fenofibrate and sirtinol

fenofibrate has been researched along with sirtinol in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (11.11)29.6817
2010's8 (88.89)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berger, SL; Brent, M; Dang, W; Howitz, K; Jackson, B; Marmorstein, R; Sanders, BD; Schreiber, SL; Taylor, AM1
Altucci, L; Farina, F; Mai, A; Néri, C; Pasco, MY; Rotili, D; Rouleau, GA1
He, B; Huang, W; Li, Y; Xie, T; You, L1
He, B; Huang, W; Li, Y; Liu, J; You, L; Zhu, H1
Forgione, M; Hailu, GS; Mai, A; Robaa, D; Rotili, D; Sippl, W1
Akhmedov, A; Breitenstein, A; Camici, GG; Elliott, PJ; Holy, EW; Lohmann, C; Lüscher, TF; Matter, CM; Spescha, R; Stein, S; Tanner, FC; Westphal, CH1
Li, YJ; Wang, YH; Zheng, GX1
Ji, M; Li, Y; Lin, Q; Lin, R; Ren, F; Wang, W; Zhang, J1
Bai, L; Ji, M; Lin, R; Lu, Y; Qiao, H; Ren, F; Wang, W; Yang, L; Zhang, J1

Reviews

1 review(s) available for fenofibrate and sirtinol

ArticleYear
Lysine Deacetylase Inhibitors in Parasites: Past, Present, and Future Perspectives.
    Journal of medicinal chemistry, 2017, 06-22, Volume: 60, Issue:12

    Topics: Animals; Antiparasitic Agents; Drug Repositioning; Helminth Proteins; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Leishmania; Plasmodium; Protozoan Proteins; Schistosoma; Toxoplasma; Trypanosoma

2017

Other Studies

8 other study(ies) available for fenofibrate and sirtinol

ArticleYear
Identification and characterization of novel sirtuin inhibitor scaffolds.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Drug Evaluation, Preclinical; Enzyme Inhibitors; Fibroblast Growth Factor 6; Fungal Proteins; Humans; Inhibitory Concentration 50; Kinetics; Sirtuins; Structure-Activity Relationship

2009
Characterization of sirtuin inhibitors in nematodes expressing a muscular dystrophy protein reveals muscle cell and behavioral protection by specific sirtinol analogues.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Animals; Animals, Genetically Modified; Benzamides; Caenorhabditis elegans; Cell Movement; Green Fluorescent Proteins; Histone Deacetylase Inhibitors; Muscle Cells; Muscular Dystrophy, Oculopharyngeal; Naphthols; Poly(A)-Binding Protein I; Sirtuins

2010
A FRET-based assay for screening SIRT5 specific modulators.
    Bioorganic & medicinal chemistry letters, 2015, Apr-15, Volume: 25, Issue:8

    Topics: Amino Acid Sequence; Coumarins; Enzyme Assays; Enzyme Inhibitors; Fluorescence Resonance Energy Transfer; Fluorescent Dyes; Kinetics; Molecular Sequence Data; p-Dimethylaminoazobenzene; Peptides; Sirtuins; Substrate Specificity

2015
A FRET-based assay for screening SIRT6 modulators.
    European journal of medicinal chemistry, 2015, Volume: 96

    Topics: Coumarins; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Enzyme Inhibitors; Fluorescence Resonance Energy Transfer; Fluorescent Dyes; Humans; Molecular Structure; Sirtuins; Structure-Activity Relationship

2015
Sirt1 inhibition promotes in vivo arterial thrombosis and tissue factor expression in stimulated cells.
    Cardiovascular research, 2011, Feb-01, Volume: 89, Issue:2

    Topics: Animals; Benzamides; Binding Sites; Cells, Cultured; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelial Cells; Enzyme Activators; Genes, Reporter; Histone Deacetylase Inhibitors; Humans; Mice; Mice, Inbred C57BL; Mice, Knockout; Mitogen-Activated Protein Kinases; Naphthalenes; Naphthols; Promoter Regions, Genetic; Pyrones; Resveratrol; RNA Interference; RNA, Messenger; Sirtuin 1; Stilbenes; Thromboplastin; Thrombosis; Transcription Factor RelA; Transfection

2011
Giardia duodenalis GlSir2.2, homolog of SIRT1, is a nuclear-located and NAD(+)-dependent deacethylase.
    Experimental parasitology, 2016, Volume: 169

    Topics: Amino Acid Sequence; Benzamides; Cell Nucleus; Fluorescent Antibody Technique, Indirect; Giardia lamblia; Group III Histone Deacetylases; Humans; Inhibitory Concentration 50; Naphthalenes; Naphthols; Niacinamide; Phylogeny; Pyrones; Sequence Alignment; Sirtuins

2016
PPARα agonist fenofibrate attenuates TNF-α-induced CD40 expression in 3T3-L1 adipocytes via the SIRT1-dependent signaling pathway.
    Experimental cell research, 2013, Jun-10, Volume: 319, Issue:10

    Topics: 3T3-L1 Cells; Adipocytes; AMP-Activated Protein Kinases; Animals; Benzamides; Blotting, Western; CD40 Antigens; Fenofibrate; Mice; Naphthols; NF-kappa B; Niacinamide; Oxazoles; PPAR alpha; Pyrrolidines; RNA, Messenger; Signal Transduction; Sirtuin 1; Thiocarbamates; Tumor Necrosis Factor-alpha; Tyrosine

2013
The protective effect of fenofibrate against TNF-α-induced CD40 expression through SIRT1-mediated deacetylation of NF-κB in endothelial cells.
    Inflammation, 2014, Volume: 37, Issue:1

    Topics: Acetylation; Antioxidants; Benzamides; CD40 Antigens; Cells, Cultured; Fenofibrate; Human Umbilical Vein Endothelial Cells; Humans; Hypolipidemic Agents; Inflammation; Naphthols; Niacinamide; Oxazoles; PPAR alpha; Pyrrolidines; RNA Interference; RNA, Small Interfering; Signal Transduction; Sirtuin 1; Thiocarbamates; Transcription Factor RelA; Tumor Necrosis Factor-alpha; Tyrosine; Up-Regulation

2014