous; Injections, Spinal; Lipids; Neurons; Nociceptors; Rats; Solubility; Spinal Cord

1990
Screening and confirmation of drugs in horse urine by using a simple column extraction procedure.
    Journal of chromatography, 1989, Jun-28, Volume: 473, Issue:1

    Topics: Animals; Chromatography, Liquid; Chromatography, Thin Layer; Etorphine; Fentanyl; Gas Chromatography-Mass Spectrometry; Horses; Mazindol; Methamphetamine; Pharmaceutical Preparations; Radioimmunoassay

1989
[Narcotics combined with low-flow nitrous oxide in open-heart surgery].
    Zhonghua wai ke za zhi [Chinese journal of surgery], 1986, Volume: 24, Issue:4

    Topics: Adolescent; Analgesics, Opioid; Anesthesia; Cardiac Surgical Procedures; Child; Etorphine; Female; Fentanyl; Heart Septal Defects, Ventricular; Humans; Male; Morphinans; Nitrous Oxide

1986
Conformation-activity relationships of opiate analgesics.
    Journal of computer-aided molecular design, 1987, Volume: 1, Issue:1

    Topics: Analgesics, Opioid; Benzimidazoles; Computer Graphics; Etorphine; Fentanyl; Models, Molecular; Molecular Conformation; Molecular Structure; Receptors, Opioid; Structure-Activity Relationship

1987
Evidence for the epsilon-type of opioid receptor in the rat vas deferens.
    Molecular pharmacology, 1985, Volume: 28, Issue:1

    Topics: Animals; Binding, Competitive; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Drug Synergism; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Etorphine; Fentanyl; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Vas Deferens

1985
Use of beta-funaltrexamine to determine mu opioid receptor involvement in the analgesic activity of various opioid ligands.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Biological Assay; Buprenorphine; Butorphanol; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Etorphine; Fentanyl; Methadone; Mice; Morphine; Muscle Contraction; Nalbuphine; Nalorphine; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, mu

1987
Effects of chemical immobilisation on the blood composition of impala (Aepyceros melampus (Lichtenstein).
    Journal of the South African Veterinary Association, 1988, Volume: 59, Issue:1

    Topics: Animals; Antelopes; Artiodactyla; Drug Combinations; Etorphine; Female; Fentanyl; Immobilization; Male; Morphinans; Thiazines; Time Factors; Xylazine

1988
[Practical advice concerning the immobilization of wild and zoo animals].
    Tierarztliche Praxis, 1985, Volume: 13, Issue:1

    Topics: Acepromazine; Animal Population Groups; Animals; Animals, Wild; Animals, Zoo; Central Nervous System Depressants; Drug Combinations; Etorphine; Fentanyl; Immobilization; Ketamine; Species Specificity; Tranquilizing Agents; Xylazine

1985
Evidence for a single opioid receptor type on the field stimulated rat vas deferens.
    Life sciences, 1981, Dec-21, Volume: 29, Issue:25

    Topics: Animals; Benzimidazoles; beta-Endorphin; Dose-Response Relationship, Drug; Electric Stimulation; Endorphins; Enkephalins; Etorphine; Fentanyl; Male; Morphine; Oxymorphone; Rats; Rats, Inbred Strains; Receptors, Opioid; Sufentanil; Vas Deferens

1981
In vivo characterization of four types of opioid binding sites in rat brain.
    Life sciences, 1983, Volume: 33 Suppl 1

    Topics: Analgesics, Opioid; Animals; Brain; Buprenorphine; Diprenorphine; Etorphine; Fentanyl; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Sufentanil; Tritium

1983
Opiates and thermoregulation in mice. I. Agonists.
    The Journal of pharmacology and experimental therapeutics, 1980, Volume: 213, Issue:2

    Topics: Animals; Benzimidazoles; Body Temperature Regulation; Codeine; Dose-Response Relationship, Drug; Etorphine; Fentanyl; Hydromorphone; Isonipecotic Acids; Levorphanol; Male; Meperidine; Methadone; Mice; Morphine; Narcotics; Oxymorphone

1980
Control of guinea pig intestinal electrolyte secretion by a delta-opiate receptor.
    Proceedings of the National Academy of Sciences of the United States of America, 1980, Volume: 77, Issue:5

    Topics: Animals; Chlorides; Electric Conductivity; Endorphins; Etorphine; Female; Fentanyl; Guinea Pigs; Intestinal Mucosa; Membrane Potentials; Morphine; Muscle, Smooth; Naloxone; Receptors, Opioid

1980
Opiate receptor binding-effect relationship: sufentanil and etorphine produce analgesia at the mu-site with low fractional receptor occupancy.
    Brain research, 1984, Jan-23, Volume: 291, Issue:2

    Topics: Animals; Brain; Diprenorphine; Drug Interactions; Etorphine; Fentanyl; Morphinans; Naloxone; Pain; Rats; Receptors, Opioid; Sufentanil

1984
Discrimination of three types of opioid binding sites in rat brain in vivo.
    Molecular pharmacology, 1984, Volume: 25, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Diprenorphine; Etorphine; Fentanyl; Male; Naloxone; Rats; Receptors, Opioid; Sufentanil

1984
Neuroleptanalgesia in the rabbit.
    Laboratory animals, 1983, Volume: 17, Issue:2

    Topics: Acidosis; Animals; Butyrophenones; Diazepam; Drug Combinations; Etorphine; Fentanyl; Hypercapnia; Methotrimeprazine; Morphinans; Neuroleptanalgesia; Rabbits; Respiration; Time Factors

1983
Effects of chemical immobilization on hematologic and serum chemical values in captive white-tailed deer.
    Journal of the American Veterinary Medical Association, 1981, Dec-01, Volume: 179, Issue:11

    Topics: Animals; Blood Chemical Analysis; Central Nervous System Depressants; Deer; Etorphine; Fentanyl; Hematocrit; Hemoglobins; Immobilization; Morphinans; Succinylcholine; Thiazines; Xylazine

1981
The effect of intrinsic efficacy on opioid tolerance.
    Anesthesiology, 1995, Volume: 82, Issue:5

    Topics: Animals; Dose-Response Relationship, Drug; Drug Tolerance; Etorphine; Fentanyl; Male; Meperidine; Mice; Morphine; Narcotics; Oxycodone

1995
Spinal and supraspinal effects of pertussis toxin on opioid analgesia.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:3

    Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Etorphine; Fentanyl; Injections, Intraventricular; Injections, Spinal; Male; Mice; Morphine; Narcotic Antagonists; Narcotics; Pain Measurement; Pertussis Toxin; Spinal Cord; Virulence Factors, Bordetella

1994
In vivo apparent pA2 analysis for naltrexone antagonism of discriminative stimulus and analgesic effects of opiate agonists in rats.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:2

    Topics: Analgesia; Animals; Benzomorphans; Buprenorphine; Discrimination, Psychological; Etorphine; Fentanyl; Male; Morphine; Nalbuphine; Naltrexone; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu

1994
Characterization and distribution of mu opioid receptors in rabbit cerebellum.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1993, Volume: 14, Issue:6

    Topics: Animals; Autoradiography; Binding Sites; Cerebellum; Etorphine; Female; Fentanyl; Male; Rabbits; Radioligand Assay; Receptors, Opioid, mu

1993
Stereochemical requirements for pseudoirreversible inhibition of opioid mu receptor binding by the 3-methylfentanyl congeners, RTI-46144 and its enantiomers: evidence for different binding domains.
    Synapse (New York, N.Y.), 1993, Volume: 15, Issue:4

    Topics: Animals; Binding Sites; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Fentanyl; Ligands; Molecular Conformation; Rats; Receptors, Opioid, mu; Stereoisomerism

1993
Opioid antagonist-induced receptor upregulation: effects of concurrent agonist administration.
    Brain research bulletin, 1994, Volume: 33, Issue:2

    Topics: Animals; Brain; Drug Combinations; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Fentanyl; Male; Mice; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid, mu; Up-Regulation

1994
Opioid receptor regulation in mice.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:1

    Topics: Analgesics; Animals; Brain; Etorphine; Fentanyl; Male; Mice; Morphine; Naloxone; Narcotics; Receptors, Opioid, mu

1993
Replacement of Gln280 by His in TM6 of the human ORL1 receptor increases affinity but reduces intrinsic activity of opioids.
    FEBS letters, 1996, Oct-14, Volume: 395, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Diprenorphine; Dynorphins; Etorphine; Fentanyl; Glutamine; Histamine; Humans; Kinetics; Ligands; Naltrexone; Narcotic Antagonists; Narcotics; Nociceptin; Nociceptin Receptor; Opioid Peptides; Receptors, Opioid

1996
Studies on the abstinence-like overshoot following reversal of the potent 19-isoamyl derivative of etorphine with naloxone. A comparison with the opioids fentanyl and alfentanil.
    Arzneimittel-Forschung, 1997, Volume: 47, Issue:1

    Topics: Alfentanil; Analgesics, Opioid; Animals; Blood Gas Analysis; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Etorphine; Fentanyl; Heart Rate; Naloxone; Narcotic Antagonists; Receptors, Opioid, mu; Substance Withdrawal Syndrome

1997
Potent reinforcing effects of dihydroetorphine in rats.
    European journal of pharmacology, 1997, Apr-18, Volume: 324, Issue:2-3

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Etorphine; Fentanyl; Heroin; Male; Morphine; Morphine Derivatives; Rats; Rats, Inbred F344; Substance Withdrawal Syndrome; Substance-Related Disorders

1997
Opioid peptide receptor studies. 7. The methylfentanyl congener RTI-4614-4 and its four enantiomers bind to different domains of the rat mu opioid receptor.
    Synapse (New York, N.Y.), 1998, Volume: 28, Issue:2

    Topics: Affinity Labels; Analgesics; Analgesics, Opioid; Animals; Binding Sites; Binding, Competitive; COS Cells; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Etorphine; Fentanyl; Melphalan; Membrane Proteins; Protein Structure, Tertiary; Radioligand Assay; Rats; Receptors, Opioid, mu; Recombinant Fusion Proteins; Stereoisomerism

1998
Anti-allodynic actions of intravenous opioids in the nerve injured rat: potential utility of heroin and dihydroetorphine against neuropathic pain.
    European journal of pharmacology, 1998, Sep-11, Volume: 357, Issue:1

    Topics: Analgesics, Opioid; Animals; Drug Evaluation; Etorphine; Fentanyl; Heroin; Infusions, Intravenous; Ligation; Male; Morphine; Nerve Compression Syndromes; Pain; Rats; Rats, Inbred F344; Spinal Nerves

1998
Human mu-opioid receptor overexpressed in baculovirus system and its pharmacological characterizations.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1998, Volume: 19, Issue:3

    Topics: Animals; Baculoviridae; Cells, Cultured; Cyclic AMP; Diprenorphine; Etorphine; Fentanyl; Gene Expression; Insecta; Radioligand Assay; Receptors, Opioid, mu; Transfection

1998
Differential binding properties of oripavines at cloned mu- and delta-opioid receptors.
    European journal of pharmacology, 1999, Aug-13, Volume: 378, Issue:3

    Topics: Analgesics, Opioid; Animals; Benzamides; Binding, Competitive; Buprenorphine; Cloning, Molecular; Diprenorphine; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Morphine; Naloxone; Piperazines; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Sulfur Radioisotopes; Thebaine; Tritium; Tumor Cells, Cultured

1999
Study on mechanism of interaction of nociceptin and opioids binding with opioid receptor-like 1 receptor.
    Acta pharmacologica Sinica, 2000, Volume: 21, Issue:6

    Topics: Binding Sites; Drug Interactions; Etorphine; Fentanyl; Models, Molecular; Molecular Conformation; Nociceptin; Nociceptin Receptor; Opioid Peptides; Receptors, Opioid

2000
Toxicology. Questions swirl over knockout gas used in hostage crisis.
    Science (New York, N.Y.), 2002, Nov-08, Volume: 298, Issue:5596

    Topics: Etorphine; Female; Fentanyl; Halothane; Humans; Male; Narcotics; Prisoners; Russia; Terrorism; Tranquilizing Agents

2002
Activity of opioid ligands in cells expressing cloned mu opioid receptors.
    BMC pharmacology, 2003, Jan-04, Volume: 3

    Topics: Azocines; beta-Endorphin; Binding, Competitive; Butorphanol; Cell Line; Colforsin; Cyclic AMP; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Humans; Hydromorphone; Ligands; Morphine; Naltrexone; Phenazocine; Radioligand Assay; Receptors, Opioid, mu; Tritium

2003
Regulation of delta-opioid receptor trafficking via mu-opioid receptor stimulation: evidence from mu-opioid receptor knock-out mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Jun-15, Volume: 23, Issue:12

    Topics: Animals; Area Under Curve; Behavior, Animal; Cell Membrane; Dose-Response Relationship, Drug; Drug Administration Schedule; Etorphine; Female; Fentanyl; Male; Methadone; Mice; Mice, Inbred C57BL; Mice, Knockout; Morphine; Narcotics; Pain Measurement; Posterior Horn Cells; Protein Transport; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu; Time; Up-Regulation

2003
Binding affinity to and dependence on some opioids in Sf9 insect cells expressing human mu-opioid receptor.
    Acta pharmacologica Sinica, 2003, Volume: 24, Issue:9

    Topics: Analgesics, Opioid; Animals; Baculoviridae; Binding, Competitive; Cells, Cultured; Cyclic AMP; Etorphine; Female; Fentanyl; Heroin; Male; Mice; Opioid-Related Disorders; Receptors, Opioid, mu; Spodoptera; Transfection

2003
Chemical immobilization of rhebok (Pelea capreolus) with carfentanil-xylazine or etorphine-xylazine.
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2004, Volume: 35, Issue:3

    Topics: Adrenergic alpha-Agonists; Analgesics, Opioid; Anesthetics, Combined; Animals; Animals, Wild; Antelopes; Carbon Dioxide; Dose-Response Relationship, Drug; Etorphine; Female; Fentanyl; Heart Rate; Hypnotics and Sedatives; Immobilization; Injections, Intramuscular; Male; Oxygen; Respiration; Time Factors; Xylazine

2004
Experience with drugs for capture and restraint of wildebeest, impala, eland and hartebeest in Kenya.
    Journal of wildlife diseases, 1976, Volume: 12, Issue:3

    Topics: Acepromazine; Animals; Animals, Wild; Antelopes; Azaperone; Dose-Response Relationship, Drug; Etorphine; Fentanyl; Hypnotics and Sedatives; Immobilization; Kenya; Xylazine

1976
Agonist-specific regulation of mu-opioid receptor desensitization and recovery from desensitization.
    Molecular pharmacology, 2008, Volume: 73, Issue:4

    Topics: Analgesics, Opioid; Animals; Down-Regulation; Electrophysiology; Enkephalins; Etorphine; Fentanyl; In Vitro Techniques; Male; Naltrexone; Oxymorphone; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu

2008
Thermal, cardiorespiratory and cortisol responses of impala (Aepyceros melampus) to chemical immobilisation with 4 different drug combinations.
    Journal of the South African Veterinary Association, 2008, Volume: 79, Issue:3

    Topics: Acepromazine; Anesthesia; Anesthetics, Combined; Animals; Antelopes; Azaperone; Body Temperature Regulation; Etorphine; Female; Fentanyl; Hydrocortisone; Hypnotics and Sedatives; Immobilization; Respiration; Time Factors; Xylazine

2008
Paradoxical relationship between RAVE (relative activity versus endocytosis) values of several opioid receptor agonists and their liability to cause dependence.
    Acta pharmacologica Sinica, 2010, Volume: 31, Issue:4

    Topics: Analgesics, Opioid; Animals; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Endocytosis; Etorphine; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Morphine; Opioid-Related Disorders; Receptors, Opioid, mu

2010
Modulating micro-opioid receptor phosphorylation switches agonist-dependent signaling as reflected in PKCepsilon activation and dendritic spine stability.
    The Journal of biological chemistry, 2011, Apr-08, Volume: 286, Issue:14

    Topics: Analgesics, Opioid; Animals; Arrestins; beta-Arrestins; Cell Line; Dendritic Spines; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Humans; Mice; Morphine; Phosphorylation; Protein Kinase C-epsilon; Receptors, Opioid, mu; Signal Transduction

2011
Differences in the characteristics of tolerance to μ-opioid receptor agonists in the colon from wild type and β-arrestin2 knockout mice.
    European journal of pharmacology, 2012, Jun-15, Volume: 685, Issue:1-3

    Topics: Analgesics, Opioid; Animals; Arrestins; beta-Arrestins; Colon; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Ileum; Ligands; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Contraction; Receptors, Opioid, mu

2012
Pulmonary gas exchange and acid-base status during immobilisation of black rhinoceroses (
    Journal of the South African Veterinary Association, 2016, Dec-02, Volume: 87, Issue:1

    Topics: Acid-Base Equilibrium; Adrenergic alpha-2 Receptor Agonists; Analgesics, Opioid; Animals; Animals, Wild; Azaperone; Dopamine Antagonists; Etorphine; Female; Fentanyl; Imidazoles; Immobilization; Male; Perissodactyla; Pulmonary Gas Exchange; Xylazine; Zimbabwe

2016
Blood acid-base status in impala (Aepyceros melampus) immobilised and maintained under total intravenous anaesthesia using two different drug protocols.
    BMC veterinary research, 2017, Aug-16, Volume: 13, Issue:1

    Topics: Acid-Base Equilibrium; Anesthesia, Intravenous; Anesthetics, Combined; Anesthetics, Dissociative; Anesthetics, Intravenous; Animals; Antelopes; Etorphine; Fentanyl; Hypnotics and Sedatives; Ketamine; Medetomidine; Propofol

2017
Comparison of thiafentanil-medetomidine to etorphine-medetomidine immobilisation of impalas (
    Journal of the South African Veterinary Association, 2017, Aug-04, Volume: 88, Issue:0

    Topics: Anesthetics, Combined; Animals; Antelopes; Butorphanol; Etorphine; Fentanyl; Hypnotics and Sedatives; Immobilization; Medetomidine

2017
A RETROSPECTIVE COMPARISON OF CHEMICAL IMMOBILIZATION WITH THIAFENTANIL, THIAFENTANIL-AZAPERONE, OR ETORPHINE-ACEPROMAZINE IN CAPTIVE PERSIAN FALLOW DEER (DAMA DAMA MESOPOTAMICA).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2017, Volume: 48, Issue:3

    Topics: Acepromazine; Analgesics, Opioid; Animals; Antipsychotic Agents; Azaperone; Deer; Etorphine; Female; Fentanyl; Hypnotics and Sedatives; Male; Restraint, Physical; Retrospective Studies

2017
Chemical capture of wild swamp buffalo (Bubalus bubalis) in tropical northern Australia using thiafentanil, etorphine and azaperone combinations.
    Australian veterinary journal, 2019, Volume: 97, Issue:1-2

    Topics: Anesthesia; Animals; Animals, Wild; Australia; Azaperone; Buffaloes; Etorphine; Fentanyl; Hypnotics and Sedatives; Immobilization

2019
Do potent immobilising-opioids induce different physiological effects in impala and blesbok?
    Journal of the South African Veterinary Association, 2020, Aug-06, Volume: 91, Issue:0

    Topics: Analgesics, Opioid; Animals; Antelopes; Cross-Over Studies; Etorphine; Female; Fentanyl; Hypnotics and Sedatives; Immobilization; Random Allocation; Species Specificity

2020
Comparison of cardiopulmonary effects of etorphine and thiafentanil administered as sole agents for immobilization of impala (Aepyceros melampus).
    Veterinary anaesthesia and analgesia, 2021, Volume: 48, Issue:1

    Topics: Analgesics, Opioid; Animals; Antelopes; Etorphine; Female; Fentanyl; Immobilization

2021
Comparison of some cardiopulmonary effects of etorphine and thiafentanil during the chemical immobilization of blesbok (Damaliscus pygargus phillipsi).
    Veterinary anaesthesia and analgesia, 2021, Volume: 48, Issue:1

    Topics: Animals; Cross-Over Studies; Etorphine; Female; Fentanyl; Hypnotics and Sedatives; Immobilization

2021
Transdermal penetration behaviour of drugs: CART-clustering, QSPR and selection of model compounds.
    Bioorganic & medicinal chemistry, 2007, Nov-15, Volume: 15, Issue:22

    Topics: Anti-Inflammatory Agents; Cell Membrane Permeability; Cluster Analysis; Drug Evaluation, Preclinical; Humans; Models, Biological; Predictive Value of Tests; Quantitative Structure-Activity Relationship; Regression Analysis; Skin; Skin Absorption

2007