felodipine and sabinene

felodipine has been researched along with sabinene in 28 studies

Research

Studies (28)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's18 (64.29)18.2507
2000's10 (35.71)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bailey, D; Bergstrand, R; Edgar, B; Johnsson, G; Regårdh, CG1
Edgar, B; Eriksson, UG; Lundahl, J; Miniscalco, A; Regårdh, CG1
Arnold, JM; Bailey, DG; Munoz, C; Spence, JD2
Chayen, R; Rosenthal, T1
Arnold, JM; Bailey, DG; Spence, JD1
Arnold, JM; Bailey, DG; Bend, JR; Spence, JD; Tran, LT2
Edgar, B; Johnsson, G; Lundahl, J; Regårdh, CG2
Abernethy, DR1
Adair, CH; Bailey, DG; Brown, MB; Fontana, RJ; Fortlage, LA; Guo, W; Janardan, SK; Lown, KS; Watkins, PB1
Feldman, EB1
Edgar, B; Johnsson, G; Lundahl, JU; Regårdh, CG1
Arnold, O; Bailey, DG; Malcolm, J; Spence, JD1
Bailey, DG; Bend, JR; Freeman, DJ; Kreeft, JH; Munoz, C1
Menke, J1
Higuchi, S; Kuroda, K; Matsuo, H; Murakami, H; Ohnishi, A; Sata, H; Sawada, Y; Takanaga, H; Urae, A1
Bailey, DG; Carruthers, SG; Dresser, GK1
Bailey, DG; Bend, JR; Dresser, GK; Freeman, DJ; Kreeft, JH; Munoz, C1
Bailey, DG; Malhotra, S; Paine, MF; Watkins, PB1
Hoffmann, R; Krisp, A1
Bailey, DG; Dresser, GK; Wacher, V; Wong, HT; Wong, S1
Bailey, DG; Bend, JR; Dresser, GK1
Bailey, DG; Cillié, D; Cohen, L; Dijkstra, HP; Goosen, TC; He, K; Hollenberg, PF; Rheeders, M; Williams, JA; Woster, PM; Yu, C1
Cao, XM; Chen, QY; Chu, XM; Guo, LQ; Li, JH; Liu, YX; Wang, X; Yamazoe, Y1

Reviews

4 review(s) available for felodipine and sabinene

ArticleYear
Grapefruit juice and drugs. How significant is the interaction?
    Clinical pharmacokinetics, 1994, Volume: 26, Issue:2

    Topics: Beverages; Biological Availability; Citrus; Dihydropyridines; Drug Interactions; Felodipine; Flavanones; Flavonoids; Half-Life; Humans; Nifedipine; Nitrendipine

1994
Grapefruits and drugs: when is statistically significant clinically significant?
    The Journal of clinical investigation, 1997, May-15, Volume: 99, Issue:10

    Topics: Animals; Aryl Hydrocarbon Hydroxylases; Beverages; Citrus; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Felodipine; Humans; Metabolic Clearance Rate; Nifedipine; Oxidoreductases, N-Demethylating; Pharmacokinetics; Smoking

1997
How grapefruit juice potentiates drug bioavailability.
    Nutrition reviews, 1997, Volume: 55, Issue:11 Pt 1

    Topics: Area Under Curve; Beverages; Biological Availability; Calcium Channel Blockers; Citrus; Down-Regulation; Drug Synergism; Felodipine; Humans

1997
Grapefruit juice-drug interactions.
    British journal of clinical pharmacology, 1998, Volume: 46, Issue:2

    Topics: Administration, Oral; Beverages; Biological Availability; Calcium Channel Blockers; Citrus; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Felodipine; Food-Drug Interactions; Humans; Intestine, Small; Mixed Function Oxygenases; Pharmacokinetics

1998

Trials

15 trial(s) available for felodipine and sabinene

ArticleYear
Interaction of citrus juices with felodipine and nifedipine.
    Lancet (London, England), 1991, Feb-02, Volume: 337, Issue:8736

    Topics: Biological Availability; Blood Pressure; Citrus; Drug Interactions; Evaluation Studies as Topic; Felodipine; Heart Rate; Humans; Hypertension; Male; Middle Aged; Nifedipine

1991
Grapefruit juice--felodipine interaction: mechanism, predictability, and effect of naringin.
    Clinical pharmacology and therapeutics, 1993, Volume: 53, Issue:6

    Topics: Adult; Beverages; Biological Availability; Citrus; Drug Interactions; Felodipine; Flavanones; Flavonoids; Humans; Male

1993
Grapefruit juice-felodipine interaction: reproducibility and characterization with the extended release drug formulation.
    British journal of clinical pharmacology, 1995, Volume: 40, Issue:2

    Topics: Adult; Analysis of Variance; Beverages; Calcium Channel Blockers; Citrus; Cross-Over Studies; Delayed-Action Preparations; Felodipine; Food-Drug Interactions; Humans; Linear Models; Male; Reproducibility of Results; White People

1995
Erythromycin-felodipine interaction: magnitude, mechanism, and comparison with grapefruit juice.
    Clinical pharmacology and therapeutics, 1996, Volume: 60, Issue:1

    Topics: Adolescent; Adult; Anti-Bacterial Agents; Beverages; Calcium Channel Blockers; Citrus; Cross-Over Studies; Cytochrome P-450 Enzyme System; Drug Interactions; Erythromycin; Felodipine; Humans; Male

1996
Relationship between time of intake of grapefruit juice and its effect on pharmacokinetics and pharmacodynamics of felodipine in healthy subjects.
    European journal of clinical pharmacology, 1995, Volume: 49, Issue:1-2

    Topics: Adult; Beverages; Blood Pressure; Calcium Channel Blockers; Citrus; Cross-Over Studies; Felodipine; Heart Rate; Humans; Male; Time Factors

1995
Effects of grapefruit juice ingestion--pharmacokinetics and haemodynamics of intravenously and orally administered felodipine in healthy men.
    European journal of clinical pharmacology, 1997, Volume: 52, Issue:2

    Topics: Administration, Oral; Adult; Beverages; Blood Pressure; Calcium Channel Blockers; Citrus; Cross-Over Studies; Drug Interactions; Felodipine; Heart Rate; Hemodynamics; Humans; Injections, Intravenous; Intestinal Absorption; Intestinal Mucosa; Intestines; Liver; Male; Tissue Distribution; Water

1997
The interaction effect of grapefruit juice is maximal after the first glass.
    European journal of clinical pharmacology, 1998, Volume: 54, Issue:1

    Topics: Adult; Beverages; Blood Pressure; Calcium Channel Blockers; Citrus; Cross-Over Studies; Dose-Response Relationship, Drug; Drug Synergism; Felodipine; Heart Rate; Humans; Male

1998
Grapefruit juice-felodipine interaction: effect of naringin and 6',7'-dihydroxybergamottin in humans.
    Clinical pharmacology and therapeutics, 1998, Volume: 64, Issue:3

    Topics: Administration, Oral; Adult; Anti-Arrhythmia Agents; Antioxidants; Area Under Curve; Beverages; Biological Availability; Calcium Channel Blockers; Citrus; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Enzyme Inhibitors; Felodipine; Flavanones; Flavonoids; Food-Drug Interactions; Furocoumarins; Humans; Male; Mixed Function Oxygenases; Reference Values

1998
Pharmacokinetic analysis of felodipine-grapefruit juice interaction based on an irreversible enzyme inhibition model.
    British journal of clinical pharmacology, 2000, Volume: 49, Issue:1

    Topics: Adult; Area Under Curve; Beverages; Biological Availability; Calcium Channel Blockers; Citrus; Computer Simulation; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Enzyme Inhibitors; Felodipine; Food-Drug Interactions; Gastrointestinal Transit; Humans; Intestinal Mucosa; Liver; Male; Metabolic Clearance Rate; Mixed Function Oxygenases; Models, Biological

2000
Grapefruit juice--felodipine interaction in the elderly.
    Clinical pharmacology and therapeutics, 2000, Volume: 68, Issue:1

    Topics: Aged; Aged, 80 and over; Antihypertensive Agents; Area Under Curve; Beverages; Blood Pressure; Citrus; Diastole; Felodipine; Female; Food-Drug Interactions; Half-Life; Heart Rate; Humans; Male; Posture; Reference Values; Systole; Time Factors

2000
Grapefruit-felodipine interaction: effect of unprocessed fruit and probable active ingredients.
    Clinical pharmacology and therapeutics, 2000, Volume: 68, Issue:5

    Topics: Administration, Oral; Adult; Antioxidants; Area Under Curve; Beverages; Citrus; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Delayed-Action Preparations; Drug Interactions; Felodipine; Female; Flavanones; Flavonoids; Furocoumarins; Half-Life; Humans; Male; Mixed Function Oxygenases; Radiation-Sensitizing Agents

2000
Seville orange juice-felodipine interaction: comparison with dilute grapefruit juice and involvement of furocoumarins.
    Clinical pharmacology and therapeutics, 2001, Volume: 69, Issue:1

    Topics: 5-Methoxypsoralen; Administration, Oral; Adult; Antihypertensive Agents; Beverages; Biological Availability; Caco-2 Cells; Citrus; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; DNA, Complementary; Enzyme Activation; Enzyme Inhibitors; Felodipine; Female; Food-Drug Interactions; Furocoumarins; Humans; Male; Methoxsalen; Mixed Function Oxygenases

2001
Evaluation of peppermint oil and ascorbyl palmitate as inhibitors of cytochrome P4503A4 activity in vitro and in vivo.
    Clinical pharmacology and therapeutics, 2002, Volume: 72, Issue:3

    Topics: Administration, Oral; Adolescent; Adult; Area Under Curve; Ascorbic Acid; Beverages; Biological Availability; Citrus; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Enzyme Activation; Enzyme Inhibitors; Felodipine; Female; Humans; Male; Mentha piperita; Microsomes, Liver; Mixed Function Oxygenases; Plant Oils

2002
Bergamottin, lime juice, and red wine as inhibitors of cytochrome P450 3A4 activity: comparison with grapefruit juice.
    Clinical pharmacology and therapeutics, 2003, Volume: 73, Issue:6

    Topics: Adult; Area Under Curve; Beverages; Biotransformation; Calcium Channel Blockers; Citrus; Citrus paradisi; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Drug Interactions; Enzyme Inhibitors; Felodipine; Female; Food-Drug Interactions; Furocoumarins; Half-Life; Humans; Male; Middle Aged; NADP; Radiation-Sensitizing Agents; Wine

2003
Bergamottin contribution to the grapefruit juice-felodipine interaction and disposition in humans.
    Clinical pharmacology and therapeutics, 2004, Volume: 76, Issue:6

    Topics: Adult; Area Under Curve; Biological Availability; Biotransformation; Calcium Channel Blockers; Capsules; Chromatography, High Pressure Liquid; Citrus; Cross-Over Studies; Delayed-Action Preparations; Felodipine; Female; Food-Drug Interactions; Furocoumarins; Humans; Male; Spectrophotometry, Ultraviolet

2004

Other Studies

9 other study(ies) available for felodipine and sabinene

ArticleYear
Acute effects of drinking grapefruit juice on the pharmacokinetics and dynamics of felodipine--and its potential clinical relevance.
    European journal of clinical pharmacology, 1992, Volume: 42, Issue:3

    Topics: Adult; Analysis of Variance; Beverages; Blood Pressure; Citrus; Felodipine; Heart Rate; Humans; Male; Middle Aged

1992
Inhibition of dihydropyridine metabolism in rat and human liver microsomes by flavonoids found in grapefruit juice.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Adult; Aged; Animals; Beverages; Citrus; Dihydropyridines; Felodipine; Flavanones; Flavonoids; Humans; Male; Microsomes, Liver; Middle Aged; Nifedipine; Quercetin; Rats; Rats, Inbred Strains; Stereoisomerism

1992
Interaction of citrus juices with felodipine and nifedipine.
    Lancet (London, England), 1991, Apr-06, Volume: 337, Issue:8745

    Topics: Beverages; Biological Availability; Citrus; Drug Interactions; Felodipine; Humans; Nifedipine

1991
Grapefruit juice interactions with drugs.
    The Medical letter on drugs and therapeutics, 1995, Aug-18, Volume: 37, Issue:955

    Topics: Beverages; Caffeine; Citrus; Cyclosporine; Estrogens; Felodipine; Food-Drug Interactions; Humans; Midazolam; Nifedipine; Terfenadine

1995
Grapefruit juice increases felodipine oral availability in humans by decreasing intestinal CYP3A protein expression.
    The Journal of clinical investigation, 1997, May-15, Volume: 99, Issue:10

    Topics: Administration, Oral; Adult; Aryl Hydrocarbon Hydroxylases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Beverages; Biopsy; Citrus; Colon; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Felodipine; Gene Expression; Humans; Intestinal Mucosa; Intestine, Small; Kinetics; Liver; Male; Mixed Function Oxygenases; Oxidoreductases, N-Demethylating; Reference Values

1997
Grapefruit juice: the untold story.
    South Dakota journal of medicine, 1998, Volume: 51, Issue:11

    Topics: Antihypertensive Agents; Beverages; Calcium Channel Blockers; Citrus; Cyclosporins; Felodipine; Food-Drug Interactions; Humans; Intestine, Small

1998
[Letter concerning the article by E.C.Bornhövd, E.Schuller, T.Bieber, A.Wollenberg: "Immunosuppressive macrolides and their use in dermatology". Der Hautarzt (2000) 51:646-654].
    Der Hautarzt; Zeitschrift fur Dermatologie, Venerologie, und verwandte Gebiete, 2001, Volume: 52, Issue:3

    Topics: Beverages; Calcium Channel Blockers; Citrus; Cyclosporine; Digestive System; Drug Interactions; Felodipine; Humans; Immunosuppressive Agents; Liver; Skin Diseases; Tacrolimus; Xenobiotics

2001
Drug interactions with grapefruit juice.
    Obstetrics and gynecology, 2005, Volume: 105, Issue:2

    Topics: Beverages; Biological Availability; Citrus; Clinical Trials as Topic; Cytochrome P-450 Enzyme System; Drug Interactions; Felodipine; Female; Humans; Male; Pharmaceutical Preparations; Risk Assessment; Sensitivity and Specificity

2005
Different roles of pummelo furanocoumarin and cytochrome P450 3A5*3 polymorphism in the fate and action of felodipine.
    Current drug metabolism, 2007, Volume: 8, Issue:6

    Topics: Adult; Beverages; Blood Pressure; Calcium Channel Blockers; Citrus; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; DNA; Felodipine; Food-Drug Interactions; Furocoumarins; Genotype; Heart Rate; Humans; Hydroxylation; Male; Microsomes, Liver; Molecular Sequence Data; Polymorphism, Genetic; Testosterone

2007