fentanyl and 3-methylfentanyl isothiocyanate

fentanyl has been researched along with 3-methylfentanyl isothiocyanate in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19907 (58.33)18.7374
1990's4 (33.33)18.2507
2000's1 (8.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blalock, JE; Bost, KL; Carr, DJ; DeCosta, BR; Jacobson, AE; Kim, CH; Rice, KC1
Bykov, V; George, C; Jacobson, AE; Kim, CH; Klee, WA; Long, JB; Mattson, MV; Rice, KC; Rothman, RB; Streaty, RA1
Blalock, JE; Carr, DJ; DeCosta, BR; Guarcello, V; Jacobson, AE; Kim, CH; Rice, KC1
Blalock, JE; Bost, KL; Carr, DJ; DeCosta, B; Jacobson, AE; Rice, KC1
Blalock, JE; Carr, DJ; deCosta, B; Jacobson, AE; Kim, CH; Rice, KC1
Burke, TR; Jacobson, AE; Klee, WA; Rice, KC; Simonds, WF1
Burke, TR; Jacobson, AE; Klee, WA; Rice, KC; Silverton, JV; Simonds, WF; Streaty, RA1
Bykov, V; Jacobson, AE; Long, JB; Rice, KC; Rothman, RB1
Chen, C; Claude, PA; Evans, CJ; Law, PY; Liu-Chen, LY; Rice, KC; Yin, J; Yu, L; Zhu, J1
Chen, KX; Chi, ZQ; Ji, RY; Jiang, HL; Rong, SB; Zhu, YC1
Bi-Yi, C; Jie, C; Wen-Qiao, J; Xin-Jian, C; You-Cheng, Z; Zhi-Qiang, C1
Hales, TG; Law, PY; Piros, ET; Prather, PL; Song, L1

Other Studies

12 other study(ies) available for fentanyl and 3-methylfentanyl isothiocyanate

ArticleYear
Anti-opioid receptor antibody recognition of a binding site on brain and leukocyte opioid receptors.
    Neuroendocrinology, 1990, Volume: 51, Issue:5

    Topics: Animals; Antibodies, Monoclonal; Brain; Chromatography, Affinity; Chromatography, Gel; Electrophoresis, Polyacrylamide Gel; Fentanyl; Immunochemistry; Indicators and Reagents; Isothiocyanates; Leukocytes; Membranes; Mice; Mice, Inbred C57BL; Receptors, Opioid; Thiocyanates; Tritium

1990
Probes for narcotic receptor mediated phenomena. 15. (3S,4S)-(+)-trans-3-methylfentanyl isothiocyanate, a potent site-directed acylating agent for the delta opioid receptors in vitro.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:6

    Topics: Acylation; Adenylyl Cyclase Inhibitors; Analgesia; Animals; Brain; Cell Membrane; Chemical Phenomena; Chemistry; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Fentanyl; Glioma; Hybrid Cells; Indicators and Reagents; Ligands; Male; Molecular Structure; Neuroblastoma; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Stereoisomerism; Structure-Activity Relationship; Tumor Cells, Cultured

1989
Opioid receptors on cells of the immune system: evidence for delta- and kappa-classes.
    The Journal of endocrinology, 1989, Volume: 122, Issue:1

    Topics: Animals; Benzeneacetamides; Cell Line; Fentanyl; Indicators and Reagents; Macrophages; Mice; Mice, Inbred C57BL; Naltrexone; Pyrrolidines; Receptors, Opioid

1989
Immunoaffinity-purified opiate receptor specifically binds the delta-class opiate receptor ligand, cis-(+)-3-methylfentanylisothiocyanate, SUPERFIT.
    FEBS letters, 1987, Nov-30, Volume: 224, Issue:2

    Topics: Animals; Cell Line; Chromatography, Affinity; Cross-Linking Reagents; Fentanyl; Immunologic Techniques; Macromolecular Substances; Mice; Molecular Weight; Receptors, Opioid; Receptors, Opioid, delta

1987
Evidence for a delta-class opioid receptor on cells of the immune system.
    Cellular immunology, 1988, Oct-01, Volume: 116, Issue:1

    Topics: Animals; Fentanyl; Humans; Leukocytes; Ligands; Mice; Molecular Weight; Oxidation-Reduction; Receptors, Opioid; Receptors, Opioid, delta; Spleen

1988
Purification of the opiate receptor of NG108-15 neuroblastoma-glioma hybrid cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:15

    Topics: Affinity Labels; Animals; Cell Line; Fentanyl; Glioma; Glycoproteins; Macromolecular Substances; Membrane Proteins; Molecular Weight; Neuroblastoma; Receptors, Opioid; Receptors, Opioid, delta

1985
Probes for narcotic receptor mediated phenomena. 12. cis-(+)-3-Methylfentanyl isothiocyanate, a potent site-directed acylating agent for delta opioid receptors. Synthesis, absolute configuration, and receptor enantioselectivity.
    Journal of medicinal chemistry, 1986, Volume: 29, Issue:6

    Topics: Acylation; Adenylyl Cyclase Inhibitors; Analgesics; Animals; Brain; Enkephalin, Methionine; Fentanyl; In Vitro Techniques; Isothiocyanates; Ligands; Mice; Molecular Conformation; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Stereoisomerism; Tritium; X-Ray Diffraction

1986
Intracerebroventricular administration of superFIT and its enantiomer to rats: evidence for in vivo acylation of [3H]DADL binding sites.
    Neuropeptides, 1987, Volume: 9, Issue:3

    Topics: Acylation; Animals; Cerebral Ventricles; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Fentanyl; Indicators and Reagents; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism

1987
Irreversible binding of cis-(+)-3-methylfentanyl isothiocyanate to the delta opioid receptor and determination of its binding domain.
    The Journal of biological chemistry, 1996, Jan-19, Volume: 271, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; CHO Cells; Cloning, Molecular; Cricetinae; Diprenorphine; Fentanyl; Indicators and Reagents; Kinetics; Mice; Models, Structural; Molecular Sequence Data; Protein Binding; Protein Structure, Secondary; Rats; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Recombinant Fusion Proteins; Sequence Homology, Amino Acid; Transfection

1996
Molecular modeling of interaction between delta opioid receptor and 3-methylfentanylisothiocyanate.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1997, Volume: 18, Issue:3

    Topics: Amino Acid Sequence; Bacteriorhodopsins; Binding Sites; Drug Interactions; Fentanyl; Ligands; Models, Molecular; Molecular Sequence Data; Receptors, Opioid, delta; Sequence Alignment

1997
Analgesic activity and selectivity of isothiocyanate derivatives of fentanyl analogs for opioid receptors.
    Life sciences, 1999, Volume: 65, Issue:15

    Topics: Amides; Analgesics, Opioid; Animals; Fentanyl; Isothiocyanates; Male; Mice; Muscle Contraction; Nociceptors; Pain Measurement; Receptors, Opioid; Receptors, Opioid, delta; Stereoisomerism; Structure-Activity Relationship; Substrate Specificity; Vas Deferens

1999
delta-Opioid receptors are more efficiently coupled to adenylyl cyclase than to L-type Ca(2+) channels in transfected rat pituitary cells.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 295, Issue:2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Alkylating Agents; Analgesics, Opioid; Animals; Barium; Calcium Channels, L-Type; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Heterotrimeric GTP-Binding Proteins; Ion Channels; Naltrexone; Pituitary Gland; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Transfection; Virulence Factors, Bordetella

2000