fentanyl and colforsin

fentanyl has been researched along with colforsin in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19901 (10.00)18.7374
1990's4 (40.00)18.2507
2000's3 (30.00)29.6817
2010's2 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Auld, DS; Austin, CP; Huang, R; Moeller, TA; Sakamuru, S; Shinn, P; Shukla, SJ; Vanleer, D; Xia, M1
Gintzler, AR; Xu, H2
Gintzler, AR; Smolens, I; Xu, H1
Butour, JL; Mazarguil, H; Meunier, JC; Moisand, C; Mollereau, C1
Grandy, DK; Hirota, K; Hirst, RA; Lambert, DG; Smart, D1
Carruthers, AM; Feniuk, W; Humphrey, PP; Jarvie, EM; Jenkins, DW; Sellers, LA1
Imanaga, K; Inoue, T; Ogawa, R; Ogura, A; Shiga, T; Wajima, Z; Yoshikawa, T1
David Clark, J; Demirci, H; Gharagozlou, P; Lameh, J1
Chi, ZQ; Liu, JG; Sun, JF; Tao, YM; Wang, YH; Xu, XJ1

Trials

1 trial(s) available for fentanyl and colforsin

ArticleYear
Intravenous colforsin daropate, a water-soluble forskolin derivative, prevents thiamylal-fentanyl-induced bronchoconstriction in humans.
    Critical care medicine, 2002, Volume: 30, Issue:4

    Topics: Adult; Airway Resistance; Anesthesia, Intravenous; Anesthetics, Intravenous; Bronchoconstriction; Bronchodilator Agents; Colforsin; Female; Fentanyl; Hemodynamics; Humans; Infusions, Intravenous; Lung Compliance; Male; Prospective Studies; Thiamylal

2002

Other Studies

9 other study(ies) available for fentanyl and colforsin

ArticleYear
Identification of clinically used drugs that activate pregnane X receptors.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:1

    Topics: Animals; Cell Line, Tumor; Cytochrome P-450 CYP3A; Drug Interactions; Hep G2 Cells; Hepatocytes; Humans; Pharmaceutical Preparations; Pregnane X Receptor; Rats; Receptors, Steroid; Small Molecule Libraries; Species Specificity; Structure-Activity Relationship; Xenobiotics

2011
Opioid enhancement of evoked [Met5]enkephalin release requires activation of cholinergic receptors: possible involvement of intracellular calcium.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Mar-01, Volume: 89, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Atropine; Calcimycin; Calcium; Colforsin; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Methionine; Enkephalins; Evoked Potentials; Fentanyl; Guinea Pigs; Hexamethonium Compounds; In Vitro Techniques; Myenteric Plexus; Naloxone; Pyrrolidines; Receptors, Muscarinic; Receptors, Opioid; Sufentanil

1992
Opioids can produce a concentration-dependent naloxone-reversible enhancement of inhibition of evoked enkephalin release.
    NIDA research monograph, 1990, Volume: 105

    Topics: Analgesics; Animals; Cholera Toxin; Colforsin; Cyclic AMP; Dynorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Methionine; Enkephalins; Fentanyl; Guinea Pigs; In Vitro Techniques; Myenteric Plexus; Naloxone; Narcotics; Parasympatholytics; Sufentanil; Thionucleotides; Virulence Factors, Bordetella

1990
Opioids can enhance and inhibit the electrically evoked release of methionine-enkephalin.
    Brain research, 1989, Dec-11, Volume: 504, Issue:1

    Topics: Action Potentials; Animals; Colforsin; Cyclic AMP; Dynorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Methionine; Enkephalins; Fentanyl; Guinea Pigs; Myenteric Plexus; Naloxone; Sufentanil

1989
Recognition and activation of the opioid receptor-like ORL 1 receptor by nociceptin, nociceptin analogs and opioids.
    European journal of pharmacology, 1997, Feb-19, Volume: 321, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Amino Acid Sequence; Analgesics, Opioid; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Enzyme Inhibitors; Fentanyl; Molecular Sequence Data; Nociceptin; Nociceptin Receptor; Opioid Peptides; Receptors, Opioid

1997
The effects of recombinant rat mu-opioid receptor activation in CHO cells on phospholipase C, [Ca2+]i and adenylyl cyclase.
    British journal of pharmacology, 1997, Volume: 120, Issue:6

    Topics: Adenylyl Cyclases; Animals; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Diprenorphine; Fentanyl; Inositol 1,4,5-Trisphosphate; Rats; Receptors, Opioid, mu; Transfection; Type C Phospholipases

1997
Adenosine A(1) receptor-mediated inhibition of protein kinase A-induced calcitonin gene-related peptide release from rat trigeminal neurons.
    Molecular pharmacology, 2001, Volume: 59, Issue:6

    Topics: Adenosine; Analgesics, Opioid; Animals; Calcitonin Gene-Related Peptide; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Drug Interactions; Fentanyl; Male; Neurons; Phenethylamines; Phosphorylation; Purinergic P1 Receptor Agonists; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Purinergic P1; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Synaptic Vesicles; Trigeminal Nerve

2001
Activity of opioid ligands in cells expressing cloned mu opioid receptors.
    BMC pharmacology, 2003, Jan-04, Volume: 3

    Topics: Azocines; beta-Endorphin; Binding, Competitive; Butorphanol; Cell Line; Colforsin; Cyclic AMP; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Humans; Hydromorphone; Ligands; Morphine; Naltrexone; Phenazocine; Radioligand Assay; Receptors, Opioid, mu; Tritium

2003
Paradoxical relationship between RAVE (relative activity versus endocytosis) values of several opioid receptor agonists and their liability to cause dependence.
    Acta pharmacologica Sinica, 2010, Volume: 31, Issue:4

    Topics: Analgesics, Opioid; Animals; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Endocytosis; Etorphine; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Morphine; Opioid-Related Disorders; Receptors, Opioid, mu

2010